Drug : Brd6368

CTRP1 Name : BRD6368

Dataset : All
Synonyms :
Targets :
Pathways : screening hit

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BRD6368 U2OS CTRP1 0.2604 33.3330
BRD6368 MCF-7 CTRP1 0.2604 33.3330
BRD6368 GAMG CTRP1 0.2603 33.3330
BRD6368 LN-229 CTRP1 0.2604 33.3330
BRD6368 SF295 CTRP1 0.2603 33.3330
BRD6368 HEC-108 CTRP1 0.2603 33.3330
BRD6368 HEC-151 CTRP1 0.2604 33.3330
BRD6368 HEC-251 CTRP1 0.2603 33.3330
BRD6368 HEC-265 CTRP1 0.2603 33.3330
BRD6368 HEC-59 CTRP1 0.2603 33.3330
BRD6368 HEC-6 CTRP1 0.2603 33.3330
BRD6368 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
BRD6368 JHUEM-2 CTRP1 0.2604 33.3330
BRD6368 KLE CTRP1 0.2603 33.3330
BRD6368 MFE-319 CTRP1 0.2603 33.3330
BRD6368 SNG-M CTRP1 0.2603 33.3330
BRD6368 AMO1 CTRP1 0.2604 33.3330
BRD6368 BL-70 CTRP1 0.2603 33.3330
BRD6368 EJM CTRP1 0.2604 33.3330
BRD6368 GDM-1 CTRP1 0.2604 33.3330
BRD6368 HT CTRP1 0.2603 33.3330
BRD6368 KMS-11 CTRP1 0.2604 33.3330
BRD6368 KU812 CTRP1 0.2603 33.3330
BRD6368 LP-1 CTRP1 0.2604 33.3330
BRD6368 MC116 CTRP1 0.2603 33.3330
BRD6368 MOLM-16 CTRP1 0.2604 33.3330
BRD6368 NOMO-1 CTRP1 0.2604 33.3330
BRD6368 NU-DUL-1 CTRP1 0.2604 33.3330
BRD6368 OCI-AML-3 CTRP1 0.2604 33.3330
BRD6368 OCI-LY10 CTRP1 0.2604 33.3330
BRD6368 P3HR-1 CTRP1 0.2603 33.3330
BRD6368 PL21 CTRP1 0.2604 33.3330
BRD6368 RPMI-8226 CTRP1 0.2604 33.3330
BRD6368 SKM-1 CTRP1 0.2604 33.3330
BRD6368 SU-DHL-4 CTRP1 0.2604 33.3330
BRD6368 SU-DHL-5 CTRP1 0.2604 33.3330
BRD6368 THP-1 CTRP1 0.2604 33.3330
BRD6368 U-937 CTRP1 0.2604 33.3330
BRD6368 WSU-DLCL2 CTRP1 0.2604 33.3330
BRD6368 RCC10RGB CTRP1 0.2604 33.3330
BRD6368 VMRC-RCW CTRP1 0.2603 33.3330
BRD6368 C2BBE1 CTRP1 0.2603 33.3330
BRD6368 CL-34 CTRP1 0.2604 33.3330
BRD6368 CL-40 CTRP1 0.2604 33.3330
BRD6368 COLO205 CTRP1 0.2603 33.3330
BRD6368 COLO320 CTRP1 0.2604 33.3330
BRD6368 COLO678 CTRP1 0.2604 33.3330
BRD6368 CW-2 CTRP1 0.2604 33.3330
BRD6368 DLD-1 CTRP1 0.2603 33.3330
BRD6368 GP2D CTRP1 0.2603 33.3330
BRD6368 HCT116 CTRP1 0.2604 33.3330
BRD6368 HCT8 CTRP1 0.2604 33.3330
BRD6368 HT115 CTRP1 0.2604 33.3330
BRD6368 HT-29 CTRP1 0.2604 33.3330
BRD6368 HT-55 CTRP1 0.2604 33.3330
BRD6368 KM12 CTRP1 0.2604 33.3330
BRD6368 LOVO CTRP1 0.2604 33.3330
BRD6368 LS123 CTRP1 0.2604 33.3330
BRD6368 LS180 CTRP1 0.2604 33.3330
BRD6368 LS411N CTRP1 0.2603 33.3330
BRD6368 LS513 CTRP1 0.2603 33.3330
BRD6368 MDST8 CTRP1 0.2604 33.3330
BRD6368 NCI-H508 CTRP1 0.2604 33.3330
BRD6368 RCM-1[HUMANESC] CTRP1 0.2604 33.3330
BRD6368 RKO CTRP1 0.2604 33.3330
BRD6368 SK-CO-1 CTRP1 0.2603 33.3330
BRD6368 SNU-1040 CTRP1 0.2604 33.3330
BRD6368 SNU-175 CTRP1 0.2604 33.3330
BRD6368 SNU-61 CTRP1 0.2604 33.3330
BRD6368 SNU-81 CTRP1 0.2604 33.3330
BRD6368 SNU-C2A CTRP1 0.2603 33.3330
BRD6368 SNU-C4 CTRP1 0.2604 33.3330
BRD6368 SNU-C5 CTRP1 0.2604 33.3330
BRD6368 SW403 CTRP1 0.2603 33.3330
BRD6368 SW48 CTRP1 0.2603 33.3330
BRD6368 SW480 CTRP1 0.2604 33.3330
BRD6368 SW620 CTRP1 0.2604 33.3330
BRD6368 SW948 CTRP1 0.2604 33.3330
BRD6368 HEP-G2 CTRP1 0.2604 33.3330
BRD6368 JHH-6 CTRP1 0.2603 33.3330
BRD6368 SNU-398 CTRP1 0.2604 33.3330
BRD6368 SNU-449 CTRP1 0.2603 33.3330
BRD6368 A-549 CTRP1 0.2603 33.3330
BRD6368 BEN CTRP1 0.2603 33.3330
BRD6368 CAL-12T CTRP1 0.2604 33.3330
BRD6368 CALU-3 CTRP1 0.2603 33.3330
BRD6368 CALU-6 CTRP1 0.2603 33.3330
BRD6368 CHAGO-K-1 CTRP1 0.2603 33.3330
BRD6368 COLO668 CTRP1 0.2603 33.3330
BRD6368 COLO699 CTRP1 0.2604 33.3330
BRD6368 COR-L23 CTRP1 0.2604 33.3330
BRD6368 COR-L279 CTRP1 0.2603 33.3330
BRD6368 COR-L51 CTRP1 0.2604 33.3330
BRD6368 COR-L88 CTRP1 0.2603 33.3330
BRD6368 DMS273 CTRP1 0.2603 33.3330
BRD6368 DV-90 CTRP1 0.2603 33.3330
BRD6368 EBC-1 CTRP1 0.2603 33.3330
BRD6368 EPLC-272H CTRP1 0.2603 33.3330
BRD6368 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
BRD6368 HCC1195 CTRP1 0.2604 33.3330
BRD6368 HCC1359 CTRP1 0.2604 33.3330
BRD6368 HCC15 CTRP1 0.2604 33.3330
BRD6368 HCC1833 CTRP1 0.2604 33.3330
BRD6368 HCC2108 CTRP1 0.2604 33.3330
BRD6368 HCC2935 CTRP1 0.2604 33.3330
BRD6368 HCC33 CTRP1 0.2603 33.3330
BRD6368 HCC4006 CTRP1 0.2604 33.3330
BRD6368 HCC44 CTRP1 0.2603 33.3330
BRD6368 HCC78 CTRP1 0.2603 33.3330
BRD6368 HCC827 CTRP1 0.2604 33.3330
BRD6368 KNS-62 CTRP1 0.2603 33.3330
BRD6368 LC-1-SQ-SF CTRP1 0.2603 33.3330
BRD6368 LCLC-103H CTRP1 0.2603 33.3330
BRD6368 LCLC-97TM1 CTRP1 0.2603 33.3330
BRD6368 LU-65 CTRP1 0.2603 33.3330
BRD6368 LU-99 CTRP1 0.2603 33.3330
BRD6368 LXF289 CTRP1 0.2603 33.3330
BRD6368 NCI-H1048 CTRP1 0.2603 33.3330
BRD6368 NCI-H1105 CTRP1 0.2604 33.3330
BRD6368 NCI-H1299 CTRP1 0.2603 33.3330
BRD6368 NCI-H1355 CTRP1 0.2603 33.3330
BRD6368 NCI-H1373 CTRP1 0.2603 33.3330
BRD6368 NCI-H1435 CTRP1 0.2603 33.3330
BRD6368 NCI-H1437 CTRP1 0.2603 33.3330
BRD6368 NCI-H1568 CTRP1 0.2603 33.3330
BRD6368 NCI-H1573 CTRP1 0.2603 33.3330
BRD6368 NCI-H1666 CTRP1 0.2603 33.3330
BRD6368 NCI-H1694 CTRP1 0.2604 33.3330
BRD6368 NCI-H1755 CTRP1 0.2604 33.3330
BRD6368 NCI-H1781 CTRP1 0.2604 33.3330
BRD6368 NCI-H1792 CTRP1 0.2603 33.3330
BRD6368 NCI-H1793 CTRP1 0.2603 33.3330
BRD6368 NCI-H1836 CTRP1 0.2604 33.3330
BRD6368 NCI-H1876 CTRP1 0.2604 33.3330
BRD6368 NCI-H1915 CTRP1 0.2603 33.3330
BRD6368 NCI-H1930 CTRP1 0.2603 33.3330
BRD6368 NCI-H1944 CTRP1 0.2603 33.3330
BRD6368 NCI-H1963 CTRP1 0.2604 33.3330
BRD6368 NCI-H1975 CTRP1 0.2603 33.3330
BRD6368 NCI-H2009 CTRP1 0.2603 33.3330
BRD6368 NCI-H2023 CTRP1 0.2604 33.3330
BRD6368 NCI-H2029 CTRP1 0.2603 33.3330
BRD6368 NCI-H2030 CTRP1 0.2604 33.3330
BRD6368 NCI-H2073 CTRP1 0.2604 33.3330
BRD6368 NCI-H2081 CTRP1 0.2604 33.3330
BRD6368 NCI-H2110 CTRP1 0.2604 33.3330
BRD6368 NCI-H2122 CTRP1 0.2604 33.3330
BRD6368 NCI-H2126 CTRP1 0.2603 33.3330
BRD6368 NCI-H2141 CTRP1 0.2604 33.3330
BRD6368 NCI-H2172 CTRP1 0.2604 33.3330
BRD6368 NCI-H2286 CTRP1 0.2603 33.3330
BRD6368 NCI-H23 CTRP1 0.2603 33.3330
BRD6368 NCI-H2342 CTRP1 0.2604 33.3330
BRD6368 NCI-H2405 CTRP1 0.2603 33.3330
BRD6368 NCI-H3255 CTRP1 0.2604 33.3330
BRD6368 NCI-H358 CTRP1 0.2603 33.3330
BRD6368 NCI-H441 CTRP1 0.2604 33.3330
BRD6368 NCI-H460 CTRP1 0.2604 33.3330
BRD6368 NCI-H522 CTRP1 0.2603 33.3330
BRD6368 NCI-H596 CTRP1 0.2604 33.3330
BRD6368 NCI-H650 CTRP1 0.2603 33.3330
BRD6368 NCI-H661 CTRP1 0.2603 33.3330
BRD6368 NCI-H727 CTRP1 0.2603 33.3330
BRD6368 NCI-H810 CTRP1 0.2603 33.3330
BRD6368 NCI-H82 CTRP1 0.2603 33.3330
BRD6368 NCI-H841 CTRP1 0.2604 33.3330
BRD6368 RERF-LC-KJ CTRP1 0.2603 33.3330
BRD6368 SCLC-21H CTRP1 0.2604 33.3330
BRD6368 SHP-77 CTRP1 0.2603 33.3330
BRD6368 SK-LU-1 CTRP1 0.2604 33.3330
BRD6368 SQ-1 CTRP1 0.2604 33.3330
BRD6368 T3M-10 CTRP1 0.2604 33.3330
BRD6368 VMRC-LCD CTRP1 0.2603 33.3330
BRD6368 KYSE-140 CTRP1 0.2603 33.3330
BRD6368 KYSE-410 CTRP1 0.2603 33.3330
BRD6368 KYSE-450 CTRP1 0.2603 33.3330
BRD6368 A2780 CTRP1 0.2604 33.3330
BRD6368 CAOV-3 CTRP1 0.2604 33.3330
BRD6368 COV318 CTRP1 0.2603 33.3330
BRD6368 COV362 CTRP1 0.2604 33.3330
BRD6368 COV434 CTRP1 0.2604 33.3330
BRD6368 COV644 CTRP1 0.2604 33.3330
BRD6368 EFO-21 CTRP1 0.2603 33.3330
BRD6368 EFO-27 CTRP1 0.2604 33.3330
BRD6368 HEYA8 CTRP1 0.2603 33.3330
BRD6368 IGROV-1 CTRP1 0.2604 33.3330
BRD6368 JHOC-5 CTRP1 0.2604 33.3330
BRD6368 JHOM-1 CTRP1 0.2604 33.3330
BRD6368 JHOS-4 CTRP1 0.2603 33.3330
BRD6368 OAW42 CTRP1 0.2604 33.3330
BRD6368 OV7 CTRP1 0.2604 33.3330
BRD6368 OV-90 CTRP1 0.2604 33.3330
BRD6368 OVCAR-4 CTRP1 0.2604 33.3330
BRD6368 OVCAR-8 CTRP1 0.2604 33.3330
BRD6368 OVK18 CTRP1 0.2604 33.3330
BRD6368 OVKATE CTRP1 0.2604 33.3330
BRD6368 OVMANA CTRP1 0.2603 33.3330
BRD6368 RKN CTRP1 0.2604 33.3330
BRD6368 RMG-I CTRP1 0.2604 33.3330
BRD6368 RMUG-S CTRP1 0.2604 33.3330
BRD6368 SK-OV-3 CTRP1 0.2603 33.3330
BRD6368 SNU-840 CTRP1 0.2604 33.3330
BRD6368 TYK-NU CTRP1 0.2604 33.3330
BRD6368 CAPAN-2 CTRP1 0.2603 33.3330
BRD6368 CFPAC-1 CTRP1 0.2603 33.3330
BRD6368 HPAC CTRP1 0.2603 33.3330
BRD6368 HUP-T4 CTRP1 0.2603 33.3330
BRD6368 KP-3 CTRP1 0.2603 33.3330
BRD6368 PANC03.27 CTRP1 0.2603 33.3330
BRD6368 PANC10.05 CTRP1 0.2603 33.3330
BRD6368 PATU8902 CTRP1 0.2603 33.3330
BRD6368 QGP-1 CTRP1 0.2603 33.3330
BRD6368 SUIT-2 CTRP1 0.2603 33.3330
BRD6368 MSTO-211H CTRP1 0.2603 33.3330
BRD6368 NCI-H2052 CTRP1 0.2603 33.3330
BRD6368 NCI-H28 CTRP1 0.2603 33.3330
BRD6368 MIAPACA-3 CTRP1 0.2603 33.3330
BRD6368 A-375 CTRP1 0.2604 33.3330
BRD6368 COLO741 CTRP1 0.2603 33.3330
BRD6368 G-361 CTRP1 0.2603 33.3330
BRD6368 HS852.T CTRP1 0.2603 33.3330
BRD6368 HS936.T CTRP1 0.2603 33.3330
BRD6368 HS944.T CTRP1 0.2603 33.3330
BRD6368 SK-MEL-1 CTRP1 0.2604 33.3330
BRD6368 SK-MEL-28 CTRP1 0.2604 33.3330
BRD6368 SK-MEL-5 CTRP1 0.2604 33.3330
BRD6368 G-401 CTRP1 0.2603 33.3330
BRD6368 HT-1080 CTRP1 0.2604 33.3330
BRD6368 AGS CTRP1 0.2604 33.3330
BRD6368 FU97 CTRP1 0.2603 33.3330
BRD6368 KE-97 CTRP1 0.2603 33.3330
BRD6368 MKN7 CTRP1 0.2603 33.3330
BRD6368 MKN74 CTRP1 0.2603 33.3330
BRD6368 NUGC-4 CTRP1 0.2603 33.3330
BRD6368 SH-10-TC CTRP1 0.2603 33.3330
BRD6368 HSC-2 CTRP1 0.2603 33.3330
BRD6368 SCC-9 CTRP1 0.2604 33.3330
BRD6368 5637 CTRP1 0.2603 33.3330
BRD6368 HT-1376 CTRP1 0.2603 33.3330
BRD6368 KMBC-2 CTRP1 0.2603 33.3330
BRD6368 RT-4 CTRP1 0.2603 33.3330
BRD6368 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.