Drug : Bix-01338

CTRP1 Name : BIX-01338

Dataset : All
Synonyms :
Targets : EHMT1;EHMT2
Pathways : inhibitor of histone lysine methyltransferase

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BIX-01338 GAMG CTRP1 0.2603 33.3330
BIX-01338 SF295 CTRP1 0.2603 33.3330
BIX-01338 HEC-108 CTRP1 0.2603 33.3330
BIX-01338 HEC-251 CTRP1 0.2603 33.3330
BIX-01338 HEC-265 CTRP1 0.2603 33.3330
BIX-01338 HEC-59 CTRP1 0.2603 33.3330
BIX-01338 HEC-6 CTRP1 0.2603 33.3330
BIX-01338 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
BIX-01338 KLE CTRP1 0.2603 33.3330
BIX-01338 MFE-319 CTRP1 0.2603 33.3330
BIX-01338 SNG-M CTRP1 0.2603 33.3330
BIX-01338 BL-70 CTRP1 0.2603 33.3330
BIX-01338 HT CTRP1 0.2603 33.3330
BIX-01338 KU812 CTRP1 0.2603 33.3330
BIX-01338 MC116 CTRP1 0.2603 33.3330
BIX-01338 P3HR-1 CTRP1 0.2603 33.3330
BIX-01338 VMRC-RCW CTRP1 0.2603 33.3330
BIX-01338 C2BBE1 CTRP1 0.2603 33.3330
BIX-01338 COLO205 CTRP1 0.2603 33.3330
BIX-01338 DLD-1 CTRP1 0.2603 33.3330
BIX-01338 GP2D CTRP1 0.2603 33.3330
BIX-01338 LS411N CTRP1 0.2603 33.3330
BIX-01338 LS513 CTRP1 0.2603 33.3330
BIX-01338 SK-CO-1 CTRP1 0.2603 33.3330
BIX-01338 SNU-C2A CTRP1 0.2603 33.3330
BIX-01338 SW403 CTRP1 0.2603 33.3330
BIX-01338 SW48 CTRP1 0.2603 33.3330
BIX-01338 JHH-6 CTRP1 0.2603 33.3330
BIX-01338 SNU-449 CTRP1 0.2603 33.3330
BIX-01338 A-549 CTRP1 0.2603 33.3330
BIX-01338 BEN CTRP1 0.2603 33.3330
BIX-01338 CALU-3 CTRP1 0.2603 33.3330
BIX-01338 CALU-6 CTRP1 0.2603 33.3330
BIX-01338 CHAGO-K-1 CTRP1 0.2603 33.3330
BIX-01338 COLO668 CTRP1 0.2603 33.3330
BIX-01338 COR-L279 CTRP1 0.2603 33.3330
BIX-01338 COR-L88 CTRP1 0.2603 33.3330
BIX-01338 DMS273 CTRP1 0.2603 33.3330
BIX-01338 DV-90 CTRP1 0.2603 33.3330
BIX-01338 EBC-1 CTRP1 0.2603 33.3330
BIX-01338 EPLC-272H CTRP1 0.2603 33.3330
BIX-01338 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
BIX-01338 HCC33 CTRP1 0.2603 33.3330
BIX-01338 HCC44 CTRP1 0.2603 33.3330
BIX-01338 HCC78 CTRP1 0.2603 33.3330
BIX-01338 KNS-62 CTRP1 0.2603 33.3330
BIX-01338 LC-1-SQ-SF CTRP1 0.2603 33.3330
BIX-01338 LCLC-103H CTRP1 0.2603 33.3330
BIX-01338 LCLC-97TM1 CTRP1 0.2603 33.3330
BIX-01338 LU-65 CTRP1 0.2603 33.3330
BIX-01338 LU-99 CTRP1 0.2603 33.3330
BIX-01338 LXF289 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1048 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1299 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1355 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1373 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1435 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1437 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1568 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1573 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1666 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1792 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1793 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1915 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1930 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1944 CTRP1 0.2603 33.3330
BIX-01338 NCI-H1975 CTRP1 0.2603 33.3330
BIX-01338 NCI-H2009 CTRP1 0.2603 33.3330
BIX-01338 NCI-H2029 CTRP1 0.2603 33.3330
BIX-01338 NCI-H2126 CTRP1 0.2603 33.3330
BIX-01338 NCI-H2286 CTRP1 0.2603 33.3330
BIX-01338 NCI-H23 CTRP1 0.2603 33.3330
BIX-01338 NCI-H2405 CTRP1 0.2603 33.3330
BIX-01338 NCI-H358 CTRP1 0.2603 33.3330
BIX-01338 NCI-H522 CTRP1 0.2603 33.3330
BIX-01338 NCI-H650 CTRP1 0.2603 33.3330
BIX-01338 NCI-H661 CTRP1 0.2603 33.3330
BIX-01338 NCI-H727 CTRP1 0.2603 33.3330
BIX-01338 NCI-H810 CTRP1 0.2603 33.3330
BIX-01338 NCI-H82 CTRP1 0.2603 33.3330
BIX-01338 RERF-LC-KJ CTRP1 0.2603 33.3330
BIX-01338 SHP-77 CTRP1 0.2603 33.3330
BIX-01338 VMRC-LCD CTRP1 0.2603 33.3330
BIX-01338 KYSE-140 CTRP1 0.2603 33.3330
BIX-01338 KYSE-410 CTRP1 0.2603 33.3330
BIX-01338 KYSE-450 CTRP1 0.2603 33.3330
BIX-01338 COV318 CTRP1 0.2603 33.3330
BIX-01338 EFO-21 CTRP1 0.2603 33.3330
BIX-01338 HEYA8 CTRP1 0.2603 33.3330
BIX-01338 JHOS-4 CTRP1 0.2603 33.3330
BIX-01338 OVMANA CTRP1 0.2603 33.3330
BIX-01338 SK-OV-3 CTRP1 0.2603 33.3330
BIX-01338 CAPAN-2 CTRP1 0.2603 33.3330
BIX-01338 CFPAC-1 CTRP1 0.2603 33.3330
BIX-01338 HPAC CTRP1 0.2603 33.3330
BIX-01338 HUP-T4 CTRP1 0.2603 33.3330
BIX-01338 KP-3 CTRP1 0.2603 33.3330
BIX-01338 PANC03.27 CTRP1 0.2603 33.3330
BIX-01338 PANC10.05 CTRP1 0.2603 33.3330
BIX-01338 PATU8902 CTRP1 0.2603 33.3330
BIX-01338 QGP-1 CTRP1 0.2603 33.3330
BIX-01338 SUIT-2 CTRP1 0.2603 33.3330
BIX-01338 MSTO-211H CTRP1 0.2603 33.3330
BIX-01338 NCI-H2052 CTRP1 0.2603 33.3330
BIX-01338 NCI-H28 CTRP1 0.2603 33.3330
BIX-01338 MIAPACA-3 CTRP1 0.2603 33.3330
BIX-01338 COLO741 CTRP1 0.2603 33.3330
BIX-01338 G-361 CTRP1 0.2603 33.3330
BIX-01338 HS852.T CTRP1 0.2603 33.3330
BIX-01338 HS936.T CTRP1 0.2603 33.3330
BIX-01338 HS944.T CTRP1 0.2603 33.3330
BIX-01338 G-401 CTRP1 0.2603 33.3330
BIX-01338 FU97 CTRP1 0.2603 33.3330
BIX-01338 KE-97 CTRP1 0.2603 33.3330
BIX-01338 MKN7 CTRP1 0.2603 33.3330
BIX-01338 MKN74 CTRP1 0.2603 33.3330
BIX-01338 NUGC-4 CTRP1 0.2603 33.3330
BIX-01338 SH-10-TC CTRP1 0.2603 33.3330
BIX-01338 HSC-2 CTRP1 0.2603 33.3330
BIX-01338 5637 CTRP1 0.2603 33.3330
BIX-01338 HT-1376 CTRP1 0.2603 33.3330
BIX-01338 KMBC-2 CTRP1 0.2603 33.3330
BIX-01338 RT-4 CTRP1 0.2603 33.3330
BIX-01338 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.