Drug : Leucascandrolide A

CTRP1 Name : leucascandrolide A

Dataset : All
Synonyms :
Targets :
Pathways : inhibitor of cellular respiration

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
leucascandrolide A U2OS CTRP1 0.0163 2.0833
leucascandrolide A MCF-7 CTRP1 0.0163 2.0833
leucascandrolide A GAMG CTRP1 0.2603 33.3330
leucascandrolide A LN-229 CTRP1 0.0163 2.0833
leucascandrolide A SF295 CTRP1 0.2603 33.3330
leucascandrolide A HEC-108 CTRP1 0.2603 33.3330
leucascandrolide A HEC-151 CTRP1 0.0163 2.0833
leucascandrolide A HEC-251 CTRP1 0.2603 33.3330
leucascandrolide A HEC-265 CTRP1 0.2603 33.3330
leucascandrolide A HEC-59 CTRP1 0.2603 33.3330
leucascandrolide A HEC-6 CTRP1 0.2603 33.3330
leucascandrolide A ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
leucascandrolide A JHUEM-2 CTRP1 0.0163 2.0833
leucascandrolide A KLE CTRP1 0.2603 33.3330
leucascandrolide A MFE-319 CTRP1 0.2603 33.3330
leucascandrolide A SNG-M CTRP1 0.2603 33.3330
leucascandrolide A AMO1 CTRP1 0.0163 2.0833
leucascandrolide A BL-70 CTRP1 0.2603 33.3330
leucascandrolide A EJM CTRP1 0.0163 2.0833
leucascandrolide A GDM-1 CTRP1 0.0163 2.0833
leucascandrolide A HT CTRP1 0.2603 33.3330
leucascandrolide A KMS-11 CTRP1 0.0163 2.0833
leucascandrolide A KU812 CTRP1 0.2603 33.3330
leucascandrolide A LP-1 CTRP1 0.0163 2.0833
leucascandrolide A MC116 CTRP1 0.2603 33.3330
leucascandrolide A MOLM-16 CTRP1 0.0163 2.0833
leucascandrolide A NOMO-1 CTRP1 0.0163 2.0833
leucascandrolide A NU-DUL-1 CTRP1 0.0163 2.0833
leucascandrolide A OCI-AML-3 CTRP1 0.0163 2.0833
leucascandrolide A OCI-LY10 CTRP1 0.0163 2.0833
leucascandrolide A P3HR-1 CTRP1 0.2603 33.3330
leucascandrolide A PL21 CTRP1 0.0163 2.0833
leucascandrolide A RPMI-8226 CTRP1 0.0163 2.0833
leucascandrolide A SKM-1 CTRP1 0.0163 2.0833
leucascandrolide A SU-DHL-4 CTRP1 0.0163 2.0833
leucascandrolide A SU-DHL-5 CTRP1 0.0163 2.0833
leucascandrolide A THP-1 CTRP1 0.0163 2.0833
leucascandrolide A U-937 CTRP1 0.0163 2.0833
leucascandrolide A WSU-DLCL2 CTRP1 0.0163 2.0833
leucascandrolide A RCC10RGB CTRP1 0.0163 2.0833
leucascandrolide A VMRC-RCW CTRP1 0.2603 33.3330
leucascandrolide A C2BBE1 CTRP1 0.2603 33.3330
leucascandrolide A CL-34 CTRP1 0.0163 2.0833
leucascandrolide A CL-40 CTRP1 0.0163 2.0833
leucascandrolide A COLO205 CTRP1 0.2603 33.3330
leucascandrolide A COLO320 CTRP1 0.0163 2.0833
leucascandrolide A COLO678 CTRP1 0.0163 2.0833
leucascandrolide A CW-2 CTRP1 0.0163 2.0833
leucascandrolide A DLD-1 CTRP1 0.2603 33.3330
leucascandrolide A GP2D CTRP1 0.2603 33.3330
leucascandrolide A HCT116 CTRP1 0.0163 2.0833
leucascandrolide A HCT8 CTRP1 0.0163 2.0833
leucascandrolide A HT115 CTRP1 0.0163 2.0833
leucascandrolide A HT-29 CTRP1 0.0163 2.0833
leucascandrolide A HT-55 CTRP1 0.0163 2.0833
leucascandrolide A KM12 CTRP1 0.0163 2.0833
leucascandrolide A LOVO CTRP1 0.0163 2.0833
leucascandrolide A LS123 CTRP1 0.0163 2.0833
leucascandrolide A LS180 CTRP1 0.0163 2.0833
leucascandrolide A LS411N CTRP1 0.2603 33.3330
leucascandrolide A LS513 CTRP1 0.2603 33.3330
leucascandrolide A MDST8 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H508 CTRP1 0.0163 2.0833
leucascandrolide A RCM-1[HUMANESC] CTRP1 0.0163 2.0833
leucascandrolide A RKO CTRP1 0.0163 2.0833
leucascandrolide A SK-CO-1 CTRP1 0.2603 33.3330
leucascandrolide A SNU-1040 CTRP1 0.0163 2.0833
leucascandrolide A SNU-175 CTRP1 0.0163 2.0833
leucascandrolide A SNU-61 CTRP1 0.0163 2.0833
leucascandrolide A SNU-81 CTRP1 0.0163 2.0833
leucascandrolide A SNU-C2A CTRP1 0.2603 33.3330
leucascandrolide A SNU-C4 CTRP1 0.0163 2.0833
leucascandrolide A SNU-C5 CTRP1 0.0163 2.0833
leucascandrolide A SW403 CTRP1 0.2603 33.3330
leucascandrolide A SW48 CTRP1 0.2603 33.3330
leucascandrolide A SW480 CTRP1 0.0163 2.0833
leucascandrolide A SW620 CTRP1 0.0163 2.0833
leucascandrolide A SW948 CTRP1 0.0163 2.0833
leucascandrolide A HEP-G2 CTRP1 0.0163 2.0833
leucascandrolide A JHH-6 CTRP1 0.2603 33.3330
leucascandrolide A SNU-398 CTRP1 0.0163 2.0833
leucascandrolide A SNU-449 CTRP1 0.2603 33.3330
leucascandrolide A A-549 CTRP1 0.2603 33.3330
leucascandrolide A BEN CTRP1 0.2603 33.3330
leucascandrolide A CAL-12T CTRP1 0.0163 2.0833
leucascandrolide A CALU-3 CTRP1 0.2603 33.3330
leucascandrolide A CALU-6 CTRP1 0.2603 33.3330
leucascandrolide A CHAGO-K-1 CTRP1 0.2603 33.3330
leucascandrolide A COLO668 CTRP1 0.2603 33.3330
leucascandrolide A COLO699 CTRP1 0.0163 2.0833
leucascandrolide A COR-L23 CTRP1 0.0163 2.0833
leucascandrolide A COR-L279 CTRP1 0.2603 33.3330
leucascandrolide A COR-L51 CTRP1 0.0163 2.0833
leucascandrolide A COR-L88 CTRP1 0.2603 33.3330
leucascandrolide A DMS273 CTRP1 0.2603 33.3330
leucascandrolide A DV-90 CTRP1 0.2603 33.3330
leucascandrolide A EBC-1 CTRP1 0.2603 33.3330
leucascandrolide A EPLC-272H CTRP1 0.2603 33.3330
leucascandrolide A HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
leucascandrolide A HCC1195 CTRP1 0.0163 2.0833
leucascandrolide A HCC1359 CTRP1 0.0163 2.0833
leucascandrolide A HCC15 CTRP1 0.0163 2.0833
leucascandrolide A HCC1833 CTRP1 0.0163 2.0833
leucascandrolide A HCC2108 CTRP1 0.0163 2.0833
leucascandrolide A HCC2935 CTRP1 0.0163 2.0833
leucascandrolide A HCC33 CTRP1 0.2603 33.3330
leucascandrolide A HCC4006 CTRP1 0.0163 2.0833
leucascandrolide A HCC44 CTRP1 0.2603 33.3330
leucascandrolide A HCC78 CTRP1 0.2603 33.3330
leucascandrolide A HCC827 CTRP1 0.0163 2.0833
leucascandrolide A KNS-62 CTRP1 0.2603 33.3330
leucascandrolide A LC-1-SQ-SF CTRP1 0.2603 33.3330
leucascandrolide A LCLC-103H CTRP1 0.2603 33.3330
leucascandrolide A LCLC-97TM1 CTRP1 0.2603 33.3330
leucascandrolide A LU-65 CTRP1 0.2603 33.3330
leucascandrolide A LU-99 CTRP1 0.2603 33.3330
leucascandrolide A LXF289 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1048 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1105 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H1299 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1355 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1373 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1435 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1437 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1568 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1573 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1666 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1694 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H1755 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H1781 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H1792 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1793 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1836 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H1876 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H1915 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1930 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1944 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H1963 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H1975 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H2009 CTRP1 0.0163 33.3330
leucascandrolide A NCI-H2023 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2029 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H2030 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2073 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2081 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2110 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2122 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2126 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H2141 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2172 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2286 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H23 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H2342 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H2405 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H3255 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H358 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H441 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H460 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H522 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H596 CTRP1 0.0163 2.0833
leucascandrolide A NCI-H650 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H661 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H727 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H810 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H82 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H841 CTRP1 0.0163 2.0833
leucascandrolide A RERF-LC-KJ CTRP1 0.2603 33.3330
leucascandrolide A SCLC-21H CTRP1 0.0163 2.0833
leucascandrolide A SHP-77 CTRP1 0.2603 33.3330
leucascandrolide A SK-LU-1 CTRP1 0.0163 2.0833
leucascandrolide A SQ-1 CTRP1 0.0163 2.0833
leucascandrolide A T3M-10 CTRP1 0.0163 2.0833
leucascandrolide A VMRC-LCD CTRP1 0.2603 33.3330
leucascandrolide A KYSE-140 CTRP1 0.2603 33.3330
leucascandrolide A KYSE-410 CTRP1 0.2603 33.3330
leucascandrolide A KYSE-450 CTRP1 0.2603 33.3330
leucascandrolide A A2780 CTRP1 0.0163 2.0833
leucascandrolide A CAOV-3 CTRP1 0.0163 2.0833
leucascandrolide A COV318 CTRP1 0.2603 33.3330
leucascandrolide A COV362 CTRP1 0.0163 2.0833
leucascandrolide A COV434 CTRP1 0.0163 2.0833
leucascandrolide A COV644 CTRP1 0.0163 2.0833
leucascandrolide A EFO-21 CTRP1 0.2603 33.3330
leucascandrolide A EFO-27 CTRP1 0.0163 2.0833
leucascandrolide A HEYA8 CTRP1 0.2603 33.3330
leucascandrolide A IGROV-1 CTRP1 0.0163 2.0833
leucascandrolide A JHOC-5 CTRP1 0.0163 2.0833
leucascandrolide A JHOM-1 CTRP1 0.0163 2.0833
leucascandrolide A JHOS-4 CTRP1 0.2603 33.3330
leucascandrolide A OAW42 CTRP1 0.0163 2.0833
leucascandrolide A OV7 CTRP1 0.0163 2.0833
leucascandrolide A OV-90 CTRP1 0.0163 2.0833
leucascandrolide A OVCAR-4 CTRP1 0.0163 2.0833
leucascandrolide A OVCAR-8 CTRP1 0.0163 2.0833
leucascandrolide A OVK18 CTRP1 0.0163 2.0833
leucascandrolide A OVKATE CTRP1 0.0163 2.0833
leucascandrolide A OVMANA CTRP1 0.2603 33.3330
leucascandrolide A RKN CTRP1 0.0163 2.0833
leucascandrolide A RMG-I CTRP1 0.0163 2.0833
leucascandrolide A RMUG-S CTRP1 0.0163 2.0833
leucascandrolide A SK-OV-3 CTRP1 0.2603 33.3330
leucascandrolide A SNU-840 CTRP1 0.0163 2.0833
leucascandrolide A TYK-NU CTRP1 0.0163 2.0833
leucascandrolide A CAPAN-2 CTRP1 0.2603 33.3330
leucascandrolide A CFPAC-1 CTRP1 0.2603 33.3330
leucascandrolide A HPAC CTRP1 0.2603 33.3330
leucascandrolide A HUP-T4 CTRP1 0.2603 33.3330
leucascandrolide A KP-3 CTRP1 0.2603 33.3330
leucascandrolide A PANC03.27 CTRP1 0.2603 33.3330
leucascandrolide A PANC10.05 CTRP1 0.2603 33.3330
leucascandrolide A PATU8902 CTRP1 0.2603 33.3330
leucascandrolide A QGP-1 CTRP1 0.2603 33.3330
leucascandrolide A SUIT-2 CTRP1 0.2603 33.3330
leucascandrolide A MSTO-211H CTRP1 0.2603 33.3330
leucascandrolide A NCI-H2052 CTRP1 0.2603 33.3330
leucascandrolide A NCI-H28 CTRP1 0.2603 33.3330
leucascandrolide A MIAPACA-3 CTRP1 0.2603 33.3330
leucascandrolide A A-375 CTRP1 0.0163 2.0833
leucascandrolide A COLO741 CTRP1 0.2603 33.3330
leucascandrolide A G-361 CTRP1 0.2603 33.3330
leucascandrolide A HS852.T CTRP1 0.2603 33.3330
leucascandrolide A HS936.T CTRP1 0.2603 33.3330
leucascandrolide A HS944.T CTRP1 0.2603 33.3330
leucascandrolide A SK-MEL-1 CTRP1 0.0163 2.0833
leucascandrolide A SK-MEL-28 CTRP1 0.0163 2.0833
leucascandrolide A SK-MEL-5 CTRP1 0.0163 2.0833
leucascandrolide A G-401 CTRP1 0.2603 33.3330
leucascandrolide A HT-1080 CTRP1 0.0163 2.0833
leucascandrolide A AGS CTRP1 0.0163 2.0833
leucascandrolide A FU97 CTRP1 0.2603 33.3330
leucascandrolide A KE-97 CTRP1 0.2603 33.3330
leucascandrolide A MKN7 CTRP1 0.2603 33.3330
leucascandrolide A MKN74 CTRP1 0.2603 33.3330
leucascandrolide A NUGC-4 CTRP1 0.2603 33.3330
leucascandrolide A SH-10-TC CTRP1 0.2603 33.3330
leucascandrolide A HSC-2 CTRP1 0.2603 33.3330
leucascandrolide A SCC-9 CTRP1 0.0163 2.0833
leucascandrolide A 5637 CTRP1 0.2603 33.3330
leucascandrolide A HT-1376 CTRP1 0.2603 33.3330
leucascandrolide A KMBC-2 CTRP1 0.2603 33.3330
leucascandrolide A RT-4 CTRP1 0.2603 33.3330
leucascandrolide A UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.