Drug : Dichloroacetic Acid

CTRP1 Name : dichloroacetic acid

Dataset : All
Synonyms :
Targets : PDK2
Pathways : inhibitor of pyruvate dehydrogenase kinase 2

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
dichloroacetic acid GAMG CTRP1 0.2603 33.3330
dichloroacetic acid SF295 CTRP1 0.2603 33.3330
dichloroacetic acid HEC-108 CTRP1 0.2603 33.3330
dichloroacetic acid HEC-251 CTRP1 0.2603 33.3330
dichloroacetic acid HEC-265 CTRP1 0.2603 33.3330
dichloroacetic acid HEC-59 CTRP1 0.2603 33.3330
dichloroacetic acid HEC-6 CTRP1 0.2603 33.3330
dichloroacetic acid ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
dichloroacetic acid KLE CTRP1 0.2603 33.3330
dichloroacetic acid MFE-319 CTRP1 0.2603 33.3330
dichloroacetic acid SNG-M CTRP1 0.2603 33.3330
dichloroacetic acid BL-70 CTRP1 0.2603 33.3330
dichloroacetic acid HT CTRP1 0.2603 33.3330
dichloroacetic acid KU812 CTRP1 0.2603 33.3330
dichloroacetic acid MC116 CTRP1 0.2603 33.3330
dichloroacetic acid P3HR-1 CTRP1 0.2603 33.3330
dichloroacetic acid VMRC-RCW CTRP1 0.2603 33.3330
dichloroacetic acid C2BBE1 CTRP1 0.2603 33.3330
dichloroacetic acid COLO205 CTRP1 0.2603 33.3330
dichloroacetic acid DLD-1 CTRP1 0.2603 33.3330
dichloroacetic acid GP2D CTRP1 0.2603 33.3330
dichloroacetic acid LS411N CTRP1 0.2603 33.3330
dichloroacetic acid LS513 CTRP1 0.2603 33.3330
dichloroacetic acid SK-CO-1 CTRP1 0.2603 33.3330
dichloroacetic acid SNU-C2A CTRP1 0.2603 33.3330
dichloroacetic acid SW403 CTRP1 0.2603 33.3330
dichloroacetic acid SW48 CTRP1 0.2603 33.3330
dichloroacetic acid JHH-6 CTRP1 0.2603 33.3330
dichloroacetic acid SNU-449 CTRP1 0.2603 33.3330
dichloroacetic acid A-549 CTRP1 0.2603 33.3330
dichloroacetic acid BEN CTRP1 0.2603 33.3330
dichloroacetic acid CALU-3 CTRP1 0.2603 33.3330
dichloroacetic acid CALU-6 CTRP1 0.2603 33.3330
dichloroacetic acid CHAGO-K-1 CTRP1 0.2603 33.3330
dichloroacetic acid COLO668 CTRP1 0.2603 33.3330
dichloroacetic acid COR-L279 CTRP1 0.2603 33.3330
dichloroacetic acid COR-L88 CTRP1 0.2603 33.3330
dichloroacetic acid DMS273 CTRP1 0.2603 33.3330
dichloroacetic acid DV-90 CTRP1 0.2603 33.3330
dichloroacetic acid EBC-1 CTRP1 0.2603 33.3330
dichloroacetic acid EPLC-272H CTRP1 0.2603 33.3330
dichloroacetic acid HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
dichloroacetic acid HCC33 CTRP1 0.2603 33.3330
dichloroacetic acid HCC44 CTRP1 0.2603 33.3330
dichloroacetic acid HCC78 CTRP1 0.2603 33.3330
dichloroacetic acid KNS-62 CTRP1 0.2603 33.3330
dichloroacetic acid LC-1-SQ-SF CTRP1 0.2603 33.3330
dichloroacetic acid LCLC-103H CTRP1 0.2603 33.3330
dichloroacetic acid LCLC-97TM1 CTRP1 0.2603 33.3330
dichloroacetic acid LU-65 CTRP1 0.2603 33.3330
dichloroacetic acid LU-99 CTRP1 0.2603 33.3330
dichloroacetic acid LXF289 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1048 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1299 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1355 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1373 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1435 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1437 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1568 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1573 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1666 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1792 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1793 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1915 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1930 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1944 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H1975 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H2009 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H2029 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H2126 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H2286 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H23 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H2405 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H358 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H522 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H650 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H661 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H727 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H810 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H82 CTRP1 0.2603 33.3330
dichloroacetic acid RERF-LC-KJ CTRP1 0.2603 33.3330
dichloroacetic acid SHP-77 CTRP1 0.2603 33.3330
dichloroacetic acid VMRC-LCD CTRP1 0.2603 33.3330
dichloroacetic acid KYSE-140 CTRP1 0.2603 33.3330
dichloroacetic acid KYSE-410 CTRP1 0.2603 33.3330
dichloroacetic acid KYSE-450 CTRP1 0.2603 33.3330
dichloroacetic acid COV318 CTRP1 0.2603 33.3330
dichloroacetic acid EFO-21 CTRP1 0.2603 33.3330
dichloroacetic acid HEYA8 CTRP1 0.2603 33.3330
dichloroacetic acid JHOS-4 CTRP1 0.2603 33.3330
dichloroacetic acid OVMANA CTRP1 0.2603 33.3330
dichloroacetic acid SK-OV-3 CTRP1 0.2603 33.3330
dichloroacetic acid CAPAN-2 CTRP1 0.2603 33.3330
dichloroacetic acid CFPAC-1 CTRP1 0.2603 33.3330
dichloroacetic acid HPAC CTRP1 0.2603 33.3330
dichloroacetic acid HUP-T4 CTRP1 0.2603 33.3330
dichloroacetic acid KP-3 CTRP1 0.2603 33.3330
dichloroacetic acid PANC03.27 CTRP1 0.2603 33.3330
dichloroacetic acid PANC10.05 CTRP1 0.2603 33.3330
dichloroacetic acid PATU8902 CTRP1 0.2603 33.3330
dichloroacetic acid QGP-1 CTRP1 0.2603 33.3330
dichloroacetic acid SUIT-2 CTRP1 0.2603 33.3330
dichloroacetic acid MSTO-211H CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H2052 CTRP1 0.2603 33.3330
dichloroacetic acid NCI-H28 CTRP1 0.2603 33.3330
dichloroacetic acid MIAPACA-3 CTRP1 0.2603 33.3330
dichloroacetic acid COLO741 CTRP1 0.2603 33.3330
dichloroacetic acid G-361 CTRP1 0.2603 33.3330
dichloroacetic acid HS852.T CTRP1 0.2603 33.3330
dichloroacetic acid HS936.T CTRP1 0.2603 33.3330
dichloroacetic acid HS944.T CTRP1 0.2603 33.3330
dichloroacetic acid G-401 CTRP1 0.2603 33.3330
dichloroacetic acid FU97 CTRP1 0.2603 33.3330
dichloroacetic acid KE-97 CTRP1 0.2603 33.3330
dichloroacetic acid MKN7 CTRP1 0.2603 33.3330
dichloroacetic acid MKN74 CTRP1 0.2603 33.3330
dichloroacetic acid NUGC-4 CTRP1 0.2603 33.3330
dichloroacetic acid SH-10-TC CTRP1 0.2603 33.3330
dichloroacetic acid HSC-2 CTRP1 0.2603 33.3330
dichloroacetic acid 5637 CTRP1 0.2603 33.3330
dichloroacetic acid HT-1376 CTRP1 0.2603 33.3330
dichloroacetic acid KMBC-2 CTRP1 0.2603 33.3330
dichloroacetic acid RT-4 CTRP1 0.2603 33.3330
dichloroacetic acid UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.