Drug : Brd63610

CTRP1 Name : BRD63610

Dataset : All
Synonyms :
Targets : NAMPT
Pathways : analog of FK866

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BRD63610 U2OS CTRP1 0.0081 1.0417
BRD63610 MCF-7 CTRP1 0.0081 1.0417
BRD63610 GAMG CTRP1 0.0027 33.3330
BRD63610 LN-229 CTRP1 0.0081 1.0417
BRD63610 SF295 CTRP1 0.2603 33.3330
BRD63610 HEC-108 CTRP1 0.0027 33.3330
BRD63610 HEC-151 CTRP1 0.0081 1.0417
BRD63610 HEC-251 CTRP1 0.2603 33.3330
BRD63610 HEC-265 CTRP1 0.2603 33.3330
BRD63610 HEC-59 CTRP1 0.0027 33.3330
BRD63610 HEC-6 CTRP1 0.2603 33.3330
BRD63610 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.0027 33.3330
BRD63610 JHUEM-2 CTRP1 0.0081 1.0417
BRD63610 KLE CTRP1 0.0027 33.3330
BRD63610 MFE-319 CTRP1 0.2603 33.3330
BRD63610 SNG-M CTRP1 0.0027 33.3330
BRD63610 AMO1 CTRP1 0.0081 1.0417
BRD63610 BL-70 CTRP1 0.0027 33.3330
BRD63610 EJM CTRP1 0.0081 1.0417
BRD63610 GDM-1 CTRP1 0.0081 1.0417
BRD63610 HT CTRP1 0.2603 33.3330
BRD63610 KMS-11 CTRP1 0.0081 1.0417
BRD63610 KU812 CTRP1 0.2603 33.3330
BRD63610 LP-1 CTRP1 0.0081 1.0417
BRD63610 MC116 CTRP1 0.2603 33.3330
BRD63610 MOLM-16 CTRP1 0.0081 1.0417
BRD63610 NOMO-1 CTRP1 0.0081 1.0417
BRD63610 NU-DUL-1 CTRP1 0.0081 1.0417
BRD63610 OCI-AML-3 CTRP1 0.0081 1.0417
BRD63610 OCI-LY10 CTRP1 0.0081 1.0417
BRD63610 P3HR-1 CTRP1 0.2603 33.3330
BRD63610 PL21 CTRP1 0.0081 1.0417
BRD63610 RPMI-8226 CTRP1 0.0081 1.0417
BRD63610 SKM-1 CTRP1 0.0081 1.0417
BRD63610 SU-DHL-4 CTRP1 0.0081 1.0417
BRD63610 SU-DHL-5 CTRP1 0.0081 1.0417
BRD63610 THP-1 CTRP1 0.0081 1.0417
BRD63610 U-937 CTRP1 0.0081 1.0417
BRD63610 WSU-DLCL2 CTRP1 0.0081 1.0417
BRD63610 RCC10RGB CTRP1 0.0081 1.0417
BRD63610 VMRC-RCW CTRP1 0.2603 33.3330
BRD63610 C2BBE1 CTRP1 0.2603 33.3330
BRD63610 CL-34 CTRP1 0.0081 1.0417
BRD63610 CL-40 CTRP1 0.0081 1.0417
BRD63610 COLO205 CTRP1 0.2603 33.3330
BRD63610 COLO320 CTRP1 0.0081 1.0417
BRD63610 COLO678 CTRP1 0.0081 1.0417
BRD63610 CW-2 CTRP1 0.0081 1.0417
BRD63610 DLD-1 CTRP1 0.2603 33.3330
BRD63610 GP2D CTRP1 0.2603 33.3330
BRD63610 HCT116 CTRP1 0.0081 1.0417
BRD63610 HCT8 CTRP1 0.0081 1.0417
BRD63610 HT115 CTRP1 0.0081 1.0417
BRD63610 HT-29 CTRP1 0.0081 1.0417
BRD63610 HT-55 CTRP1 0.0081 1.0417
BRD63610 KM12 CTRP1 0.0081 1.0417
BRD63610 LOVO CTRP1 0.0081 1.0417
BRD63610 LS123 CTRP1 0.0081 1.0417
BRD63610 LS180 CTRP1 0.0081 1.0417
BRD63610 LS411N CTRP1 0.2603 33.3330
BRD63610 LS513 CTRP1 0.2603 33.3330
BRD63610 MDST8 CTRP1 0.0081 1.0417
BRD63610 NCI-H508 CTRP1 0.0081 1.0417
BRD63610 RCM-1[HUMANESC] CTRP1 0.0081 1.0417
BRD63610 RKO CTRP1 0.0081 1.0417
BRD63610 SK-CO-1 CTRP1 0.2603 33.3330
BRD63610 SNU-1040 CTRP1 0.0081 1.0417
BRD63610 SNU-175 CTRP1 0.0081 1.0417
BRD63610 SNU-61 CTRP1 0.0081 1.0417
BRD63610 SNU-81 CTRP1 0.0081 1.0417
BRD63610 SNU-C2A CTRP1 0.2603 33.3330
BRD63610 SNU-C4 CTRP1 0.0081 1.0417
BRD63610 SNU-C5 CTRP1 0.0081 1.0417
BRD63610 SW403 CTRP1 0.2603 33.3330
BRD63610 SW48 CTRP1 0.2603 33.3330
BRD63610 SW480 CTRP1 0.0081 1.0417
BRD63610 SW620 CTRP1 0.0081 1.0417
BRD63610 SW948 CTRP1 0.0081 1.0417
BRD63610 HEP-G2 CTRP1 0.0081 1.0417
BRD63610 JHH-6 CTRP1 0.0027 33.3330
BRD63610 SNU-398 CTRP1 0.0081 1.0417
BRD63610 SNU-449 CTRP1 0.0027 33.3330
BRD63610 A-549 CTRP1 0.2603 33.3330
BRD63610 BEN CTRP1 0.2603 33.3330
BRD63610 CAL-12T CTRP1 0.0081 1.0417
BRD63610 CALU-3 CTRP1 0.2603 33.3330
BRD63610 CALU-6 CTRP1 0.2603 33.3330
BRD63610 CHAGO-K-1 CTRP1 0.2603 33.3330
BRD63610 COLO668 CTRP1 0.0027 33.3330
BRD63610 COLO699 CTRP1 0.0081 1.0417
BRD63610 COR-L23 CTRP1 0.0081 1.0417
BRD63610 COR-L279 CTRP1 0.2603 33.3330
BRD63610 COR-L51 CTRP1 0.0081 1.0417
BRD63610 COR-L88 CTRP1 0.2603 33.3330
BRD63610 DMS273 CTRP1 0.2603 33.3330
BRD63610 DV-90 CTRP1 0.2603 33.3330
BRD63610 EBC-1 CTRP1 0.2603 33.3330
BRD63610 EPLC-272H CTRP1 0.2603 33.3330
BRD63610 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
BRD63610 HCC1195 CTRP1 0.0081 1.0417
BRD63610 HCC1359 CTRP1 0.0081 1.0417
BRD63610 HCC15 CTRP1 0.0081 1.0417
BRD63610 HCC1833 CTRP1 0.0081 1.0417
BRD63610 HCC2108 CTRP1 0.0081 1.0417
BRD63610 HCC2935 CTRP1 0.0081 1.0417
BRD63610 HCC33 CTRP1 0.2603 33.3330
BRD63610 HCC4006 CTRP1 0.0081 1.0417
BRD63610 HCC44 CTRP1 0.2603 33.3330
BRD63610 HCC78 CTRP1 0.2603 33.3330
BRD63610 HCC827 CTRP1 0.0081 1.0417
BRD63610 KNS-62 CTRP1 0.2603 33.3330
BRD63610 LC-1-SQ-SF CTRP1 0.2603 33.3330
BRD63610 LCLC-103H CTRP1 0.2603 33.3330
BRD63610 LCLC-97TM1 CTRP1 0.2603 33.3330
BRD63610 LU-65 CTRP1 0.2603 33.3330
BRD63610 LU-99 CTRP1 0.2603 33.3330
BRD63610 LXF289 CTRP1 0.0027 33.3330
BRD63610 NCI-H1048 CTRP1 0.2603 33.3330
BRD63610 NCI-H1105 CTRP1 0.0081 1.0417
BRD63610 NCI-H1299 CTRP1 0.2603 33.3330
BRD63610 NCI-H1355 CTRP1 0.2603 33.3330
BRD63610 NCI-H1373 CTRP1 0.2603 33.3330
BRD63610 NCI-H1435 CTRP1 0.0027 33.3330
BRD63610 NCI-H1437 CTRP1 0.2603 33.3330
BRD63610 NCI-H1568 CTRP1 0.2603 33.3330
BRD63610 NCI-H1573 CTRP1 0.2603 33.3330
BRD63610 NCI-H1666 CTRP1 0.2603 33.3330
BRD63610 NCI-H1694 CTRP1 0.0081 1.0417
BRD63610 NCI-H1755 CTRP1 0.0081 1.0417
BRD63610 NCI-H1781 CTRP1 0.0081 1.0417
BRD63610 NCI-H1792 CTRP1 0.2603 33.3330
BRD63610 NCI-H1793 CTRP1 0.2603 33.3330
BRD63610 NCI-H1836 CTRP1 0.0081 1.0417
BRD63610 NCI-H1876 CTRP1 0.0081 1.0417
BRD63610 NCI-H1915 CTRP1 0.0027 33.3330
BRD63610 NCI-H1930 CTRP1 0.0027 33.3330
BRD63610 NCI-H1944 CTRP1 0.2603 33.3330
BRD63610 NCI-H1963 CTRP1 0.0081 1.0417
BRD63610 NCI-H1975 CTRP1 0.2603 33.3330
BRD63610 NCI-H2009 CTRP1 0.2603 33.3330
BRD63610 NCI-H2023 CTRP1 0.0081 1.0417
BRD63610 NCI-H2029 CTRP1 0.2603 33.3330
BRD63610 NCI-H2030 CTRP1 0.0081 1.0417
BRD63610 NCI-H2073 CTRP1 0.0081 1.0417
BRD63610 NCI-H2081 CTRP1 0.0081 1.0417
BRD63610 NCI-H2110 CTRP1 0.0081 1.0417
BRD63610 NCI-H2122 CTRP1 0.0081 1.0417
BRD63610 NCI-H2126 CTRP1 0.2603 33.3330
BRD63610 NCI-H2141 CTRP1 0.0081 1.0417
BRD63610 NCI-H2172 CTRP1 0.0081 1.0417
BRD63610 NCI-H2286 CTRP1 0.0027 33.3330
BRD63610 NCI-H23 CTRP1 0.2603 33.3330
BRD63610 NCI-H2342 CTRP1 0.0081 1.0417
BRD63610 NCI-H2405 CTRP1 0.2603 33.3330
BRD63610 NCI-H3255 CTRP1 0.0081 1.0417
BRD63610 NCI-H358 CTRP1 0.2603 33.3330
BRD63610 NCI-H441 CTRP1 0.0081 1.0417
BRD63610 NCI-H460 CTRP1 0.0081 1.0417
BRD63610 NCI-H522 CTRP1 0.2603 33.3330
BRD63610 NCI-H596 CTRP1 0.0081 1.0417
BRD63610 NCI-H650 CTRP1 0.2603 33.3330
BRD63610 NCI-H661 CTRP1 0.2603 33.3330
BRD63610 NCI-H727 CTRP1 0.2603 33.3330
BRD63610 NCI-H810 CTRP1 0.2603 33.3330
BRD63610 NCI-H82 CTRP1 0.2603 33.3330
BRD63610 NCI-H841 CTRP1 0.0081 1.0417
BRD63610 RERF-LC-KJ CTRP1 0.0027 33.3330
BRD63610 SCLC-21H CTRP1 0.0081 1.0417
BRD63610 SHP-77 CTRP1 0.2603 33.3330
BRD63610 SK-LU-1 CTRP1 0.0081 1.0417
BRD63610 SQ-1 CTRP1 0.0081 1.0417
BRD63610 T3M-10 CTRP1 0.0081 1.0417
BRD63610 VMRC-LCD CTRP1 0.2603 33.3330
BRD63610 KYSE-140 CTRP1 0.2603 33.3330
BRD63610 KYSE-410 CTRP1 0.2603 33.3330
BRD63610 KYSE-450 CTRP1 0.2603 33.3330
BRD63610 A2780 CTRP1 0.0081 1.0417
BRD63610 CAOV-3 CTRP1 0.0081 1.0417
BRD63610 COV318 CTRP1 0.0027 33.3330
BRD63610 COV362 CTRP1 0.0081 1.0417
BRD63610 COV434 CTRP1 0.0081 1.0417
BRD63610 COV644 CTRP1 0.0081 1.0417
BRD63610 EFO-21 CTRP1 0.2603 33.3330
BRD63610 EFO-27 CTRP1 0.0081 1.0417
BRD63610 HEYA8 CTRP1 0.2603 33.3330
BRD63610 IGROV-1 CTRP1 0.0081 1.0417
BRD63610 JHOC-5 CTRP1 0.0081 1.0417
BRD63610 JHOM-1 CTRP1 0.0081 1.0417
BRD63610 JHOS-4 CTRP1 0.0027 33.3330
BRD63610 OAW42 CTRP1 0.0081 1.0417
BRD63610 OV7 CTRP1 0.0081 1.0417
BRD63610 OV-90 CTRP1 0.0081 1.0417
BRD63610 OVCAR-4 CTRP1 0.0081 1.0417
BRD63610 OVCAR-8 CTRP1 0.0081 1.0417
BRD63610 OVK18 CTRP1 0.0081 1.0417
BRD63610 OVKATE CTRP1 0.0081 1.0417
BRD63610 OVMANA CTRP1 0.0027 33.3330
BRD63610 RKN CTRP1 0.0081 1.0417
BRD63610 RMG-I CTRP1 0.0081 1.0417
BRD63610 RMUG-S CTRP1 0.0081 1.0417
BRD63610 SK-OV-3 CTRP1 0.2603 33.3330
BRD63610 SNU-840 CTRP1 0.0081 1.0417
BRD63610 TYK-NU CTRP1 0.0081 1.0417
BRD63610 CAPAN-2 CTRP1 0.2603 33.3330
BRD63610 CFPAC-1 CTRP1 0.2603 33.3330
BRD63610 HPAC CTRP1 0.2603 33.3330
BRD63610 HUP-T4 CTRP1 0.2603 33.3330
BRD63610 KP-3 CTRP1 0.2603 33.3330
BRD63610 PANC03.27 CTRP1 0.2603 33.3330
BRD63610 PANC10.05 CTRP1 0.2603 33.3330
BRD63610 PATU8902 CTRP1 0.0027 33.3330
BRD63610 QGP-1 CTRP1 0.2603 33.3330
BRD63610 SUIT-2 CTRP1 0.2603 33.3330
BRD63610 MSTO-211H CTRP1 0.2603 33.3330
BRD63610 NCI-H2052 CTRP1 0.2603 33.3330
BRD63610 NCI-H28 CTRP1 0.2603 33.3330
BRD63610 MIAPACA-3 CTRP1 0.0027 33.3330
BRD63610 A-375 CTRP1 0.0081 1.0417
BRD63610 COLO741 CTRP1 0.2603 33.3330
BRD63610 G-361 CTRP1 0.2603 33.3330
BRD63610 HS852.T CTRP1 0.0027 33.3330
BRD63610 HS936.T CTRP1 0.2603 33.3330
BRD63610 HS944.T CTRP1 0.2603 33.3330
BRD63610 SK-MEL-1 CTRP1 0.0081 1.0417
BRD63610 SK-MEL-28 CTRP1 0.0081 1.0417
BRD63610 SK-MEL-5 CTRP1 0.0081 1.0417
BRD63610 G-401 CTRP1 0.2603 33.3330
BRD63610 HT-1080 CTRP1 0.0081 1.0417
BRD63610 AGS CTRP1 0.0081 1.0417
BRD63610 FU97 CTRP1 0.2603 33.3330
BRD63610 KE-97 CTRP1 0.2603 33.3330
BRD63610 MKN7 CTRP1 0.2603 33.3330
BRD63610 MKN74 CTRP1 0.0027 33.3330
BRD63610 NUGC-4 CTRP1 0.2603 33.3330
BRD63610 SH-10-TC CTRP1 0.2603 33.3330
BRD63610 HSC-2 CTRP1 0.2603 33.3330
BRD63610 SCC-9 CTRP1 0.0081 1.0417
BRD63610 5637 CTRP1 0.2603 33.3330
BRD63610 HT-1376 CTRP1 0.2603 33.3330
BRD63610 KMBC-2 CTRP1 0.2603 33.3330
BRD63610 RT-4 CTRP1 0.2603 33.3330
BRD63610 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.