Drug : Pt-630

CTRP1 Name : PT-630

Dataset : All
Synonyms :
Targets : FAP
Pathways : inhibitor of fibroblast activation protein

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
PT-630 MCF-7 CTRP1 0.2604 33.3330
PT-630 GAMG CTRP1 0.2603 33.3330
PT-630 LN-229 CTRP1 0.2604 33.3330
PT-630 SF295 CTRP1 0.2603 33.3330
PT-630 HEC-108 CTRP1 0.2603 33.3330
PT-630 HEC-151 CTRP1 0.1302 33.3330
PT-630 HEC-251 CTRP1 0.2603 33.3330
PT-630 HEC-265 CTRP1 0.2603 33.3330
PT-630 HEC-59 CTRP1 0.2603 33.3330
PT-630 HEC-6 CTRP1 0.2603 33.3330
PT-630 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
PT-630 JHUEM-2 CTRP1 0.2604 33.3330
PT-630 KLE CTRP1 0.2603 33.3330
PT-630 MFE-319 CTRP1 0.2603 33.3330
PT-630 SNG-M CTRP1 0.2603 33.3330
PT-630 AMO1 CTRP1 0.1302 33.3330
PT-630 BL-70 CTRP1 0.2603 33.3330
PT-630 EJM CTRP1 0.2604 33.3330
PT-630 GDM-1 CTRP1 0.2604 33.3330
PT-630 HT CTRP1 0.2603 33.3330
PT-630 KMS-11 CTRP1 0.1302 33.3330
PT-630 KU812 CTRP1 0.2603 33.3330
PT-630 LP-1 CTRP1 0.1302 33.3330
PT-630 MC116 CTRP1 0.2603 33.3330
PT-630 MOLM-16 CTRP1 0.2604 33.3330
PT-630 NOMO-1 CTRP1 0.2604 33.3330
PT-630 NU-DUL-1 CTRP1 0.2604 33.3330
PT-630 OCI-AML-3 CTRP1 0.2604 33.3330
PT-630 OCI-LY10 CTRP1 0.1302 33.3330
PT-630 P3HR-1 CTRP1 0.2603 33.3330
PT-630 PL21 CTRP1 0.2604 33.3330
PT-630 RPMI-8226 CTRP1 0.2604 33.3330
PT-630 SKM-1 CTRP1 0.2604 33.3330
PT-630 SU-DHL-4 CTRP1 0.2604 33.3330
PT-630 SU-DHL-5 CTRP1 0.2604 33.3330
PT-630 THP-1 CTRP1 0.2604 33.3330
PT-630 U-937 CTRP1 0.2604 33.3330
PT-630 WSU-DLCL2 CTRP1 0.2604 33.3330
PT-630 VMRC-RCW CTRP1 0.2603 33.3330
PT-630 C2BBE1 CTRP1 0.2603 33.3330
PT-630 CL-34 CTRP1 0.2604 33.3330
PT-630 CL-40 CTRP1 0.2604 33.3330
PT-630 COLO205 CTRP1 0.2603 33.3330
PT-630 COLO320 CTRP1 0.2604 33.3330
PT-630 COLO678 CTRP1 0.2604 33.3330
PT-630 CW-2 CTRP1 0.2604 33.3330
PT-630 DLD-1 CTRP1 0.2603 33.3330
PT-630 GP2D CTRP1 0.2603 33.3330
PT-630 HCT116 CTRP1 0.2604 33.3330
PT-630 HCT8 CTRP1 0.2604 33.3330
PT-630 HT115 CTRP1 0.2604 33.3330
PT-630 HT-29 CTRP1 0.2604 33.3330
PT-630 HT-55 CTRP1 0.2604 33.3330
PT-630 KM12 CTRP1 0.2604 33.3330
PT-630 LOVO CTRP1 0.2604 33.3330
PT-630 LS123 CTRP1 0.2604 33.3330
PT-630 LS180 CTRP1 0.1302 33.3330
PT-630 LS411N CTRP1 0.2603 33.3330
PT-630 LS513 CTRP1 0.2603 33.3330
PT-630 MDST8 CTRP1 0.2604 33.3330
PT-630 NCI-H508 CTRP1 0.2604 33.3330
PT-630 RCM-1[HUMANESC] CTRP1 0.2604 33.3330
PT-630 RKO CTRP1 0.2604 33.3330
PT-630 SK-CO-1 CTRP1 0.2603 33.3330
PT-630 SNU-1040 CTRP1 0.2604 33.3330
PT-630 SNU-175 CTRP1 0.2604 33.3330
PT-630 SNU-61 CTRP1 0.2604 33.3330
PT-630 SNU-81 CTRP1 0.2604 33.3330
PT-630 SNU-C2A CTRP1 0.2603 33.3330
PT-630 SNU-C4 CTRP1 0.2604 33.3330
PT-630 SNU-C5 CTRP1 0.2604 33.3330
PT-630 SW403 CTRP1 0.2603 33.3330
PT-630 SW48 CTRP1 0.2603 33.3330
PT-630 SW480 CTRP1 0.2604 33.3330
PT-630 SW620 CTRP1 0.2604 33.3330
PT-630 SW948 CTRP1 0.2604 33.3330
PT-630 HEP-G2 CTRP1 0.2604 33.3330
PT-630 JHH-6 CTRP1 0.2603 33.3330
PT-630 SNU-398 CTRP1 0.1302 33.3330
PT-630 SNU-449 CTRP1 0.2603 33.3330
PT-630 A-549 CTRP1 0.2603 33.3330
PT-630 BEN CTRP1 0.2603 33.3330
PT-630 CAL-12T CTRP1 0.2604 33.3330
PT-630 CALU-3 CTRP1 0.2603 33.3330
PT-630 CALU-6 CTRP1 0.2603 33.3330
PT-630 CHAGO-K-1 CTRP1 0.2603 33.3330
PT-630 COLO668 CTRP1 0.2603 33.3330
PT-630 COLO699 CTRP1 0.2604 33.3330
PT-630 COR-L23 CTRP1 0.2604 33.3330
PT-630 COR-L279 CTRP1 0.2603 33.3330
PT-630 COR-L51 CTRP1 0.1302 33.3330
PT-630 COR-L88 CTRP1 0.2603 33.3330
PT-630 DMS273 CTRP1 0.2603 33.3330
PT-630 DV-90 CTRP1 0.2603 33.3330
PT-630 EBC-1 CTRP1 0.2603 33.3330
PT-630 EPLC-272H CTRP1 0.2603 33.3330
PT-630 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
PT-630 HCC1195 CTRP1 0.2604 33.3330
PT-630 HCC1359 CTRP1 0.2604 33.3330
PT-630 HCC15 CTRP1 0.2604 33.3330
PT-630 HCC1833 CTRP1 0.2604 33.3330
PT-630 HCC2108 CTRP1 0.2604 33.3330
PT-630 HCC2935 CTRP1 0.2604 33.3330
PT-630 HCC33 CTRP1 0.2603 33.3330
PT-630 HCC4006 CTRP1 0.2604 33.3330
PT-630 HCC44 CTRP1 0.2603 33.3330
PT-630 HCC78 CTRP1 0.2603 33.3330
PT-630 HCC827 CTRP1 0.2604 33.3330
PT-630 KNS-62 CTRP1 0.2603 33.3330
PT-630 LC-1-SQ-SF CTRP1 0.2603 33.3330
PT-630 LCLC-103H CTRP1 0.2603 33.3330
PT-630 LCLC-97TM1 CTRP1 0.2603 33.3330
PT-630 LU-65 CTRP1 0.2603 33.3330
PT-630 LU-99 CTRP1 0.2603 33.3330
PT-630 LXF289 CTRP1 0.2603 33.3330
PT-630 NCI-H1048 CTRP1 0.2603 33.3330
PT-630 NCI-H1105 CTRP1 0.2604 33.3330
PT-630 NCI-H1299 CTRP1 0.2603 33.3330
PT-630 NCI-H1355 CTRP1 0.2603 33.3330
PT-630 NCI-H1373 CTRP1 0.2603 33.3330
PT-630 NCI-H1435 CTRP1 0.2603 33.3330
PT-630 NCI-H1437 CTRP1 0.2603 33.3330
PT-630 NCI-H1568 CTRP1 0.2603 33.3330
PT-630 NCI-H1573 CTRP1 0.2603 33.3330
PT-630 NCI-H1666 CTRP1 0.2603 33.3330
PT-630 NCI-H1694 CTRP1 0.2604 33.3330
PT-630 NCI-H1755 CTRP1 0.2604 33.3330
PT-630 NCI-H1781 CTRP1 0.2604 33.3330
PT-630 NCI-H1792 CTRP1 0.2603 33.3330
PT-630 NCI-H1793 CTRP1 0.2603 33.3330
PT-630 NCI-H1836 CTRP1 0.2604 33.3330
PT-630 NCI-H1876 CTRP1 0.2604 33.3330
PT-630 NCI-H1915 CTRP1 0.2603 33.3330
PT-630 NCI-H1930 CTRP1 0.2603 33.3330
PT-630 NCI-H1944 CTRP1 0.2603 33.3330
PT-630 NCI-H1963 CTRP1 0.1302 33.3330
PT-630 NCI-H1975 CTRP1 0.2603 33.3330
PT-630 NCI-H2009 CTRP1 0.2603 33.3330
PT-630 NCI-H2023 CTRP1 0.2604 33.3330
PT-630 NCI-H2029 CTRP1 0.2603 33.3330
PT-630 NCI-H2030 CTRP1 0.2604 33.3330
PT-630 NCI-H2073 CTRP1 0.2604 33.3330
PT-630 NCI-H2081 CTRP1 0.2604 33.3330
PT-630 NCI-H2110 CTRP1 0.2604 33.3330
PT-630 NCI-H2122 CTRP1 0.2604 33.3330
PT-630 NCI-H2126 CTRP1 0.2603 33.3330
PT-630 NCI-H2141 CTRP1 0.1302 33.3330
PT-630 NCI-H2172 CTRP1 0.2604 33.3330
PT-630 NCI-H2286 CTRP1 0.2603 33.3330
PT-630 NCI-H23 CTRP1 0.2603 33.3330
PT-630 NCI-H2342 CTRP1 0.2604 33.3330
PT-630 NCI-H2405 CTRP1 0.2603 33.3330
PT-630 NCI-H3255 CTRP1 0.2604 33.3330
PT-630 NCI-H358 CTRP1 0.2603 33.3330
PT-630 NCI-H441 CTRP1 0.2604 33.3330
PT-630 NCI-H460 CTRP1 0.2604 33.3330
PT-630 NCI-H522 CTRP1 0.2603 33.3330
PT-630 NCI-H596 CTRP1 0.2604 33.3330
PT-630 NCI-H650 CTRP1 0.2603 33.3330
PT-630 NCI-H661 CTRP1 0.2603 33.3330
PT-630 NCI-H727 CTRP1 0.2603 33.3330
PT-630 NCI-H810 CTRP1 0.2603 33.3330
PT-630 NCI-H82 CTRP1 0.2603 33.3330
PT-630 NCI-H841 CTRP1 0.2604 33.3330
PT-630 RERF-LC-KJ CTRP1 0.2603 33.3330
PT-630 SCLC-21H CTRP1 0.1302 33.3330
PT-630 SHP-77 CTRP1 0.2603 33.3330
PT-630 SK-LU-1 CTRP1 0.2604 33.3330
PT-630 SQ-1 CTRP1 0.2604 33.3330
PT-630 T3M-10 CTRP1 0.2604 33.3330
PT-630 VMRC-LCD CTRP1 0.2603 33.3330
PT-630 KYSE-140 CTRP1 0.2603 33.3330
PT-630 KYSE-410 CTRP1 0.2603 33.3330
PT-630 KYSE-450 CTRP1 0.2603 33.3330
PT-630 A2780 CTRP1 0.1302 33.3330
PT-630 CAOV-3 CTRP1 0.2604 33.3330
PT-630 COV318 CTRP1 0.2603 33.3330
PT-630 COV362 CTRP1 0.2604 33.3330
PT-630 COV434 CTRP1 0.2604 33.3330
PT-630 COV644 CTRP1 0.2604 33.3330
PT-630 EFO-21 CTRP1 0.2603 33.3330
PT-630 EFO-27 CTRP1 0.2604 33.3330
PT-630 HEYA8 CTRP1 0.2603 33.3330
PT-630 IGROV-1 CTRP1 0.1302 33.3330
PT-630 JHOC-5 CTRP1 0.2604 33.3330
PT-630 JHOM-1 CTRP1 0.2604 33.3330
PT-630 JHOS-4 CTRP1 0.2603 33.3330
PT-630 OAW42 CTRP1 0.2604 33.3330
PT-630 OV7 CTRP1 0.2604 33.3330
PT-630 OV-90 CTRP1 0.2604 33.3330
PT-630 OVCAR-4 CTRP1 0.1302 33.3330
PT-630 OVCAR-8 CTRP1 0.1302 33.3330
PT-630 OVK18 CTRP1 0.2604 33.3330
PT-630 OVKATE CTRP1 0.1302 33.3330
PT-630 OVMANA CTRP1 0.2603 33.3330
PT-630 RKN CTRP1 0.1302 33.3330
PT-630 RMG-I CTRP1 0.2604 33.3330
PT-630 RMUG-S CTRP1 0.2604 33.3330
PT-630 SK-OV-3 CTRP1 0.2603 33.3330
PT-630 SNU-840 CTRP1 0.2604 33.3330
PT-630 TYK-NU CTRP1 0.2604 33.3330
PT-630 CAPAN-2 CTRP1 0.2603 33.3330
PT-630 CFPAC-1 CTRP1 0.2603 33.3330
PT-630 HPAC CTRP1 0.2603 33.3330
PT-630 HUP-T4 CTRP1 0.2603 33.3330
PT-630 KP-3 CTRP1 0.2603 33.3330
PT-630 PANC03.27 CTRP1 0.2603 33.3330
PT-630 PANC10.05 CTRP1 0.2603 33.3330
PT-630 PATU8902 CTRP1 0.2603 33.3330
PT-630 QGP-1 CTRP1 0.2603 33.3330
PT-630 SUIT-2 CTRP1 0.2603 33.3330
PT-630 MSTO-211H CTRP1 0.2603 33.3330
PT-630 NCI-H2052 CTRP1 0.2603 33.3330
PT-630 NCI-H28 CTRP1 0.2603 33.3330
PT-630 MIAPACA-3 CTRP1 0.2603 33.3330
PT-630 A-375 CTRP1 0.2604 33.3330
PT-630 COLO741 CTRP1 0.2603 33.3330
PT-630 G-361 CTRP1 0.2603 33.3330
PT-630 HS852.T CTRP1 0.2603 33.3330
PT-630 HS936.T CTRP1 0.2603 33.3330
PT-630 HS944.T CTRP1 0.2603 33.3330
PT-630 SK-MEL-1 CTRP1 0.2604 33.3330
PT-630 SK-MEL-28 CTRP1 0.2604 33.3330
PT-630 SK-MEL-5 CTRP1 0.2604 33.3330
PT-630 G-401 CTRP1 0.2603 33.3330
PT-630 HT-1080 CTRP1 0.2604 33.3330
PT-630 AGS CTRP1 0.1302 33.3330
PT-630 FU97 CTRP1 0.2603 33.3330
PT-630 KE-97 CTRP1 0.2603 33.3330
PT-630 MKN7 CTRP1 0.2603 33.3330
PT-630 MKN74 CTRP1 0.2603 33.3330
PT-630 NUGC-4 CTRP1 0.2603 33.3330
PT-630 SH-10-TC CTRP1 0.2603 33.3330
PT-630 HSC-2 CTRP1 0.2603 33.3330
PT-630 SCC-9 CTRP1 0.1302 33.3330
PT-630 5637 CTRP1 0.2603 33.3330
PT-630 HT-1376 CTRP1 0.2603 33.3330
PT-630 KMBC-2 CTRP1 0.2603 33.3330
PT-630 RT-4 CTRP1 0.2603 33.3330
PT-630 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.