Drug : Bms-191011

CTRP1 Name : BMS-191011

Dataset : All
Synonyms :
Targets : KCNMA1;KCNMB1
Pathways : opener of large-conductance Ca2+-activated potassium (BK/Maxi-K) channels

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BMS-191011 U2OS CTRP1 0.2604 33.3330
BMS-191011 MCF-7 CTRP1 0.2604 33.3330
BMS-191011 GAMG CTRP1 0.2603 33.3330
BMS-191011 LN-229 CTRP1 0.2604 33.3330
BMS-191011 SF295 CTRP1 0.2603 33.3330
BMS-191011 HEC-108 CTRP1 0.2603 33.3330
BMS-191011 HEC-151 CTRP1 0.2604 33.3330
BMS-191011 HEC-251 CTRP1 0.2603 33.3330
BMS-191011 HEC-265 CTRP1 0.2603 33.3330
BMS-191011 HEC-59 CTRP1 0.2603 33.3330
BMS-191011 HEC-6 CTRP1 0.2603 33.3330
BMS-191011 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
BMS-191011 JHUEM-2 CTRP1 0.2604 33.3330
BMS-191011 KLE CTRP1 0.2603 33.3330
BMS-191011 MFE-319 CTRP1 0.2603 33.3330
BMS-191011 SNG-M CTRP1 0.2603 33.3330
BMS-191011 AMO1 CTRP1 0.2604 33.3330
BMS-191011 BL-70 CTRP1 0.2603 33.3330
BMS-191011 EJM CTRP1 0.2604 33.3330
BMS-191011 GDM-1 CTRP1 0.2604 33.3330
BMS-191011 HT CTRP1 0.2603 33.3330
BMS-191011 KMS-11 CTRP1 0.2604 33.3330
BMS-191011 KU812 CTRP1 0.2603 33.3330
BMS-191011 LP-1 CTRP1 0.2604 33.3330
BMS-191011 MC116 CTRP1 0.2603 33.3330
BMS-191011 MOLM-16 CTRP1 0.2604 33.3330
BMS-191011 NOMO-1 CTRP1 0.2604 33.3330
BMS-191011 NU-DUL-1 CTRP1 0.2604 33.3330
BMS-191011 OCI-AML-3 CTRP1 0.2604 33.3330
BMS-191011 OCI-LY10 CTRP1 0.2604 33.3330
BMS-191011 P3HR-1 CTRP1 0.2603 33.3330
BMS-191011 PL21 CTRP1 0.2604 33.3330
BMS-191011 RPMI-8226 CTRP1 0.2604 33.3330
BMS-191011 SKM-1 CTRP1 0.2604 33.3330
BMS-191011 SU-DHL-4 CTRP1 0.2604 33.3330
BMS-191011 SU-DHL-5 CTRP1 0.2604 33.3330
BMS-191011 THP-1 CTRP1 0.2604 33.3330
BMS-191011 U-937 CTRP1 0.2604 33.3330
BMS-191011 WSU-DLCL2 CTRP1 0.2604 33.3330
BMS-191011 RCC10RGB CTRP1 0.2604 33.3330
BMS-191011 VMRC-RCW CTRP1 0.2603 33.3330
BMS-191011 C2BBE1 CTRP1 0.2603 33.3330
BMS-191011 CL-34 CTRP1 0.2604 33.3330
BMS-191011 CL-40 CTRP1 0.2604 33.3330
BMS-191011 COLO205 CTRP1 0.2603 33.3330
BMS-191011 COLO320 CTRP1 0.2604 16.6670
BMS-191011 COLO678 CTRP1 0.2604 33.3330
BMS-191011 CW-2 CTRP1 0.2604 33.3330
BMS-191011 DLD-1 CTRP1 0.2603 33.3330
BMS-191011 GP2D CTRP1 0.2603 33.3330
BMS-191011 HCT116 CTRP1 0.2604 33.3330
BMS-191011 HCT8 CTRP1 0.2604 33.3330
BMS-191011 HT115 CTRP1 0.2604 33.3330
BMS-191011 HT-29 CTRP1 0.2604 33.3330
BMS-191011 HT-55 CTRP1 0.2604 33.3330
BMS-191011 KM12 CTRP1 0.2604 33.3330
BMS-191011 LOVO CTRP1 0.2604 33.3330
BMS-191011 LS123 CTRP1 0.2604 33.3330
BMS-191011 LS180 CTRP1 0.2604 33.3330
BMS-191011 LS411N CTRP1 0.2603 33.3330
BMS-191011 LS513 CTRP1 0.2603 33.3330
BMS-191011 MDST8 CTRP1 0.2604 33.3330
BMS-191011 NCI-H508 CTRP1 0.2604 33.3330
BMS-191011 RCM-1[HUMANESC] CTRP1 0.2604 33.3330
BMS-191011 RKO CTRP1 0.2604 33.3330
BMS-191011 SK-CO-1 CTRP1 0.2603 33.3330
BMS-191011 SNU-1040 CTRP1 0.2604 33.3330
BMS-191011 SNU-175 CTRP1 0.2604 33.3330
BMS-191011 SNU-61 CTRP1 0.2604 33.3330
BMS-191011 SNU-81 CTRP1 0.2604 33.3330
BMS-191011 SNU-C2A CTRP1 0.2603 33.3330
BMS-191011 SNU-C4 CTRP1 0.2604 33.3330
BMS-191011 SNU-C5 CTRP1 0.2604 33.3330
BMS-191011 SW403 CTRP1 0.2603 33.3330
BMS-191011 SW48 CTRP1 0.2603 33.3330
BMS-191011 SW480 CTRP1 0.2604 33.3330
BMS-191011 SW620 CTRP1 0.2604 33.3330
BMS-191011 SW948 CTRP1 0.2604 33.3330
BMS-191011 HEP-G2 CTRP1 0.2604 33.3330
BMS-191011 JHH-6 CTRP1 0.2603 33.3330
BMS-191011 SNU-398 CTRP1 0.2604 33.3330
BMS-191011 SNU-449 CTRP1 0.2603 33.3330
BMS-191011 A-549 CTRP1 0.2603 33.3330
BMS-191011 BEN CTRP1 0.2603 33.3330
BMS-191011 CAL-12T CTRP1 0.2604 33.3330
BMS-191011 CALU-3 CTRP1 0.2603 33.3330
BMS-191011 CALU-6 CTRP1 0.2603 33.3330
BMS-191011 CHAGO-K-1 CTRP1 0.2603 33.3330
BMS-191011 COLO668 CTRP1 0.2603 33.3330
BMS-191011 COLO699 CTRP1 0.2604 33.3330
BMS-191011 COR-L23 CTRP1 0.2604 33.3330
BMS-191011 COR-L279 CTRP1 0.2603 33.3330
BMS-191011 COR-L51 CTRP1 0.2604 33.3330
BMS-191011 COR-L88 CTRP1 0.2603 33.3330
BMS-191011 DMS273 CTRP1 0.2603 33.3330
BMS-191011 DV-90 CTRP1 0.2603 33.3330
BMS-191011 EBC-1 CTRP1 0.2603 33.3330
BMS-191011 EPLC-272H CTRP1 0.2603 33.3330
BMS-191011 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
BMS-191011 HCC1195 CTRP1 0.2604 33.3330
BMS-191011 HCC1359 CTRP1 0.2604 33.3330
BMS-191011 HCC15 CTRP1 0.2604 33.3330
BMS-191011 HCC1833 CTRP1 0.2604 33.3330
BMS-191011 HCC2108 CTRP1 0.2604 33.3330
BMS-191011 HCC2935 CTRP1 0.2604 33.3330
BMS-191011 HCC33 CTRP1 0.2603 33.3330
BMS-191011 HCC4006 CTRP1 0.2604 33.3330
BMS-191011 HCC44 CTRP1 0.2603 33.3330
BMS-191011 HCC78 CTRP1 0.2603 33.3330
BMS-191011 HCC827 CTRP1 0.2604 33.3330
BMS-191011 KNS-62 CTRP1 0.2603 33.3330
BMS-191011 LC-1-SQ-SF CTRP1 0.2603 33.3330
BMS-191011 LCLC-103H CTRP1 0.2603 33.3330
BMS-191011 LCLC-97TM1 CTRP1 0.2603 33.3330
BMS-191011 LU-65 CTRP1 0.2603 33.3330
BMS-191011 LU-99 CTRP1 0.2603 33.3330
BMS-191011 LXF289 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1048 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1105 CTRP1 0.2604 33.3330
BMS-191011 NCI-H1299 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1355 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1373 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1435 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1437 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1568 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1573 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1666 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1694 CTRP1 0.2604 33.3330
BMS-191011 NCI-H1755 CTRP1 0.2604 33.3330
BMS-191011 NCI-H1781 CTRP1 0.2604 33.3330
BMS-191011 NCI-H1792 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1793 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1836 CTRP1 0.2604 33.3330
BMS-191011 NCI-H1876 CTRP1 0.2604 33.3330
BMS-191011 NCI-H1915 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1930 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1944 CTRP1 0.2603 33.3330
BMS-191011 NCI-H1963 CTRP1 0.2604 33.3330
BMS-191011 NCI-H1975 CTRP1 0.2603 33.3330
BMS-191011 NCI-H2009 CTRP1 0.2603 33.3330
BMS-191011 NCI-H2023 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2029 CTRP1 0.2603 33.3330
BMS-191011 NCI-H2030 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2073 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2081 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2110 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2122 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2126 CTRP1 0.2603 33.3330
BMS-191011 NCI-H2141 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2172 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2286 CTRP1 0.2603 33.3330
BMS-191011 NCI-H23 CTRP1 0.2603 33.3330
BMS-191011 NCI-H2342 CTRP1 0.2604 33.3330
BMS-191011 NCI-H2405 CTRP1 0.2603 33.3330
BMS-191011 NCI-H3255 CTRP1 0.2604 33.3330
BMS-191011 NCI-H358 CTRP1 0.2603 33.3330
BMS-191011 NCI-H441 CTRP1 0.2604 33.3330
BMS-191011 NCI-H460 CTRP1 0.2604 33.3330
BMS-191011 NCI-H522 CTRP1 0.2603 33.3330
BMS-191011 NCI-H596 CTRP1 0.2604 33.3330
BMS-191011 NCI-H650 CTRP1 0.2603 33.3330
BMS-191011 NCI-H661 CTRP1 0.2603 33.3330
BMS-191011 NCI-H727 CTRP1 0.2603 33.3330
BMS-191011 NCI-H810 CTRP1 0.2603 33.3330
BMS-191011 NCI-H82 CTRP1 0.2603 33.3330
BMS-191011 NCI-H841 CTRP1 0.2604 33.3330
BMS-191011 RERF-LC-KJ CTRP1 0.2603 33.3330
BMS-191011 SCLC-21H CTRP1 0.2604 33.3330
BMS-191011 SHP-77 CTRP1 0.2603 33.3330
BMS-191011 SK-LU-1 CTRP1 0.2604 33.3330
BMS-191011 SQ-1 CTRP1 0.2604 33.3330
BMS-191011 T3M-10 CTRP1 0.2604 33.3330
BMS-191011 VMRC-LCD CTRP1 0.2603 33.3330
BMS-191011 KYSE-140 CTRP1 0.2603 33.3330
BMS-191011 KYSE-410 CTRP1 0.2603 33.3330
BMS-191011 KYSE-450 CTRP1 0.2603 33.3330
BMS-191011 A2780 CTRP1 0.2604 33.3330
BMS-191011 CAOV-3 CTRP1 0.2604 33.3330
BMS-191011 COV318 CTRP1 0.2603 33.3330
BMS-191011 COV362 CTRP1 0.2604 33.3330
BMS-191011 COV434 CTRP1 0.2604 33.3330
BMS-191011 COV644 CTRP1 0.2604 33.3330
BMS-191011 EFO-21 CTRP1 0.2603 33.3330
BMS-191011 EFO-27 CTRP1 0.2604 33.3330
BMS-191011 HEYA8 CTRP1 0.2603 33.3330
BMS-191011 IGROV-1 CTRP1 0.2604 33.3330
BMS-191011 JHOC-5 CTRP1 0.2604 33.3330
BMS-191011 JHOM-1 CTRP1 0.2604 33.3330
BMS-191011 JHOS-4 CTRP1 0.2603 33.3330
BMS-191011 OAW42 CTRP1 0.2604 33.3330
BMS-191011 OV7 CTRP1 0.2604 33.3330
BMS-191011 OV-90 CTRP1 0.2604 33.3330
BMS-191011 OVCAR-4 CTRP1 0.2604 33.3330
BMS-191011 OVCAR-8 CTRP1 0.2604 33.3330
BMS-191011 OVK18 CTRP1 0.2604 33.3330
BMS-191011 OVKATE CTRP1 0.2604 33.3330
BMS-191011 OVMANA CTRP1 0.2603 33.3330
BMS-191011 RKN CTRP1 0.2604 33.3330
BMS-191011 RMG-I CTRP1 0.2604 33.3330
BMS-191011 RMUG-S CTRP1 0.2604 33.3330
BMS-191011 SK-OV-3 CTRP1 0.2603 33.3330
BMS-191011 SNU-840 CTRP1 0.2604 33.3330
BMS-191011 TYK-NU CTRP1 0.2604 33.3330
BMS-191011 CAPAN-2 CTRP1 0.2603 33.3330
BMS-191011 CFPAC-1 CTRP1 0.2603 33.3330
BMS-191011 HPAC CTRP1 0.2603 33.3330
BMS-191011 HUP-T4 CTRP1 0.2603 33.3330
BMS-191011 KP-3 CTRP1 0.2603 33.3330
BMS-191011 PANC03.27 CTRP1 0.2603 33.3330
BMS-191011 PANC10.05 CTRP1 0.2603 33.3330
BMS-191011 PATU8902 CTRP1 0.2603 33.3330
BMS-191011 QGP-1 CTRP1 0.2603 33.3330
BMS-191011 SUIT-2 CTRP1 0.2603 33.3330
BMS-191011 MSTO-211H CTRP1 0.2603 33.3330
BMS-191011 NCI-H2052 CTRP1 0.2603 33.3330
BMS-191011 NCI-H28 CTRP1 0.2603 33.3330
BMS-191011 MIAPACA-3 CTRP1 0.2603 33.3330
BMS-191011 A-375 CTRP1 0.2604 33.3330
BMS-191011 COLO741 CTRP1 0.2603 33.3330
BMS-191011 G-361 CTRP1 0.2603 33.3330
BMS-191011 HS852.T CTRP1 0.2603 33.3330
BMS-191011 HS936.T CTRP1 0.2603 33.3330
BMS-191011 HS944.T CTRP1 0.2603 33.3330
BMS-191011 SK-MEL-1 CTRP1 0.2604 33.3330
BMS-191011 SK-MEL-28 CTRP1 0.2604 33.3330
BMS-191011 SK-MEL-5 CTRP1 0.2604 33.3330
BMS-191011 G-401 CTRP1 0.2603 33.3330
BMS-191011 HT-1080 CTRP1 0.2604 33.3330
BMS-191011 AGS CTRP1 0.2604 33.3330
BMS-191011 FU97 CTRP1 0.2603 33.3330
BMS-191011 KE-97 CTRP1 0.2603 33.3330
BMS-191011 MKN7 CTRP1 0.2603 33.3330
BMS-191011 MKN74 CTRP1 0.2603 33.3330
BMS-191011 NUGC-4 CTRP1 0.2603 33.3330
BMS-191011 SH-10-TC CTRP1 0.2603 33.3330
BMS-191011 HSC-2 CTRP1 0.2603 33.3330
BMS-191011 SCC-9 CTRP1 0.2604 33.3330
BMS-191011 5637 CTRP1 0.2603 33.3330
BMS-191011 HT-1376 CTRP1 0.2603 33.3330
BMS-191011 KMBC-2 CTRP1 0.2603 33.3330
BMS-191011 RT-4 CTRP1 0.2603 33.3330
BMS-191011 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.