Drug : Tki258

CCLE Name : TKI258

Dataset : All
Synonyms :
Targets : Multitargeted RTK inhibitor
Pathways :

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
TKI258 1321N1 CCLE 0.0025 8.0000
TKI258 22RV1 CCLE 0.0025 8.0000
TKI258 42-MG-BA CCLE 0.0025 8.0000
TKI258 5637 CCLE 0.0025 8.0000
TKI258 639V CCLE 0.0025 8.0000
TKI258 697 CCLE 0.0025 8.0000
TKI258 769-P CCLE 0.0025 8.0000
TKI258 786-O CCLE 0.0025 8.0000
TKI258 8305C CCLE 0.0025 8.0000
TKI258 8505C CCLE 0.0025 8.0000
TKI258 8-MG-BA CCLE 0.0025 8.0000
TKI258 A-172 CCLE 0.0025 8.0000
TKI258 A-204 CCLE 0.0025 8.0000
TKI258 A2058 CCLE 0.0025 8.0000
TKI258 A-253 CCLE 0.0025 8.0000
TKI258 A2780 CCLE 0.0025 8.0000
TKI258 A-375 CCLE 0.0025 8.0000
TKI258 A-549 CCLE 0.0025 8.0000
TKI258 A-673 CCLE 0.0025 8.0000
TKI258 ACHN CCLE 0.0025 8.0000
TKI258 ALL-SIL CCLE 0.0025 8.0000
TKI258 AMO1 CCLE 0.0025 8.0000
TKI258 AN3-CA CCLE 0.0025 8.0000
TKI258 ASPC-1 CCLE 0.0025 8.0000
TKI258 AU565 CCLE 0.0025 8.0000
TKI258 AZ-521 CCLE 0.0025 8.0000
TKI258 B-CPAP CCLE 0.0025 8.0000
TKI258 BDCM CCLE 0.0025 8.0000
TKI258 BFTC-909 CCLE 0.0025 8.0000
TKI258 BGC-823 CCLE 0.0025 8.0000
TKI258 BL-41 CCLE 0.0025 8.0000
TKI258 BL-70 CCLE 0.0025 8.0000
TKI258 BT-20 CCLE 0.0025 8.0000
TKI258 BT-474 CCLE 0.0025 8.0000
TKI258 BT-549 CCLE 0.0025 8.0000
TKI258 BXPC-3 CCLE 0.0025 8.0000
TKI258 C2BBE1 CCLE 0.0025 8.0000
TKI258 C32[HUMANMELANOMA] CCLE 0.0025 8.0000
TKI258 HEP-G2-C3A CCLE 0.0025 8.0000
TKI258 CAKI-2 CCLE 0.0025 8.0000
TKI258 CAL-12T CCLE 0.0025 8.0000
TKI258 CAL-27 CCLE 0.0025 8.0000
TKI258 CAL-78 CCLE 0.0025 8.0000
TKI258 CAL-85-1 CCLE 0.0025 8.0000
TKI258 CALU-1 CCLE 0.0025 8.0000
TKI258 CALU-3 CCLE 0.0025 8.0000
TKI258 CALU-6 CCLE 0.0025 8.0000
TKI258 CAMA-1 CCLE 0.0025 8.0000
TKI258 CAPAN-2 CCLE 0.0025 8.0000
TKI258 CAS-1 CCLE 0.0025 8.0000
TKI258 CCK-81 CCLE 0.0025 8.0000
TKI258 CHL-1 CCLE 0.0025 8.0000
TKI258 CHP-212 CCLE 0.0025 8.0000
TKI258 CI-1 CCLE 0.0025 8.0000
TKI258 CMK-86 CCLE 0.0025 8.0000
TKI258 COLO201 CCLE 0.0025 8.0000
TKI258 COLO205 CCLE 0.0025 8.0000
TKI258 COLO320 CCLE 0.0025 8.0000
TKI258 COLO677 CCLE 0.0025 8.0000
TKI258 COLO678 CCLE 0.0025 8.0000
TKI258 COLO679 CCLE 0.0025 8.0000
TKI258 COLO699 CCLE 0.0025 8.0000
TKI258 COLO741 CCLE 0.0025 8.0000
TKI258 COR-L105 CCLE 0.0025 8.0000
TKI258 COR-L23 CCLE 0.0025 8.0000
TKI258 COV318 CCLE 0.0025 8.0000
TKI258 COV504 CCLE 0.0025 8.0000
TKI258 DAOY CCLE 0.0025 8.0000
TKI258 DBTRG-05MG CCLE 0.0025 8.0000
TKI258 DEL CCLE 0.0025 8.0000
TKI258 DETROIT562 CCLE 0.0025 8.0000
TKI258 DK-MG CCLE 0.0025 8.0000
TKI258 DMS114 CCLE 0.0025 8.0000
TKI258 DOHH2 CCLE 0.0025 8.0000
TKI258 DOV13 CCLE 0.0025 8.0000
TKI258 DU145 CCLE 0.0025 8.0000
TKI258 DV-90 CCLE 0.0025 8.0000
TKI258 EB1 CCLE 0.0025 8.0000
TKI258 EB2 CCLE 0.0025 8.0000
TKI258 EBC-1 CCLE 0.0025 8.0000
TKI258 EFE-184 CCLE 0.0025 8.0000
TKI258 EFM-19 CCLE 0.0025 8.0000
TKI258 EFO-21 CCLE 0.0025 8.0000
TKI258 EFO-27 CCLE 0.0025 8.0000
TKI258 EM-2 CCLE 0.0025 8.0000
TKI258 EN CCLE 0.0025 8.0000
TKI258 ES-2 CCLE 0.0025 8.0000
TKI258 ESS-1 CCLE 0.0025 8.0000
TKI258 F-36P CCLE 0.0025 8.0000
TKI258 FADU CCLE 0.0025 8.0000
TKI258 FU97 CCLE 0.0025 8.0000
TKI258 FU-OV-1 CCLE 0.0025 8.0000
TKI258 G-361 CCLE 0.0025 8.0000
TKI258 G-401 CCLE 0.0025 8.0000
TKI258 G-402 CCLE 0.0025 8.0000
TKI258 GAMG CCLE 0.0025 8.0000
TKI258 GB-1 CCLE 0.0025 8.0000
TKI258 GCIY CCLE 0.0025 8.0000
TKI258 GCT CCLE 0.0025 8.0000
TKI258 GI-1 CCLE 0.0025 8.0000
TKI258 GLC-82 CCLE 0.0025 8.0000
TKI258 GMS-10 CCLE 0.0025 8.0000
TKI258 GRANTA-519 CCLE 0.0025 8.0000
TKI258 H4 CCLE 0.0025 8.0000
TKI258 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CCLE 0.0025 8.0000
TKI258 HCC1187 CCLE 0.0025 8.0000
TKI258 HCC1395 CCLE 0.0025 8.0000
TKI258 HCC15 CCLE 0.0025 8.0000
TKI258 HCC1569 CCLE 0.0025 8.0000
TKI258 HCC1806 CCLE 0.0025 8.0000
TKI258 HCC1954 CCLE 0.0025 8.0000
TKI258 HCC2935 CCLE 0.0025 8.0000
TKI258 HCC4006 CCLE 0.0025 8.0000
TKI258 HCC44 CCLE 0.0025 8.0000
TKI258 HCC-56 CCLE 0.0025 8.0000
TKI258 HCC70 CCLE 0.0025 8.0000
TKI258 HCC78 CCLE 0.0025 8.0000
TKI258 HCC827 CCLE 0.0025 8.0000
TKI258 HCT116 CCLE 0.0025 8.0000
TKI258 HCT15 CCLE 0.0025 8.0000
TKI258 HD-MY-Z CCLE 0.0025 8.0000
TKI258 HDQ-P1 CCLE 0.0025 8.0000
TKI258 HEC-151 CCLE 0.0025 8.0000
TKI258 HEC-1-A CCLE 0.0025 8.0000
TKI258 HEC-1-B CCLE 0.0080 8.0000
TKI258 HEC-251 CCLE 0.0025 8.0000
TKI258 HEC-265 CCLE 0.0025 8.0000
TKI258 HEC-59 CCLE 0.0025 8.0000
TKI258 HEC-6 CCLE 0.0025 8.0000
TKI258 HEL92.1.7 CCLE 0.0025 8.0000
TKI258 HEP3B2.1-7 CCLE 0.0025 8.0000
TKI258 HEP-G2 CCLE 0.0025 8.0000
TKI258 HEYA8 CCLE 0.0025 8.0000
TKI258 HGC-27 CCLE 0.0025 8.0000
TKI258 HH[HUMANLYMPHOMA] CCLE 0.0025 8.0000
TKI258 HLE CCLE 0.0025 8.0000
TKI258 HLF CCLE 0.0025 8.0000
TKI258 HMC-1-8 CCLE 0.0025 8.0000
TKI258 HMCB CCLE 0.0025 8.0000
TKI258 HOS CCLE 0.0025 8.0000
TKI258 HPAC CCLE 0.0025 8.0000
TKI258 HPAF-II CCLE 0.0025 8.0000
TKI258 HS229.T CCLE 0.0025 8.0000
TKI258 HS294T CCLE 0.0025 8.0000
TKI258 HS578T CCLE 0.0025 8.0000
TKI258 HS683 CCLE 0.0025 8.0000
TKI258 HS695T CCLE 0.0025 8.0000
TKI258 HS729.T CCLE 0.0025 8.0000
TKI258 HS739.T CCLE 0.0025 8.0000
TKI258 HS746.T CCLE 0.0025 8.0000
TKI258 HS766T CCLE 0.0025 8.0000
TKI258 HS840.T CCLE 0.0025 8.0000
TKI258 HS852.T CCLE 0.0025 8.0000
TKI258 HS895.T CCLE 0.0025 8.0000
TKI258 HS936.T CCLE 0.0025 8.0000
TKI258 HS939.T CCLE 0.0025 8.0000
TKI258 HS944.T CCLE 0.0025 8.0000
TKI258 HSC-2 CCLE 0.0025 8.0000
TKI258 HT CCLE 0.0025 8.0000
TKI258 HT-1080 CCLE 0.0025 8.0000
TKI258 HT-1197 CCLE 0.0025 8.0000
TKI258 HT-1376 CCLE 0.0025 8.0000
TKI258 HT-144 CCLE 0.0025 8.0000
TKI258 HT-29 CCLE 0.0025 8.0000
TKI258 HUCC-T1 CCLE 0.0025 8.0000
TKI258 HUH-1 CCLE 0.0025 8.0000
TKI258 HUP-T3 CCLE 0.0025 8.0000
TKI258 HUP-T4 CCLE 0.0025 8.0000
TKI258 HUT78 CCLE 0.0025 8.0000
TKI258 IA-LM CCLE 0.0025 8.0000
TKI258 IGR-37 CCLE 0.0025 8.0000
TKI258 IGR-39 CCLE 0.0025 8.0000
TKI258 IGROV-1 CCLE 0.0025 8.0000
TKI258 IM95 CCLE 0.0025 8.0000
TKI258 IMR-32 CCLE 0.0025 8.0000
TKI258 IPC-298 CCLE 0.0025 8.0000
TKI258 ISHIKAWA(HERAKLIO)02ER- CCLE 0.0025 8.0000
TKI258 IST-MES1 CCLE 0.0025 8.0000
TKI258 IST-MES2 CCLE 0.0025 8.0000
TKI258 J82 CCLE 0.0025 8.0000
TKI258 JHH-2 CCLE 0.0025 8.0000
TKI258 JHH-4 CCLE 0.0025 8.0000
TKI258 JHH-5 CCLE 0.0025 8.0000
TKI258 JHH-6 CCLE 0.0025 8.0000
TKI258 JHH-7 CCLE 0.0025 8.0000
TKI258 JHOS-2 CCLE 0.0025 8.0000
TKI258 JHOS-4 CCLE 0.0025 8.0000
TKI258 JHUEM-2 CCLE 0.0025 8.0000
TKI258 JM-1 CCLE 0.0025 8.0000
TKI258 JMSU-1 CCLE 0.0025 8.0000
TKI258 JURKAT CCLE 0.0025 8.0000
TKI258 JVM-3 CCLE 0.0025 8.0000
TKI258 K029AX CCLE 0.0025 8.0000
TKI258 KALS-1 CCLE 0.0025 8.0000
TKI258 KARPAS-299 CCLE 0.0025 8.0000
TKI258 KARPAS-422 CCLE 0.0025 8.0000
TKI258 KARPAS-620 CCLE 0.0025 8.0000
TKI258 KASUMI-2 CCLE 0.0025 8.0000
TKI258 KCI-MOH1 CCLE 0.0025 8.0000
TKI258 KCL-22 CCLE 0.0025 8.0000
TKI258 KE-39 CCLE 0.0025 8.0000
TKI258 KE-97 CCLE 0.0025 8.0000
TKI258 KELLY CCLE 0.0025 8.0000
TKI258 KG-1 CCLE 0.0025 8.0000
TKI258 KHM-1B CCLE 0.0025 8.0000
TKI258 KLE CCLE 0.0025 8.0000
TKI258 KMBC-2 CCLE 0.0025 8.0000
TKI258 KMM-1 CCLE 0.0025 8.0000
TKI258 KMRC-1 CCLE 0.0025 8.0000
TKI258 KMRC-2 CCLE 0.0025 8.0000
TKI258 KMS-11 CCLE 0.0025 8.0000
TKI258 KMS-12-BM CCLE 0.0025 8.0000
TKI258 KMS-26 CCLE 0.0025 8.0000
TKI258 KMS-34 CCLE 0.0025 8.0000
TKI258 KNS-42 CCLE 0.0025 8.0000
TKI258 KNS-60 CCLE 0.0025 8.0000
TKI258 KNS-62 CCLE 0.0025 8.0000
TKI258 KNS-81 CCLE 0.0025 8.0000
TKI258 KO52 CCLE 0.0025 8.0000
TKI258 KP-1N CCLE 0.0025 8.0000
TKI258 KP-1NL CCLE 0.0025 8.0000
TKI258 KP-2 CCLE 0.0025 8.0000
TKI258 KP-3 CCLE 0.0025 8.0000
TKI258 KP-4 CCLE 0.0025 8.0000
TKI258 KP-N-SI9S CCLE 0.0025 8.0000
TKI258 KU812 CCLE 0.0025 8.0000
TKI258 KURAMOCHI CCLE 0.0025 8.0000
TKI258 KYM-1 CCLE 0.0025 8.0000
TKI258 KYSE-140 CCLE 0.0025 8.0000
TKI258 KYSE-150 CCLE 0.0025 8.0000
TKI258 KYSE-180 CCLE 0.0025 8.0000
TKI258 KYSE-30 CCLE 0.0025 8.0000
TKI258 KYSE-410 CCLE 0.0025 8.0000
TKI258 KYSE-450 CCLE 0.0025 8.0000
TKI258 KYSE-510 CCLE 0.0025 8.0000
TKI258 KYSE-520 CCLE 0.0025 8.0000
TKI258 KYSE-70 CCLE 0.0025 8.0000
TKI258 L3.3 CCLE 0.0025 8.0000
TKI258 L-363 CCLE 0.0025 8.0000
TKI258 L-428 CCLE 0.0025 8.0000
TKI258 LC-1-SQ-SF CCLE 0.0025 8.0000
TKI258 LCLC-103H CCLE 0.0025 8.0000
TKI258 LN-18 CCLE 0.0025 8.0000
TKI258 LN-229 CCLE 0.0025 8.0000
TKI258 LOU-NH91 CCLE 0.0025 8.0000
TKI258 LOX-IMVI CCLE 0.0025 8.0000
TKI258 LP-1 CCLE 0.0025 8.0000
TKI258 LS123 CCLE 0.0025 8.0000
TKI258 LS411N CCLE 0.0025 8.0000
TKI258 LS513 CCLE 0.0025 8.0000
TKI258 LU-99 CCLE 0.0025 8.0000
TKI258 LUDLU-1 CCLE 0.0025 8.0000
TKI258 M059J CCLE 0.0025 8.0000
TKI258 MALME-3M CCLE 0.0025 8.0000
TKI258 MDA-MB-157 CCLE 0.0025 8.0000
TKI258 MC116 CCLE 0.0025 8.0000
TKI258 MCAS CCLE 0.0025 8.0000
TKI258 MCF-7 CCLE 0.0025 8.0000
TKI258 MDA-MB-175-VII CCLE 0.0025 8.0000
TKI258 MDA-MB-415 CCLE 0.0025 8.0000
TKI258 MDA-MB-435S CCLE 0.0025 8.0000
TKI258 MDA-MB-436 CCLE 0.0025 8.0000
TKI258 MDA-MB-453 CCLE 0.0025 8.0000
TKI258 MDA-MB-468 CCLE 0.0025 8.0000
TKI258 MEC-1 CCLE 0.0025 8.0000
TKI258 MEG-01 CCLE 0.0025 8.0000
TKI258 MELHO CCLE 0.0025 8.0000
TKI258 MES-SA CCLE 0.0025 8.0000
TKI258 MEWO CCLE 0.0025 8.0000
TKI258 MFE-280 CCLE 0.0025 8.0000
TKI258 MFE-296 CCLE 0.0025 8.0000
TKI258 MFE-319 CCLE 0.0025 8.0000
TKI258 MG-63 CCLE 0.0025 8.0000
TKI258 MHH-ES-1 CCLE 0.0025 8.0000
TKI258 MIAPACA-2 CCLE 0.0025 8.0000
TKI258 MINO CCLE 0.0025 8.0000
TKI258 MJ CCLE 0.0025 8.0000
TKI258 MKN45 CCLE 0.0025 8.0000
TKI258 MKN7 CCLE 0.0025 8.0000
TKI258 MKN74 CCLE 0.0025 8.0000
TKI258 MOG-G-CCM CCLE 0.0025 8.0000
TKI258 MOLP-8 CCLE 0.0025 8.0000
TKI258 MOLT-16 CCLE 0.0025 8.0000
TKI258 MONO-MAC-1 CCLE 0.0025 8.0000
TKI258 MOR-CPR CCLE 0.0025 8.0000
TKI258 MPP89 CCLE 0.0025 8.0000
TKI258 MSTO-211H CCLE 0.0025 8.0000
TKI258 NCI-H1048 CCLE 0.0025 8.0000
TKI258 NCI-H1092 CCLE 0.0025 8.0000
TKI258 NCI-H1155 CCLE 0.0025 8.0000
TKI258 NCI-H1184 CCLE 0.0025 8.0000
TKI258 NCI-H1299 CCLE 0.0025 8.0000
TKI258 NCI-H1339 CCLE 0.0025 8.0000
TKI258 NCI-H1341 CCLE 0.0025 8.0000
TKI258 NCI-H1355 CCLE 0.0025 8.0000
TKI258 NCI-H1373 CCLE 0.0025 8.0000
TKI258 NCI-H1563 CCLE 0.0025 8.0000
TKI258 NCI-H1568 CCLE 0.0025 8.0000
TKI258 NCI-H1573 CCLE 0.0025 8.0000
TKI258 NCI-H1581 CCLE 0.0025 8.0000
TKI258 NCI-H1648 CCLE 0.0025 8.0000
TKI258 NCI-H1650 CCLE 0.0025 8.0000
TKI258 NCI-H1651 CCLE 0.0025 8.0000
TKI258 NCI-H1666 CCLE 0.0025 8.0000
TKI258 NCI-H1693 CCLE 0.0025 8.0000
TKI258 NCI-H1694 CCLE 0.0025 8.0000
TKI258 NCI-H1703 CCLE 0.0025 8.0000
TKI258 NCI-H1792 CCLE 0.0025 8.0000
TKI258 NCI-H1793 CCLE 0.0025 8.0000
TKI258 NCI-H1869 CCLE 0.0025 8.0000
TKI258 NCI-H1915 CCLE 0.0025 8.0000
TKI258 NCI-H1944 CCLE 0.0025 8.0000
TKI258 NCI-H1975 CCLE 0.0025 8.0000
TKI258 NCI-H2009 CCLE 0.0025 8.0000
TKI258 NCI-H2023 CCLE 0.0025 8.0000
TKI258 NCI-H2030 CCLE 0.0025 8.0000
TKI258 NCI-H2052 CCLE 0.0025 8.0000
TKI258 NCI-H2085 CCLE 0.0025 8.0000
TKI258 NCI-H2087 CCLE 0.0025 8.0000
TKI258 NCI-H211 CCLE 0.0025 8.0000
TKI258 NCI-H2122 CCLE 0.0025 8.0000
TKI258 NCI-H2170 CCLE 0.0025 8.0000
TKI258 NCI-H2172 CCLE 0.0025 8.0000
TKI258 NCI-H2228 CCLE 0.0025 8.0000
TKI258 NCI-H226 CCLE 0.0025 8.0000
TKI258 NCI-H2286 CCLE 0.0025 8.0000
TKI258 NCI-H23 CCLE 0.0025 8.0000
TKI258 NCI-H2444 CCLE 0.0025 8.0000
TKI258 NCI-H2452 CCLE 0.0025 8.0000
TKI258 NCI-H28 CCLE 0.0025 8.0000
TKI258 NCI-H322 CCLE 0.0025 8.0000
TKI258 NCI-H3255 CCLE 0.0025 8.0000
TKI258 NCI-H358 CCLE 0.0025 8.0000
TKI258 NCI-H441 CCLE 0.0025 8.0000
TKI258 NCI-H460 CCLE 0.0025 8.0000
TKI258 NCI-H520 CCLE 0.0025 8.0000
TKI258 NCI-H522 CCLE 0.0025 8.0000
TKI258 NCI-H647 CCLE 0.0025 8.0000
TKI258 NCI-H650 CCLE 0.0025 8.0000
TKI258 NCI-H661 CCLE 0.0025 8.0000
TKI258 NCI-H727 CCLE 0.0025 8.0000
TKI258 NCI-H747 CCLE 0.0025 8.0000
TKI258 NCI-H810 CCLE 0.0025 8.0000
TKI258 NCI-N87 CCLE 0.0025 8.0000
TKI258 NCO2 CCLE 0.0025 8.0000
TKI258 OVCAR-3 CCLE 0.0025 8.0000
TKI258 NUGC-3 CCLE 0.0025 8.0000
TKI258 NUGC-4 CCLE 0.0025 8.0000
TKI258 OC314 CCLE 0.0025 8.0000
TKI258 OC315 CCLE 0.0025 8.0000
TKI258 OC316 CCLE 0.0025 8.0000
TKI258 OCI-AML-2 CCLE 0.0025 8.0000
TKI258 OCI-AML-5 CCLE 0.0025 8.0000
TKI258 OCI-LY10 CCLE 0.0025 8.0000
TKI258 OCUM-1 CCLE 0.0025 8.0000
TKI258 OE21 CCLE 0.0025 8.0000
TKI258 OE33 CCLE 0.0025 8.0000
TKI258 ONCO-DG-1 CCLE 0.0025 8.0000
TKI258 ONS-76 CCLE 0.0025 8.0000
TKI258 OPM-2 CCLE 0.0025 8.0000
TKI258 OV-90 CCLE 0.0025 8.0000
TKI258 OVCAR-4 CCLE 0.0025 8.0000
TKI258 OVCAR-8 CCLE 0.0025 8.0000
TKI258 OVMANA CCLE 0.0025 8.0000
TKI258 OVSAHO CCLE 0.0025 8.0000
TKI258 OVTOKO CCLE 0.0025 8.0000
TKI258 P12-ICHIKAWA CCLE 0.0025 8.0000
TKI258 P31-FUJ CCLE 0.0025 8.0000
TKI258 P3HR-1 CCLE 0.0025 8.0000
TKI258 PANC02.03 CCLE 0.0025 8.0000
TKI258 PANC03.27 CCLE 0.0025 8.0000
TKI258 PANC04.03 CCLE 0.0025 8.0000
TKI258 PANC10.05 CCLE 0.0025 8.0000
TKI258 PATU8902 CCLE 0.0025 8.0000
TKI258 PC-14 CCLE 0.0025 8.0000
TKI258 PC-3 CCLE 0.0025 8.0000
TKI258 PFEIFFER CCLE 0.0025 8.0000
TKI258 PK-1 CCLE 0.0025 8.0000
TKI258 PK-45H CCLE 0.0025 8.0000
TKI258 PK-59 CCLE 0.0025 8.0000
TKI258 PL45 CCLE 0.0025 8.0000
TKI258 PLC-PRF-5 CCLE 0.0025 8.0000
TKI258 PSN1 CCLE 0.0025 8.0000
TKI258 QGP-1 CCLE 0.0025 8.0000
TKI258 RAJI CCLE 0.0025 8.0000
TKI258 RD CCLE 0.0025 8.0000
TKI258 REH CCLE 0.0025 8.0000
TKI258 RERF-GC-1B CCLE 0.0025 8.0000
TKI258 RERF-LC-A1 CCLE 0.0025 8.0000
TKI258 RERF-LC-MS CCLE 0.0025 8.0000
TKI258 RKN CCLE 0.0025 8.0000
TKI258 RKO CCLE 0.0025 8.0000
TKI258 RL95-2 CCLE 0.0025 8.0000
TKI258 RPMI-7951 CCLE 0.0025 8.0000
TKI258 RPMI-8402 CCLE 0.0025 8.0000
TKI258 RT-112 CCLE 0.0025 8.0000
TKI258 RT-4 CCLE 0.0025 8.0000
TKI258 RVH-421 CCLE 0.0025 8.0000
TKI258 SAOS-2 CCLE 0.0025 8.0000
TKI258 SBC-5 CCLE 0.0025 8.0000
TKI258 SCABER CCLE 0.0025 8.0000
TKI258 SCC-9 CCLE 0.0025 8.0000
TKI258 SF126 CCLE 0.0025 8.0000
TKI258 SF295 CCLE 0.0025 8.0000
TKI258 SF8657 CCLE 0.0025 8.0000
TKI258 SH-10-TC CCLE 0.0025 8.0000
TKI258 SHP-77 CCLE 0.0025 8.0000
TKI258 SIG-M5 CCLE 0.0025 8.0000
TKI258 SIMA CCLE 0.0025 8.0000
TKI258 RH30 CCLE 0.0025 8.0000
TKI258 SJSA-1 CCLE 0.0025 8.0000
TKI258 SK-BR-3 CCLE 0.0025 8.0000
TKI258 SK-CO-1 CCLE 0.0025 8.0000
TKI258 SK-ES-1 CCLE 0.0025 8.0000
TKI258 SK-HEP-1 CCLE 0.0025 8.0000
TKI258 SK-LMS-1 CCLE 0.0025 8.0000
TKI258 SK-LU-1 CCLE 0.0025 8.0000
TKI258 SK-MEL-2 CCLE 0.0025 8.0000
TKI258 SK-MEL-24 CCLE 0.0025 8.0000
TKI258 SK-MEL-30 CCLE 0.0025 8.0000
TKI258 SK-MEL-31 CCLE 0.0025 8.0000
TKI258 SK-MEL-5 CCLE 0.0025 8.0000
TKI258 SK-MES-1 CCLE 0.0025 8.0000
TKI258 SK-MM-2 CCLE 0.0025 8.0000
TKI258 SK-N-AS CCLE 0.0025 8.0000
TKI258 SK-N-BE(2) CCLE 0.0025 8.0000
TKI258 SK-N-DZ CCLE 0.0025 8.0000
TKI258 SK-N-FI CCLE 0.0025 8.0000
TKI258 SK-N-SH CCLE 0.0025 8.0000
TKI258 SK-OV-3 CCLE 0.0025 8.0000
TKI258 SNG-M CCLE 0.0025 8.0000
TKI258 SNU-1 CCLE 0.0025 8.0000
TKI258 SNU-16 CCLE 0.0025 8.0000
TKI258 SNU-182 CCLE 0.0025 8.0000
TKI258 SNU-387 CCLE 0.0025 8.0000
TKI258 SNU-398 CCLE 0.0025 8.0000
TKI258 SNU-423 CCLE 0.0025 8.0000
TKI258 SNU-449 CCLE 0.0025 8.0000
TKI258 SNU-475 CCLE 0.0025 8.0000
TKI258 SNU-C2A CCLE 0.0025 8.0000
TKI258 SNU-C2B CCLE 0.0025 8.0000
TKI258 SQ-1 CCLE 0.0025 8.0000
TKI258 SU.86.86 CCLE 0.0025 8.0000
TKI258 SU-DHL-10 CCLE 0.0025 8.0000
TKI258 SU-DHL-4 CCLE 0.0025 8.0000
TKI258 SU-DHL-6 CCLE 0.0025 8.0000
TKI258 SU-DHL-8 CCLE 0.0025 8.0000
TKI258 SUIT-2 CCLE 0.0025 8.0000
TKI258 SUP-M2 CCLE 0.0025 8.0000
TKI258 SUP-T1 CCLE 0.0025 8.0000
TKI258 SW1088 CCLE 0.0025 8.0000
TKI258 SW1271 CCLE 0.0025 8.0000
TKI258 SW1353 CCLE 0.0025 8.0000
TKI258 SW1417 CCLE 0.0025 8.0000
TKI258 SW1573 CCLE 0.0025 8.0000
TKI258 SW1990 CCLE 0.0025 8.0000
TKI258 SW403 CCLE 0.0025 8.0000
TKI258 SW48 CCLE 0.0025 8.0000
TKI258 SW480 CCLE 0.0025 8.0000
TKI258 SW579 CCLE 0.0025 8.0000
TKI258 SW620 CCLE 0.0025 8.0000
TKI258 SW780 CCLE 0.0025 8.0000
TKI258 SW900 CCLE 0.0025 8.0000
TKI258 T24 CCLE 0.0025 8.0000
TKI258 T3M-10 CCLE 0.0025 8.0000
TKI258 T-47D CCLE 0.0025 8.0000
TKI258 T84 CCLE 0.0025 8.0000
TKI258 T98G CCLE 0.0025 8.0000
TKI258 TC-71 CCLE 0.0025 8.0000
TKI258 TCCSUP CCLE 0.0025 8.0000
TKI258 TE-1 CCLE 0.0025 8.0000
TKI258 TE-11 CCLE 0.0025 8.0000
TKI258 TE-15 CCLE 0.0025 8.0000
TKI258 TE-5 CCLE 0.0025 8.0000
TKI258 TE617.T CCLE 0.0025 8.0000
TKI258 TE-9 CCLE 0.0025 8.0000
TKI258 TEN CCLE 0.0025 8.0000
TKI258 TOLEDO CCLE 0.0025 8.0000
TKI258 TOV-112D CCLE 0.0025 8.0000
TKI258 TOV-21G CCLE 0.0025 8.0000
TKI258 TT2609-C02 CCLE 0.0025 8.0000
TKI258 TYK-NU CCLE 0.0025 8.0000
TKI258 U-118MG CCLE 0.0025 8.0000
TKI258 U2OS CCLE 0.0025 8.0000
TKI258 U-87MGATCC CCLE 0.0025 8.0000
TKI258 U-937 CCLE 0.0025 8.0000
TKI258 UACC-257 CCLE 0.0025 8.0000
TKI258 UACC-62 CCLE 0.0025 8.0000
TKI258 UACC-812 CCLE 0.0025 8.0000
TKI258 UM-UC-3 CCLE 0.0025 8.0000
TKI258 VMRC-LCD CCLE 0.0025 8.0000
TKI258 VMRC-RCW CCLE 0.0025 8.0000
TKI258 VMRC-RCZ CCLE 0.0025 8.0000
TKI258 WM115 CCLE 0.0025 8.0000
TKI258 WM1799 CCLE 0.0025 8.0000
TKI258 WM266-4 CCLE 0.0025 8.0000
TKI258 WM793 CCLE 0.0025 8.0000
TKI258 WM88 CCLE 0.0025 8.0000
TKI258 WM983B CCLE 0.0025 8.0000
TKI258 YKG-1 CCLE 0.0025 8.0000
TKI258 ZR-75-1 CCLE 0.0025 8.0000
TKI258 ZR-75-30 CCLE 0.0025 8.0000
TKI258 SCC-25 CCLE 0.0025 8.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.