Drug : Ly-2157299

CTRP2 Name : LY-2157299

Dataset : All
Synonyms :
Targets : TGFBR1
Pathways : inhibitor of the transforming growth factor beta type 1 receptor

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

:


Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
LY-2157299 CAS-1 CTRP2 0.0020 66.0000
LY-2157299 KPL-1 CTRP2 0.0020 66.0000
LY-2157299 MKN1 CTRP2 0.0020 66.0000
LY-2157299 253J-BV CTRP2 0.0020 66.0000
LY-2157299 BFTC-905 CTRP2 0.0020 66.0000
LY-2157299 BFTC-909 CTRP2 0.0020 66.0000
LY-2157299 CADO-ES1 CTRP2 0.0020 66.0000
LY-2157299 CAL-120 CTRP2 0.0020 66.0000
LY-2157299 CAL-29 CTRP2 0.0020 66.0000
LY-2157299 CAL-62 CTRP2 0.0020 66.0000
LY-2157299 HUCC-T1 CTRP2 0.0020 66.0000
LY-2157299 NMC-G1 CTRP2 0.0020 66.0000
LY-2157299 RPMI-7951 CTRP2 0.0020 66.0000
LY-2157299 253J CTRP2 0.0020 66.0000
LY-2157299 ALL-SIL CTRP2 0.0020 66.0000
LY-2157299 HDQ-P1 CTRP2 0.0020 66.0000
LY-2157299 SNU-245 CTRP2 0.0020 66.0000
LY-2157299 SNU-489 CTRP2 0.0020 66.0000
LY-2157299 SNU-626 CTRP2 0.0020 66.0000
LY-2157299 SNU-738 CTRP2 0.0020 66.0000
LY-2157299 SNU-878 CTRP2 0.0020 66.0000
LY-2157299 TUHR4TKB CTRP2 0.0020 66.0000
LY-2157299 ACC-MESO-1 CTRP2 0.0020 66.0000
LY-2157299 B-CPAP CTRP2 0.0020 66.0000
LY-2157299 CGTH-W-1 CTRP2 0.0020 66.0000
LY-2157299 COLO680N CTRP2 0.0020 66.0000
LY-2157299 ECC12 CTRP2 0.0020 66.0000
LY-2157299 HCC95 CTRP2 0.0020 66.0000
LY-2157299 JMSU-1 CTRP2 0.0020 66.0000
LY-2157299 RH41 CTRP2 0.0020 66.0000
LY-2157299 WSU-DLCL2 CTRP2 0.0020 66.0000
LY-2157299 23132-87 CTRP2 0.0020 66.0000
LY-2157299 8305C CTRP2 0.0020 66.0000
LY-2157299 BHY CTRP2 0.0020 66.0000
LY-2157299 GSU CTRP2 0.0020 66.0000
LY-2157299 JIMT-1 CTRP2 0.0020 66.0000
LY-2157299 KMRC-20 CTRP2 0.0020 66.0000
LY-2157299 OUMS-23 CTRP2 0.0020 66.0000
LY-2157299 SNU-1076 CTRP2 0.0020 66.0000
LY-2157299 SNU-1196 CTRP2 0.0020 66.0000
LY-2157299 SNU-8 CTRP2 0.0020 66.0000
LY-2157299 A-375 CTRP2 0.0020 66.0000
LY-2157299 A-549 CTRP2 0.0020 66.0000
LY-2157299 NCI-H2009 CTRP2 0.0020 66.0000
LY-2157299 SNU-201 CTRP2 0.0020 66.0000
LY-2157299 SUIT-2 CTRP2 0.0020 66.0000
LY-2157299 SNU-1079 CTRP2 0.0020 66.0000
LY-2157299 DEL CTRP2 0.0020 66.0000
LY-2157299 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP2 0.0020 66.0000
LY-2157299 HCC15 CTRP2 0.0020 66.0000
LY-2157299 KP-4 CTRP2 0.0020 66.0000
LY-2157299 LU-99 CTRP2 0.0020 66.0000
LY-2157299 NCI-H1155 CTRP2 0.0020 66.0000
LY-2157299 NCI-H1581 CTRP2 0.0020 66.0000
LY-2157299 NCI-H2106 CTRP2 0.0020 66.0000
LY-2157299 NCI-H358 CTRP2 0.0020 66.0000
LY-2157299 DLD-1 CTRP2 0.0020 66.0000
LY-2157299 EM-2 CTRP2 0.0020 66.0000
LY-2157299 JURL-MK1 CTRP2 0.0020 66.0000
LY-2157299 P12-ICHIKAWA CTRP2 0.0020 66.0000
LY-2157299 KE-37 CTRP2 0.0020 66.0000
LY-2157299 KMS-21-BM CTRP2 0.0020 66.0000
LY-2157299 LI-7 CTRP2 0.0020 66.0000
LY-2157299 MHH-NB-11 CTRP2 0.0020 66.0000
LY-2157299 MOLM-13 CTRP2 0.0020 66.0000
LY-2157299 NCI-H1975 CTRP2 0.0020 66.0000
LY-2157299 NCI-H28 CTRP2 0.0020 66.0000
LY-2157299 639V CTRP2 0.0020 66.0000
LY-2157299 BXPC-3 CTRP2 0.0020 66.0000
LY-2157299 CML-T1 CTRP2 0.0020 66.0000
LY-2157299 GSS CTRP2 0.0020 66.0000
LY-2157299 HCC366 CTRP2 0.0020 66.0000
LY-2157299 KURAMOCHI CTRP2 0.0020 66.0000
LY-2157299 LS411N CTRP2 0.0020 66.0000
LY-2157299 LS513 CTRP2 0.0020 66.0000
LY-2157299 ONCO-DG-1 CTRP2 0.0020 66.0000
LY-2157299 ONS-76 CTRP2 0.0020 66.0000
LY-2157299 SK-CO-1 CTRP2 0.0020 66.0000
LY-2157299 SW48 CTRP2 0.0020 66.0000
LY-2157299 VM-CUB-1 CTRP2 0.0020 66.0000
LY-2157299 BEN CTRP2 0.0020 66.0000
LY-2157299 CFPAC-1 CTRP2 0.0020 66.0000
LY-2157299 HCC78 CTRP2 0.0020 66.0000
LY-2157299 HT CTRP2 0.0020 66.0000
LY-2157299 KU-19-19 CTRP2 0.0020 66.0000
LY-2157299 NCI-H1299 CTRP2 0.0020 66.0000
LY-2157299 NCI-H727 CTRP2 0.0020 66.0000
LY-2157299 NCO2 CTRP2 0.0020 66.0000
LY-2157299 OVTOKO CTRP2 0.0020 66.0000
LY-2157299 P31-FUJ CTRP2 0.0020 66.0000
LY-2157299 PEER CTRP2 0.0020 66.0000
LY-2157299 RPMI-8402 CTRP2 0.0020 66.0000
LY-2157299 SHP-77 CTRP2 0.0020 66.0000
LY-2157299 SNU-1077 CTRP2 0.0020 66.0000
LY-2157299 SNU-620 CTRP2 0.0020 66.0000
LY-2157299 SU-DHL-1 CTRP2 0.0020 66.0000
LY-2157299 COLO205 CTRP2 0.0020 66.0000
LY-2157299 EHEB CTRP2 0.0020 66.0000
LY-2157299 KI-JK CTRP2 0.0020 66.0000
LY-2157299 KMM-1 CTRP2 0.0020 66.0000
LY-2157299 LCLC-103H CTRP2 0.0020 66.0000
LY-2157299 MKN45 CTRP2 0.0020 66.0000
LY-2157299 NCI-H2405 CTRP2 0.0020 66.0000
LY-2157299 NCI-H650 CTRP2 0.0020 66.0000
LY-2157299 OS-RC-2 CTRP2 0.0020 66.0000
LY-2157299 OVSAHO CTRP2 0.0020 66.0000
LY-2157299 QGP-1 CTRP2 0.0020 66.0000
LY-2157299 RL95-2 CTRP2 0.0020 66.0000
LY-2157299 SNU-1041 CTRP2 0.0020 66.0000
LY-2157299 SNU-1066 CTRP2 0.0020 66.0000
LY-2157299 SW1353 CTRP2 0.0020 66.0000
LY-2157299 SNU-213 CTRP2 0.0020 66.0000
LY-2157299 8505C CTRP2 0.0020 66.0000
LY-2157299 CALU-3 CTRP2 0.0020 66.0000
LY-2157299 DAOY CTRP2 0.0020 66.0000
LY-2157299 GB-1 CTRP2 0.0020 66.0000
LY-2157299 HCC1171 CTRP2 0.0020 66.0000
LY-2157299 HCC44 CTRP2 0.0020 66.0000
LY-2157299 NCI-H211 CTRP2 0.0020 66.0000
LY-2157299 RERF-LC-A1 CTRP2 0.0020 66.0000
LY-2157299 SBC-5 CTRP2 0.0020 66.0000
LY-2157299 SF126 CTRP2 0.0020 66.0000
LY-2157299 SNU-119 CTRP2 0.0020 66.0000
LY-2157299 SNU-182 CTRP2 0.0020 66.0000
LY-2157299 TCCSUP CTRP2 0.0020 66.0000
LY-2157299 CAMA-1 CTRP2 0.0020 66.0000
LY-2157299 DETROIT562 CTRP2 0.0020 66.0000
LY-2157299 HEC-1-B CTRP2 0.0020 66.0000
LY-2157299 HEP3B2.1-7 CTRP2 0.0020 66.0000
LY-2157299 HSC-3 CTRP2 0.0020 66.0000
LY-2157299 MCF-7 CTRP2 0.0020 66.0000
LY-2157299 SNU-1105 CTRP2 0.0020 66.0000
LY-2157299 U-87MGATCC CTRP2 0.0020 66.0000
LY-2157299 22RV1 CTRP2 0.0020 66.0000
LY-2157299 769-P CTRP2 0.0020 66.0000
LY-2157299 COLO699 CTRP2 0.0020 66.0000
LY-2157299 DOV13 CTRP2 0.0020 66.0000
LY-2157299 ES2 CTRP2 0.0020 66.0000
LY-2157299 HCC1806 CTRP2 0.0020 66.0000
LY-2157299 HCC1954 CTRP2 0.0020 66.0000
LY-2157299 HPAF-II CTRP2 0.0020 66.0000
LY-2157299 KHM-1B CTRP2 0.0020 66.0000
LY-2157299 OVISE CTRP2 0.0020 66.0000
LY-2157299 JVM-3 CTRP2 0.0020 66.0000
LY-2157299 SNU-C2A CTRP2 0.0020 66.0000
LY-2157299 U2OS CTRP2 0.0020 66.0000
LY-2157299 5637 CTRP2 0.0020 66.0000
LY-2157299 CAL-12T CTRP2 0.0020 66.0000
LY-2157299 HCC1588 CTRP2 0.0020 66.0000
LY-2157299 HCC1833 CTRP2 0.0020 66.0000
LY-2157299 HCC2279 CTRP2 0.0020 66.0000
LY-2157299 KE-97 CTRP2 0.0020 66.0000
LY-2157299 KP-3 CTRP2 0.0020 66.0000
LY-2157299 KU812 CTRP2 0.0020 66.0000
LY-2157299 KYSE-140 CTRP2 0.0020 66.0000
LY-2157299 NALM-6 CTRP2 0.0020 66.0000
LY-2157299 NUGC-4 CTRP2 0.0020 66.0000
LY-2157299 TT CTRP2 0.0020 66.0000
LY-2157299 AGS CTRP2 0.0020 66.0000
LY-2157299 HCT116 CTRP2 0.0020 66.0000
LY-2157299 HEC-108 CTRP2 0.0020 66.0000
LY-2157299 HEC-59 CTRP2 0.0020 66.0000
LY-2157299 HMC-1-8 CTRP2 0.0020 66.0000
LY-2157299 HT-29 CTRP2 0.0020 66.0000
LY-2157299 ISHIKAWA(HERAKLIO)02ER- CTRP2 0.0020 66.0000
LY-2157299 JHOC-5 CTRP2 0.0020 66.0000
LY-2157299 KYSE-180 CTRP2 0.0020 66.0000
LY-2157299 LS180 CTRP2 0.0020 66.0000
LY-2157299 MELHO CTRP2 0.0020 66.0000
LY-2157299 MHH-ES-1 CTRP2 0.0020 66.0000
LY-2157299 MOR-CPR CTRP2 0.0020 66.0000
LY-2157299 NCI-H460 CTRP2 0.0020 66.0000
LY-2157299 HCC2108 CTRP2 0.0020 66.0000
LY-2157299 HCC827 CTRP2 0.0020 66.0000
LY-2157299 HEC-251 CTRP2 0.0020 66.0000
LY-2157299 HEC-265 CTRP2 0.0020 66.0000
LY-2157299 HEC-6 CTRP2 0.0020 66.0000
LY-2157299 HEL CTRP2 0.0020 66.0000
LY-2157299 JHUEM-2 CTRP2 0.0020 66.0000
LY-2157299 JURKAT CTRP2 0.0020 66.0000
LY-2157299 JVM-2 CTRP2 0.0020 66.0000
LY-2157299 KCL-22 CTRP2 0.0020 66.0000
LY-2157299 KE-39 CTRP2 0.0020 66.0000
LY-2157299 KM-H2 CTRP2 0.0020 66.0000
LY-2157299 LAMA-84 CTRP2 0.0020 66.0000
LY-2157299 NCI-H2030 CTRP2 0.0020 66.0000
LY-2157299 SNU-719 CTRP2 0.0020 66.0000
LY-2157299 KMS-27 CTRP2 0.0020 66.0000
LY-2157299 NCI-H1838 CTRP2 0.0020 66.0000
LY-2157299 NCI-H196 CTRP2 0.0020 66.0000
LY-2157299 NCI-H292 CTRP2 0.0020 66.0000
LY-2157299 SK-MEL-1 CTRP2 0.0020 66.0000
LY-2157299 HCC1937 CTRP2 0.0020 66.0000
LY-2157299 HDLM-2 CTRP2 0.0020 66.0000
LY-2157299 SNU-1272 CTRP2 0.0020 66.0000
LY-2157299 SNU-308 CTRP2 0.0020 66.0000
LY-2157299 SNU-478 CTRP2 0.0020 66.0000
LY-2157299 BHT-101 CTRP2 0.0020 66.0000
LY-2157299 CAL-51 CTRP2 0.0020 66.0000
LY-2157299 HCC1395 CTRP2 0.0020 66.0000
LY-2157299 HT115 CTRP2 0.0020 66.0000
LY-2157299 LN-18 CTRP2 0.0020 66.0000
LY-2157299 LN-229 CTRP2 0.0020 66.0000
LY-2157299 NCI-H2291 CTRP2 0.0020 66.0000
LY-2157299 RERF-LC-AD1 CTRP2 0.0020 66.0000
LY-2157299 SNU-1214 CTRP2 0.0020 66.0000
LY-2157299 SNU-46 CTRP2 0.0020 66.0000
LY-2157299 SNU-5 CTRP2 0.0020 66.0000
LY-2157299 SNU-668 CTRP2 0.0020 66.0000
LY-2157299 SNU-899 CTRP2 0.0020 66.0000
LY-2157299 TE-10 CTRP2 0.0020 66.0000
LY-2157299 TE-9 CTRP2 0.0020 66.0000
LY-2157299 YD-10B CTRP2 0.0020 66.0000
LY-2157299 YD-15 CTRP2 0.0020 66.0000
LY-2157299 YD-38 CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.