Drug : Sitagliptin

CTRP2 Name : sitagliptin

Dataset : All
Synonyms :
Targets : DPP4
Pathways : inhibitor of dipetidyl peptidase-4

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
sitagliptin CAS-1 CTRP2 0.0020 66.0000
sitagliptin KPL-1 CTRP2 0.0020 66.0000
sitagliptin MKN1 CTRP2 0.0020 66.0000
sitagliptin 253J-BV CTRP2 0.0020 66.0000
sitagliptin BFTC-905 CTRP2 0.0020 66.0000
sitagliptin BFTC-909 CTRP2 0.0020 66.0000
sitagliptin CAL-29 CTRP2 0.0020 66.0000
sitagliptin CAL-62 CTRP2 0.0020 66.0000
sitagliptin HUCC-T1 CTRP2 0.0020 66.0000
sitagliptin NMC-G1 CTRP2 0.0020 66.0000
sitagliptin RPMI-7951 CTRP2 0.0020 66.0000
sitagliptin 253J CTRP2 0.0020 66.0000
sitagliptin ALL-SIL CTRP2 0.0020 66.0000
sitagliptin HDQ-P1 CTRP2 0.0020 66.0000
sitagliptin SNU-489 CTRP2 0.0020 66.0000
sitagliptin SNU-626 CTRP2 0.0020 66.0000
sitagliptin SNU-738 CTRP2 0.0020 66.0000
sitagliptin SNU-878 CTRP2 0.0020 66.0000
sitagliptin TUHR4TKB CTRP2 0.0020 66.0000
sitagliptin ACC-MESO-1 CTRP2 0.0020 66.0000
sitagliptin B-CPAP CTRP2 0.0020 66.0000
sitagliptin CGTH-W-1 CTRP2 0.0020 66.0000
sitagliptin COLO680N CTRP2 0.0020 66.0000
sitagliptin ECC12 CTRP2 0.0020 66.0000
sitagliptin HCC95 CTRP2 0.0020 66.0000
sitagliptin JMSU-1 CTRP2 0.0020 66.0000
sitagliptin RH41 CTRP2 0.0020 66.0000
sitagliptin SNU-175 CTRP2 0.0020 66.0000
sitagliptin WSU-DLCL2 CTRP2 0.0020 66.0000
sitagliptin 23132-87 CTRP2 0.0020 33.0000
sitagliptin 8305C CTRP2 0.0020 33.0000
sitagliptin BHY CTRP2 0.0020 66.0000
sitagliptin GSU CTRP2 0.0020 66.0000
sitagliptin JIMT-1 CTRP2 0.0020 66.0000
sitagliptin KMRC-20 CTRP2 0.0020 66.0000
sitagliptin OUMS-23 CTRP2 0.0020 66.0000
sitagliptin SNU-1076 CTRP2 0.0020 33.0000
sitagliptin SNU-1196 CTRP2 0.0020 66.0000
sitagliptin SNU-8 CTRP2 0.0020 66.0000
sitagliptin A-375 CTRP2 0.0020 33.0000
sitagliptin A-549 CTRP2 0.0020 33.0000
sitagliptin NCI-H2009 CTRP2 0.0020 33.0000
sitagliptin SNU-201 CTRP2 0.0020 33.0000
sitagliptin SUIT-2 CTRP2 0.0020 66.0000
sitagliptin SNU-1079 CTRP2 0.0020 33.0000
sitagliptin DEL CTRP2 0.0020 66.0000
sitagliptin HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP2 0.0020 66.0000
sitagliptin HCC15 CTRP2 0.0020 66.0000
sitagliptin KP-4 CTRP2 0.0020 66.0000
sitagliptin LU-99 CTRP2 0.0020 66.0000
sitagliptin NCI-H1155 CTRP2 0.0020 66.0000
sitagliptin NCI-H1581 CTRP2 0.0020 66.0000
sitagliptin NCI-H2106 CTRP2 0.0020 66.0000
sitagliptin NCI-H358 CTRP2 0.0020 66.0000
sitagliptin DLD-1 CTRP2 0.0020 66.0000
sitagliptin EM-2 CTRP2 0.0020 66.0000
sitagliptin JURL-MK1 CTRP2 0.0020 66.0000
sitagliptin P12-ICHIKAWA CTRP2 0.0020 66.0000
sitagliptin KE-37 CTRP2 0.0020 66.0000
sitagliptin KMS-21-BM CTRP2 0.0020 66.0000
sitagliptin LI-7 CTRP2 0.0020 66.0000
sitagliptin MHH-NB-11 CTRP2 0.0020 66.0000
sitagliptin MOLM-13 CTRP2 0.0020 66.0000
sitagliptin NCI-H28 CTRP2 0.0020 66.0000
sitagliptin 639V CTRP2 0.0020 66.0000
sitagliptin BXPC-3 CTRP2 0.0020 66.0000
sitagliptin CML-T1 CTRP2 0.0020 66.0000
sitagliptin GSS CTRP2 0.0020 66.0000
sitagliptin HCC366 CTRP2 0.0020 66.0000
sitagliptin KURAMOCHI CTRP2 0.0020 66.0000
sitagliptin LS411N CTRP2 0.0020 66.0000
sitagliptin LS513 CTRP2 0.0020 66.0000
sitagliptin ONCO-DG-1 CTRP2 0.0020 66.0000
sitagliptin ONS-76 CTRP2 0.0020 66.0000
sitagliptin SK-CO-1 CTRP2 0.0020 66.0000
sitagliptin SW48 CTRP2 0.0020 66.0000
sitagliptin VM-CUB-1 CTRP2 0.0020 66.0000
sitagliptin BEN CTRP2 0.0020 66.0000
sitagliptin CFPAC-1 CTRP2 0.0020 66.0000
sitagliptin HCC78 CTRP2 0.0020 66.0000
sitagliptin HT CTRP2 0.0020 66.0000
sitagliptin KU-19-19 CTRP2 0.0020 66.0000
sitagliptin NCI-H1299 CTRP2 0.0020 66.0000
sitagliptin NCI-H727 CTRP2 0.0020 66.0000
sitagliptin NCO2 CTRP2 0.0020 66.0000
sitagliptin OVTOKO CTRP2 0.0020 66.0000
sitagliptin P31-FUJ CTRP2 0.0020 66.0000
sitagliptin PEER CTRP2 0.0020 66.0000
sitagliptin RPMI-8402 CTRP2 0.0020 66.0000
sitagliptin SHP-77 CTRP2 0.0020 66.0000
sitagliptin SNU-1077 CTRP2 0.0020 66.0000
sitagliptin SNU-620 CTRP2 0.0020 66.0000
sitagliptin SU-DHL-1 CTRP2 0.0020 66.0000
sitagliptin COLO205 CTRP2 0.0020 66.0000
sitagliptin EHEB CTRP2 0.0020 66.0000
sitagliptin KI-JK CTRP2 0.0020 66.0000
sitagliptin KMM-1 CTRP2 0.0020 66.0000
sitagliptin LCLC-103H CTRP2 0.0020 66.0000
sitagliptin MKN45 CTRP2 0.0020 66.0000
sitagliptin NCI-H2405 CTRP2 0.0020 66.0000
sitagliptin NCI-H650 CTRP2 0.0020 66.0000
sitagliptin OS-RC-2 CTRP2 0.0020 66.0000
sitagliptin OVSAHO CTRP2 0.0020 66.0000
sitagliptin RL95-2 CTRP2 0.0020 66.0000
sitagliptin SNU-1041 CTRP2 0.0020 66.0000
sitagliptin SNU-1066 CTRP2 0.0020 66.0000
sitagliptin SW1353 CTRP2 0.0020 66.0000
sitagliptin SNU-213 CTRP2 0.0020 66.0000
sitagliptin 8505C CTRP2 0.0020 66.0000
sitagliptin CALU-3 CTRP2 0.0020 66.0000
sitagliptin DAOY CTRP2 0.0020 66.0000
sitagliptin GB-1 CTRP2 0.0020 66.0000
sitagliptin HCC1171 CTRP2 0.0020 66.0000
sitagliptin HCC44 CTRP2 0.0020 66.0000
sitagliptin NCI-H211 CTRP2 0.0020 66.0000
sitagliptin RERF-LC-A1 CTRP2 0.0020 66.0000
sitagliptin SBC-5 CTRP2 0.0020 66.0000
sitagliptin SF126 CTRP2 0.0020 66.0000
sitagliptin SNU-119 CTRP2 0.0020 66.0000
sitagliptin SNU-81 CTRP2 0.0020 66.0000
sitagliptin SNU-182 CTRP2 0.0020 66.0000
sitagliptin TCCSUP CTRP2 0.0020 66.0000
sitagliptin CAMA-1 CTRP2 0.0020 66.0000
sitagliptin DETROIT562 CTRP2 0.0020 66.0000
sitagliptin HEC-1-B CTRP2 0.0020 66.0000
sitagliptin HEP3B2.1-7 CTRP2 0.0020 66.0000
sitagliptin HSC-3 CTRP2 0.0020 66.0000
sitagliptin MCF-7 CTRP2 0.0020 66.0000
sitagliptin SNU-1105 CTRP2 0.0020 66.0000
sitagliptin U-87MGATCC CTRP2 0.0020 66.0000
sitagliptin JVM-3 CTRP2 0.0020 33.0000
sitagliptin 5637 CTRP2 0.0020 66.0000
sitagliptin CAL-12T CTRP2 0.0020 66.0000
sitagliptin HCC1588 CTRP2 0.0020 66.0000
sitagliptin HCC1833 CTRP2 0.0020 66.0000
sitagliptin HCC2279 CTRP2 0.0020 66.0000
sitagliptin KE-97 CTRP2 0.0020 66.0000
sitagliptin KP-3 CTRP2 0.0020 66.0000
sitagliptin KU812 CTRP2 0.0020 66.0000
sitagliptin KYSE-140 CTRP2 0.0020 66.0000
sitagliptin NALM-6 CTRP2 0.0020 66.0000
sitagliptin NUGC-4 CTRP2 0.0020 66.0000
sitagliptin TT CTRP2 0.0020 66.0000
sitagliptin AGS CTRP2 0.0020 66.0000
sitagliptin HCT116 CTRP2 0.0020 66.0000
sitagliptin HEC-108 CTRP2 0.0020 66.0000
sitagliptin HEC-59 CTRP2 0.0020 66.0000
sitagliptin HMC-1-8 CTRP2 0.0020 66.0000
sitagliptin HT-29 CTRP2 0.0020 66.0000
sitagliptin ISHIKAWA(HERAKLIO)02ER- CTRP2 0.0020 66.0000
sitagliptin JHOC-5 CTRP2 0.0020 66.0000
sitagliptin KYSE-180 CTRP2 0.0020 66.0000
sitagliptin LS180 CTRP2 0.0020 66.0000
sitagliptin MELHO CTRP2 0.0020 66.0000
sitagliptin MHH-ES-1 CTRP2 0.0020 66.0000
sitagliptin MOR-CPR CTRP2 0.0020 66.0000
sitagliptin NCI-H460 CTRP2 0.0020 66.0000
sitagliptin HCC2108 CTRP2 0.0020 66.0000
sitagliptin HCC827 CTRP2 0.0020 66.0000
sitagliptin HEC-251 CTRP2 0.0020 66.0000
sitagliptin HEC-265 CTRP2 0.0020 66.0000
sitagliptin HEC-6 CTRP2 0.0020 66.0000
sitagliptin HEL CTRP2 0.0020 66.0000
sitagliptin JHUEM-2 CTRP2 0.0020 66.0000
sitagliptin JURKAT CTRP2 0.0020 66.0000
sitagliptin KCL-22 CTRP2 0.0020 66.0000
sitagliptin KE-39 CTRP2 0.0020 66.0000
sitagliptin KM-H2 CTRP2 0.0020 66.0000
sitagliptin LAMA-84 CTRP2 0.0020 66.0000
sitagliptin NCI-H2030 CTRP2 0.0020 66.0000
sitagliptin SNU-719 CTRP2 0.0020 66.0000
sitagliptin KLE CTRP2 0.0020 66.0000
sitagliptin KMS-26 CTRP2 0.0020 66.0000
sitagliptin KMS-27 CTRP2 0.0020 66.0000
sitagliptin NCI-H1838 CTRP2 0.0020 66.0000
sitagliptin NCI-H196 CTRP2 0.0020 66.0000
sitagliptin NCI-H292 CTRP2 0.0020 66.0000
sitagliptin SK-MEL-1 CTRP2 0.0020 66.0000
sitagliptin HCC1937 CTRP2 0.0020 66.0000
sitagliptin HDLM-2 CTRP2 0.0020 66.0000
sitagliptin HUH-28 CTRP2 0.0020 66.0000
sitagliptin MV4-11 CTRP2 0.0020 66.0000
sitagliptin NCI-H526 CTRP2 0.0020 66.0000
sitagliptin NCI-H69 CTRP2 0.0020 66.0000
sitagliptin NCI-H929 CTRP2 0.0020 66.0000
sitagliptin NCI-N87 CTRP2 0.0020 66.0000
sitagliptin PF-382 CTRP2 0.0020 66.0000
sitagliptin SF295 CTRP2 0.0020 66.0000
sitagliptin SNU-1272 CTRP2 0.0020 66.0000
sitagliptin SNU-308 CTRP2 0.0020 66.0000
sitagliptin SNU-478 CTRP2 0.0020 66.0000
sitagliptin BHT-101 CTRP2 0.0020 66.0000
sitagliptin CAL-148 CTRP2 0.0020 66.0000
sitagliptin CAL-51 CTRP2 0.0020 66.0000
sitagliptin HCC1395 CTRP2 0.0020 66.0000
sitagliptin HT115 CTRP2 0.0020 66.0000
sitagliptin LN-18 CTRP2 0.0020 66.0000
sitagliptin LN-229 CTRP2 0.0020 66.0000
sitagliptin NCI-H1734 CTRP2 0.0020 66.0000
sitagliptin NCI-H2291 CTRP2 0.0020 66.0000
sitagliptin RERF-LC-AD1 CTRP2 0.0020 66.0000
sitagliptin SNU-1214 CTRP2 0.0020 66.0000
sitagliptin SNU-46 CTRP2 0.0020 66.0000
sitagliptin SNU-466 CTRP2 0.0020 66.0000
sitagliptin SNU-5 CTRP2 0.0020 66.0000
sitagliptin SNU-668 CTRP2 0.0020 66.0000
sitagliptin SNU-899 CTRP2 0.0020 66.0000
sitagliptin TE-10 CTRP2 0.0020 66.0000
sitagliptin TE-9 CTRP2 0.0020 66.0000
sitagliptin YD-10B CTRP2 0.0020 66.0000
sitagliptin YD-15 CTRP2 0.0020 66.0000
sitagliptin YD-38 CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.