Drug : Zileuton

CTRP1 Name : zileuton

Dataset : All
Synonyms :
Targets : ALOX5
Pathways : inhibitor of 5-lipoxygenase

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
zileuton MCF-7 CTRP1 4.1667 533.3300
zileuton GAMG CTRP1 0.2603 33.3330
zileuton LN-229 CTRP1 4.1667 533.3300
zileuton SF295 CTRP1 0.2603 33.3330
zileuton HEC-108 CTRP1 0.2603 33.3330
zileuton HEC-151 CTRP1 4.1667 533.3300
zileuton HEC-251 CTRP1 0.2603 33.3330
zileuton HEC-265 CTRP1 0.2603 33.3330
zileuton HEC-59 CTRP1 0.2603 33.3330
zileuton HEC-6 CTRP1 0.2603 33.3330
zileuton ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
zileuton JHUEM-2 CTRP1 4.1667 533.3300
zileuton KLE CTRP1 0.2603 33.3330
zileuton MFE-319 CTRP1 0.2603 33.3330
zileuton SNG-M CTRP1 0.2603 33.3330
zileuton AMO1 CTRP1 4.1667 533.3300
zileuton BL-70 CTRP1 0.2603 33.3330
zileuton EJM CTRP1 4.1667 533.3300
zileuton GDM-1 CTRP1 4.1667 533.3300
zileuton HT CTRP1 0.2603 33.3330
zileuton KMS-11 CTRP1 4.1667 533.3300
zileuton KU812 CTRP1 0.2603 33.3330
zileuton LP-1 CTRP1 4.1667 533.3300
zileuton MC116 CTRP1 0.2603 33.3330
zileuton MOLM-16 CTRP1 4.1667 533.3300
zileuton NOMO-1 CTRP1 4.1667 533.3300
zileuton NU-DUL-1 CTRP1 4.1667 533.3300
zileuton OCI-AML-3 CTRP1 4.1667 533.3300
zileuton OCI-LY10 CTRP1 4.1667 533.3300
zileuton P3HR-1 CTRP1 0.2603 33.3330
zileuton PL21 CTRP1 4.1667 533.3300
zileuton RPMI-8226 CTRP1 4.1667 533.3300
zileuton SKM-1 CTRP1 4.1667 533.3300
zileuton SU-DHL-4 CTRP1 4.1667 533.3300
zileuton SU-DHL-5 CTRP1 4.1667 533.3300
zileuton THP-1 CTRP1 4.1667 533.3300
zileuton U-937 CTRP1 4.1667 533.3300
zileuton WSU-DLCL2 CTRP1 4.1667 533.3300
zileuton RCC10RGB CTRP1 4.1667 533.3300
zileuton VMRC-RCW CTRP1 0.2603 33.3330
zileuton C2BBE1 CTRP1 0.2603 33.3330
zileuton CL-34 CTRP1 4.1667 533.3300
zileuton CL-40 CTRP1 4.1667 533.3300
zileuton COLO205 CTRP1 0.2603 33.3330
zileuton COLO320 CTRP1 4.1667 533.3300
zileuton COLO678 CTRP1 4.1667 533.3300
zileuton CW-2 CTRP1 4.1667 533.3300
zileuton DLD-1 CTRP1 0.2603 33.3330
zileuton GP2D CTRP1 0.2603 33.3330
zileuton HCT116 CTRP1 4.1667 533.3300
zileuton HCT8 CTRP1 4.1667 533.3300
zileuton HT115 CTRP1 4.1667 533.3300
zileuton HT-29 CTRP1 4.1667 533.3300
zileuton HT-55 CTRP1 4.1667 533.3300
zileuton KM12 CTRP1 4.1667 533.3300
zileuton LOVO CTRP1 4.1667 533.3300
zileuton LS123 CTRP1 4.1667 533.3300
zileuton LS180 CTRP1 4.1667 533.3300
zileuton LS411N CTRP1 0.2603 33.3330
zileuton LS513 CTRP1 0.2603 33.3330
zileuton MDST8 CTRP1 4.1667 533.3300
zileuton NCI-H508 CTRP1 4.1667 533.3300
zileuton RCM-1[HUMANESC] CTRP1 4.1667 533.3300
zileuton RKO CTRP1 4.1667 533.3300
zileuton SK-CO-1 CTRP1 0.2603 33.3330
zileuton SNU-1040 CTRP1 4.1667 533.3300
zileuton SNU-175 CTRP1 4.1667 533.3300
zileuton SNU-61 CTRP1 4.1667 533.3300
zileuton SNU-81 CTRP1 4.1667 533.3300
zileuton SNU-C2A CTRP1 0.2603 33.3330
zileuton SNU-C4 CTRP1 4.1667 533.3300
zileuton SNU-C5 CTRP1 4.1667 533.3300
zileuton SW403 CTRP1 0.2603 33.3330
zileuton SW48 CTRP1 0.2603 33.3330
zileuton SW480 CTRP1 4.1667 533.3300
zileuton SW620 CTRP1 4.1667 533.3300
zileuton SW948 CTRP1 4.1667 533.3300
zileuton HEP-G2 CTRP1 4.1667 533.3300
zileuton JHH-6 CTRP1 0.2603 33.3330
zileuton SNU-398 CTRP1 4.1667 533.3300
zileuton SNU-449 CTRP1 0.2603 33.3330
zileuton A-549 CTRP1 0.2603 33.3330
zileuton BEN CTRP1 0.2603 33.3330
zileuton CAL-12T CTRP1 4.1667 533.3300
zileuton CALU-3 CTRP1 0.2603 33.3330
zileuton CALU-6 CTRP1 0.2603 33.3330
zileuton CHAGO-K-1 CTRP1 0.2603 33.3330
zileuton COLO668 CTRP1 0.2603 33.3330
zileuton COLO699 CTRP1 4.1667 533.3300
zileuton COR-L23 CTRP1 4.1667 533.3300
zileuton COR-L279 CTRP1 0.2603 33.3330
zileuton COR-L51 CTRP1 4.1667 533.3300
zileuton COR-L88 CTRP1 0.2603 33.3330
zileuton DMS273 CTRP1 0.2603 33.3330
zileuton DV-90 CTRP1 0.2603 33.3330
zileuton EBC-1 CTRP1 0.2603 33.3330
zileuton EPLC-272H CTRP1 0.2603 33.3330
zileuton HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
zileuton HCC1195 CTRP1 4.1667 533.3300
zileuton HCC1359 CTRP1 4.1667 533.3300
zileuton HCC15 CTRP1 4.1667 533.3300
zileuton HCC1833 CTRP1 4.1667 533.3300
zileuton HCC2108 CTRP1 4.1667 533.3300
zileuton HCC2935 CTRP1 4.1667 533.3300
zileuton HCC33 CTRP1 0.2603 33.3330
zileuton HCC4006 CTRP1 4.1667 533.3300
zileuton HCC44 CTRP1 0.2603 33.3330
zileuton HCC78 CTRP1 0.2603 33.3330
zileuton HCC827 CTRP1 4.1667 533.3300
zileuton KNS-62 CTRP1 0.2603 33.3330
zileuton LC-1-SQ-SF CTRP1 0.2603 33.3330
zileuton LCLC-103H CTRP1 0.2603 33.3330
zileuton LCLC-97TM1 CTRP1 0.2603 33.3330
zileuton LU-65 CTRP1 0.2603 33.3330
zileuton LU-99 CTRP1 0.2603 33.3330
zileuton LXF289 CTRP1 0.2603 33.3330
zileuton NCI-H1048 CTRP1 0.2603 33.3330
zileuton NCI-H1105 CTRP1 4.1667 533.3300
zileuton NCI-H1299 CTRP1 0.2603 33.3330
zileuton NCI-H1355 CTRP1 0.2603 33.3330
zileuton NCI-H1373 CTRP1 0.2603 33.3330
zileuton NCI-H1435 CTRP1 0.2603 33.3330
zileuton NCI-H1437 CTRP1 0.2603 33.3330
zileuton NCI-H1568 CTRP1 0.2603 33.3330
zileuton NCI-H1573 CTRP1 0.2603 33.3330
zileuton NCI-H1666 CTRP1 0.2603 33.3330
zileuton NCI-H1694 CTRP1 4.1667 533.3300
zileuton NCI-H1755 CTRP1 4.1667 533.3300
zileuton NCI-H1781 CTRP1 4.1667 533.3300
zileuton NCI-H1792 CTRP1 0.2603 33.3330
zileuton NCI-H1793 CTRP1 0.2603 33.3330
zileuton NCI-H1836 CTRP1 4.1667 533.3300
zileuton NCI-H1876 CTRP1 4.1667 533.3300
zileuton NCI-H1915 CTRP1 0.2603 33.3330
zileuton NCI-H1930 CTRP1 0.2603 33.3330
zileuton NCI-H1944 CTRP1 0.2603 33.3330
zileuton NCI-H1963 CTRP1 4.1667 533.3300
zileuton NCI-H1975 CTRP1 0.2603 33.3330
zileuton NCI-H2009 CTRP1 0.2603 33.3330
zileuton NCI-H2023 CTRP1 4.1667 533.3300
zileuton NCI-H2029 CTRP1 0.2603 33.3330
zileuton NCI-H2030 CTRP1 4.1667 533.3300
zileuton NCI-H2073 CTRP1 4.1667 533.3300
zileuton NCI-H2081 CTRP1 4.1667 533.3300
zileuton NCI-H2110 CTRP1 4.1667 533.3300
zileuton NCI-H2122 CTRP1 4.1667 533.3300
zileuton NCI-H2126 CTRP1 0.2603 33.3330
zileuton NCI-H2141 CTRP1 4.1667 533.3300
zileuton NCI-H2172 CTRP1 4.1667 533.3300
zileuton NCI-H2286 CTRP1 0.2603 33.3330
zileuton NCI-H23 CTRP1 0.2603 33.3330
zileuton NCI-H2342 CTRP1 4.1667 533.3300
zileuton NCI-H2405 CTRP1 0.2603 33.3330
zileuton NCI-H3255 CTRP1 4.1667 533.3300
zileuton NCI-H358 CTRP1 0.2603 33.3330
zileuton NCI-H441 CTRP1 4.1667 533.3300
zileuton NCI-H460 CTRP1 4.1667 533.3300
zileuton NCI-H522 CTRP1 0.2603 33.3330
zileuton NCI-H596 CTRP1 4.1667 533.3300
zileuton NCI-H650 CTRP1 0.2603 33.3330
zileuton NCI-H661 CTRP1 0.2603 33.3330
zileuton NCI-H727 CTRP1 0.2603 33.3330
zileuton NCI-H810 CTRP1 0.2603 33.3330
zileuton NCI-H82 CTRP1 0.2603 33.3330
zileuton NCI-H841 CTRP1 4.1667 533.3300
zileuton RERF-LC-KJ CTRP1 0.2603 33.3330
zileuton SCLC-21H CTRP1 4.1667 533.3300
zileuton SHP-77 CTRP1 0.2603 33.3330
zileuton SK-LU-1 CTRP1 4.1667 533.3300
zileuton SQ-1 CTRP1 4.1667 533.3300
zileuton T3M-10 CTRP1 4.1667 533.3300
zileuton VMRC-LCD CTRP1 0.2603 33.3330
zileuton KYSE-140 CTRP1 0.2603 33.3330
zileuton KYSE-410 CTRP1 0.2603 33.3330
zileuton KYSE-450 CTRP1 0.2603 33.3330
zileuton A2780 CTRP1 4.1667 533.3300
zileuton CAOV-3 CTRP1 4.1667 533.3300
zileuton COV318 CTRP1 0.2603 33.3330
zileuton COV362 CTRP1 4.1667 533.3300
zileuton COV434 CTRP1 4.1667 533.3300
zileuton COV644 CTRP1 4.1667 533.3300
zileuton EFO-21 CTRP1 0.2603 33.3330
zileuton EFO-27 CTRP1 4.1667 533.3300
zileuton HEYA8 CTRP1 0.2603 33.3330
zileuton IGROV-1 CTRP1 4.1667 533.3300
zileuton JHOC-5 CTRP1 4.1667 533.3300
zileuton JHOM-1 CTRP1 4.1667 533.3300
zileuton JHOS-4 CTRP1 0.2603 33.3330
zileuton OAW42 CTRP1 4.1667 533.3300
zileuton OV7 CTRP1 4.1667 533.3300
zileuton OV-90 CTRP1 4.1667 533.3300
zileuton OVCAR-4 CTRP1 4.1667 533.3300
zileuton OVCAR-8 CTRP1 4.1667 533.3300
zileuton OVK18 CTRP1 4.1667 533.3300
zileuton OVKATE CTRP1 4.1667 533.3300
zileuton OVMANA CTRP1 0.2603 33.3330
zileuton RKN CTRP1 4.1667 533.3300
zileuton RMG-I CTRP1 4.1667 533.3300
zileuton RMUG-S CTRP1 4.1667 533.3300
zileuton SK-OV-3 CTRP1 0.2603 33.3330
zileuton SNU-840 CTRP1 4.1667 533.3300
zileuton TYK-NU CTRP1 4.1667 533.3300
zileuton CAPAN-2 CTRP1 0.2603 33.3330
zileuton CFPAC-1 CTRP1 0.2603 33.3330
zileuton HPAC CTRP1 0.2603 33.3330
zileuton HUP-T4 CTRP1 0.2603 33.3330
zileuton KP-3 CTRP1 0.2603 33.3330
zileuton PANC03.27 CTRP1 0.2603 33.3330
zileuton PANC10.05 CTRP1 0.2603 33.3330
zileuton PATU8902 CTRP1 0.2603 33.3330
zileuton QGP-1 CTRP1 0.2603 33.3330
zileuton SUIT-2 CTRP1 0.2603 33.3330
zileuton MSTO-211H CTRP1 0.2603 33.3330
zileuton NCI-H2052 CTRP1 0.2603 33.3330
zileuton NCI-H28 CTRP1 0.2603 33.3330
zileuton MIAPACA-3 CTRP1 0.2603 33.3330
zileuton A-375 CTRP1 4.1667 533.3300
zileuton COLO741 CTRP1 0.2603 33.3330
zileuton G-361 CTRP1 0.2603 33.3330
zileuton HS852.T CTRP1 0.2603 33.3330
zileuton HS936.T CTRP1 0.2603 33.3330
zileuton HS944.T CTRP1 0.2603 33.3330
zileuton SK-MEL-1 CTRP1 4.1667 533.3300
zileuton SK-MEL-28 CTRP1 4.1667 533.3300
zileuton SK-MEL-5 CTRP1 4.1667 533.3300
zileuton G-401 CTRP1 0.2603 33.3330
zileuton HT-1080 CTRP1 4.1667 533.3300
zileuton AGS CTRP1 4.1667 533.3300
zileuton FU97 CTRP1 0.2603 33.3330
zileuton KE-97 CTRP1 0.2603 33.3330
zileuton MKN7 CTRP1 0.2603 33.3330
zileuton MKN74 CTRP1 0.2603 33.3330
zileuton NUGC-4 CTRP1 0.2603 33.3330
zileuton SH-10-TC CTRP1 0.2603 33.3330
zileuton HSC-2 CTRP1 0.2603 33.3330
zileuton SCC-9 CTRP1 4.1667 533.3300
zileuton 5637 CTRP1 0.2603 33.3330
zileuton HT-1376 CTRP1 0.2603 33.3330
zileuton KMBC-2 CTRP1 0.2603 33.3330
zileuton RT-4 CTRP1 0.2603 33.3330
zileuton UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.