Drug : Maraviroc

CTRP1 Name : maraviroc

Dataset : All
Synonyms :
Targets : CCR5
Pathways : negative allosteric modulator of chemokine (C-C motif) receptor 5

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
maraviroc U2OS CTRP1 0.2604 33.3330
maraviroc MCF-7 CTRP1 0.2604 33.3330
maraviroc GAMG CTRP1 0.2603 33.3330
maraviroc LN-229 CTRP1 0.2604 33.3330
maraviroc SF295 CTRP1 0.2603 33.3330
maraviroc HEC-108 CTRP1 0.2603 33.3330
maraviroc HEC-151 CTRP1 0.2604 33.3330
maraviroc HEC-251 CTRP1 0.2603 33.3330
maraviroc HEC-265 CTRP1 0.2603 33.3330
maraviroc HEC-59 CTRP1 0.2603 33.3330
maraviroc HEC-6 CTRP1 0.2603 33.3330
maraviroc ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
maraviroc JHUEM-2 CTRP1 0.2604 33.3330
maraviroc KLE CTRP1 0.2603 33.3330
maraviroc MFE-319 CTRP1 0.2603 33.3330
maraviroc SNG-M CTRP1 0.2603 33.3330
maraviroc AMO1 CTRP1 0.2604 33.3330
maraviroc BL-70 CTRP1 0.2603 33.3330
maraviroc EJM CTRP1 0.2604 33.3330
maraviroc GDM-1 CTRP1 0.2604 33.3330
maraviroc HT CTRP1 0.2603 33.3330
maraviroc KMS-11 CTRP1 0.2604 33.3330
maraviroc KU812 CTRP1 0.2603 33.3330
maraviroc LP-1 CTRP1 0.2604 33.3330
maraviroc MC116 CTRP1 0.2603 33.3330
maraviroc MOLM-16 CTRP1 0.2604 33.3330
maraviroc NOMO-1 CTRP1 0.2604 33.3330
maraviroc NU-DUL-1 CTRP1 0.2604 33.3330
maraviroc OCI-AML-3 CTRP1 0.2604 33.3330
maraviroc OCI-LY10 CTRP1 0.2604 33.3330
maraviroc P3HR-1 CTRP1 0.2603 33.3330
maraviroc PL21 CTRP1 0.2604 33.3330
maraviroc RPMI-8226 CTRP1 0.2604 33.3330
maraviroc SKM-1 CTRP1 0.2604 33.3330
maraviroc SU-DHL-4 CTRP1 0.2604 33.3330
maraviroc SU-DHL-5 CTRP1 0.2604 33.3330
maraviroc THP-1 CTRP1 0.2604 33.3330
maraviroc U-937 CTRP1 0.2604 33.3330
maraviroc WSU-DLCL2 CTRP1 0.2604 33.3330
maraviroc RCC10RGB CTRP1 0.2604 33.3330
maraviroc VMRC-RCW CTRP1 0.2603 33.3330
maraviroc C2BBE1 CTRP1 0.2603 33.3330
maraviroc CL-34 CTRP1 0.2604 33.3330
maraviroc CL-40 CTRP1 0.2604 33.3330
maraviroc COLO205 CTRP1 0.2603 33.3330
maraviroc COLO320 CTRP1 0.2604 33.3330
maraviroc COLO678 CTRP1 0.2604 33.3330
maraviroc CW-2 CTRP1 0.2604 33.3330
maraviroc DLD-1 CTRP1 0.2603 33.3330
maraviroc GP2D CTRP1 0.2603 33.3330
maraviroc HCT116 CTRP1 0.2604 33.3330
maraviroc HCT8 CTRP1 0.2604 33.3330
maraviroc HT115 CTRP1 0.2604 33.3330
maraviroc HT-29 CTRP1 0.2604 33.3330
maraviroc HT-55 CTRP1 0.2604 33.3330
maraviroc KM12 CTRP1 0.2604 33.3330
maraviroc LOVO CTRP1 0.2604 33.3330
maraviroc LS123 CTRP1 0.2604 33.3330
maraviroc LS180 CTRP1 0.2604 33.3330
maraviroc LS411N CTRP1 0.2603 33.3330
maraviroc LS513 CTRP1 0.2603 33.3330
maraviroc MDST8 CTRP1 0.2604 33.3330
maraviroc NCI-H508 CTRP1 0.2604 33.3330
maraviroc RCM-1[HUMANESC] CTRP1 0.2604 33.3330
maraviroc RKO CTRP1 0.2604 33.3330
maraviroc SK-CO-1 CTRP1 0.2603 33.3330
maraviroc SNU-1040 CTRP1 0.2604 33.3330
maraviroc SNU-175 CTRP1 0.2604 33.3330
maraviroc SNU-61 CTRP1 0.2604 33.3330
maraviroc SNU-81 CTRP1 0.2604 33.3330
maraviroc SNU-C2A CTRP1 0.2603 33.3330
maraviroc SNU-C4 CTRP1 0.2604 33.3330
maraviroc SNU-C5 CTRP1 0.2604 33.3330
maraviroc SW403 CTRP1 0.2603 33.3330
maraviroc SW48 CTRP1 0.2603 33.3330
maraviroc SW480 CTRP1 0.2604 33.3330
maraviroc SW620 CTRP1 0.2604 33.3330
maraviroc SW948 CTRP1 0.2604 33.3330
maraviroc HEP-G2 CTRP1 0.2604 33.3330
maraviroc JHH-6 CTRP1 0.2603 33.3330
maraviroc SNU-398 CTRP1 0.2604 33.3330
maraviroc SNU-449 CTRP1 0.2603 33.3330
maraviroc A-549 CTRP1 0.2603 33.3330
maraviroc BEN CTRP1 0.2603 33.3330
maraviroc CAL-12T CTRP1 0.2604 33.3330
maraviroc CALU-3 CTRP1 0.2603 33.3330
maraviroc CALU-6 CTRP1 0.2603 33.3330
maraviroc CHAGO-K-1 CTRP1 0.2603 33.3330
maraviroc COLO668 CTRP1 0.2603 33.3330
maraviroc COLO699 CTRP1 0.2604 33.3330
maraviroc COR-L23 CTRP1 0.2604 33.3330
maraviroc COR-L279 CTRP1 0.2603 33.3330
maraviroc COR-L51 CTRP1 0.2604 33.3330
maraviroc COR-L88 CTRP1 0.2603 33.3330
maraviroc DMS273 CTRP1 0.2603 33.3330
maraviroc DV-90 CTRP1 0.2603 33.3330
maraviroc EBC-1 CTRP1 0.2603 33.3330
maraviroc EPLC-272H CTRP1 0.2603 33.3330
maraviroc HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
maraviroc HCC1195 CTRP1 0.2604 33.3330
maraviroc HCC1359 CTRP1 0.2604 33.3330
maraviroc HCC15 CTRP1 0.2604 33.3330
maraviroc HCC1833 CTRP1 0.2604 33.3330
maraviroc HCC2108 CTRP1 0.2604 33.3330
maraviroc HCC2935 CTRP1 0.2604 33.3330
maraviroc HCC33 CTRP1 0.2603 33.3330
maraviroc HCC4006 CTRP1 0.2604 33.3330
maraviroc HCC44 CTRP1 0.2603 33.3330
maraviroc HCC78 CTRP1 0.2603 33.3330
maraviroc HCC827 CTRP1 0.2604 33.3330
maraviroc KNS-62 CTRP1 0.2603 33.3330
maraviroc LC-1-SQ-SF CTRP1 0.2603 33.3330
maraviroc LCLC-103H CTRP1 0.2603 33.3330
maraviroc LCLC-97TM1 CTRP1 0.2603 33.3330
maraviroc LU-65 CTRP1 0.2603 33.3330
maraviroc LU-99 CTRP1 0.2603 33.3330
maraviroc LXF289 CTRP1 0.2603 33.3330
maraviroc NCI-H1048 CTRP1 0.2603 33.3330
maraviroc NCI-H1105 CTRP1 0.2604 33.3330
maraviroc NCI-H1299 CTRP1 0.2603 33.3330
maraviroc NCI-H1355 CTRP1 0.2603 33.3330
maraviroc NCI-H1373 CTRP1 0.2603 33.3330
maraviroc NCI-H1435 CTRP1 0.2603 33.3330
maraviroc NCI-H1437 CTRP1 0.2603 33.3330
maraviroc NCI-H1568 CTRP1 0.2603 33.3330
maraviroc NCI-H1573 CTRP1 0.2603 33.3330
maraviroc NCI-H1666 CTRP1 0.2603 33.3330
maraviroc NCI-H1694 CTRP1 0.2604 33.3330
maraviroc NCI-H1755 CTRP1 0.2604 33.3330
maraviroc NCI-H1781 CTRP1 0.2604 33.3330
maraviroc NCI-H1792 CTRP1 0.2603 33.3330
maraviroc NCI-H1793 CTRP1 0.2603 33.3330
maraviroc NCI-H1836 CTRP1 0.2604 33.3330
maraviroc NCI-H1876 CTRP1 0.2604 33.3330
maraviroc NCI-H1915 CTRP1 0.2603 33.3330
maraviroc NCI-H1930 CTRP1 0.2603 33.3330
maraviroc NCI-H1944 CTRP1 0.2603 33.3330
maraviroc NCI-H1963 CTRP1 0.2604 33.3330
maraviroc NCI-H1975 CTRP1 0.2603 33.3330
maraviroc NCI-H2009 CTRP1 0.2603 33.3330
maraviroc NCI-H2023 CTRP1 0.2604 33.3330
maraviroc NCI-H2029 CTRP1 0.2603 33.3330
maraviroc NCI-H2030 CTRP1 0.2604 33.3330
maraviroc NCI-H2073 CTRP1 0.2604 33.3330
maraviroc NCI-H2081 CTRP1 0.2604 33.3330
maraviroc NCI-H2110 CTRP1 0.2604 33.3330
maraviroc NCI-H2122 CTRP1 0.2604 33.3330
maraviroc NCI-H2126 CTRP1 0.2603 33.3330
maraviroc NCI-H2141 CTRP1 0.2604 33.3330
maraviroc NCI-H2172 CTRP1 0.2604 33.3330
maraviroc NCI-H2286 CTRP1 0.2603 33.3330
maraviroc NCI-H23 CTRP1 0.2603 33.3330
maraviroc NCI-H2342 CTRP1 0.2604 33.3330
maraviroc NCI-H2405 CTRP1 0.2603 33.3330
maraviroc NCI-H3255 CTRP1 0.2604 33.3330
maraviroc NCI-H358 CTRP1 0.2603 33.3330
maraviroc NCI-H441 CTRP1 0.2604 33.3330
maraviroc NCI-H460 CTRP1 0.2604 33.3330
maraviroc NCI-H522 CTRP1 0.2603 33.3330
maraviroc NCI-H596 CTRP1 0.2604 33.3330
maraviroc NCI-H650 CTRP1 0.2603 33.3330
maraviroc NCI-H661 CTRP1 0.2603 33.3330
maraviroc NCI-H727 CTRP1 0.2603 33.3330
maraviroc NCI-H810 CTRP1 0.2603 33.3330
maraviroc NCI-H82 CTRP1 0.2603 33.3330
maraviroc NCI-H841 CTRP1 0.2604 33.3330
maraviroc RERF-LC-KJ CTRP1 0.2603 33.3330
maraviroc SCLC-21H CTRP1 0.2604 33.3330
maraviroc SHP-77 CTRP1 0.2603 33.3330
maraviroc SK-LU-1 CTRP1 0.2604 33.3330
maraviroc SQ-1 CTRP1 0.2604 33.3330
maraviroc T3M-10 CTRP1 0.2604 33.3330
maraviroc VMRC-LCD CTRP1 0.2603 33.3330
maraviroc KYSE-140 CTRP1 0.2603 33.3330
maraviroc KYSE-410 CTRP1 0.2603 33.3330
maraviroc KYSE-450 CTRP1 0.2603 33.3330
maraviroc A2780 CTRP1 0.2604 33.3330
maraviroc CAOV-3 CTRP1 0.2604 33.3330
maraviroc COV318 CTRP1 0.2603 33.3330
maraviroc COV362 CTRP1 0.2604 33.3330
maraviroc COV434 CTRP1 0.2604 33.3330
maraviroc COV644 CTRP1 0.2604 33.3330
maraviroc EFO-21 CTRP1 0.2603 33.3330
maraviroc EFO-27 CTRP1 0.2604 33.3330
maraviroc HEYA8 CTRP1 0.2603 33.3330
maraviroc IGROV-1 CTRP1 0.2604 33.3330
maraviroc JHOC-5 CTRP1 0.2604 33.3330
maraviroc JHOM-1 CTRP1 0.2604 33.3330
maraviroc JHOS-4 CTRP1 0.2603 33.3330
maraviroc OAW42 CTRP1 0.2604 33.3330
maraviroc OV7 CTRP1 0.2604 33.3330
maraviroc OV-90 CTRP1 0.2604 33.3330
maraviroc OVCAR-4 CTRP1 0.2604 33.3330
maraviroc OVCAR-8 CTRP1 0.2604 33.3330
maraviroc OVK18 CTRP1 0.2604 33.3330
maraviroc OVKATE CTRP1 0.2604 33.3330
maraviroc OVMANA CTRP1 0.2603 33.3330
maraviroc RKN CTRP1 0.2604 33.3330
maraviroc RMG-I CTRP1 0.2604 33.3330
maraviroc RMUG-S CTRP1 0.2604 33.3330
maraviroc SK-OV-3 CTRP1 0.2603 33.3330
maraviroc SNU-840 CTRP1 0.2604 33.3330
maraviroc TYK-NU CTRP1 0.2604 33.3330
maraviroc CAPAN-2 CTRP1 0.2603 33.3330
maraviroc CFPAC-1 CTRP1 0.2603 33.3330
maraviroc HPAC CTRP1 0.2603 33.3330
maraviroc HUP-T4 CTRP1 0.2603 33.3330
maraviroc KP-3 CTRP1 0.2603 33.3330
maraviroc PANC03.27 CTRP1 0.2603 33.3330
maraviroc PANC10.05 CTRP1 0.2603 33.3330
maraviroc PATU8902 CTRP1 0.2603 33.3330
maraviroc QGP-1 CTRP1 0.2603 33.3330
maraviroc SUIT-2 CTRP1 0.2603 33.3330
maraviroc MSTO-211H CTRP1 0.2603 33.3330
maraviroc NCI-H2052 CTRP1 0.2603 33.3330
maraviroc NCI-H28 CTRP1 0.2603 33.3330
maraviroc MIAPACA-3 CTRP1 0.2603 33.3330
maraviroc A-375 CTRP1 0.2604 33.3330
maraviroc COLO741 CTRP1 0.2603 33.3330
maraviroc G-361 CTRP1 0.2603 33.3330
maraviroc HS852.T CTRP1 0.2603 33.3330
maraviroc HS936.T CTRP1 0.2603 33.3330
maraviroc HS944.T CTRP1 0.2603 33.3330
maraviroc SK-MEL-1 CTRP1 0.2604 33.3330
maraviroc SK-MEL-28 CTRP1 0.2604 33.3330
maraviroc SK-MEL-5 CTRP1 0.2604 33.3330
maraviroc G-401 CTRP1 0.2603 33.3330
maraviroc HT-1080 CTRP1 0.2604 33.3330
maraviroc AGS CTRP1 0.2604 33.3330
maraviroc FU97 CTRP1 0.2603 33.3330
maraviroc KE-97 CTRP1 0.2603 33.3330
maraviroc MKN7 CTRP1 0.2603 33.3330
maraviroc MKN74 CTRP1 0.2603 33.3330
maraviroc NUGC-4 CTRP1 0.2603 33.3330
maraviroc SH-10-TC CTRP1 0.2603 33.3330
maraviroc HSC-2 CTRP1 0.2603 33.3330
maraviroc SCC-9 CTRP1 0.2604 33.3330
maraviroc 5637 CTRP1 0.2603 33.3330
maraviroc HT-1376 CTRP1 0.2603 33.3330
maraviroc KMBC-2 CTRP1 0.2603 33.3330
maraviroc RT-4 CTRP1 0.2603 33.3330
maraviroc UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.