Drug : Brd7137

CTRP1 Name : BRD7137

Dataset : All
Synonyms :
Targets :
Pathways : screening hit

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

:


Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BRD7137 U2OS CTRP1 0.2604 33.3330
BRD7137 MCF-7 CTRP1 0.2604 33.3330
BRD7137 GAMG CTRP1 0.2603 33.3330
BRD7137 LN-229 CTRP1 0.2604 33.3330
BRD7137 SF295 CTRP1 0.2603 33.3330
BRD7137 HEC-108 CTRP1 0.2603 33.3330
BRD7137 HEC-151 CTRP1 0.2604 33.3330
BRD7137 HEC-251 CTRP1 0.2603 33.3330
BRD7137 HEC-265 CTRP1 0.2603 33.3330
BRD7137 HEC-59 CTRP1 0.2603 33.3330
BRD7137 HEC-6 CTRP1 0.2603 33.3330
BRD7137 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
BRD7137 JHUEM-2 CTRP1 0.2604 33.3330
BRD7137 KLE CTRP1 0.2603 33.3330
BRD7137 MFE-319 CTRP1 0.2603 33.3330
BRD7137 SNG-M CTRP1 0.2603 33.3330
BRD7137 AMO1 CTRP1 0.2604 33.3330
BRD7137 BL-70 CTRP1 0.2603 33.3330
BRD7137 EJM CTRP1 0.2604 33.3330
BRD7137 GDM-1 CTRP1 0.2604 33.3330
BRD7137 HT CTRP1 0.2603 33.3330
BRD7137 KMS-11 CTRP1 0.2604 33.3330
BRD7137 KU812 CTRP1 0.2603 33.3330
BRD7137 LP-1 CTRP1 0.2604 33.3330
BRD7137 MC116 CTRP1 0.2603 33.3330
BRD7137 MOLM-16 CTRP1 0.2604 33.3330
BRD7137 NOMO-1 CTRP1 0.2604 33.3330
BRD7137 NU-DUL-1 CTRP1 0.2604 33.3330
BRD7137 OCI-AML-3 CTRP1 0.2604 33.3330
BRD7137 OCI-LY10 CTRP1 0.2604 33.3330
BRD7137 P3HR-1 CTRP1 0.2603 33.3330
BRD7137 PL21 CTRP1 0.2604 33.3330
BRD7137 RPMI-8226 CTRP1 0.2604 33.3330
BRD7137 SKM-1 CTRP1 0.2604 33.3330
BRD7137 SU-DHL-4 CTRP1 0.2604 33.3330
BRD7137 SU-DHL-5 CTRP1 0.2604 33.3330
BRD7137 THP-1 CTRP1 0.2604 33.3330
BRD7137 U-937 CTRP1 0.2604 33.3330
BRD7137 WSU-DLCL2 CTRP1 0.2604 33.3330
BRD7137 RCC10RGB CTRP1 0.2604 33.3330
BRD7137 VMRC-RCW CTRP1 0.2603 33.3330
BRD7137 C2BBE1 CTRP1 0.2603 33.3330
BRD7137 CL-34 CTRP1 0.2604 33.3330
BRD7137 CL-40 CTRP1 0.2604 33.3330
BRD7137 COLO205 CTRP1 0.2603 33.3330
BRD7137 COLO320 CTRP1 0.2604 33.3330
BRD7137 COLO678 CTRP1 0.2604 33.3330
BRD7137 CW-2 CTRP1 0.2604 33.3330
BRD7137 DLD-1 CTRP1 0.2603 33.3330
BRD7137 GP2D CTRP1 0.2603 33.3330
BRD7137 HCT116 CTRP1 0.2604 33.3330
BRD7137 HCT8 CTRP1 0.2604 33.3330
BRD7137 HT115 CTRP1 0.2604 33.3330
BRD7137 HT-29 CTRP1 0.2604 33.3330
BRD7137 HT-55 CTRP1 0.2604 33.3330
BRD7137 KM12 CTRP1 0.2604 33.3330
BRD7137 LOVO CTRP1 0.2604 33.3330
BRD7137 LS123 CTRP1 0.2604 33.3330
BRD7137 LS180 CTRP1 0.2604 33.3330
BRD7137 LS411N CTRP1 0.2603 33.3330
BRD7137 LS513 CTRP1 0.2603 33.3330
BRD7137 MDST8 CTRP1 0.2604 33.3330
BRD7137 NCI-H508 CTRP1 0.2604 33.3330
BRD7137 RCM-1[HUMANESC] CTRP1 0.2604 33.3330
BRD7137 RKO CTRP1 0.2604 33.3330
BRD7137 SK-CO-1 CTRP1 0.2603 33.3330
BRD7137 SNU-1040 CTRP1 0.2604 33.3330
BRD7137 SNU-175 CTRP1 0.2604 33.3330
BRD7137 SNU-61 CTRP1 0.2604 33.3330
BRD7137 SNU-81 CTRP1 0.2604 33.3330
BRD7137 SNU-C2A CTRP1 0.2603 33.3330
BRD7137 SNU-C4 CTRP1 0.2604 33.3330
BRD7137 SNU-C5 CTRP1 0.2604 33.3330
BRD7137 SW403 CTRP1 0.2603 33.3330
BRD7137 SW48 CTRP1 0.2603 33.3330
BRD7137 SW480 CTRP1 0.2604 33.3330
BRD7137 SW620 CTRP1 0.2604 33.3330
BRD7137 SW948 CTRP1 0.2604 33.3330
BRD7137 HEP-G2 CTRP1 0.2604 33.3330
BRD7137 JHH-6 CTRP1 0.2603 33.3330
BRD7137 SNU-398 CTRP1 0.2604 33.3330
BRD7137 SNU-449 CTRP1 0.2603 33.3330
BRD7137 A-549 CTRP1 0.2603 33.3330
BRD7137 BEN CTRP1 0.2603 33.3330
BRD7137 CAL-12T CTRP1 0.2604 33.3330
BRD7137 CALU-3 CTRP1 0.2603 33.3330
BRD7137 CALU-6 CTRP1 0.2603 33.3330
BRD7137 CHAGO-K-1 CTRP1 0.2603 33.3330
BRD7137 COLO668 CTRP1 0.2603 33.3330
BRD7137 COLO699 CTRP1 0.2604 33.3330
BRD7137 COR-L23 CTRP1 0.2604 33.3330
BRD7137 COR-L279 CTRP1 0.2603 33.3330
BRD7137 COR-L51 CTRP1 0.2604 33.3330
BRD7137 COR-L88 CTRP1 0.2603 33.3330
BRD7137 DMS273 CTRP1 0.2603 33.3330
BRD7137 DV-90 CTRP1 0.2603 33.3330
BRD7137 EBC-1 CTRP1 0.2603 33.3330
BRD7137 EPLC-272H CTRP1 0.2603 33.3330
BRD7137 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
BRD7137 HCC1195 CTRP1 0.2604 33.3330
BRD7137 HCC1359 CTRP1 0.2604 33.3330
BRD7137 HCC15 CTRP1 0.2604 33.3330
BRD7137 HCC1833 CTRP1 0.2604 33.3330
BRD7137 HCC2108 CTRP1 0.2604 33.3330
BRD7137 HCC2935 CTRP1 0.2604 33.3330
BRD7137 HCC33 CTRP1 0.2603 33.3330
BRD7137 HCC4006 CTRP1 0.2604 33.3330
BRD7137 HCC44 CTRP1 0.2603 33.3330
BRD7137 HCC78 CTRP1 0.2603 33.3330
BRD7137 HCC827 CTRP1 0.2604 33.3330
BRD7137 KNS-62 CTRP1 0.2603 33.3330
BRD7137 LC-1-SQ-SF CTRP1 0.2603 33.3330
BRD7137 LCLC-103H CTRP1 0.2603 33.3330
BRD7137 LCLC-97TM1 CTRP1 0.2603 33.3330
BRD7137 LU-65 CTRP1 0.2603 33.3330
BRD7137 LU-99 CTRP1 0.2603 33.3330
BRD7137 LXF289 CTRP1 0.2603 33.3330
BRD7137 NCI-H1048 CTRP1 0.2603 33.3330
BRD7137 NCI-H1105 CTRP1 0.2604 33.3330
BRD7137 NCI-H1299 CTRP1 0.2603 33.3330
BRD7137 NCI-H1355 CTRP1 0.2603 33.3330
BRD7137 NCI-H1373 CTRP1 0.2603 33.3330
BRD7137 NCI-H1435 CTRP1 0.2603 33.3330
BRD7137 NCI-H1437 CTRP1 0.2603 33.3330
BRD7137 NCI-H1568 CTRP1 0.2603 33.3330
BRD7137 NCI-H1573 CTRP1 0.2603 33.3330
BRD7137 NCI-H1666 CTRP1 0.2603 33.3330
BRD7137 NCI-H1694 CTRP1 0.2604 33.3330
BRD7137 NCI-H1755 CTRP1 0.2604 33.3330
BRD7137 NCI-H1781 CTRP1 0.2604 33.3330
BRD7137 NCI-H1792 CTRP1 0.2603 33.3330
BRD7137 NCI-H1793 CTRP1 0.2603 33.3330
BRD7137 NCI-H1836 CTRP1 0.2604 33.3330
BRD7137 NCI-H1876 CTRP1 0.2604 33.3330
BRD7137 NCI-H1915 CTRP1 0.2603 33.3330
BRD7137 NCI-H1930 CTRP1 0.2603 33.3330
BRD7137 NCI-H1944 CTRP1 0.2603 33.3330
BRD7137 NCI-H1963 CTRP1 0.2604 33.3330
BRD7137 NCI-H1975 CTRP1 0.2603 33.3330
BRD7137 NCI-H2009 CTRP1 0.2603 33.3330
BRD7137 NCI-H2023 CTRP1 0.2604 33.3330
BRD7137 NCI-H2029 CTRP1 0.2603 33.3330
BRD7137 NCI-H2030 CTRP1 0.2604 33.3330
BRD7137 NCI-H2073 CTRP1 0.2604 33.3330
BRD7137 NCI-H2081 CTRP1 0.2604 33.3330
BRD7137 NCI-H2110 CTRP1 0.2604 33.3330
BRD7137 NCI-H2122 CTRP1 0.2604 33.3330
BRD7137 NCI-H2126 CTRP1 0.2603 33.3330
BRD7137 NCI-H2141 CTRP1 0.2604 33.3330
BRD7137 NCI-H2172 CTRP1 0.2604 33.3330
BRD7137 NCI-H2286 CTRP1 0.2603 33.3330
BRD7137 NCI-H23 CTRP1 0.2603 33.3330
BRD7137 NCI-H2342 CTRP1 0.2604 33.3330
BRD7137 NCI-H2405 CTRP1 0.2603 33.3330
BRD7137 NCI-H3255 CTRP1 0.2604 33.3330
BRD7137 NCI-H358 CTRP1 0.2603 33.3330
BRD7137 NCI-H441 CTRP1 0.2604 33.3330
BRD7137 NCI-H460 CTRP1 0.2604 33.3330
BRD7137 NCI-H522 CTRP1 0.2603 33.3330
BRD7137 NCI-H596 CTRP1 0.2604 33.3330
BRD7137 NCI-H650 CTRP1 0.2603 33.3330
BRD7137 NCI-H661 CTRP1 0.2603 33.3330
BRD7137 NCI-H727 CTRP1 0.2603 33.3330
BRD7137 NCI-H810 CTRP1 0.2603 33.3330
BRD7137 NCI-H82 CTRP1 0.2603 33.3330
BRD7137 NCI-H841 CTRP1 0.2604 33.3330
BRD7137 RERF-LC-KJ CTRP1 0.2603 33.3330
BRD7137 SCLC-21H CTRP1 0.2604 33.3330
BRD7137 SHP-77 CTRP1 0.2603 33.3330
BRD7137 SK-LU-1 CTRP1 0.2604 33.3330
BRD7137 SQ-1 CTRP1 0.2604 33.3330
BRD7137 T3M-10 CTRP1 0.2604 33.3330
BRD7137 VMRC-LCD CTRP1 0.2603 33.3330
BRD7137 KYSE-140 CTRP1 0.2603 33.3330
BRD7137 KYSE-410 CTRP1 0.2603 33.3330
BRD7137 KYSE-450 CTRP1 0.2603 33.3330
BRD7137 A2780 CTRP1 0.2604 33.3330
BRD7137 CAOV-3 CTRP1 0.2604 33.3330
BRD7137 COV318 CTRP1 0.2603 33.3330
BRD7137 COV362 CTRP1 0.2604 33.3330
BRD7137 COV434 CTRP1 0.2604 33.3330
BRD7137 COV644 CTRP1 0.2604 33.3330
BRD7137 EFO-21 CTRP1 0.2603 33.3330
BRD7137 EFO-27 CTRP1 0.2604 33.3330
BRD7137 HEYA8 CTRP1 0.2603 33.3330
BRD7137 IGROV-1 CTRP1 0.2604 33.3330
BRD7137 JHOC-5 CTRP1 0.2604 33.3330
BRD7137 JHOM-1 CTRP1 0.2604 33.3330
BRD7137 JHOS-4 CTRP1 0.2603 33.3330
BRD7137 OAW42 CTRP1 0.2604 33.3330
BRD7137 OV7 CTRP1 0.2604 33.3330
BRD7137 OV-90 CTRP1 0.2604 33.3330
BRD7137 OVCAR-4 CTRP1 0.2604 33.3330
BRD7137 OVCAR-8 CTRP1 0.2604 33.3330
BRD7137 OVK18 CTRP1 0.2604 33.3330
BRD7137 OVKATE CTRP1 0.2604 33.3330
BRD7137 OVMANA CTRP1 0.2603 33.3330
BRD7137 RKN CTRP1 0.2604 33.3330
BRD7137 RMG-I CTRP1 0.2604 33.3330
BRD7137 RMUG-S CTRP1 0.2604 33.3330
BRD7137 SK-OV-3 CTRP1 0.2603 33.3330
BRD7137 SNU-840 CTRP1 0.2604 33.3330
BRD7137 TYK-NU CTRP1 0.2604 33.3330
BRD7137 CAPAN-2 CTRP1 0.2603 33.3330
BRD7137 CFPAC-1 CTRP1 0.2603 33.3330
BRD7137 HPAC CTRP1 0.2603 33.3330
BRD7137 HUP-T4 CTRP1 0.2603 33.3330
BRD7137 KP-3 CTRP1 0.2603 33.3330
BRD7137 PANC03.27 CTRP1 0.2603 33.3330
BRD7137 PANC10.05 CTRP1 0.2603 33.3330
BRD7137 PATU8902 CTRP1 0.2603 33.3330
BRD7137 QGP-1 CTRP1 0.2603 33.3330
BRD7137 SUIT-2 CTRP1 0.2603 33.3330
BRD7137 MSTO-211H CTRP1 0.2603 33.3330
BRD7137 NCI-H2052 CTRP1 0.2603 33.3330
BRD7137 NCI-H28 CTRP1 0.2603 33.3330
BRD7137 MIAPACA-3 CTRP1 0.2603 33.3330
BRD7137 A-375 CTRP1 0.2604 33.3330
BRD7137 COLO741 CTRP1 0.2603 33.3330
BRD7137 G-361 CTRP1 0.2603 33.3330
BRD7137 HS852.T CTRP1 0.2603 33.3330
BRD7137 HS936.T CTRP1 0.2603 33.3330
BRD7137 HS944.T CTRP1 0.2603 33.3330
BRD7137 SK-MEL-1 CTRP1 0.2604 33.3330
BRD7137 SK-MEL-28 CTRP1 0.2604 33.3330
BRD7137 SK-MEL-5 CTRP1 0.2604 33.3330
BRD7137 G-401 CTRP1 0.2603 33.3330
BRD7137 HT-1080 CTRP1 0.2604 33.3330
BRD7137 AGS CTRP1 0.2604 33.3330
BRD7137 FU97 CTRP1 0.2603 33.3330
BRD7137 KE-97 CTRP1 0.2603 33.3330
BRD7137 MKN7 CTRP1 0.2603 33.3330
BRD7137 MKN74 CTRP1 0.2603 33.3330
BRD7137 NUGC-4 CTRP1 0.2603 33.3330
BRD7137 SH-10-TC CTRP1 0.2603 33.3330
BRD7137 HSC-2 CTRP1 0.2603 33.3330
BRD7137 SCC-9 CTRP1 0.2604 33.3330
BRD7137 5637 CTRP1 0.2603 33.3330
BRD7137 HT-1376 CTRP1 0.2603 33.3330
BRD7137 KMBC-2 CTRP1 0.2603 33.3330
BRD7137 RT-4 CTRP1 0.2603 33.3330
BRD7137 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.