Drug : Fluoropyruvate

CTRP1 Name : fluoropyruvate

Dataset : All
Synonyms :
Targets : PDHX
Pathways : inhibitor of pyruvate dehydrogenase complex

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
fluoropyruvate MCF-7 CTRP1 1.1562 148.0000
fluoropyruvate GAMG CTRP1 0.2890 37.0000
fluoropyruvate LN-229 CTRP1 1.1562 148.0000
fluoropyruvate SF295 CTRP1 0.2890 37.0000
fluoropyruvate HEC-108 CTRP1 0.2890 37.0000
fluoropyruvate HEC-151 CTRP1 1.1562 148.0000
fluoropyruvate HEC-251 CTRP1 0.2890 37.0000
fluoropyruvate HEC-265 CTRP1 0.2890 37.0000
fluoropyruvate HEC-59 CTRP1 0.2890 37.0000
fluoropyruvate HEC-6 CTRP1 0.2890 37.0000
fluoropyruvate ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2890 37.0000
fluoropyruvate JHUEM-2 CTRP1 1.1562 148.0000
fluoropyruvate KLE CTRP1 0.2890 37.0000
fluoropyruvate MFE-319 CTRP1 0.2890 37.0000
fluoropyruvate SNG-M CTRP1 0.2890 37.0000
fluoropyruvate AMO1 CTRP1 1.1562 148.0000
fluoropyruvate BL-70 CTRP1 0.2890 37.0000
fluoropyruvate EJM CTRP1 1.1562 148.0000
fluoropyruvate GDM-1 CTRP1 1.1562 148.0000
fluoropyruvate HT CTRP1 0.2890 37.0000
fluoropyruvate KMS-11 CTRP1 1.1562 148.0000
fluoropyruvate KU812 CTRP1 0.2890 37.0000
fluoropyruvate LP-1 CTRP1 1.1562 148.0000
fluoropyruvate MC116 CTRP1 0.2890 37.0000
fluoropyruvate MOLM-16 CTRP1 1.1562 148.0000
fluoropyruvate NOMO-1 CTRP1 1.1562 148.0000
fluoropyruvate NU-DUL-1 CTRP1 1.1562 148.0000
fluoropyruvate OCI-AML-3 CTRP1 1.1562 148.0000
fluoropyruvate OCI-LY10 CTRP1 1.1562 148.0000
fluoropyruvate P3HR-1 CTRP1 0.2890 37.0000
fluoropyruvate PL21 CTRP1 1.1562 148.0000
fluoropyruvate RPMI-8226 CTRP1 1.1562 148.0000
fluoropyruvate SKM-1 CTRP1 1.1562 148.0000
fluoropyruvate SU-DHL-4 CTRP1 1.1562 148.0000
fluoropyruvate SU-DHL-5 CTRP1 1.1562 148.0000
fluoropyruvate THP-1 CTRP1 1.1562 148.0000
fluoropyruvate U-937 CTRP1 1.1562 148.0000
fluoropyruvate WSU-DLCL2 CTRP1 1.1562 148.0000
fluoropyruvate RCC10RGB CTRP1 1.1562 148.0000
fluoropyruvate VMRC-RCW CTRP1 0.2890 37.0000
fluoropyruvate C2BBE1 CTRP1 0.2890 37.0000
fluoropyruvate CL-34 CTRP1 1.1562 148.0000
fluoropyruvate CL-40 CTRP1 1.1562 148.0000
fluoropyruvate COLO205 CTRP1 0.2890 37.0000
fluoropyruvate COLO320 CTRP1 1.1562 148.0000
fluoropyruvate COLO678 CTRP1 1.1562 148.0000
fluoropyruvate CW-2 CTRP1 1.1562 148.0000
fluoropyruvate DLD-1 CTRP1 0.2890 37.0000
fluoropyruvate GP2D CTRP1 0.2890 37.0000
fluoropyruvate HCT116 CTRP1 1.1562 148.0000
fluoropyruvate HCT8 CTRP1 1.1562 148.0000
fluoropyruvate HT115 CTRP1 1.1562 148.0000
fluoropyruvate HT-29 CTRP1 1.1562 148.0000
fluoropyruvate HT-55 CTRP1 1.1562 148.0000
fluoropyruvate KM12 CTRP1 1.1562 148.0000
fluoropyruvate LOVO CTRP1 1.1562 148.0000
fluoropyruvate LS123 CTRP1 1.1562 148.0000
fluoropyruvate LS180 CTRP1 1.1562 148.0000
fluoropyruvate LS411N CTRP1 0.2890 37.0000
fluoropyruvate LS513 CTRP1 0.2890 37.0000
fluoropyruvate MDST8 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H508 CTRP1 1.1562 148.0000
fluoropyruvate RCM-1[HUMANESC] CTRP1 1.1562 148.0000
fluoropyruvate RKO CTRP1 1.1562 148.0000
fluoropyruvate SK-CO-1 CTRP1 0.2890 37.0000
fluoropyruvate SNU-1040 CTRP1 1.1562 148.0000
fluoropyruvate SNU-175 CTRP1 1.1562 148.0000
fluoropyruvate SNU-61 CTRP1 1.1562 148.0000
fluoropyruvate SNU-81 CTRP1 1.1562 148.0000
fluoropyruvate SNU-C2A CTRP1 0.2890 37.0000
fluoropyruvate SNU-C4 CTRP1 1.1562 148.0000
fluoropyruvate SNU-C5 CTRP1 1.1562 148.0000
fluoropyruvate SW403 CTRP1 0.2890 37.0000
fluoropyruvate SW48 CTRP1 0.2890 37.0000
fluoropyruvate SW480 CTRP1 1.1562 148.0000
fluoropyruvate SW620 CTRP1 1.1562 148.0000
fluoropyruvate SW948 CTRP1 1.1562 148.0000
fluoropyruvate HEP-G2 CTRP1 1.1562 148.0000
fluoropyruvate JHH-6 CTRP1 0.2890 37.0000
fluoropyruvate SNU-398 CTRP1 1.1562 148.0000
fluoropyruvate SNU-449 CTRP1 0.2890 37.0000
fluoropyruvate A-549 CTRP1 0.2890 37.0000
fluoropyruvate BEN CTRP1 0.2890 37.0000
fluoropyruvate CAL-12T CTRP1 1.1562 148.0000
fluoropyruvate CALU-3 CTRP1 0.2890 37.0000
fluoropyruvate CALU-6 CTRP1 0.2890 37.0000
fluoropyruvate CHAGO-K-1 CTRP1 0.2890 37.0000
fluoropyruvate COLO668 CTRP1 0.2890 37.0000
fluoropyruvate COLO699 CTRP1 1.1562 148.0000
fluoropyruvate COR-L23 CTRP1 1.1562 148.0000
fluoropyruvate COR-L279 CTRP1 0.2890 37.0000
fluoropyruvate COR-L51 CTRP1 1.1562 148.0000
fluoropyruvate COR-L88 CTRP1 0.2890 37.0000
fluoropyruvate DMS273 CTRP1 0.2890 37.0000
fluoropyruvate DV-90 CTRP1 0.2890 37.0000
fluoropyruvate EBC-1 CTRP1 0.2890 37.0000
fluoropyruvate EPLC-272H CTRP1 0.2890 37.0000
fluoropyruvate HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2890 37.0000
fluoropyruvate HCC1195 CTRP1 1.1562 148.0000
fluoropyruvate HCC1359 CTRP1 1.1562 148.0000
fluoropyruvate HCC15 CTRP1 1.1562 148.0000
fluoropyruvate HCC1833 CTRP1 1.1562 148.0000
fluoropyruvate HCC2108 CTRP1 1.1562 148.0000
fluoropyruvate HCC2935 CTRP1 1.1562 148.0000
fluoropyruvate HCC33 CTRP1 0.2890 37.0000
fluoropyruvate HCC4006 CTRP1 1.1562 148.0000
fluoropyruvate HCC44 CTRP1 0.2890 37.0000
fluoropyruvate HCC78 CTRP1 0.2890 37.0000
fluoropyruvate HCC827 CTRP1 1.1562 148.0000
fluoropyruvate KNS-62 CTRP1 0.2890 37.0000
fluoropyruvate LC-1-SQ-SF CTRP1 0.2890 37.0000
fluoropyruvate LCLC-103H CTRP1 0.2890 37.0000
fluoropyruvate LCLC-97TM1 CTRP1 0.2890 37.0000
fluoropyruvate LU-65 CTRP1 0.2890 37.0000
fluoropyruvate LU-99 CTRP1 0.2890 37.0000
fluoropyruvate LXF289 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1048 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1105 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H1299 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1355 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1373 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1435 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1437 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1568 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1573 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1666 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1694 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H1755 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H1781 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H1792 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1793 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1836 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H1876 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H1915 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1930 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1944 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H1963 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H1975 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H2009 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H2023 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2029 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H2030 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2073 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2081 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2110 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2122 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2126 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H2141 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2172 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2286 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H23 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H2342 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H2405 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H3255 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H358 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H441 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H460 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H522 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H596 CTRP1 1.1562 148.0000
fluoropyruvate NCI-H650 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H661 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H727 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H810 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H82 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H841 CTRP1 1.1562 148.0000
fluoropyruvate RERF-LC-KJ CTRP1 0.2890 37.0000
fluoropyruvate SCLC-21H CTRP1 1.1562 148.0000
fluoropyruvate SHP-77 CTRP1 0.2890 37.0000
fluoropyruvate SK-LU-1 CTRP1 1.1562 148.0000
fluoropyruvate SQ-1 CTRP1 1.1562 148.0000
fluoropyruvate T3M-10 CTRP1 1.1562 148.0000
fluoropyruvate VMRC-LCD CTRP1 0.2890 37.0000
fluoropyruvate KYSE-140 CTRP1 0.2890 37.0000
fluoropyruvate KYSE-410 CTRP1 0.2890 37.0000
fluoropyruvate KYSE-450 CTRP1 0.2890 37.0000
fluoropyruvate A2780 CTRP1 1.1562 148.0000
fluoropyruvate CAOV-3 CTRP1 1.1562 148.0000
fluoropyruvate COV318 CTRP1 0.2890 37.0000
fluoropyruvate COV362 CTRP1 1.1562 148.0000
fluoropyruvate COV434 CTRP1 1.1562 148.0000
fluoropyruvate COV644 CTRP1 1.1562 148.0000
fluoropyruvate EFO-21 CTRP1 0.2890 37.0000
fluoropyruvate EFO-27 CTRP1 1.1562 148.0000
fluoropyruvate HEYA8 CTRP1 0.2890 37.0000
fluoropyruvate IGROV-1 CTRP1 1.1562 148.0000
fluoropyruvate JHOC-5 CTRP1 1.1562 148.0000
fluoropyruvate JHOM-1 CTRP1 1.1562 148.0000
fluoropyruvate JHOS-4 CTRP1 0.2890 37.0000
fluoropyruvate OAW42 CTRP1 1.1562 148.0000
fluoropyruvate OV7 CTRP1 1.1562 148.0000
fluoropyruvate OV-90 CTRP1 1.1562 148.0000
fluoropyruvate OVCAR-4 CTRP1 1.1562 148.0000
fluoropyruvate OVCAR-8 CTRP1 1.1562 148.0000
fluoropyruvate OVK18 CTRP1 1.1562 148.0000
fluoropyruvate OVKATE CTRP1 1.1562 148.0000
fluoropyruvate OVMANA CTRP1 0.2890 37.0000
fluoropyruvate RKN CTRP1 1.1562 148.0000
fluoropyruvate RMG-I CTRP1 1.1562 148.0000
fluoropyruvate RMUG-S CTRP1 1.1562 148.0000
fluoropyruvate SK-OV-3 CTRP1 0.2890 37.0000
fluoropyruvate SNU-840 CTRP1 1.1562 148.0000
fluoropyruvate TYK-NU CTRP1 1.1562 148.0000
fluoropyruvate CAPAN-2 CTRP1 0.2890 37.0000
fluoropyruvate CFPAC-1 CTRP1 0.2890 37.0000
fluoropyruvate HPAC CTRP1 0.2890 37.0000
fluoropyruvate HUP-T4 CTRP1 0.2890 37.0000
fluoropyruvate KP-3 CTRP1 0.2890 37.0000
fluoropyruvate PANC03.27 CTRP1 0.2890 37.0000
fluoropyruvate PANC10.05 CTRP1 0.2890 37.0000
fluoropyruvate PATU8902 CTRP1 0.2890 37.0000
fluoropyruvate QGP-1 CTRP1 0.2890 37.0000
fluoropyruvate SUIT-2 CTRP1 0.2890 37.0000
fluoropyruvate MSTO-211H CTRP1 0.2890 37.0000
fluoropyruvate NCI-H2052 CTRP1 0.2890 37.0000
fluoropyruvate NCI-H28 CTRP1 0.2890 37.0000
fluoropyruvate MIAPACA-3 CTRP1 0.2890 37.0000
fluoropyruvate A-375 CTRP1 1.1562 148.0000
fluoropyruvate COLO741 CTRP1 0.2890 37.0000
fluoropyruvate G-361 CTRP1 0.2890 37.0000
fluoropyruvate HS852.T CTRP1 0.2890 37.0000
fluoropyruvate HS936.T CTRP1 0.2890 37.0000
fluoropyruvate HS944.T CTRP1 0.2890 37.0000
fluoropyruvate SK-MEL-1 CTRP1 1.1562 148.0000
fluoropyruvate SK-MEL-28 CTRP1 1.1562 148.0000
fluoropyruvate SK-MEL-5 CTRP1 1.1562 148.0000
fluoropyruvate G-401 CTRP1 0.2890 37.0000
fluoropyruvate HT-1080 CTRP1 1.1562 148.0000
fluoropyruvate AGS CTRP1 1.1562 148.0000
fluoropyruvate FU97 CTRP1 0.2890 37.0000
fluoropyruvate KE-97 CTRP1 0.2890 37.0000
fluoropyruvate MKN7 CTRP1 0.2890 37.0000
fluoropyruvate MKN74 CTRP1 0.2890 37.0000
fluoropyruvate NUGC-4 CTRP1 0.2890 37.0000
fluoropyruvate SH-10-TC CTRP1 0.2890 37.0000
fluoropyruvate HSC-2 CTRP1 0.2890 37.0000
fluoropyruvate SCC-9 CTRP1 1.1562 148.0000
fluoropyruvate 5637 CTRP1 0.2890 37.0000
fluoropyruvate HT-1376 CTRP1 0.2890 37.0000
fluoropyruvate KMBC-2 CTRP1 0.2890 37.0000
fluoropyruvate RT-4 CTRP1 0.2890 37.0000
fluoropyruvate UM-UC-3 CTRP1 0.2890 37.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.