Cell Line : A-549

Cellosaurus Index : CVCL_0023
Cellosaurus ID : A-549

CCLE Name : A549_LUNG
CTRP1 Name , CTRP2 Name , GDSC1 Name , GDSC2 Name : A549

Cancer Type : lung
Dataset : All

Drug Response Information

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Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including cell line name, drug name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Cellosaurus ID Drug Name Original Dataset(s) Min Dose Max Dose Dose-response
A-549 (-)-gallocatechin-3-monogallate CTRP1 0.2890 37.0000
A-549 (5Z)-7-Oxozeaenol GDSC1 0.0391 10.0000
A-549 123138 GDSC2 0.0010 1.0000
A-549 123829 GDSC2 0.0030 3.0000
A-549 150412 GDSC2 0.0030 3.0000
A-549 16-beta-bromoandrosterone CTRP2,CTRP1 0.0011 37.0000
A-549 16,16-dimethylprostaglandin-E2 CTRP1 0.2603 33.3330
A-549 1S,3R-RSL-3 CTRP2 0.0010 33.0000
A-549 2-bromopyruvate CTRP1 0.2603 37.0000
A-549 2-deoxyglucose CTRP1 0.2890 37.0080
A-549 2-fluoropalmitic acid CTRP1 0.2890 37.0000
A-549 2,4-dideoxy-DC-45-A2 CTRP1 0.2603 33.3330
A-549 3-chloro-L-alanine CTRP1 0.2603 33.3330
A-549 3-Cl-AHPC CTRP2 0.0020 66.0000
A-549 4-IPP CTRP1 0.2603 33.3330
A-549 4-methylfasudil CTRP1 0.2603 33.3330
A-549 5-azacytidine GDSC2 0.0200 20.0000
A-549 5-benzyl-9-tert-butyl-paullone CTRP1 0.2603 33.3330
A-549 5-Fluorouracil GDSC1,GDSC2 0.0200 32.0000
A-549 50869 GDSC2 0.0030 3.0000
A-549 6-diazo-5-oxo-L-norleucine CTRP1 0.2603 33.3330
A-549 6-NBDG CTRP1 0.2603 33.3330
A-549 615590 GDSC2 0.0030 3.0000
A-549 630600 GDSC2 0.0030 3.0000
A-549 667880 GDSC2 0.0030 3.0000
A-549 7-nitroindazole CTRP1 0.2603 33.3330
A-549 720427 GDSC2 0.0030 3.0000
A-549 729189 GDSC2 0.0030 3.0000
A-549 741909 GDSC2 0.0010 1.0000
A-549 743380 GDSC2 0.0010 1.0000
A-549 765771 GDSC2 0.0030 3.0000
A-549 776928 GDSC2 0.0300 30.0000
A-549 965-D2 GDSC1 0.0391 10.0000
A-549 968 CTRP2 0.0020 66.0000
A-549 993-D2 GDSC1 0.0391 10.0000
A-549 A-366 GDSC2 0.0100 10.0000
A-549 A-804598 CTRP2 0.0020 66.0000
A-549 A-83-01 GDSC1 0.0781 20.0000
A-549 AA-COCF3 CTRP2,CTRP1 0.0081 270.0000
A-549 ABH CTRP1 0.2890 37.0000
A-549 abiraterone CTRP2 0.0005 17.0000
A-549 ABT-751 CTRP1 0.2603 33.3330
A-549 ABT737 GDSC2,CTRP2,CTRP1 0.0011 37.0000
A-549 AC55649 CTRP2,CTRP1 0.0010 33.3330
A-549 Acetalax GDSC2 0.0300 30.0000
A-549 ACY-1215 GDSC1 0.0781 20.0000
A-549 AEW541 CCLE 0.0025 8.0000
A-549 Afatinib GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 Afuresertib GDSC2 0.0100 10.0000
A-549 AGI-5198 GDSC2 0.0100 10.0000
A-549 AGI-6780 GDSC1,GDSC2 0.0020 10.0000
A-549 AGK-2 GDSC2,CTRP2,CTRP1 0.0010 33.3330
A-549 AICA Ribonucleotide GDSC1 7.8125 2000.0000
A-549 AKT inhibitor VIII GDSC1 0.0100 10.2400
A-549 Alda-1 CTRP1 0.2603 33.3330
A-549 Alectinib GDSC1 0.0200 5.1200
A-549 Alisertib GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 alisertib:navitoclax (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 Alpelisib GDSC2,CTRP2 0.0020 66.0000
A-549 alpha-cyano-4-hydroxycinnamic acid CTRP1 0.2603 33.3330
A-549 alpha-lipoic acid GDSC2 0.1211 121.0000
A-549 AM-580 CTRP2,CTRP1 0.0160 530.0000
A-549 AMG-319 GDSC2 0.0100 10.0000
A-549 Amuvatinib GDSC1 0.0781 20.0000
A-549 apicidin CTRP2 0.0010 33.0000
A-549 Apitolisib GDSC1 0.0781 20.0000
A-549 AR-42 GDSC1 0.0200 5.1200
A-549 Ara-G GDSC1 0.0781 20.0000
A-549 ARRY-520 GDSC1 0.0010 0.2560
A-549 AS601245 GDSC1 0.0312 8.0000
A-549 AS605240 GDSC1 0.0400 20.0000
A-549 ascorbate (vitamin C) GDSC2 2.0011 2000.0000
A-549 ASN 05257430 CTRP2,CTRP1 0.0011 37.0000
A-549 aspirin CTRP1 0.2603 33.3330
A-549 AST-1306 GDSC1 0.0781 20.0000
A-549 AT-406 CTRP2 0.0020 66.0000
A-549 AT-7519 GDSC1 0.0400 10.2400
A-549 AT13148 GDSC2 0.0100 10.0000
A-549 AT7867 GDSC1,CTRP2 0.0020 66.0000
A-549 austocystin D CTRP2,CTRP1 0.0011 37.0000
A-549 Avagacestat GDSC1,GDSC2 0.0100 10.2400
A-549 avrainvillamide CTRP2,CTRP1 0.0010 33.3330
A-549 Axitinib GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 AZ-3146 CTRP2 0.0020 66.0000
A-549 AZ20 GDSC1 0.0391 10.0000
A-549 AZ6102 GDSC2 0.0100 10.0000
A-549 AZ960 GDSC2 0.0100 10.0000
A-549 azacitidine CTRP2 0.0020 66.0000
A-549 AZD-7545 CTRP2,CTRP1 0.0023 74.0000
A-549 AZD1208 GDSC1,GDSC2 0.0100 10.0000
A-549 AZD1332 GDSC1,GDSC2 0.0100 10.0000
A-549 AZD1480 GDSC1 0.0098 2.5000
A-549 AZD2014 GDSC1,GDSC2 0.0100 10.0000
A-549 AZD3514 GDSC1 0.0391 10.0000
A-549 AZD3759 GDSC2 0.0010 1.0000
A-549 AZD4547 GDSC1,GDSC2,CTRP2 0.0010 66.0000
A-549 AZD4877 GDSC1 0.0002 0.6250
A-549 AZD5153 GDSC2 0.0100 10.0000
A-549 AZD5363 GDSC2 0.0100 10.0000
A-549 AZD5438 GDSC1,GDSC2 0.0100 10.0000
A-549 AZD5582 GDSC1,GDSC2 0.0100 10.0000
A-549 AZD5991 GDSC2 0.0100 10.0000
A-549 AZD6094 GDSC1 0.0098 2.5000
A-549 AZD6482 GDSC1,CTRP2 0.0020 66.0000
A-549 AZD6738 GDSC1,GDSC2 0.0100 10.0000
A-549 AZD7762 GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 AZD7969 GDSC1 0.0391 10.0000
A-549 AZD8055 GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 AZD8186 GDSC1,GDSC2 0.0098 10.0000
A-549 AZD8835 GDSC1 0.0391 10.0000
A-549 AZD8931 GDSC1 0.0391 10.0000
A-549 B02 CTRP2 0.0041 130.0000
A-549 BAM7 GDSC1 0.0781 20.0000
A-549 barasertib CTRP2 0.0020 66.0000
A-549 bardoxolone methyl CTRP2 0.0020 66.0000
A-549 batimastat CTRP1 0.2890 37.0000
A-549 Bax channel blocker CTRP2,CTRP1 0.0010 33.3330
A-549 BAY ACCi GDSC1 0.0391 10.0000
A-549 BAY AKT1 GDSC1 0.0391 10.0000
A-549 BAY-61-3606 GDSC1 0.0312 8.0000
A-549 BAY-HDAC11_1 GDSC1 0.0391 10.0000
A-549 BAY-HDAC11_2 GDSC1 0.0391 10.0000
A-549 BAY-HDAC11_4 GDSC1 0.0391 10.0000
A-549 BAY-MPS-combo 2 (paclitaxel 1 uM) GDSC1 0.0039 1.0000
A-549 BAY-MPS-combo-1 (paclitaxel 5 uM) GDSC1 0.0039 1.0000
A-549 BAY-MPS1 GDSC1 0.0117 3.0000
A-549 BDF00022089a GDSC2 0.0050 5.0000
A-549 BDILV000379a GDSC2 0.0050 5.0000
A-549 BDOCA000347a GDSC2 0.0020 2.0000
A-549 BDP-00009066 GDSC2 0.0100 10.0000
A-549 BEC CTRP2,CTRP1 0.0081 270.0000
A-549 Belinostat GDSC1 0.0781 20.0000
A-549 BEN GDSC2 0.0300 30.0000
A-549 bendamustine CTRP2 0.0020 66.0000
A-549 betulinic acid CTRP2 0.0020 66.0000
A-549 Bexarotene GDSC1,CTRP2 0.0020 66.0000
A-549 BI-2536 GDSC2,CTRP2 0.0010 33.0000
A-549 BIBF-1120 GDSC1 0.0781 20.0000
A-549 BIBR-1532 GDSC2,CTRP2 0.0081 270.0000
A-549 Bicalutamide GDSC1 0.0040 10.0000
A-549 birinapant CTRP2 0.0020 66.0000
A-549 bistramide A CTRP1 0.2517 32.2330
A-549 BIX-01294 CTRP2,CTRP1 0.0010 33.3330
A-549 BIX-01338 CTRP1 0.2603 33.3330
A-549 BIX02189 GDSC1 0.0781 20.0000
A-549 blebbistatin CTRP2,CTRP1 0.0041 130.0000
A-549 Bleomycin GDSC1,GDSC2 0.0020 64.0000
A-549 Bleomycin (10 uM) GDSC1 0.0391 10.0000
A-549 Bleomycin (50 uM) GDSC1,GDSC2 0.0400 50.0000
A-549 bleomycin A2 CTRP2 0.0020 66.0000
A-549 BMS-191011 CTRP1 0.2603 33.3330
A-549 BMS-195614 CTRP2 0.0020 66.0000
A-549 BMS-270394 CTRP2 0.0020 66.0000
A-549 BMS-345541 GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 BMS-536924 GDSC1,GDSC2,CTRP2,CTRP1 0.0011 37.0000
A-549 BMS-641988 CTRP1 0.2890 37.0000
A-549 BMS-754807 GDSC1,GDSC2,CTRP2 0.0010 33.0000
A-549 Bortezomib GDSC2,CTRP2,CTRP1 0.0000 33.3330
A-549 Bosutinib GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 bovinocidin CTRP1 0.2603 33.3330
A-549 BPD-00008900 GDSC2 0.0100 10.0000
A-549 BPTES GDSC1 0.0391 10.0000
A-549 BRD-A02303741 CTRP2 0.0017 55.0000
A-549 BRD-A02303741:carboplatin (1:1 mol-mol) CTRP2 0.0020 66.0000
A-549 BRD-A02303741:navitoclax (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 BRD-A71883111 CTRP2 0.0010 33.0000
A-549 BRD-A94377914 CTRP2 0.0010 33.0000
A-549 BRD-K02251932 CTRP2 0.0020 66.0000
A-549 BRD-K02492147 CTRP2 0.0020 66.0000
A-549 BRD-K03536150 CTRP2 0.0020 66.0000
A-549 BRD-K03911514 CTRP2 0.0020 66.0000
A-549 BRD-K04800985 CTRP2 0.0020 66.0000
A-549 BRD-K07442505 CTRP2 0.0020 66.0000
A-549 BRD-K09344309 CTRP2 0.0010 33.0000
A-549 BRD-K09587429 CTRP2 0.0020 66.0000
A-549 BRD-K11533227 CTRP2 0.0020 66.0000
A-549 BRD-K13185470 CTRP2 0.0020 66.0000
A-549 BRD-K13999467 CTRP2 0.0020 66.0000
A-549 BRD-K14844214 CTRP2 0.0020 66.0000
A-549 BRD-K16130065 CTRP2 0.0020 66.0000
A-549 BRD-K16147474 CTRP2 0.0020 66.0000
A-549 BRD-K17060750 CTRP2 0.0020 66.0000
A-549 BRD-K19103580 CTRP2 0.0020 66.0000
A-549 BRD-K20514654 CTRP2 0.0020 66.0000
A-549 BRD-K24690302 CTRP2 0.0020 66.0000
A-549 BRD-K26531177 CTRP2 0.0100 330.0000
A-549 BRD-K27188169 CTRP2 0.0020 66.0000
A-549 BRD-K27188169:navitoclax (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 BRD-K27224038 CTRP2 0.0020 66.0000
A-549 BRD-K27986637 CTRP2 0.0020 66.0000
A-549 BRD-K28456706 CTRP2 0.0020 66.0000
A-549 BRD-K29086754 CTRP2 0.0020 66.0000
A-549 BRD-K29313308 CTRP2 0.0020 66.0000
A-549 BRD-K30019337 CTRP2 0.0020 66.0000
A-549 BRD-K33199242 CTRP2 0.0020 66.0000
A-549 BRD-K34099515 CTRP2 0.0020 66.0000
A-549 BRD-K34222889 CTRP2 0.0020 66.0000
A-549 BRD-K34485477 CTRP2 0.0010 33.0000
A-549 BRD-K35604418 CTRP2 0.0020 66.0000
A-549 BRD-K37390332 CTRP2 0.0010 33.0000
A-549 BRD-K41334119 CTRP2 0.0020 66.0000
A-549 BRD-K41597374 CTRP2 0.0020 66.0000
A-549 BRD-K44224150 CTRP2 0.0010 34.0000
A-549 BRD-K45681478 CTRP2 0.0020 66.0000
A-549 BRD-K48334597 CTRP2 0.0020 66.0000
A-549 BRD-K49290616 CTRP2 0.0020 66.0000
A-549 BRD-K50799972 CTRP2 0.0020 66.0000
A-549 BRD-K51490254 CTRP2 0.0020 66.0000
A-549 BRD-K52037352 CTRP2 0.0020 66.0000
A-549 BRD-K55116708 CTRP2 0.0020 66.0000
A-549 BRD-K55473186 CTRP2 0.0020 66.0000
A-549 BRD-K58730230 CTRP2 0.0020 66.0000
A-549 BRD-K61166597 CTRP2 0.0020 66.0000
A-549 BRD-K63431240 CTRP2 0.0020 66.0000
A-549 BRD-K64610608 CTRP2 0.0010 33.0000
A-549 BRD-K66453893 CTRP2 0.0020 66.0000
A-549 BRD-K66532283 CTRP2 0.0020 66.0000
A-549 BRD-K70511574 CTRP2 0.0020 66.0000
A-549 BRD-K71781559 CTRP2 0.0020 66.0000
A-549 BRD-K71935468 CTRP2 0.0025 83.0000
A-549 BRD-K75293299 CTRP2 0.0020 66.0000
A-549 BRD-K78574327 CTRP2 0.0020 66.0000
A-549 BRD-K79669418 CTRP2 0.0020 66.0000
A-549 BRD-K80183349 CTRP2 0.0020 66.0000
A-549 BRD-K84807411 CTRP2 0.0020 66.0000
A-549 BRD-K85133207 CTRP2 0.0020 66.0000
A-549 BRD-K86535717 CTRP2 0.0020 66.0000
A-549 BRD-K88742110 CTRP2 0.0020 66.0000
A-549 BRD-K92856060 CTRP2 0.0010 33.0000
A-549 BRD-K94991378 CTRP2 0.0025 83.0000
A-549 BRD-K96431673 CTRP2 0.0020 66.0000
A-549 BRD-K96970199 CTRP2 0.0020 66.0000
A-549 BRD-K97651142 CTRP2 0.0020 66.0000
A-549 BRD-K99584050 CTRP2 0.0020 66.0000
A-549 BRD-M00053801 CTRP2 0.0020 66.0000
A-549 BRD1812 CTRP2,CTRP1 0.0020 66.0000
A-549 BRD1835 CTRP2 0.0041 130.0000
A-549 BRD2649 CTRP1 0.2603 33.3330
A-549 BRD4132 CTRP2 0.0049 160.0000
A-549 BRD4770 CTRP2 0.0010 33.0000
A-549 BRD55319 CTRP2,CTRP1 0.0011 37.0000
A-549 BRD6340 CTRP2 0.0010 33.0000
A-549 BRD63610 CTRP1 0.2603 33.3330
A-549 BRD6368 CTRP1 0.2603 33.3330
A-549 BRD6430 CTRP2 0.0010 33.0000
A-549 BRD7137 CTRP1 0.2603 33.3330
A-549 BRD8899 CTRP2 0.0010 33.0000
A-549 BRD8958 CTRP2,CTRP1 0.0020 66.0000
A-549 BRD9647 CTRP2 0.0010 33.0000
A-549 BRD9786 CTRP1 0.2603 33.3330
A-549 BRD9876 CTRP2 0.0041 130.0000
A-549 brefeldin A CTRP2,CTRP1 0.0011 37.0000
A-549 brivanib CTRP2 0.0020 66.0000
A-549 Brivanib, BMS-540215 GDSC1 0.0781 20.0000
A-549 Bromosporine GDSC2 0.0020 2.0000
A-549 Bryostatin 1 GDSC1 0.0000 0.0080
A-549 Buparlisib GDSC2 0.0100 10.0000
A-549 BX-912 GDSC1 0.0400 10.2400
A-549 BX795 GDSC1 0.0195 5.0000
A-549 C-75 GDSC1 0.0781 20.0000
A-549 C6-ceramide CTRP2 0.0020 66.0000
A-549 Cabozantinib GDSC1,CTRP2 0.0020 66.0000
A-549 Camptothecin GDSC2 0.0001 0.1000
A-549 canertinib CTRP2 0.0020 66.0000
A-549 CAP-232, TT-232, TLN-232 GDSC1 0.0781 20.0000
A-549 Capivasertib GDSC1 0.1172 30.0000
A-549 capsaicin CTRP1 0.2603 33.3330
A-549 Carboplatin CTRP2 0.0020 66.0000
A-549 carboplatin:etoposide (40:17 mol-mol) CTRP2 0.0014 47.0000
A-549 carboplatin:UNC0638 (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 Carmustine GDSC2 0.0300 30.0000
A-549 CAY10566 GDSC1 0.0100 2.5600
A-549 CAY10576 CTRP2 0.0020 66.0000
A-549 CAY10594 CTRP2,CTRP1 0.0020 66.0000
A-549 CAY10603 GDSC1 0.0781 20.0000
A-549 CAY10618 CTRP2 0.0010 33.0000
A-549 CCT-018159 GDSC1 0.0391 10.0000
A-549 CCT007093 GDSC1,GDSC2 0.0100 10.0000
A-549 CCT036477 CTRP2 0.0010 33.0000
A-549 CCT245232 GDSC1 0.0008 0.2000
A-549 CCT245467 GDSC1 0.0008 0.2000
A-549 CD-1530 CTRP2,CTRP1 0.0041 130.0000
A-549 CD-437 CTRP2,CTRP1 0.0011 37.0000
A-549 CD532 GDSC1 0.0200 5.1200
A-549 CDK9_5038 GDSC2 0.0030 3.0000
A-549 CDK9_5576 GDSC2 0.0100 10.0000
A-549 Cediranib GDSC2 0.0100 10.0000
A-549 ceranib-2 CTRP2 0.0020 66.0000
A-549 cerulenin CTRP2,CTRP1 0.0045 150.0000
A-549 Cetuximab GDSC1 0.2570 65.8000
A-549 Ch-55 CTRP2 0.0020 66.0000
A-549 CHEMBL1222381 CTRP2,CTRP1 0.0081 270.0000
A-549 CHEMBL374350 CTRP2,CTRP1 0.0010 33.3330
A-549 CHEMBL399379 CTRP1 0.2603 33.3330
A-549 CHIR-99021 GDSC1,CTRP2 0.0024 80.0000
A-549 chlorambucil CTRP2 0.0081 270.0000
A-549 CHM-1 CTRP2 0.0005 16.0000
A-549 CI-1033 GDSC1 0.0781 20.0000
A-549 CI-1040 GDSC1 0.0391 10.0000
A-549 CI-976 CTRP2,CTRP1 0.0081 270.0000
A-549 ciclopirox CTRP2 0.0020 66.0000
A-549 ciclosporin CTRP2,CTRP1 0.0010 33.3330
A-549 CID-5951923 CTRP2 0.0020 66.0000
A-549 CIL41 CTRP2 0.0049 160.0000
A-549 CIL55 CTRP2 0.0003 10.0000
A-549 CIL55A CTRP2 0.0024 80.0000
A-549 CIL56 CTRP2 0.0001 2.5000
A-549 CIL70 CTRP2 0.0012 40.0000
A-549 cimetidine CTRP2 0.0081 270.0000
A-549 Cisplatin GDSC1,GDSC2 0.0040 10.0000
A-549 clofarabine CTRP2 0.0020 66.0000
A-549 COL-3 CTRP2 0.0020 66.0000
A-549 Compound 10b CTRP1 0.2890 37.0000
A-549 Compound 110 CTRP1 0.2890 37.0000
A-549 Compound 12 CTRP1 0.2890 37.0000
A-549 Compound 1541A CTRP2,CTRP1 0.0011 37.0000
A-549 compound 1B CTRP2 0.0020 66.0000
A-549 Compound 2 CTRP1 0.2603 33.3330
A-549 Compound 23 citrate CTRP2,CTRP1 0.0010 33.3330
A-549 Compound 4 CTRP1 0.2603 33.3330
A-549 Compound 44 CTRP1 0.2603 33.3330
A-549 Compound 7d-cis CTRP2,CTRP1 0.0010 33.3330
A-549 CP466722 GDSC1 0.0625 16.0000
A-549 CP724714 GDSC1 0.0400 10.2400
A-549 CPI-613 GDSC1 1.0000 256.0000
A-549 CPI-637 GDSC2 0.0100 10.0000
A-549 CR-1-31B CTRP2 0.0010 33.0000
A-549 Crizotinib GDSC2,CTRP2,CCLE 0.0010 66.0000
A-549 crizotinib:PLX-4032 (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 CRT0105446 GDSC1 0.0391 10.0000
A-549 CRT0105950 GDSC1 0.0391 10.0000
A-549 CRT0160829 GDSC1 0.0781 20.0000
A-549 CT7033-2 GDSC2 0.0100 10.0000
A-549 cucurbitacin I CTRP2 0.0010 33.0000
A-549 CUDC-101 GDSC1 0.0200 5.1200
A-549 curcumin CTRP2 0.0051 170.0000
A-549 CX-5461 GDSC1 0.0400 10.2400
A-549 cyanoquinoline 11 CTRP2,CTRP1 0.0041 130.0000
A-549 Cyclophosphamide GDSC2,CTRP2 0.0041 130.0000
A-549 Cytarabine GDSC1,GDSC2 0.0020 2.0000
A-549 cytarabine hydrochloride CTRP2 0.0020 66.0000
A-549 cytochalasin B CTRP2,CTRP1 0.0010 33.3330
A-549 cytosporone B CTRP1 0.2603 33.3330
A-549 CZC24832 GDSC2 0.0100 10.0000
A-549 Dabrafenib GDSC1,GDSC2 0.0100 10.0000
A-549 Dacarbazine GDSC2,CTRP2 0.0020 66.0000
A-549 Dacinostat GDSC1 0.0040 1.0240
A-549 Dactinomycin GDSC2 0.0000 0.8000
A-549 Dactolisib GDSC1,GDSC2,CTRP2 0.0003 17.0000
A-549 dalcetrapib CTRP1 0.2587 33.1000
A-549 Daporinad GDSC1,GDSC2,CTRP2,CTRP1 0.0000 33.3330
A-549 darinaparsin CTRP2 0.0010 33.0000
A-549 Dasatinib GDSC2,CTRP2 0.0010 66.0000
A-549 DBeQ CTRP2 0.0020 66.0000
A-549 DC-45-A2 CTRP1 0.2890 37.0000
A-549 Decitabine CTRP2 0.0020 66.0000
A-549 decitabine:carboplatin (1:1 mol-mol) CTRP2 0.0020 66.0000
A-549 decitabine:navitoclax (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 dexamethasone CTRP2,CTRP1 0.0010 33.3330
A-549 DG-041 CTRP1 0.2603 33.3330
A-549 dichloroacetic acid CTRP1 0.2603 33.3330
A-549 Dihydrorotenone GDSC2 0.0010 1.0000
A-549 Dinaciclib GDSC2 0.0010 1.0000
A-549 DL-TBOA CTRP1 0.2603 33.3330
A-549 DMOG GDSC1 15.6250 4000.0000
A-549 Docetaxel GDSC1,GDSC2 0.0000 3.0000
A-549 docetaxel:tanespimycin (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 Doramapimod GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 Doxorubicin GDSC1,CTRP2 0.0020 66.0000
A-549 doxorubicin:navitoclax (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 Dyrk1b_0191 GDSC1 0.0391 10.0000
A-549 eEF2K Inhibitor, A-484954 GDSC1 0.0781 20.0000
A-549 eflornithine CTRP1 0.2890 37.0000
A-549 Eg5_9814 GDSC2 0.0001 0.1000
A-549 EHT-1864 GDSC1,GDSC2 0.0100 10.0000
A-549 ELCPK CTRP2 0.0000 0.4000
A-549 Elephantin GDSC2 0.0200 20.0000
A-549 Elesclomol GDSC1 0.0008 0.2000
A-549 elocalcitol CTRP2 0.0020 66.0000
A-549 Embelin GDSC1 0.1250 32.0000
A-549 Entinostat GDSC2,CTRP2 0.0020 66.0000
A-549 Entospletinib GDSC2 0.0100 10.0000
A-549 Enzastaurin GDSC1 0.0400 20.0000
A-549 EphB4_9721 GDSC1 0.0391 10.0000
A-549 epigallocatechin-3-monogallate CTRP2 0.0090 300.0000
A-549 Epirubicin GDSC2 0.0010 1.0000
A-549 Epothilone B GDSC1 0.0001 0.0320
A-549 EPZ004777 GDSC2 0.0100 10.0000
A-549 EPZ5676 GDSC2 0.0100 10.0000
A-549 erastin CTRP2 0.0020 66.0000
A-549 ERK_2440 GDSC2 0.0100 10.0000
A-549 ERK_6604 GDSC2 0.0100 10.0000
A-549 Erlotinib GDSC2,CTRP2,CCLE 0.0020 66.0000
A-549 erlotinib:PLX-4032 (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 ethylidene glucose CTRP1 0.2603 33.3330
A-549 etomoxir CTRP2,CTRP1 0.0090 300.0000
A-549 Etoposide GDSC1,CTRP2 0.0009 28.0000
A-549 ETP-45835 GDSC1 0.0781 20.0000
A-549 ETP-46464 CTRP2 0.0020 66.0000
A-549 fatostatin CTRP1 0.2603 33.3330
A-549 Fedratinib GDSC1,CTRP2,CTRP1 0.0011 37.0000
A-549 FEN1_3940 GDSC1 0.0391 10.0000
A-549 FGFR_0939 GDSC1 0.0098 2.5000
A-549 FGFR_3831 GDSC1 0.0391 10.0000
A-549 FGIN-1-27 CTRP2 0.0010 33.0000
A-549 FH535 GDSC1 0.1250 32.0000
A-549 fingolimod CTRP2 0.0020 66.0000
A-549 Flavopiridol GDSC1 0.0100 2.5600
A-549 Fludarabine GDSC2 0.0200 20.0000
A-549 fluoropyruvate CTRP1 0.2890 37.0000
A-549 fluorouracil CTRP2 0.0041 130.0000
A-549 fluvastatin CTRP2 0.0020 66.0000
A-549 FMK GDSC1 0.0400 20.0000
A-549 FMK-PA CTRP1 0.2890 37.0000
A-549 Foretinib GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 fosfomycin CTRP1 0.2603 33.3330
A-549 FQI-1 CTRP2 0.0010 33.0000
A-549 FQI-2 CTRP2 0.0010 33.0000
A-549 FR-180204 GDSC1 0.0781 20.0000
A-549 FS106 GDSC1 0.0391 10.0000
A-549 FS112 GDSC1 0.0195 10.0000
A-549 FSC231 CTRP2 0.0081 270.0000
A-549 FTI-277 GDSC1 0.0040 1.0240
A-549 FTY-720 GDSC1 0.0781 20.0000
A-549 Fulvestrant GDSC1,GDSC2 0.0010 10.0000
A-549 fumagillol CTRP1 0.2603 33.3330
A-549 fumonisin B1 CTRP2 0.0150 500.0000
A-549 FY012 GDSC1 0.0391 10.0000
A-549 FY026 GDSC1 0.0391 10.0000
A-549 FY069 GDSC1 0.0391 10.0000
A-549 Gallibiscoquinazole GDSC2 0.0010 1.0000
A-549 GANT-61 CTRP2 0.0020 66.0000
A-549 GDC-0879 CTRP2 0.0020 66.0000
A-549 GDC0810 GDSC2 0.0100 10.0000
A-549 Gefitinib GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 Gemcitabine GDSC1,GDSC2,CTRP2,CTRP1 0.0001 37.0000
A-549 Genentech Cpd 10 GDSC1 0.0400 10.2400
A-549 glibenclamide CTRP1 0.2603 33.3330
A-549 glutathione GDSC2 0.6403 640.0000
A-549 Gly-Gly-PALO CTRP1 0.2603 33.3330
A-549 GMX-1778 CTRP2,CTRP1 0.0000 33.3330
A-549 GNE-317 GDSC2 0.0100 10.0000
A-549 gossypol CTRP2,CTRP1 0.0011 37.0000
A-549 GSK-3 inhibitor IX CTRP2 0.0020 66.0000
A-549 GSK-J4 GDSC1 0.1172 30.0000
A-549 GSK-LSD1 GDSC2 0.0010 1.0000
A-549 GSK-LSD1-2HCl GDSC2 0.0010 1.0000
A-549 GSK1059615 GDSC1,CTRP2 0.0010 33.0000
A-549 GSK1070916 GDSC1 0.0100 10.2400
A-549 GSK1904529A GDSC1,GDSC2 0.0040 10.0000
A-549 GSK2110183B GDSC2 0.0030 3.0000
A-549 GSK2256098C GDSC2 0.0030 3.0000
A-549 GSK2276186C GDSC2 0.0100 10.0000
A-549 GSK2578215A GDSC2 0.0100 10.0000
A-549 GSK2606414 GDSC2 0.0100 10.0000
A-549 GSK2636771 CTRP2 0.0020 66.0000
A-549 GSK269962A GDSC1 0.0195 5.0000
A-549 GSK2801 GDSC2 0.0100 10.0000
A-549 GSK2830371 GDSC2 0.0100 10.0000
A-549 GSK2830371A GDSC2 0.0030 10.0000
A-549 GSK3337463A GDSC2 0.0100 10.0000
A-549 GSK343 GDSC2 0.0010 10.0000
A-549 GSK4112 CTRP2 0.0020 66.0000
A-549 GSK429286A GDSC1 0.0400 20.0000
A-549 GSK461364 CTRP2 0.0020 66.0000
A-549 GSK591 GDSC2 0.0100 10.0000
A-549 GSK626616AC GDSC2 0.0001 0.1000
A-549 GSK650394 GDSC1 0.0625 16.0000
A-549 GSK690693 GDSC1 0.0400 10.2400
A-549 GW-2580 GDSC1 0.0781 20.0000
A-549 GW-405833 CTRP2,CTRP1 0.0041 130.0000
A-549 GW441756 GDSC1,GDSC2 0.0020 2.0000
A-549 GW843682X CTRP2,CTRP1 0.0010 33.3330
A-549 HBX-41108 CTRP2 0.0020 66.0000
A-549 HC-067047 CTRP2 0.0020 66.0000
A-549 HG-5-113-01 GDSC1 0.0391 10.0000
A-549 HG-5-88-01 GDSC1 0.0391 10.0000
A-549 HG-6-71-01 GDSC1 0.0391 10.0000
A-549 HG6-64-1 GDSC1 0.0200 5.1200
A-549 HKMTI-1-005 GDSC2 0.0100 10.0000
A-549 HLI 373 CTRP2 0.0010 33.0000
A-549 hyperforin CTRP2 0.0020 66.0000
A-549 I-BET-762 GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 I-BET151 GDSC1,CTRP2 0.0020 66.0000
A-549 I-BRD9 GDSC2 0.0100 10.0000
A-549 I-CBP112 GDSC1 0.0391 10.0000
A-549 IAP_5620 GDSC1,GDSC2 0.0100 10.0000
A-549 IAP_7638 GDSC1 0.0391 10.0000
A-549 Ibrutinib GDSC2,CTRP2 0.0020 66.0000
A-549 IC-87114 GDSC1,CTRP2 0.0020 66.0000
A-549 ICL-SIRT078 GDSC2 0.0100 10.0000
A-549 ICL1100013 GDSC1 0.0781 20.0000
A-549 idarubicin CTRP1 0.2603 33.3330
A-549 Idelalisib GDSC1,CTRP2 0.0020 66.0000
A-549 ifosfamide CTRP2 0.0020 66.0000
A-549 IGF1R_3801 GDSC2 0.0100 10.0000
A-549 IGFR_3801 GDSC1 0.0391 10.0000
A-549 Imatinib CTRP2 0.0020 66.0000
A-549 IMD-0354 GDSC1 0.0781 20.0000
A-549 importazole CTRP2 0.0061 200.0000
A-549 indisulam CTRP2,CTRP1 0.0010 33.3330
A-549 IOX2 GDSC1 0.0004 0.1000
A-549 IPA-3 GDSC1 0.1250 32.0000
A-549 Ipatasertib GDSC2 0.0100 10.0000
A-549 IPR-456 CTRP2 0.0020 66.0000
A-549 IRAK4_4710 GDSC2 0.0100 10.0000
A-549 Irinotecan GDSC2,CCLE 0.0025 10.0000
A-549 iso-DC-45-A2 CTRP1 0.2603 33.3330
A-549 isoevodiamine CTRP2 0.0010 33.0000
A-549 isoliquiritigenin CTRP2 0.0010 33.0000
A-549 isonicotinohydroxamic acid CTRP2 0.0010 33.0000
A-549 ISOX CTRP2 0.0010 33.0000
A-549 ISOX:bortezomib (250:1 mol-mol) CTRP2 0.0005 17.0000
A-549 Ispinesib Mesylate GDSC1 0.0005 0.1280
A-549 itraconazole CTRP2,CTRP1 0.0005 33.3330
A-549 IU1 CTRP2 0.0020 66.0000
A-549 IWP-2 GDSC2 0.0010 1.0000
A-549 JAK_8517 GDSC2 0.0100 10.0000
A-549 JAK1_3715 GDSC1 0.0391 10.0000
A-549 JAK1_8709 GDSC2 0.0100 10.0000
A-549 JAK3_7406 GDSC1 0.0391 10.0000
A-549 JNJ38877605 GDSC1 0.0781 20.0000
A-549 JNK Inhibitor VIII GDSC1,GDSC2 0.0100 10.0000
A-549 JNK-9L GDSC1 0.0200 5.1200
A-549 JQ-1:carboplatin (1:1 mol-mol) CTRP2 0.0020 66.0000
A-549 JQ-1:MK-0752 (1:1 mol-mol) CTRP2 0.0020 66.0000
A-549 JQ-1:navitoclax (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 JQ-1:UNC0638 (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 JQ-1:vorinostat (2:1 mol-mol) CTRP2 0.0015 50.0000
A-549 JQ1 GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 JQ12 GDSC1 0.0200 5.1200
A-549 JW-480 CTRP2 0.0020 66.0000
A-549 JW-55 CTRP2 0.0020 66.0000
A-549 JW-7-24-1 GDSC1 0.0400 10.2400
A-549 JW-74 CTRP2 0.0020 66.0000
A-549 JZL-184 CTRP1 0.2890 37.0000
A-549 kb NB 142-70 GDSC1 0.0781 20.0000
A-549 KH-CB19 CTRP2 0.0005 17.0000
A-549 KHS101 CTRP2 0.0020 66.0000
A-549 Ki8751 CTRP2 0.0020 66.0000
A-549 KIN001-042 GDSC1 0.0400 10.2400
A-549 KIN001-236 GDSC1 0.0400 10.2400
A-549 KIN001-244 GDSC1 0.0781 20.0000
A-549 KIN001-260 GDSC1 0.0781 20.0000
A-549 KIN001-266 GDSC1 0.0781 20.0000
A-549 KIN001-270 GDSC1 0.0781 20.0000
A-549 kinetin riboside CTRP1 0.2603 33.3330
A-549 Ko-143 CTRP2,CTRP1 0.0041 130.0000
A-549 Kobe2602 GDSC1 0.0781 20.0000
A-549 KPT185 CTRP2 0.0020 66.0000
A-549 KRAS (G12C) Inhibitor-12 GDSC2 0.0200 20.0000
A-549 KU 0060648 CTRP2 0.0010 33.0000
A-549 KU-0063794 CTRP2 0.0020 66.0000
A-549 KU-55933 GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 KU-60019 GDSC1,CTRP2 0.0020 66.0000
A-549 KW-2449 CTRP2 0.0020 66.0000
A-549 KX2-391 CTRP2 0.0020 66.0000
A-549 L-685458 CTRP2,CTRP1,CCLE 0.0011 37.0000
A-549 L-Oxonoreleagnine GDSC2 0.0030 3.0000
A-549 Lapatinib GDSC2,CTRP2,CCLE 0.0020 66.0000
A-549 LBH-589 CTRP2 0.0020 66.0000
A-549 LBW242 CCLE 0.0025 8.0000
A-549 LCL161 GDSC1,GDSC2 0.0100 10.0000
A-549 LDN-193189 GDSC1,CTRP1 0.0400 33.3330
A-549 LE-135 CTRP2,CTRP1 0.0020 66.0000
A-549 Leflunomide GDSC2 0.1001 100.0000
A-549 Lenalidomide GDSC1,GDSC2,CTRP1 0.0100 37.0000
A-549 Lenvatinib CTRP2 0.0020 66.0000
A-549 leptomycin B CTRP2 0.0020 66.0000
A-549 Lestaurtinib GDSC1,GDSC2 0.0020 2.0000
A-549 leucascandrolide A CTRP1 0.2603 33.3330
A-549 LFM-A13 GDSC1 0.0625 16.0000
A-549 LGK974 GDSC1,GDSC2 0.0050 10.0000
A-549 LIMK1 inhibitor BMS4 GDSC1 0.0781 20.0000
A-549 Linifanib GDSC1,CTRP2 0.0020 66.0000
A-549 Linsitinib GDSC1,GDSC2,CTRP2 0.0010 33.0000
A-549 LJI308 GDSC2 0.0100 10.0000
A-549 LMB_AB1 GDSC2 0.0100 10.0000
A-549 LMB_AB2 GDSC2 0.0100 10.0000
A-549 LMB_AB3 GDSC2 0.0100 10.0000
A-549 LMP744 GDSC2 0.0030 3.0000
A-549 lomeguatrib CTRP2 0.0020 66.0000
A-549 lonidamine CTRP1 0.2890 37.0000
A-549 losartan CTRP1 0.2603 33.3330
A-549 lovastatin acid CTRP2,CTRP1 0.0041 130.0000
A-549 LRRK2-IN-1 CTRP2 0.0020 66.0000
A-549 Luminespib GDSC1,GDSC2 0.0003 1.0000
A-549 LY-2157299 CTRP2 0.0020 66.0000
A-549 LY-2183240 CTRP2,CTRP1 0.0010 33.3330
A-549 LY-2365109 CTRP1 0.2603 33.3330
A-549 LY2109761 GDSC2 0.0100 10.0000
A-549 m-3M3-FBS CTRP1 0.2603 33.3330
A-549 manumycin A CTRP2 0.0009 30.0000
A-549 maraviroc CTRP1 0.2603 33.3330
A-549 marinopyrrole A CTRP2 0.0020 66.0000
A-549 Masitinib GDSC1,CTRP2 0.0020 66.0000
A-549 MCT1_6447 GDSC1 0.0391 10.0000
A-549 MCT4_1422 GDSC1 0.0391 10.0000
A-549 Mdivi-1 CTRP2 0.0020 66.0000
A-549 Merck60 CTRP2,CTRP1 0.0010 33.3330
A-549 MetAP2 Inhibitor, A832234 GDSC1 0.0100 2.5600
A-549 Methotrexate GDSC1,GDSC2,CTRP2 0.0008 66.0000
A-549 methylstat CTRP2 0.0020 66.0000
A-549 MG-132 GDSC2 0.0156 4.0000
A-549 MGCD-265 CTRP2 0.0020 66.0000
A-549 MI-1 CTRP2 0.0010 33.0000
A-549 Midostaurin GDSC1 0.0020 0.5120
A-549 MIM1 GDSC1,GDSC2 0.0100 40.0000
A-549 MIRA-1 GDSC2,CTRP2 0.0020 66.0000
A-549 Mirin GDSC1,GDSC2 0.1001 100.0000
A-549 mitomycin CTRP2 0.0015 50.0000
A-549 Mitomycin-C GDSC1 0.0625 16.0000
A-549 Mitoxantrone GDSC2 0.0030 3.0000
A-549 MK-0752 CTRP2 0.0020 66.0000
A-549 MK-1775 GDSC2,CTRP2,CTRP1 0.0010 33.3330
A-549 MK-2206 GDSC1,GDSC2,CTRP2 0.0010 33.0000
A-549 MK-591 CTRP1 0.2603 33.3330
A-549 MK-8776 GDSC2 0.0050 5.0000
A-549 ML006 CTRP2,CTRP1 0.0160 530.0000
A-549 ML007 CTRP1 0.2890 37.0000
A-549 ML013 CTRP1 0.2603 33.3330
A-549 ML030 CTRP2,CTRP1 0.0020 66.0000
A-549 ML037 CTRP1 0.2603 33.3330
A-549 ML038 CTRP1 0.2603 33.3330
A-549 ML039 CTRP1 0.2603 33.3330
A-549 ML050 CTRP2,CTRP1 0.0020 66.0000
A-549 ML101 CTRP1 0.2890 37.0000
A-549 ML162 CTRP2 0.0010 33.0000
A-549 ML203 CTRP2,CTRP1 0.0011 37.0000
A-549 ML210 CTRP2 0.0010 33.0000
A-549 ML239 CTRP2 0.0020 66.0000
A-549 ML258 CTRP2 0.0020 66.0000
A-549 ML311 CTRP2 0.0010 66.0000
A-549 ML312 CTRP2 0.0020 66.0000
A-549 ML320 CTRP2 0.0020 66.0000
A-549 ML323 GDSC2 0.0200 20.0000
A-549 ML334 diastereomer CTRP2 0.0041 130.0000
A-549 MLN2238 CTRP2 0.0010 33.0000
A-549 MN-64 GDSC2 0.0100 10.0000
A-549 momelotinib CTRP2 0.0020 66.0000
A-549 Motesanib GDSC1,GDSC2 0.0078 10.0000
A-549 MPS-1-IN-1 GDSC1 0.0781 20.0000
A-549 Mycophenolic acid GDSC2 0.0100 10.0000
A-549 myricetin CTRP2 0.0020 66.0000
A-549 myriocin CTRP2 0.0010 33.0000
A-549 N-acetyl cysteine GDSC2 2.0011 2000.0000
A-549 N-oxalyl-D-phenylalanine CTRP1 0.2603 33.3330
A-549 N22899-6-C1 GDSC1 0.0391 10.0000
A-549 N23918-95-7 GDSC1 0.0391 10.0000
A-549 N24798-49-A1 GDSC1 0.0391 10.0000
A-549 N25720-51-A1 GDSC2 0.0100 10.0000
A-549 N27922-53-1 GDSC2 0.0100 10.0000
A-549 N29087-69-1 GDSC2 0.0100 10.0000
A-549 N30652-18-1 GDSC2 0.0100 10.0000
A-549 N5-iminoethyl-L-ornithine CTRP1 0.2603 33.3330
A-549 N9-isopropylolomoucine CTRP2 0.0120 400.0000
A-549 nakiterpiosin CTRP2,CTRP1 0.0010 33.3330
A-549 narciclasine CTRP2 0.0010 33.0000
A-549 Navitoclax GDSC1,GDSC2,CTRP2,CTRP1 0.0010 33.3330
A-549 navitoclax:birinapant (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 navitoclax:gemcitabine (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 navitoclax:MST-312 (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 navitoclax:piperlongumine (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 navitoclax:pluripotin (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 navitoclax:PLX-4032 (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 navitoclax:sorafenib (1:1 mol-mol) CTRP2 0.0015 50.0000
A-549 necrostatin-1 CTRP2,CTRP1 0.0160 530.0000
A-549 necrostatin-7 CTRP2 0.0020 66.0000
A-549 necrosulfonamide CTRP2 0.0020 66.0000
A-549 Nelarabine GDSC2,CTRP2 0.0020 66.0000
A-549 neopeltolide CTRP2,CTRP1 0.0010 33.3330
A-549 neratinib CTRP2 0.0010 33.0000
A-549 NG-25 GDSC1 0.0391 10.2400
A-549 niclosamide CTRP2 0.0010 33.0000
A-549 nifedipine CTRP1 0.2603 33.3330
A-549 Nilotinib GDSC1,GDSC2,CTRP2,CCLE 0.0020 66.0000
A-549 nintedanib CTRP2 0.0020 66.0000
A-549 Niraparib GDSC2 0.0100 10.0000
A-549 NPC-26 CTRP2 0.0012 40.0000
A-549 NPK76-II-72-1 GDSC1 0.0400 10.2400
A-549 NSC 74859 CTRP2,CTRP1 0.0160 530.0000
A-549 NSC-207895 GDSC1 0.0781 20.0000
A-549 NSC-87877 GDSC1 0.0625 16.0000
A-549 NSC23766 CTRP2,CTRP1 0.0160 530.0000
A-549 NSC30930 CTRP2 0.0020 66.0000
A-549 NSC319726 GDSC1 0.0010 0.2560
A-549 NSC48300 CTRP2 0.0020 66.0000
A-549 NSC632839 CTRP2,CTRP1 0.0010 33.3330
A-549 NSC95397 CTRP2,CTRP1 0.0010 33.3330
A-549 NU7441 GDSC1,GDSC2 0.0078 10.0000
A-549 Nutlin-3a CTRP1,CCLE,GDSC1,GDSC2,CTRP2 0.0025 150.0000
A-549 NVP-231 CTRP2 0.0020 66.0000
A-549 NVP-ADW742 GDSC2,CTRP2 0.0020 66.0000
A-549 NVP-AUY922 CTRP1 0.2603 33.3330
A-549 NVP-BHG712 GDSC1 0.0400 10.2400
A-549 NVP-BSK805 CTRP2 0.0020 66.0000
A-549 NVP-TAE684 CTRP2,CCLE 0.0020 66.0000
A-549 Obatoclax Mesylate GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 OF-1 GDSC2 0.0100 10.0000
A-549 Olaparib GDSC1,GDSC2,CTRP2,CTRP1 0.0045 150.0000
A-549 oligomycin A CTRP2,CTRP1 0.0010 33.3330
A-549 omacetaxine mepesuccinate CTRP2 0.0020 66.0000
A-549 Omipalisib GDSC1 0.0005 0.1280
A-549 orteronel CTRP1 0.2603 33.3330
A-549 OSI-027 GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 OSI-930 GDSC1,CTRP2 0.0020 66.0000
A-549 Osimertinib GDSC2 0.0010 1.0000
A-549 OSU-03012 GDSC1 0.0625 16.0000
A-549 OSW-1 CTRP1 0.2603 33.3330
A-549 OTX015 GDSC2 0.0100 10.0000
A-549 ouabain CTRP2 0.0081 270.0000
A-549 Oxaliplatin GDSC2,CTRP2 0.0020 66.0000
A-549 oxythiamine CTRP1 0.2603 33.3330
A-549 P-0850 CTRP1 0.2603 33.3330
A-549 P22077 GDSC2 0.0100 10.0000
A-549 PAC-1 GDSC1,CTRP2,CTRP1 0.0010 33.3330
A-549 Paclitaxel GDSC2,CTRP2,CCLE 0.0000 66.0000
A-549 PAK_5339 GDSC2 0.0300 30.0000
A-549 Palbociclib GDSC1,GDSC2,CCLE 0.0025 10.0000
A-549 palmostatin B CTRP2 0.0020 66.0000
A-549 pandacostat CTRP2,CTRP1 0.0010 33.0000
A-549 panduratin A CTRP1 0.2603 33.3330
A-549 Panobinostat GDSC1,CCLE 0.0025 8.0000
A-549 parbendazole CTRP2 0.0020 66.0000
A-549 PARP_0108 GDSC1 0.0098 2.5000
A-549 PARP_9482 GDSC1 0.0098 2.5000
A-549 PARP_9495 GDSC1 0.0098 2.5000
A-549 Parthenolide CTRP2,CTRP1 0.0020 66.0000
A-549 Pazopanib GDSC1,CTRP2 0.0020 66.0000
A-549 PBD-288 GDSC2 0.0050 5.0000
A-549 PCI-34051 GDSC2 0.0100 10.0000
A-549 PD 153035 CTRP2 0.0010 33.0000
A-549 PD0325901 GDSC1,GDSC2,CCLE 0.0003 8.0000
A-549 PD173074 GDSC1,GDSC2 0.0020 10.0000
A-549 PD318088 CTRP2 0.0020 66.0000
A-549 PDMP CTRP2 0.0065 210.0000
A-549 Pelitinib GDSC1 0.0098 2.5000
A-549 Pemetrexed GDSC1,CTRP1 0.0100 37.0000
A-549 Pevonedistat GDSC1,GDSC2,CTRP2,CTRP1 0.0011 37.0000
A-549 PF-00299804 GDSC1 0.0781 20.0000
A-549 PF-184 CTRP2 0.0020 66.0000
A-549 PF-3845 CTRP1 0.2603 33.3330
A-549 PF-4708671 GDSC1 0.0391 10.0000
A-549 PF-562271 GDSC1 0.0100 2.5600
A-549 PF-573228 CTRP2 0.0020 66.0000
A-549 PF-750 CTRP2,CTRP1 0.0081 270.0000
A-549 PFI-1 GDSC1,GDSC2 0.0100 10.0000
A-549 PFI3 GDSC1,GDSC2 0.0100 10.0000
A-549 PHA-665752 CCLE 0.0025 8.0000
A-549 PHA-793887 GDSC1,CTRP2 0.0020 66.0000
A-549 Phenformin GDSC1 15.6250 4000.0000
A-549 phloretin CTRP2,CTRP1 0.0180 590.0000
A-549 PI-103 GDSC1,CTRP2,CTRP1 0.0011 37.0000
A-549 PI3Ka_4409 GDSC1 0.0391 10.0000
A-549 Picolinici-acid GDSC2 0.0100 10.0000
A-549 Pictilisib GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 pifithrin-alpha CTRP2 0.0071 230.0000
A-549 pifithrin-mu CTRP2,CTRP1 0.0010 33.3330
A-549 PIK-75 CTRP1 0.2890 37.0000
A-549 PIK-93 GDSC1,CTRP2 0.0020 66.0000
A-549 Pilaralisib GDSC1 0.0781 20.0000
A-549 Piperlongumine GDSC1,CTRP2,CTRP1 0.0010 33.3330
A-549 piperlongumine:MST-312 (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 pitstop2 CTRP2 0.0020 66.0000
A-549 PL-DI CTRP2 0.0020 66.0000
A-549 Platin CTRP2 0.0020 66.0000
A-549 PLK_6522 GDSC1 0.0024 0.6250
A-549 pluripotin CTRP2,CTRP1 0.0010 33.3330
A-549 PLX-4032 CTRP2 0.0010 33.0000
A-549 PLX-4720 GDSC1,GDSC2,CTRP2,CCLE 0.0010 33.0000
A-549 Podophyllotoxin bromide GDSC2 0.0010 1.0000
A-549 POMHEX GDSC2 0.0100 10.0000
A-549 Ponatinib GDSC1 0.0020 0.5120
A-549 PP-30 CTRP1 0.2890 37.0000
A-549 PRIMA-1 CTRP2,CTRP1 0.0051 170.0000
A-549 PRIMA-1MET GDSC2,CTRP2 0.0010 33.0000
A-549 PRL-3 Inhibitor I CTRP2,CTRP1 0.0041 130.0000
A-549 procarbazine CTRP2 0.0020 66.0000
A-549 prochlorperazine CTRP2 0.0020 66.0000
A-549 PRT062607 GDSC2 0.0100 10.0000
A-549 PT-630 CTRP1 0.2603 33.3330
A-549 purmorphamine CTRP2,CTRP1 0.0046 150.0000
A-549 PX-12 CTRP2 0.0030 100.0000
A-549 PYR-41 CTRP2 0.0020 66.0000
A-549 pyrazolanthrone CTRP2 0.0020 66.0000
A-549 Pyridostatin GDSC2 0.0100 10.0000
A-549 QL-VIII-58 GDSC1 0.0391 10.0000
A-549 QL-X-138 GDSC1 0.0400 10.2400
A-549 QL-XI-92 GDSC1 0.0400 10.2400
A-549 QL-XII-47 GDSC1 0.0391 10.2400
A-549 QL-XII-61 GDSC1 0.0391 10.0000
A-549 QS11 GDSC1,CTRP2 0.0010 33.0000
A-549 quinoclamine CTRP1 0.2890 37.0000
A-549 Quizartinib GDSC1,CTRP2 0.0020 66.0000
A-549 R428 CTRP2 0.0020 17.0000
A-549 racemic-2,4-dideoxy-DC-45-A2 CTRP1 0.2890 37.0000
A-549 RAF_9304 GDSC1 0.0391 10.0000
A-549 RAF265 CTRP2,CCLE 0.0020 66.0000
A-549 Rapamycin GDSC2,CTRP2,CTRP1 0.0000 37.0000
A-549 Refametinib GDSC1,GDSC2 0.0100 10.0000
A-549 Regorafenib CTRP2 0.0020 66.0000
A-549 Remodelin GDSC2 0.0500 50.0000
A-549 Repligen 136 CTRP2 0.0020 66.0000
A-549 RepSox CTRP1 0.2603 33.3330
A-549 RG-108 CTRP2,CTRP1 0.0081 270.0000
A-549 Ribociclib GDSC2 0.0020 2.0000
A-549 rigosertib CTRP2 0.0020 66.0000
A-549 RITA CTRP2,CTRP1 0.0010 33.3330
A-549 Ro-28-1675 CTRP1 0.2603 33.3330
A-549 RO-3306 GDSC1,GDSC2 0.0100 10.0000
A-549 Romidepsin GDSC2 0.0000 0.0100
A-549 rosiglitazone CTRP1 0.2603 33.3330
A-549 rotenone CTRP1 0.2603 33.3330
A-549 rTRAIL GDSC1 0.0004 0.1000
A-549 RU-SKI 43 GDSC1 0.0781 20.0000
A-549 Rucaparib GDSC1,GDSC2 0.0050 5.0000
A-549 Ruxolitinib GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 RVX-208 GDSC2 0.0100 10.0000
A-549 Sabutoclax GDSC2 0.0100 10.0000
A-549 salermide CTRP2 0.0120 400.0000
A-549 salermide:PLX-4032 (12:1 mol-mol) CTRP2 0.0066 220.0000
A-549 Sapitinib GDSC2 0.0050 10.0000
A-549 Saracatinib CTRP2,CCLE 0.0020 66.0000
A-549 Savolitinib GDSC2 0.0010 1.0000
A-549 SB-225002 CTRP2,CTRP1 0.0011 37.0000
A-549 SB-431542 CTRP2 0.0020 66.0000
A-549 SB-525334 CTRP2 0.0020 66.0000
A-549 SB-743921 CTRP2 0.0010 33.0000
A-549 SB216763 GDSC1,GDSC2 0.0100 10.0000
A-549 SB505124 GDSC1 0.0391 20.0000
A-549 SB52334 GDSC1 0.0781 20.0000
A-549 SB590885 GDSC1,GDSC2 0.0050 5.0000
A-549 SCH-529074 CTRP2 0.0010 33.0000
A-549 SCH-79797 CTRP2,CTRP1 0.0011 37.0000
A-549 SCH772984 GDSC2 0.0050 5.0000
A-549 Schweinfurthin A GDSC2 0.0010 1.0000
A-549 Selisistat GDSC1,CTRP2 0.0024 80.0000
A-549 Selumetinib GDSC1,GDSC2,CTRP2,CCLE 0.0025 270.0000
A-549 selumetinib:BRD-A02303741 (4:1 mol-mol) CTRP2 0.0051 170.0000
A-549 selumetinib:decitabine (4:1 mol-mol) CTRP2 0.0051 170.0000
A-549 selumetinib:GDC-0941 (4:1 mol-mol) CTRP2 0.0051 170.0000
A-549 selumetinib:JQ-1 (4:1 mol-mol) CTRP2 0.0051 170.0000
A-549 selumetinib:MK-2206 (8:1 mol-mol) CTRP2 0.0046 150.0000
A-549 selumetinib:navitoclax (8:1 mol-mol) CTRP2 0.0046 150.0000
A-549 selumetinib:piperlongumine (8:1 mol-mol) CTRP2 0.0046 150.0000
A-549 selumetinib:PLX-4032 (8:1 mol-mol) CTRP2 0.0046 150.0000
A-549 selumetinib:tretinoin (2:1 mol-mol) CTRP2 0.0061 200.0000
A-549 selumetinib:UNC0638 (4:1 mol-mol) CTRP2 0.0051 170.0000
A-549 selumetinib:vorinostat (8:1 mol-mol) CTRP2 0.0046 150.0000
A-549 semagacestat CTRP2 0.0020 66.0000
A-549 Sepantronium bromide GDSC1,GDSC2,CTRP2 0.0000 10.0000
A-549 Serdemetan GDSC1,GDSC2,CTRP2,CTRP1 0.0010 33.3330
A-549 serdemetan:SCH-529074 (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 SGC-CBP30 GDSC2 0.0050 5.0000
A-549 SGC0946 GDSC1,GDSC2 0.0005 0.5000
A-549 SGX-523 CTRP2 0.0020 66.0000
A-549 Shikonin GDSC1 0.0625 16.0000
A-549 SID 26681509 CTRP2,CTRP1 0.0090 300.0000
A-549 sildenafil CTRP2,CTRP1 0.0160 530.0000
A-549 silmitasertib CTRP2 0.0020 66.0000
A-549 simvastatin CTRP2,CTRP1 0.0010 33.3330
A-549 Sinularin GDSC2 0.0030 3.0000
A-549 sirolimus:bortezomib (250:1 mol-mol) CTRP2 0.0005 17.0000
A-549 sitagliptin CTRP2 0.0020 33.0000
A-549 SJ-172550 CTRP2,CTRP1 0.0010 37.0000
A-549 SKI-II CTRP2,CTRP1 0.0041 130.0000
A-549 SL0101 GDSC1 0.0391 10.0000
A-549 SMER-3 CTRP2 0.0020 66.0000
A-549 SN-38 GDSC1,GDSC2,CTRP2,CTRP1 0.0000 37.0000
A-549 SNS-032 CTRP2 0.0020 66.0000
A-549 SNX-2112 GDSC1,CTRP2,CTRP1 0.0010 33.3330
A-549 SNX-2112:bortezomib (250:1 mol-mol) CTRP2 0.0005 17.0000
A-549 Sorafenib GDSC2,CTRP2,CCLE 0.0020 66.0000
A-549 sotrastaurin CTRP2 0.0020 66.0000
A-549 sparfosic acid CTRP1 0.2603 33.3330
A-549 spautin-1 CTRP2 0.0020 66.0000
A-549 Sphingosine Kinase 1 Inhibitor II GDSC1,CTRP2 0.0010 33.0000
A-549 SR-II-138A CTRP2,CTRP1 0.0010 33.3330
A-549 SR1001 CTRP2 0.0020 66.0000
A-549 Staurosporine GDSC2,CTRP2 0.0001 3.3000
A-549 StemRegenin 1 CTRP2 0.0020 66.0000
A-549 STF-31 CTRP2 0.0020 66.0000
A-549 STF-62247 GDSC1 0.0400 10.2400
A-549 SU11274 GDSC1,CTRP2 0.0020 66.0000
A-549 Sunitinib CTRP2 0.0020 66.0000
A-549 T-5345967 CTRP2,CTRP1 0.0160 530.0000
A-549 T0901317 GDSC1 0.0400 10.2400
A-549 tacedinaline CTRP2 0.0010 33.0000
A-549 tacrolimus CTRP2,CTRP1 0.0023 74.0000
A-549 TAF1_5496 GDSC2 0.0100 10.0000
A-549 TAK-715 GDSC1 0.0400 20.0000
A-549 Talazoparib GDSC1,GDSC2 0.0100 10.0000
A-549 tamatinib CTRP2 0.0010 33.0000
A-549 Tamoxifen GDSC1,GDSC2,CTRP2 0.0030 100.0000
A-549 tandutinib CTRP2 0.0020 66.0000
A-549 Tanespimycin CTRP1,CCLE,GDSC1,GDSC2,CTRP2 0.0010 37.0000
A-549 tanespimycin:bortezomib (250:1 mol-mol) CTRP2 0.0005 17.0000
A-549 tanespimycin:gemcitabine (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 TANK_1366 GDSC1 0.0098 2.5000
A-549 Taselisib GDSC2 0.0040 10.0000
A-549 Telomerase Inhibitor IX GDSC2,CTRP2,CTRP1 0.0010 37.0000
A-549 Temozolomide GDSC1,GDSC2,CTRP2 0.0020 66.0000
A-549 Temsirolimus GDSC1,GDSC2,CTRP2 0.0008 66.0000
A-549 Teniposide GDSC2,CTRP2 0.0010 33.0000
A-549 Tenovin-6 GDSC1 0.0781 20.0000
A-549 TG-100-115 CTRP2 0.0020 66.0000
A-549 TGX-115 CTRP1 0.2603 33.3330
A-549 TGX221 CTRP2 0.0020 66.0000
A-549 Thapsigargin GDSC1 0.0020 0.5120
A-549 THR-101 GDSC2 0.0100 10.0000
A-549 THR-102 GDSC2 0.0100 10.0000
A-549 THR-103 GDSC2 0.0100 10.0000
A-549 THZ-1-87 GDSC1 0.0391 10.0000
A-549 THZ-2-102-1 GDSC1 0.0098 2.5000
A-549 THZ-2-49 GDSC1 0.0781 20.0000
A-549 THZ-2-98-01 GDSC1 0.0391 10.0000
A-549 tigecycline CTRP2 0.0020 66.0000
A-549 Tipifarnib GDSC1 0.0625 16.0000
A-549 tipifarnib-P1 CTRP2,CTRP1 0.0010 33.3330
A-549 tipifarnib-P2 CTRP2,CTRP1 0.0010 33.3330
A-549 Tivozanib GDSC1,CTRP2,CTRP1 0.0005 33.3330
A-549 TKI258 CCLE 0.0025 8.0000
A-549 TL-1-85 GDSC1 0.0400 10.2400
A-549 TL-2-105 GDSC1 0.0200 10.2400
A-549 Topotecan GDSC2,CTRP2,CCLE 0.0020 66.0000
A-549 Torin 2 GDSC1 0.0781 20.0000
A-549 torin2 GDSC1 0.0391 10.0000
A-549 tosedostat CTRP2 0.0081 270.0000
A-549 Tozasertib CTRP1 0.2603 33.3330
A-549 TPCA-1 GDSC1,CTRP2 0.0020 66.0000
A-549 Trametinib GDSC1,GDSC2 0.0010 1.0000
A-549 Tretinoin GDSC1,CTRP2,CTRP1 0.0041 130.0000
A-549 tretinoin:carboplatin (2:1 mol-mol) CTRP2 0.0030 100.0000
A-549 tretinoin:navitoclax (4:1 mol-mol) CTRP2 0.0025 83.0000
A-549 triacsin C CTRP1 0.2603 33.3330
A-549 Trichostatin A GDSC1 0.0040 1.0240
A-549 trifluoperazine CTRP2 0.0010 33.0000
A-549 triptolide CTRP2,CTRP1 0.0000 33.3330
A-549 TTK_3146 GDSC1 0.0391 10.0000
A-549 Tubastatin A GDSC1,CTRP2 0.0010 33.0000
A-549 TW 37 GDSC1,GDSC2,CTRP2 0.0010 33.0000
A-549 TWS119 GDSC1 0.0781 20.0000
A-549 ubistatin B CTRP1 0.2603 33.3330
A-549 Ulixertinib GDSC2 0.0020 10.0000
A-549 ULK1_4989 GDSC2 0.0300 30.0000
A-549 UMI-77 GDSC2 0.0100 10.0000
A-549 UNC0321 CTRP2 0.0010 33.0000
A-549 UNC0379 GDSC2 0.0100 10.0000
A-549 UNC0638 GDSC1,GDSC2,CTRP2 0.0010 40.0000
A-549 UNC0638:navitoclax (1:1 mol-mol) CTRP2 0.0010 33.0000
A-549 UNC0642 GDSC1 0.0020 0.5000
A-549 UNC1215 GDSC1 0.0039 1.0000
A-549 Uprosertib GDSC2 0.0100 10.0000
A-549 VAF-347 CTRP2 0.0020 66.0000
A-549 valdecoxib CTRP2,CTRP1 0.0180 600.0000
A-549 vandetanib CTRP2 0.0020 66.0000
A-549 VE-822 GDSC2 0.0050 5.0000
A-549 VE821 GDSC2 0.0100 10.0000
A-549 Veliparib GDSC1,GDSC2,CTRP2 0.0010 33.0000
A-549 Venetoclax GDSC2,CTRP2 0.0010 66.0000
A-549 Venotoclax GDSC1 0.0010 0.2560
A-549 VER-155008 CTRP2,CTRP1 0.0011 37.0000
A-549 Vinblastine GDSC1,GDSC2 0.0001 0.1000
A-549 Vincristine GDSC2,CTRP2 0.0030 130.0000
A-549 Vinorelbine GDSC1,GDSC2 0.0001 0.1000
A-549 Vismodegib GDSC1,GDSC2,CTRP1 0.0100 33.3330
A-549 VNLG-124 GDSC1 0.0200 5.1200
A-549 vorapaxar CTRP2 0.0020 66.0000
A-549 Vorinostat GDSC1,GDSC2,CTRP2,CTRP1 0.0010 37.0000
A-549 vorinostat:carboplatin (1:1 mol-mol) CTRP2 0.0020 66.0000
A-549 vorinostat:navitoclax (4:1 mol-mol) CTRP2 0.0010 33.0000
A-549 Voxtalisib GDSC1 0.0781 20.0000
A-549 VSP34_8731 GDSC2 0.0300 30.0000
A-549 VTP-A GDSC2 0.0010 1.0000
A-549 VTP-B GDSC2 0.0010 1.0000
A-549 VU0155056 CTRP2 0.0020 66.0000
A-549 VX-11e GDSC1,GDSC2 0.0100 10.0000
A-549 VX-702 GDSC1 0.0078 2.0000
A-549 WAY-362450 CTRP2 0.0020 66.0000
A-549 Wee1 Inhibitor GDSC1,GDSC2 0.0078 10.0000
A-549 WEHI-539 GDSC2 0.0100 10.0000
A-549 WHI-P97 GDSC1 0.0400 10.2400
A-549 WIKI4 GDSC2 0.0100 10.0000
A-549 Wnt-C59 GDSC1,GDSC2 0.0100 10.0000
A-549 WP1130 CTRP2 0.0020 66.0000
A-549 WT-161 CTRP1 0.2603 33.3330
A-549 WYE-125132 GDSC1 0.0400 10.2400
A-549 WZ3105 GDSC1 0.0050 1.2800
A-549 WZ4002 CTRP2 0.0010 33.0000
A-549 WZ4003 GDSC2 0.0100 10.0000
A-549 WZ8040 CTRP2 0.0020 66.0000
A-549 XAV939 GDSC1,GDSC2,CTRP1 0.0100 37.0000
A-549 XL765 CTRP2 0.0020 66.0000
A-549 XMD11-50 GDSC1 0.0391 10.0000
A-549 XMD11-85h GDSC1 0.0391 10.0000
A-549 XMD13-2 GDSC1 0.0400 10.2400
A-549 XMD14-99 GDSC1 0.0400 10.2400
A-549 XMD15-27 GDSC1 0.0400 10.2400
A-549 XMD8-92 GDSC1 0.0391 10.0000
A-549 Y-39983 GDSC1 0.0781 20.0000
A-549 YK-4-279 GDSC1,GDSC2,CTRP2 0.0010 33.0000
A-549 YL54 CTRP2 0.0020 66.0000
A-549 YM-022 CTRP1 0.2603 33.3330
A-549 YM201636 GDSC1 0.0200 5.1200
A-549 ZD-6474 CCLE 0.0025 8.0000
A-549 zebularine CTRP2,CTRP1 0.0180 590.0000
A-549 ZG-10 GDSC1 0.0391 10.0000
A-549 Zibotentan GDSC1 0.0781 20.0000
A-549 zileuton CTRP1 0.2603 33.3330
A-549 ZL049 GDSC1 0.0391 10.0000
A-549 ZL109 GDSC1 0.0391 10.0000
A-549 ZM447439 GDSC1,GDSC2 0.0100 10.0000
A-549 Zoledronate GDSC2 0.0020 2.0000
A-549 ZSTK474 GDSC1,CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Drugs with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Drugs with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Drugs with highest and lowest AUC