Drug : Mk-591

CTRP1 Name : MK-591

Dataset : All
Synonyms :
Targets : ALOX5AP
Pathways : inhibitor of arachidonate 5-lipoxygenase-activating protein (FLAP)

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
MK-591 U2OS CTRP1 2.0833 266.6700
MK-591 MCF-7 CTRP1 2.0833 266.6700
MK-591 GAMG CTRP1 0.2603 33.3330
MK-591 LN-229 CTRP1 2.0833 266.6700
MK-591 SF295 CTRP1 0.2603 33.3330
MK-591 HEC-108 CTRP1 0.2603 33.3330
MK-591 HEC-151 CTRP1 2.0833 266.6700
MK-591 HEC-251 CTRP1 0.2603 33.3330
MK-591 HEC-265 CTRP1 0.2603 33.3330
MK-591 HEC-59 CTRP1 0.2603 33.3330
MK-591 HEC-6 CTRP1 0.2603 33.3330
MK-591 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
MK-591 JHUEM-2 CTRP1 2.0833 266.6700
MK-591 KLE CTRP1 0.2603 33.3330
MK-591 MFE-319 CTRP1 0.2603 33.3330
MK-591 SNG-M CTRP1 0.2603 33.3330
MK-591 AMO1 CTRP1 2.0833 266.6700
MK-591 BL-70 CTRP1 0.2603 33.3330
MK-591 EJM CTRP1 2.0833 266.6700
MK-591 GDM-1 CTRP1 2.0833 266.6700
MK-591 HT CTRP1 0.2603 33.3330
MK-591 KMS-11 CTRP1 2.0833 266.6700
MK-591 KU812 CTRP1 0.2603 33.3330
MK-591 LP-1 CTRP1 2.0833 266.6700
MK-591 MC116 CTRP1 0.2603 33.3330
MK-591 MOLM-16 CTRP1 2.0833 266.6700
MK-591 NOMO-1 CTRP1 2.0833 266.6700
MK-591 NU-DUL-1 CTRP1 2.0833 266.6700
MK-591 OCI-AML-3 CTRP1 2.0833 266.6700
MK-591 OCI-LY10 CTRP1 2.0833 266.6700
MK-591 P3HR-1 CTRP1 0.2603 33.3330
MK-591 PL21 CTRP1 2.0833 266.6700
MK-591 RPMI-8226 CTRP1 2.0833 266.6700
MK-591 SKM-1 CTRP1 2.0833 266.6700
MK-591 SU-DHL-4 CTRP1 2.0833 266.6700
MK-591 SU-DHL-5 CTRP1 2.0833 266.6700
MK-591 THP-1 CTRP1 2.0833 266.6700
MK-591 U-937 CTRP1 2.0833 266.6700
MK-591 WSU-DLCL2 CTRP1 2.0833 266.6700
MK-591 RCC10RGB CTRP1 2.0833 266.6700
MK-591 VMRC-RCW CTRP1 0.2603 33.3330
MK-591 C2BBE1 CTRP1 0.2603 33.3330
MK-591 CL-34 CTRP1 2.0833 266.6700
MK-591 CL-40 CTRP1 2.0833 266.6700
MK-591 COLO205 CTRP1 0.2603 33.3330
MK-591 COLO320 CTRP1 2.0833 266.6700
MK-591 COLO678 CTRP1 2.0833 266.6700
MK-591 CW-2 CTRP1 2.0833 266.6700
MK-591 DLD-1 CTRP1 0.2603 33.3330
MK-591 GP2D CTRP1 0.2603 33.3330
MK-591 HCT116 CTRP1 2.0833 266.6700
MK-591 HCT8 CTRP1 2.0833 266.6700
MK-591 HT115 CTRP1 2.0833 266.6700
MK-591 HT-29 CTRP1 2.0833 266.6700
MK-591 HT-55 CTRP1 2.0833 266.6700
MK-591 KM12 CTRP1 2.0833 266.6700
MK-591 LOVO CTRP1 2.0833 266.6700
MK-591 LS123 CTRP1 2.0833 266.6700
MK-591 LS180 CTRP1 2.0833 266.6700
MK-591 LS411N CTRP1 0.2603 33.3330
MK-591 LS513 CTRP1 0.2603 33.3330
MK-591 MDST8 CTRP1 2.0833 266.6700
MK-591 NCI-H508 CTRP1 2.0833 266.6700
MK-591 RCM-1[HUMANESC] CTRP1 2.0833 266.6700
MK-591 RKO CTRP1 2.0833 266.6700
MK-591 SK-CO-1 CTRP1 0.2603 33.3330
MK-591 SNU-1040 CTRP1 2.0833 266.6700
MK-591 SNU-175 CTRP1 2.0833 266.6700
MK-591 SNU-61 CTRP1 2.0833 266.6700
MK-591 SNU-81 CTRP1 2.0833 266.6700
MK-591 SNU-C2A CTRP1 0.2603 33.3330
MK-591 SNU-C4 CTRP1 2.0833 266.6700
MK-591 SNU-C5 CTRP1 2.0833 266.6700
MK-591 SW403 CTRP1 0.2603 33.3330
MK-591 SW48 CTRP1 0.2603 33.3330
MK-591 SW480 CTRP1 2.0833 266.6700
MK-591 SW620 CTRP1 2.0833 266.6700
MK-591 SW948 CTRP1 2.0833 266.6700
MK-591 HEP-G2 CTRP1 2.0833 266.6700
MK-591 JHH-6 CTRP1 0.2603 33.3330
MK-591 SNU-398 CTRP1 2.0833 266.6700
MK-591 SNU-449 CTRP1 0.2603 33.3330
MK-591 A-549 CTRP1 0.2603 33.3330
MK-591 BEN CTRP1 0.2603 33.3330
MK-591 CAL-12T CTRP1 2.0833 266.6700
MK-591 CALU-3 CTRP1 0.2603 33.3330
MK-591 CALU-6 CTRP1 0.2603 33.3330
MK-591 CHAGO-K-1 CTRP1 0.2603 33.3330
MK-591 COLO668 CTRP1 0.2603 33.3330
MK-591 COLO699 CTRP1 2.0833 266.6700
MK-591 COR-L23 CTRP1 2.0833 266.6700
MK-591 COR-L279 CTRP1 0.2603 33.3330
MK-591 COR-L51 CTRP1 2.0833 266.6700
MK-591 COR-L88 CTRP1 0.2603 33.3330
MK-591 DMS273 CTRP1 0.2603 33.3330
MK-591 DV-90 CTRP1 0.2603 33.3330
MK-591 EBC-1 CTRP1 0.2603 33.3330
MK-591 EPLC-272H CTRP1 0.2603 33.3330
MK-591 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
MK-591 HCC1195 CTRP1 2.0833 266.6700
MK-591 HCC1359 CTRP1 2.0833 266.6700
MK-591 HCC15 CTRP1 2.0833 266.6700
MK-591 HCC1833 CTRP1 2.0833 266.6700
MK-591 HCC2108 CTRP1 2.0833 266.6700
MK-591 HCC2935 CTRP1 2.0833 266.6700
MK-591 HCC33 CTRP1 0.2603 33.3330
MK-591 HCC4006 CTRP1 2.0833 266.6700
MK-591 HCC44 CTRP1 0.2603 33.3330
MK-591 HCC78 CTRP1 0.2603 33.3330
MK-591 HCC827 CTRP1 2.0833 266.6700
MK-591 KNS-62 CTRP1 0.2603 33.3330
MK-591 LC-1-SQ-SF CTRP1 0.2603 33.3330
MK-591 LCLC-103H CTRP1 0.2603 33.3330
MK-591 LCLC-97TM1 CTRP1 0.2603 33.3330
MK-591 LU-65 CTRP1 0.2603 33.3330
MK-591 LU-99 CTRP1 0.2603 33.3330
MK-591 LXF289 CTRP1 0.2603 33.3330
MK-591 NCI-H1048 CTRP1 0.2603 33.3330
MK-591 NCI-H1105 CTRP1 2.0833 266.6700
MK-591 NCI-H1299 CTRP1 0.2603 33.3330
MK-591 NCI-H1355 CTRP1 0.2603 33.3330
MK-591 NCI-H1373 CTRP1 0.2603 33.3330
MK-591 NCI-H1435 CTRP1 0.2603 33.3330
MK-591 NCI-H1437 CTRP1 0.2603 33.3330
MK-591 NCI-H1568 CTRP1 0.2603 33.3330
MK-591 NCI-H1573 CTRP1 0.2603 33.3330
MK-591 NCI-H1666 CTRP1 0.2603 33.3330
MK-591 NCI-H1694 CTRP1 2.0833 266.6700
MK-591 NCI-H1755 CTRP1 2.0833 266.6700
MK-591 NCI-H1781 CTRP1 2.0833 266.6700
MK-591 NCI-H1792 CTRP1 0.2603 33.3330
MK-591 NCI-H1793 CTRP1 0.2603 33.3330
MK-591 NCI-H1836 CTRP1 2.0833 266.6700
MK-591 NCI-H1876 CTRP1 2.0833 266.6700
MK-591 NCI-H1915 CTRP1 0.2603 33.3330
MK-591 NCI-H1930 CTRP1 0.2603 33.3330
MK-591 NCI-H1944 CTRP1 0.2603 33.3330
MK-591 NCI-H1963 CTRP1 2.0833 266.6700
MK-591 NCI-H1975 CTRP1 0.2603 33.3330
MK-591 NCI-H2009 CTRP1 0.2603 33.3330
MK-591 NCI-H2023 CTRP1 2.0833 266.6700
MK-591 NCI-H2029 CTRP1 0.2603 33.3330
MK-591 NCI-H2030 CTRP1 2.0833 266.6700
MK-591 NCI-H2073 CTRP1 2.0833 266.6700
MK-591 NCI-H2081 CTRP1 2.0833 266.6700
MK-591 NCI-H2110 CTRP1 2.0833 266.6700
MK-591 NCI-H2122 CTRP1 2.0833 266.6700
MK-591 NCI-H2126 CTRP1 0.2603 33.3330
MK-591 NCI-H2141 CTRP1 2.0833 266.6700
MK-591 NCI-H2172 CTRP1 2.0833 266.6700
MK-591 NCI-H2286 CTRP1 0.2603 33.3330
MK-591 NCI-H23 CTRP1 0.2603 33.3330
MK-591 NCI-H2342 CTRP1 2.0833 266.6700
MK-591 NCI-H2405 CTRP1 0.2603 33.3330
MK-591 NCI-H3255 CTRP1 2.0833 266.6700
MK-591 NCI-H358 CTRP1 0.2603 33.3330
MK-591 NCI-H441 CTRP1 2.0833 266.6700
MK-591 NCI-H460 CTRP1 2.0833 266.6700
MK-591 NCI-H522 CTRP1 0.2603 33.3330
MK-591 NCI-H596 CTRP1 2.0833 266.6700
MK-591 NCI-H650 CTRP1 0.2603 33.3330
MK-591 NCI-H661 CTRP1 0.2603 33.3330
MK-591 NCI-H727 CTRP1 0.2603 33.3330
MK-591 NCI-H810 CTRP1 0.2603 33.3330
MK-591 NCI-H82 CTRP1 0.2603 33.3330
MK-591 NCI-H841 CTRP1 2.0833 266.6700
MK-591 RERF-LC-KJ CTRP1 0.2603 33.3330
MK-591 SCLC-21H CTRP1 2.0833 266.6700
MK-591 SHP-77 CTRP1 0.2603 33.3330
MK-591 SK-LU-1 CTRP1 2.0833 266.6700
MK-591 SQ-1 CTRP1 2.0833 266.6700
MK-591 T3M-10 CTRP1 2.0833 266.6700
MK-591 VMRC-LCD CTRP1 0.2603 33.3330
MK-591 KYSE-140 CTRP1 0.2603 33.3330
MK-591 KYSE-410 CTRP1 0.2603 33.3330
MK-591 KYSE-450 CTRP1 0.2603 33.3330
MK-591 A2780 CTRP1 2.0833 266.6700
MK-591 CAOV-3 CTRP1 2.0833 266.6700
MK-591 COV318 CTRP1 0.2603 33.3330
MK-591 COV362 CTRP1 2.0833 266.6700
MK-591 COV434 CTRP1 2.0833 266.6700
MK-591 COV644 CTRP1 2.0833 266.6700
MK-591 EFO-21 CTRP1 0.2603 33.3330
MK-591 EFO-27 CTRP1 2.0833 266.6700
MK-591 HEYA8 CTRP1 0.2603 33.3330
MK-591 IGROV-1 CTRP1 2.0833 266.6700
MK-591 JHOC-5 CTRP1 2.0833 266.6700
MK-591 JHOM-1 CTRP1 2.0833 266.6700
MK-591 JHOS-4 CTRP1 0.2603 33.3330
MK-591 OAW42 CTRP1 2.0833 266.6700
MK-591 OV7 CTRP1 2.0833 266.6700
MK-591 OV-90 CTRP1 2.0833 266.6700
MK-591 OVCAR-4 CTRP1 2.0833 266.6700
MK-591 OVCAR-8 CTRP1 2.0833 266.6700
MK-591 OVK18 CTRP1 2.0833 266.6700
MK-591 OVKATE CTRP1 2.0833 266.6700
MK-591 OVMANA CTRP1 0.2603 33.3330
MK-591 RKN CTRP1 2.0833 266.6700
MK-591 RMG-I CTRP1 2.0833 266.6700
MK-591 RMUG-S CTRP1 2.0833 266.6700
MK-591 SK-OV-3 CTRP1 0.2603 33.3330
MK-591 SNU-840 CTRP1 2.0833 266.6700
MK-591 TYK-NU CTRP1 2.0833 266.6700
MK-591 CAPAN-2 CTRP1 0.2603 33.3330
MK-591 CFPAC-1 CTRP1 0.2603 33.3330
MK-591 HPAC CTRP1 0.2603 33.3330
MK-591 HUP-T4 CTRP1 0.2603 33.3330
MK-591 KP-3 CTRP1 0.2603 33.3330
MK-591 PANC03.27 CTRP1 0.2603 33.3330
MK-591 PANC10.05 CTRP1 0.2603 33.3330
MK-591 PATU8902 CTRP1 0.2603 33.3330
MK-591 QGP-1 CTRP1 0.2603 33.3330
MK-591 SUIT-2 CTRP1 0.2603 33.3330
MK-591 MSTO-211H CTRP1 0.2603 33.3330
MK-591 NCI-H2052 CTRP1 0.2603 33.3330
MK-591 NCI-H28 CTRP1 0.2603 33.3330
MK-591 MIAPACA-3 CTRP1 0.2603 33.3330
MK-591 A-375 CTRP1 2.0833 266.6700
MK-591 COLO741 CTRP1 0.2603 33.3330
MK-591 G-361 CTRP1 0.2603 33.3330
MK-591 HS852.T CTRP1 0.2603 33.3330
MK-591 HS936.T CTRP1 0.2603 33.3330
MK-591 HS944.T CTRP1 0.2603 33.3330
MK-591 SK-MEL-1 CTRP1 2.0833 266.6700
MK-591 SK-MEL-28 CTRP1 2.0833 266.6700
MK-591 SK-MEL-5 CTRP1 2.0833 266.6700
MK-591 G-401 CTRP1 0.2603 33.3330
MK-591 HT-1080 CTRP1 2.0833 266.6700
MK-591 AGS CTRP1 2.0833 266.6700
MK-591 FU97 CTRP1 0.2603 33.3330
MK-591 KE-97 CTRP1 0.2603 33.3330
MK-591 MKN7 CTRP1 0.2603 33.3330
MK-591 MKN74 CTRP1 0.2603 33.3330
MK-591 NUGC-4 CTRP1 0.2603 33.3330
MK-591 SH-10-TC CTRP1 0.2603 33.3330
MK-591 HSC-2 CTRP1 0.2603 33.3330
MK-591 SCC-9 CTRP1 2.0833 266.6700
MK-591 5637 CTRP1 0.2603 33.3330
MK-591 HT-1376 CTRP1 0.2603 33.3330
MK-591 KMBC-2 CTRP1 0.2603 33.3330
MK-591 RT-4 CTRP1 0.2603 33.3330
MK-591 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.