Drug : Fatostatin

CTRP1 Name : fatostatin

Dataset : All
Synonyms :
Targets : SREBF1;SREBF2
Pathways : inhibitor of sterol regulatory element binding transcription factor 1 and 2 signaling

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
fatostatin U2OS CTRP1 0.2604 33.3330
fatostatin MCF-7 CTRP1 0.2604 33.3330
fatostatin GAMG CTRP1 0.2603 33.3330
fatostatin LN-229 CTRP1 0.2604 33.3330
fatostatin SF295 CTRP1 0.2603 33.3330
fatostatin HEC-108 CTRP1 0.2603 33.3330
fatostatin HEC-151 CTRP1 0.2604 33.3330
fatostatin HEC-251 CTRP1 0.2603 33.3330
fatostatin HEC-265 CTRP1 0.2603 33.3330
fatostatin HEC-59 CTRP1 0.2603 33.3330
fatostatin HEC-6 CTRP1 0.2603 33.3330
fatostatin ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
fatostatin JHUEM-2 CTRP1 0.2604 33.3330
fatostatin KLE CTRP1 0.2603 33.3330
fatostatin MFE-319 CTRP1 0.2603 33.3330
fatostatin SNG-M CTRP1 0.2603 33.3330
fatostatin AMO1 CTRP1 0.2604 33.3330
fatostatin BL-70 CTRP1 0.2603 33.3330
fatostatin EJM CTRP1 0.2604 33.3330
fatostatin GDM-1 CTRP1 0.2604 33.3330
fatostatin HT CTRP1 0.2603 33.3330
fatostatin KMS-11 CTRP1 0.2604 33.3330
fatostatin KU812 CTRP1 0.2603 33.3330
fatostatin LP-1 CTRP1 0.2604 33.3330
fatostatin MC116 CTRP1 0.2603 33.3330
fatostatin MOLM-16 CTRP1 0.2604 33.3330
fatostatin NOMO-1 CTRP1 0.2604 33.3330
fatostatin NU-DUL-1 CTRP1 0.2604 33.3330
fatostatin OCI-AML-3 CTRP1 0.2604 33.3330
fatostatin OCI-LY10 CTRP1 0.2604 33.3330
fatostatin P3HR-1 CTRP1 0.2603 33.3330
fatostatin PL21 CTRP1 0.2604 33.3330
fatostatin RPMI-8226 CTRP1 0.2604 33.3330
fatostatin SKM-1 CTRP1 0.2604 33.3330
fatostatin SU-DHL-4 CTRP1 0.2604 33.3330
fatostatin SU-DHL-5 CTRP1 0.2604 33.3330
fatostatin THP-1 CTRP1 0.2604 33.3330
fatostatin U-937 CTRP1 0.2604 33.3330
fatostatin WSU-DLCL2 CTRP1 0.2604 33.3330
fatostatin RCC10RGB CTRP1 0.2604 33.3330
fatostatin VMRC-RCW CTRP1 0.2603 33.3330
fatostatin C2BBE1 CTRP1 0.2603 33.3330
fatostatin CL-34 CTRP1 0.2604 33.3330
fatostatin CL-40 CTRP1 0.2604 33.3330
fatostatin COLO205 CTRP1 0.2603 33.3330
fatostatin COLO320 CTRP1 0.2604 33.3330
fatostatin COLO678 CTRP1 0.2604 33.3330
fatostatin CW-2 CTRP1 0.2604 33.3330
fatostatin DLD-1 CTRP1 0.2603 33.3330
fatostatin GP2D CTRP1 0.2603 33.3330
fatostatin HCT116 CTRP1 0.2604 33.3330
fatostatin HCT8 CTRP1 0.2604 33.3330
fatostatin HT115 CTRP1 0.2604 33.3330
fatostatin HT-29 CTRP1 0.2604 33.3330
fatostatin HT-55 CTRP1 0.2604 33.3330
fatostatin KM12 CTRP1 0.2604 33.3330
fatostatin LOVO CTRP1 0.2604 33.3330
fatostatin LS123 CTRP1 0.2604 33.3330
fatostatin LS180 CTRP1 0.2604 33.3330
fatostatin LS411N CTRP1 0.2603 33.3330
fatostatin LS513 CTRP1 0.2603 33.3330
fatostatin MDST8 CTRP1 0.2604 33.3330
fatostatin NCI-H508 CTRP1 0.2604 33.3330
fatostatin RCM-1[HUMANESC] CTRP1 0.2604 33.3330
fatostatin RKO CTRP1 0.2604 33.3330
fatostatin SK-CO-1 CTRP1 0.2603 33.3330
fatostatin SNU-1040 CTRP1 0.2604 33.3330
fatostatin SNU-175 CTRP1 0.2604 33.3330
fatostatin SNU-61 CTRP1 0.2604 33.3330
fatostatin SNU-81 CTRP1 0.2604 33.3330
fatostatin SNU-C2A CTRP1 0.2603 33.3330
fatostatin SNU-C4 CTRP1 0.2604 33.3330
fatostatin SNU-C5 CTRP1 0.2604 33.3330
fatostatin SW403 CTRP1 0.2603 33.3330
fatostatin SW48 CTRP1 0.2603 33.3330
fatostatin SW480 CTRP1 0.2604 33.3330
fatostatin SW620 CTRP1 0.2604 33.3330
fatostatin SW948 CTRP1 0.2604 33.3330
fatostatin HEP-G2 CTRP1 0.2604 33.3330
fatostatin JHH-6 CTRP1 0.2603 33.3330
fatostatin SNU-398 CTRP1 0.2604 33.3330
fatostatin SNU-449 CTRP1 0.2603 33.3330
fatostatin A-549 CTRP1 0.2603 33.3330
fatostatin BEN CTRP1 0.2603 33.3330
fatostatin CAL-12T CTRP1 0.2604 33.3330
fatostatin CALU-3 CTRP1 0.2603 33.3330
fatostatin CALU-6 CTRP1 0.2603 33.3330
fatostatin CHAGO-K-1 CTRP1 0.2603 33.3330
fatostatin COLO668 CTRP1 0.2603 33.3330
fatostatin COLO699 CTRP1 0.2604 33.3330
fatostatin COR-L23 CTRP1 0.2604 33.3330
fatostatin COR-L279 CTRP1 0.2603 33.3330
fatostatin COR-L51 CTRP1 0.2604 33.3330
fatostatin COR-L88 CTRP1 0.2603 33.3330
fatostatin DMS273 CTRP1 0.2603 33.3330
fatostatin DV-90 CTRP1 0.2603 33.3330
fatostatin EBC-1 CTRP1 0.2603 33.3330
fatostatin EPLC-272H CTRP1 0.2603 33.3330
fatostatin HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
fatostatin HCC1195 CTRP1 0.2604 33.3330
fatostatin HCC1359 CTRP1 0.2604 33.3330
fatostatin HCC15 CTRP1 0.2604 33.3330
fatostatin HCC1833 CTRP1 0.2604 33.3330
fatostatin HCC2108 CTRP1 0.2604 33.3330
fatostatin HCC2935 CTRP1 0.2604 33.3330
fatostatin HCC33 CTRP1 0.2603 33.3330
fatostatin HCC4006 CTRP1 0.2604 33.3330
fatostatin HCC44 CTRP1 0.2603 33.3330
fatostatin HCC78 CTRP1 0.2603 33.3330
fatostatin HCC827 CTRP1 0.2604 33.3330
fatostatin KNS-62 CTRP1 0.2603 33.3330
fatostatin LC-1-SQ-SF CTRP1 0.2603 33.3330
fatostatin LCLC-103H CTRP1 0.2603 33.3330
fatostatin LCLC-97TM1 CTRP1 0.2603 33.3330
fatostatin LU-65 CTRP1 0.2603 33.3330
fatostatin LU-99 CTRP1 0.2603 33.3330
fatostatin LXF289 CTRP1 0.2603 33.3330
fatostatin NCI-H1048 CTRP1 0.2603 33.3330
fatostatin NCI-H1105 CTRP1 0.2604 33.3330
fatostatin NCI-H1299 CTRP1 0.2603 33.3330
fatostatin NCI-H1355 CTRP1 0.2603 33.3330
fatostatin NCI-H1373 CTRP1 0.2603 33.3330
fatostatin NCI-H1435 CTRP1 0.2603 33.3330
fatostatin NCI-H1437 CTRP1 0.2603 33.3330
fatostatin NCI-H1568 CTRP1 0.2603 33.3330
fatostatin NCI-H1573 CTRP1 0.2603 33.3330
fatostatin NCI-H1666 CTRP1 0.2603 33.3330
fatostatin NCI-H1694 CTRP1 0.2604 33.3330
fatostatin NCI-H1755 CTRP1 0.2604 33.3330
fatostatin NCI-H1781 CTRP1 0.2604 33.3330
fatostatin NCI-H1792 CTRP1 0.2603 33.3330
fatostatin NCI-H1793 CTRP1 0.2603 33.3330
fatostatin NCI-H1836 CTRP1 0.2604 33.3330
fatostatin NCI-H1876 CTRP1 0.2604 33.3330
fatostatin NCI-H1915 CTRP1 0.2603 33.3330
fatostatin NCI-H1930 CTRP1 0.2603 33.3330
fatostatin NCI-H1944 CTRP1 0.2603 33.3330
fatostatin NCI-H1963 CTRP1 0.2604 33.3330
fatostatin NCI-H1975 CTRP1 0.2603 33.3330
fatostatin NCI-H2009 CTRP1 0.2603 33.3330
fatostatin NCI-H2023 CTRP1 0.2604 33.3330
fatostatin NCI-H2029 CTRP1 0.2603 33.3330
fatostatin NCI-H2030 CTRP1 0.2604 33.3330
fatostatin NCI-H2073 CTRP1 0.2604 33.3330
fatostatin NCI-H2081 CTRP1 0.2604 33.3330
fatostatin NCI-H2110 CTRP1 0.2604 33.3330
fatostatin NCI-H2122 CTRP1 0.2604 33.3330
fatostatin NCI-H2126 CTRP1 0.2603 33.3330
fatostatin NCI-H2141 CTRP1 0.2604 33.3330
fatostatin NCI-H2172 CTRP1 0.2604 33.3330
fatostatin NCI-H2286 CTRP1 0.2603 33.3330
fatostatin NCI-H23 CTRP1 0.2603 33.3330
fatostatin NCI-H2342 CTRP1 0.2604 33.3330
fatostatin NCI-H2405 CTRP1 0.2603 33.3330
fatostatin NCI-H3255 CTRP1 0.2604 33.3330
fatostatin NCI-H358 CTRP1 0.2603 33.3330
fatostatin NCI-H441 CTRP1 0.2604 33.3330
fatostatin NCI-H460 CTRP1 0.2604 33.3330
fatostatin NCI-H522 CTRP1 0.2603 33.3330
fatostatin NCI-H596 CTRP1 0.2604 33.3330
fatostatin NCI-H650 CTRP1 0.2603 33.3330
fatostatin NCI-H661 CTRP1 0.2603 33.3330
fatostatin NCI-H727 CTRP1 0.2603 33.3330
fatostatin NCI-H810 CTRP1 0.2603 33.3330
fatostatin NCI-H82 CTRP1 0.2603 33.3330
fatostatin NCI-H841 CTRP1 0.2604 33.3330
fatostatin RERF-LC-KJ CTRP1 0.2603 33.3330
fatostatin SCLC-21H CTRP1 0.2604 33.3330
fatostatin SHP-77 CTRP1 0.2603 33.3330
fatostatin SK-LU-1 CTRP1 0.2604 33.3330
fatostatin SQ-1 CTRP1 0.2604 33.3330
fatostatin T3M-10 CTRP1 0.2604 33.3330
fatostatin VMRC-LCD CTRP1 0.2603 33.3330
fatostatin KYSE-140 CTRP1 0.2603 33.3330
fatostatin KYSE-410 CTRP1 0.2603 33.3330
fatostatin KYSE-450 CTRP1 0.2603 33.3330
fatostatin A2780 CTRP1 0.2604 33.3330
fatostatin CAOV-3 CTRP1 0.2604 33.3330
fatostatin COV318 CTRP1 0.2603 33.3330
fatostatin COV362 CTRP1 0.2604 33.3330
fatostatin COV434 CTRP1 0.2604 33.3330
fatostatin COV644 CTRP1 0.2604 33.3330
fatostatin EFO-21 CTRP1 0.2603 33.3330
fatostatin EFO-27 CTRP1 0.2604 33.3330
fatostatin HEYA8 CTRP1 0.2603 33.3330
fatostatin IGROV-1 CTRP1 0.2604 33.3330
fatostatin JHOC-5 CTRP1 0.2604 33.3330
fatostatin JHOM-1 CTRP1 0.2604 33.3330
fatostatin JHOS-4 CTRP1 0.2603 33.3330
fatostatin OAW42 CTRP1 0.2604 33.3330
fatostatin OV7 CTRP1 0.2604 33.3330
fatostatin OV-90 CTRP1 0.2604 33.3330
fatostatin OVCAR-4 CTRP1 0.2604 33.3330
fatostatin OVCAR-8 CTRP1 0.2604 33.3330
fatostatin OVK18 CTRP1 0.2604 33.3330
fatostatin OVKATE CTRP1 0.2604 33.3330
fatostatin OVMANA CTRP1 0.2603 33.3330
fatostatin RKN CTRP1 0.2604 33.3330
fatostatin RMG-I CTRP1 0.2604 33.3330
fatostatin RMUG-S CTRP1 0.2604 33.3330
fatostatin SK-OV-3 CTRP1 0.2603 33.3330
fatostatin SNU-840 CTRP1 0.2604 33.3330
fatostatin TYK-NU CTRP1 0.2604 33.3330
fatostatin CAPAN-2 CTRP1 0.2603 33.3330
fatostatin CFPAC-1 CTRP1 0.2603 33.3330
fatostatin HPAC CTRP1 0.2603 33.3330
fatostatin HUP-T4 CTRP1 0.2603 33.3330
fatostatin KP-3 CTRP1 0.2603 33.3330
fatostatin PANC03.27 CTRP1 0.2603 33.3330
fatostatin PANC10.05 CTRP1 0.2603 33.3330
fatostatin PATU8902 CTRP1 0.2603 33.3330
fatostatin QGP-1 CTRP1 0.2603 33.3330
fatostatin SUIT-2 CTRP1 0.2603 33.3330
fatostatin MSTO-211H CTRP1 0.2603 33.3330
fatostatin NCI-H2052 CTRP1 0.2603 33.3330
fatostatin NCI-H28 CTRP1 0.2603 33.3330
fatostatin MIAPACA-3 CTRP1 0.2603 33.3330
fatostatin A-375 CTRP1 0.2604 33.3330
fatostatin COLO741 CTRP1 0.2603 33.3330
fatostatin G-361 CTRP1 0.2603 33.3330
fatostatin HS852.T CTRP1 0.2603 33.3330
fatostatin HS936.T CTRP1 0.2603 33.3330
fatostatin HS944.T CTRP1 0.2603 33.3330
fatostatin SK-MEL-1 CTRP1 0.2604 33.3330
fatostatin SK-MEL-28 CTRP1 0.2604 33.3330
fatostatin SK-MEL-5 CTRP1 0.2604 33.3330
fatostatin G-401 CTRP1 0.2603 33.3330
fatostatin HT-1080 CTRP1 0.2604 33.3330
fatostatin AGS CTRP1 0.2604 33.3330
fatostatin FU97 CTRP1 0.2603 33.3330
fatostatin KE-97 CTRP1 0.2603 33.3330
fatostatin MKN7 CTRP1 0.2603 33.3330
fatostatin MKN74 CTRP1 0.2603 33.3330
fatostatin NUGC-4 CTRP1 0.2603 33.3330
fatostatin SH-10-TC CTRP1 0.2603 33.3330
fatostatin HSC-2 CTRP1 0.2603 33.3330
fatostatin SCC-9 CTRP1 0.2604 33.3330
fatostatin 5637 CTRP1 0.2603 33.3330
fatostatin HT-1376 CTRP1 0.2603 33.3330
fatostatin KMBC-2 CTRP1 0.2603 33.3330
fatostatin RT-4 CTRP1 0.2603 33.3330
fatostatin UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.