Drug : Brd-K58730230

CTRP2 Name : BRD-K58730230

Dataset : All
Synonyms :
Targets :
Pathways : stapled helical peptide

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BRD-K58730230 CAS-1 CTRP2 0.0020 66.0000
BRD-K58730230 KPL-1 CTRP2 0.0020 66.0000
BRD-K58730230 MKN1 CTRP2 0.0020 66.0000
BRD-K58730230 253J-BV CTRP2 0.0020 66.0000
BRD-K58730230 BFTC-905 CTRP2 0.0020 66.0000
BRD-K58730230 BFTC-909 CTRP2 0.0020 66.0000
BRD-K58730230 CAL-29 CTRP2 0.0020 66.0000
BRD-K58730230 CAL-62 CTRP2 0.0020 66.0000
BRD-K58730230 HUCC-T1 CTRP2 0.0020 66.0000
BRD-K58730230 NMC-G1 CTRP2 0.0020 66.0000
BRD-K58730230 RPMI-7951 CTRP2 0.0020 66.0000
BRD-K58730230 253J CTRP2 0.0020 66.0000
BRD-K58730230 HDQ-P1 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-489 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-626 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-738 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-878 CTRP2 0.0020 66.0000
BRD-K58730230 TUHR4TKB CTRP2 0.0020 66.0000
BRD-K58730230 ACC-MESO-1 CTRP2 0.0020 66.0000
BRD-K58730230 B-CPAP CTRP2 0.0020 66.0000
BRD-K58730230 CGTH-W-1 CTRP2 0.0020 66.0000
BRD-K58730230 COLO680N CTRP2 0.0020 66.0000
BRD-K58730230 ECC12 CTRP2 0.0020 66.0000
BRD-K58730230 HCC95 CTRP2 0.0020 66.0000
BRD-K58730230 JMSU-1 CTRP2 0.0020 66.0000
BRD-K58730230 RH41 CTRP2 0.0020 66.0000
BRD-K58730230 WSU-DLCL2 CTRP2 0.0020 66.0000
BRD-K58730230 23132-87 CTRP2 0.0020 66.0000
BRD-K58730230 8305C CTRP2 0.0020 66.0000
BRD-K58730230 BHY CTRP2 0.0020 66.0000
BRD-K58730230 GSU CTRP2 0.0020 66.0000
BRD-K58730230 JIMT-1 CTRP2 0.0020 66.0000
BRD-K58730230 KMRC-20 CTRP2 0.0020 66.0000
BRD-K58730230 OUMS-23 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-1076 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-1196 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-8 CTRP2 0.0020 66.0000
BRD-K58730230 A-375 CTRP2 0.0020 66.0000
BRD-K58730230 A-549 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H2009 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-201 CTRP2 0.0020 66.0000
BRD-K58730230 SUIT-2 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-1079 CTRP2 0.0020 66.0000
BRD-K58730230 COLO741 CTRP2 0.0020 66.0000
BRD-K58730230 DEL CTRP2 0.0020 66.0000
BRD-K58730230 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP2 0.0020 66.0000
BRD-K58730230 HCC15 CTRP2 0.0020 66.0000
BRD-K58730230 KP-4 CTRP2 0.0020 66.0000
BRD-K58730230 LU-99 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H1155 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H1581 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H2106 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H358 CTRP2 0.0020 66.0000
BRD-K58730230 DLD-1 CTRP2 0.0020 66.0000
BRD-K58730230 EM-2 CTRP2 0.0020 66.0000
BRD-K58730230 JURL-MK1 CTRP2 0.0020 66.0000
BRD-K58730230 P12-ICHIKAWA CTRP2 0.0020 66.0000
BRD-K58730230 KE-37 CTRP2 0.0020 66.0000
BRD-K58730230 KMS-21-BM CTRP2 0.0020 66.0000
BRD-K58730230 LI-7 CTRP2 0.0020 66.0000
BRD-K58730230 MOLM-13 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H28 CTRP2 0.0020 66.0000
BRD-K58730230 639V CTRP2 0.0020 66.0000
BRD-K58730230 BXPC-3 CTRP2 0.0020 66.0000
BRD-K58730230 CML-T1 CTRP2 0.0020 66.0000
BRD-K58730230 GSS CTRP2 0.0020 66.0000
BRD-K58730230 HCC366 CTRP2 0.0020 66.0000
BRD-K58730230 KURAMOCHI CTRP2 0.0020 66.0000
BRD-K58730230 LS411N CTRP2 0.0020 66.0000
BRD-K58730230 LS513 CTRP2 0.0020 66.0000
BRD-K58730230 ONCO-DG-1 CTRP2 0.0020 66.0000
BRD-K58730230 ONS-76 CTRP2 0.0020 66.0000
BRD-K58730230 SK-CO-1 CTRP2 0.0020 66.0000
BRD-K58730230 SW48 CTRP2 0.0020 66.0000
BRD-K58730230 VM-CUB-1 CTRP2 0.0020 66.0000
BRD-K58730230 BEN CTRP2 0.0020 66.0000
BRD-K58730230 CFPAC-1 CTRP2 0.0020 66.0000
BRD-K58730230 HCC78 CTRP2 0.0020 66.0000
BRD-K58730230 HT CTRP2 0.0020 66.0000
BRD-K58730230 KU-19-19 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H1299 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H727 CTRP2 0.0020 66.0000
BRD-K58730230 NCO2 CTRP2 0.0020 66.0000
BRD-K58730230 OVTOKO CTRP2 0.0020 66.0000
BRD-K58730230 P31-FUJ CTRP2 0.0020 66.0000
BRD-K58730230 PEER CTRP2 0.0020 66.0000
BRD-K58730230 RPMI-8402 CTRP2 0.0020 66.0000
BRD-K58730230 SHP-77 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-1077 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-620 CTRP2 0.0020 66.0000
BRD-K58730230 SU-DHL-1 CTRP2 0.0020 66.0000
BRD-K58730230 COLO205 CTRP2 0.0020 66.0000
BRD-K58730230 EHEB CTRP2 0.0020 66.0000
BRD-K58730230 KI-JK CTRP2 0.0020 66.0000
BRD-K58730230 KMM-1 CTRP2 0.0020 66.0000
BRD-K58730230 LCLC-103H CTRP2 0.0020 66.0000
BRD-K58730230 MKN45 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H2405 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H650 CTRP2 0.0020 66.0000
BRD-K58730230 OS-RC-2 CTRP2 0.0020 66.0000
BRD-K58730230 OVSAHO CTRP2 0.0020 66.0000
BRD-K58730230 QGP-1 CTRP2 0.0020 66.0000
BRD-K58730230 RL95-2 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-1041 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-1066 CTRP2 0.0020 66.0000
BRD-K58730230 SW1353 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-213 CTRP2 0.0020 66.0000
BRD-K58730230 8505C CTRP2 0.0020 66.0000
BRD-K58730230 CALU-3 CTRP2 0.0020 66.0000
BRD-K58730230 DAOY CTRP2 0.0020 66.0000
BRD-K58730230 GB-1 CTRP2 0.0020 66.0000
BRD-K58730230 HCC1171 CTRP2 0.0020 66.0000
BRD-K58730230 HCC44 CTRP2 0.0020 66.0000
BRD-K58730230 NCI-H211 CTRP2 0.0020 66.0000
BRD-K58730230 RERF-LC-A1 CTRP2 0.0020 66.0000
BRD-K58730230 SBC-5 CTRP2 0.0020 66.0000
BRD-K58730230 SF126 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-119 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-81 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-182 CTRP2 0.0020 66.0000
BRD-K58730230 TCCSUP CTRP2 0.0020 66.0000
BRD-K58730230 CAMA-1 CTRP2 0.0020 66.0000
BRD-K58730230 DETROIT562 CTRP2 0.0020 66.0000
BRD-K58730230 HEC-1-B CTRP2 0.0020 66.0000
BRD-K58730230 HEP3B2.1-7 CTRP2 0.0020 66.0000
BRD-K58730230 HSC-3 CTRP2 0.0020 66.0000
BRD-K58730230 MCF-7 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-1105 CTRP2 0.0020 33.0000
BRD-K58730230 U-87MGATCC CTRP2 0.0020 66.0000
BRD-K58730230 22RV1 CTRP2 0.0020 33.0000
BRD-K58730230 769-P CTRP2 0.0020 33.0000
BRD-K58730230 COLO699 CTRP2 0.0020 66.0000
BRD-K58730230 DOV13 CTRP2 0.0020 66.0000
BRD-K58730230 ES2 CTRP2 0.0020 33.0000
BRD-K58730230 HCC1806 CTRP2 0.0020 66.0000
BRD-K58730230 HCC1954 CTRP2 0.0020 33.0000
BRD-K58730230 HPAF-II CTRP2 0.0020 33.0000
BRD-K58730230 KHM-1B CTRP2 0.0020 66.0000
BRD-K58730230 OVISE CTRP2 0.0020 66.0000
BRD-K58730230 JVM-3 CTRP2 0.0020 66.0000
BRD-K58730230 SNU-C2A CTRP2 0.0020 66.0000
BRD-K58730230 U2OS CTRP2 0.0020 33.0000
BRD-K58730230 5637 CTRP2 0.0020 33.0000
BRD-K58730230 CAL-12T CTRP2 0.0020 66.0000
BRD-K58730230 DMS79 CTRP2 0.0020 33.0000
BRD-K58730230 HCC1588 CTRP2 0.0020 33.0000
BRD-K58730230 HCC1833 CTRP2 0.0020 33.0000
BRD-K58730230 HCC2279 CTRP2 0.0020 33.0000
BRD-K58730230 KE-97 CTRP2 0.0020 33.0000
BRD-K58730230 KP-3 CTRP2 0.0020 33.0000
BRD-K58730230 KU812 CTRP2 0.0020 66.0000
BRD-K58730230 KYSE-140 CTRP2 0.0020 33.0000
BRD-K58730230 NALM-6 CTRP2 0.0020 33.0000
BRD-K58730230 NUGC-4 CTRP2 0.0020 66.0000
BRD-K58730230 TT CTRP2 0.0020 33.0000
BRD-K58730230 AGS CTRP2 0.0020 33.0000
BRD-K58730230 HCT116 CTRP2 0.0020 33.0000
BRD-K58730230 HEC-108 CTRP2 0.0020 33.0000
BRD-K58730230 HEC-59 CTRP2 0.0020 33.0000
BRD-K58730230 HMC-1-8 CTRP2 0.0020 33.0000
BRD-K58730230 HT-29 CTRP2 0.0020 33.0000
BRD-K58730230 ISHIKAWA(HERAKLIO)02ER- CTRP2 0.0020 33.0000
BRD-K58730230 JHOC-5 CTRP2 0.0020 66.0000
BRD-K58730230 KYSE-180 CTRP2 0.0020 33.0000
BRD-K58730230 LS180 CTRP2 0.0020 33.0000
BRD-K58730230 MELHO CTRP2 0.0020 33.0000
BRD-K58730230 MHH-ES-1 CTRP2 0.0020 66.0000
BRD-K58730230 MOR-CPR CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H460 CTRP2 0.0020 33.0000
BRD-K58730230 HCC2108 CTRP2 0.0020 33.0000
BRD-K58730230 HCC827 CTRP2 0.0020 33.0000
BRD-K58730230 HEC-251 CTRP2 0.0020 33.0000
BRD-K58730230 HEC-265 CTRP2 0.0020 66.0000
BRD-K58730230 HEC-6 CTRP2 0.0020 33.0000
BRD-K58730230 HEL CTRP2 0.0020 33.0000
BRD-K58730230 JHUEM-2 CTRP2 0.0020 33.0000
BRD-K58730230 JURKAT CTRP2 0.0020 33.0000
BRD-K58730230 KCL-22 CTRP2 0.0020 66.0000
BRD-K58730230 KE-39 CTRP2 0.0020 33.0000
BRD-K58730230 KM-H2 CTRP2 0.0020 33.0000
BRD-K58730230 LAMA-84 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H2030 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-719 CTRP2 0.0020 33.0000
BRD-K58730230 HCC1569 CTRP2 0.0020 33.0000
BRD-K58730230 KLE CTRP2 0.0020 33.0000
BRD-K58730230 KMS-26 CTRP2 0.0020 33.0000
BRD-K58730230 KMS-27 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H1838 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H196 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H292 CTRP2 0.0020 33.0000
BRD-K58730230 SK-MEL-1 CTRP2 0.0020 33.0000
BRD-K58730230 HCC1937 CTRP2 0.0020 33.0000
BRD-K58730230 HDLM-2 CTRP2 0.0020 33.0000
BRD-K58730230 HUH-28 CTRP2 0.0020 33.0000
BRD-K58730230 MV4-11 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H526 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H69 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H929 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-N87 CTRP2 0.0020 33.0000
BRD-K58730230 PF-382 CTRP2 0.0020 33.0000
BRD-K58730230 SF295 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-1272 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-308 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-478 CTRP2 0.0020 33.0000
BRD-K58730230 BHT-101 CTRP2 0.0020 33.0000
BRD-K58730230 CAL-148 CTRP2 0.0020 33.0000
BRD-K58730230 CAL-51 CTRP2 0.0020 33.0000
BRD-K58730230 HCC1395 CTRP2 0.0020 33.0000
BRD-K58730230 HT115 CTRP2 0.0020 33.0000
BRD-K58730230 LN-18 CTRP2 0.0020 33.0000
BRD-K58730230 LN-229 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H1734 CTRP2 0.0020 33.0000
BRD-K58730230 NCI-H2291 CTRP2 0.0020 33.0000
BRD-K58730230 RERF-LC-AD1 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-1214 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-46 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-466 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-5 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-668 CTRP2 0.0020 33.0000
BRD-K58730230 SNU-899 CTRP2 0.0020 33.0000
BRD-K58730230 TE-10 CTRP2 0.0020 33.0000
BRD-K58730230 TE-9 CTRP2 0.0020 33.0000
BRD-K58730230 YD-10B CTRP2 0.0020 33.0000
BRD-K58730230 YD-15 CTRP2 0.0020 33.0000
BRD-K58730230 YD-38 CTRP2 0.0020 33.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.