Drug : Cytosporone B

CTRP1 Name : cytosporone B

Dataset : All
Synonyms :
Targets : NR4A1
Pathways : agonist of Nur77

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

:


Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
cytosporone B U2OS CTRP1 0.2604 33.3330
cytosporone B MCF-7 CTRP1 0.2604 33.3330
cytosporone B GAMG CTRP1 0.2603 33.3330
cytosporone B LN-229 CTRP1 0.2604 33.3330
cytosporone B SF295 CTRP1 0.2603 33.3330
cytosporone B HEC-108 CTRP1 0.2603 33.3330
cytosporone B HEC-151 CTRP1 0.2604 33.3330
cytosporone B HEC-251 CTRP1 0.2603 33.3330
cytosporone B HEC-265 CTRP1 0.2603 33.3330
cytosporone B HEC-59 CTRP1 0.2603 33.3330
cytosporone B HEC-6 CTRP1 0.2603 33.3330
cytosporone B ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
cytosporone B JHUEM-2 CTRP1 0.2604 33.3330
cytosporone B KLE CTRP1 0.2603 33.3330
cytosporone B MFE-319 CTRP1 0.2603 33.3330
cytosporone B SNG-M CTRP1 0.2603 33.3330
cytosporone B AMO1 CTRP1 0.2604 33.3330
cytosporone B BL-70 CTRP1 0.2603 33.3330
cytosporone B EJM CTRP1 0.2604 33.3330
cytosporone B GDM-1 CTRP1 0.2604 33.3330
cytosporone B HT CTRP1 0.2603 33.3330
cytosporone B KMS-11 CTRP1 0.2604 33.3330
cytosporone B KU812 CTRP1 0.2603 33.3330
cytosporone B LP-1 CTRP1 0.2604 33.3330
cytosporone B MC116 CTRP1 0.2603 33.3330
cytosporone B MOLM-16 CTRP1 0.2604 33.3330
cytosporone B NOMO-1 CTRP1 0.2604 33.3330
cytosporone B NU-DUL-1 CTRP1 0.2604 33.3330
cytosporone B OCI-AML-3 CTRP1 0.2604 33.3330
cytosporone B OCI-LY10 CTRP1 0.2604 33.3330
cytosporone B P3HR-1 CTRP1 0.2603 33.3330
cytosporone B PL21 CTRP1 0.2604 33.3330
cytosporone B RPMI-8226 CTRP1 0.2604 33.3330
cytosporone B SKM-1 CTRP1 0.2604 33.3330
cytosporone B SU-DHL-4 CTRP1 0.2604 33.3330
cytosporone B SU-DHL-5 CTRP1 0.2604 33.3330
cytosporone B THP-1 CTRP1 0.2604 33.3330
cytosporone B U-937 CTRP1 0.2604 33.3330
cytosporone B WSU-DLCL2 CTRP1 0.2604 33.3330
cytosporone B RCC10RGB CTRP1 0.2604 33.3330
cytosporone B VMRC-RCW CTRP1 0.2603 33.3330
cytosporone B C2BBE1 CTRP1 0.2603 33.3330
cytosporone B CL-34 CTRP1 0.2604 33.3330
cytosporone B CL-40 CTRP1 0.2604 33.3330
cytosporone B COLO205 CTRP1 0.2603 33.3330
cytosporone B COLO320 CTRP1 0.2604 33.3330
cytosporone B COLO678 CTRP1 0.2604 33.3330
cytosporone B CW-2 CTRP1 0.2604 33.3330
cytosporone B DLD-1 CTRP1 0.2603 33.3330
cytosporone B GP2D CTRP1 0.2603 33.3330
cytosporone B HCT116 CTRP1 0.2604 33.3330
cytosporone B HCT8 CTRP1 0.2604 33.3330
cytosporone B HT115 CTRP1 0.2604 33.3330
cytosporone B HT-29 CTRP1 0.2604 33.3330
cytosporone B HT-55 CTRP1 0.2604 33.3330
cytosporone B KM12 CTRP1 0.2604 33.3330
cytosporone B LOVO CTRP1 0.2604 33.3330
cytosporone B LS123 CTRP1 0.2604 33.3330
cytosporone B LS180 CTRP1 0.2604 33.3330
cytosporone B LS411N CTRP1 0.2603 33.3330
cytosporone B LS513 CTRP1 0.2603 33.3330
cytosporone B MDST8 CTRP1 0.2604 33.3330
cytosporone B NCI-H508 CTRP1 0.2604 33.3330
cytosporone B RCM-1[HUMANESC] CTRP1 0.2604 33.3330
cytosporone B RKO CTRP1 0.2604 33.3330
cytosporone B SK-CO-1 CTRP1 0.2603 33.3330
cytosporone B SNU-1040 CTRP1 0.2604 33.3330
cytosporone B SNU-175 CTRP1 0.2604 33.3330
cytosporone B SNU-61 CTRP1 0.2604 33.3330
cytosporone B SNU-81 CTRP1 0.2604 33.3330
cytosporone B SNU-C2A CTRP1 0.2603 33.3330
cytosporone B SNU-C4 CTRP1 0.2604 33.3330
cytosporone B SNU-C5 CTRP1 0.2604 33.3330
cytosporone B SW403 CTRP1 0.2603 33.3330
cytosporone B SW48 CTRP1 0.2603 33.3330
cytosporone B SW480 CTRP1 0.2604 33.3330
cytosporone B SW620 CTRP1 0.2604 33.3330
cytosporone B SW948 CTRP1 0.2604 33.3330
cytosporone B HEP-G2 CTRP1 0.2604 33.3330
cytosporone B JHH-6 CTRP1 0.2603 33.3330
cytosporone B SNU-398 CTRP1 0.2604 33.3330
cytosporone B SNU-449 CTRP1 0.2603 33.3330
cytosporone B A-549 CTRP1 0.2603 33.3330
cytosporone B BEN CTRP1 0.2603 33.3330
cytosporone B CAL-12T CTRP1 0.2604 33.3330
cytosporone B CALU-3 CTRP1 0.2603 33.3330
cytosporone B CALU-6 CTRP1 0.2603 33.3330
cytosporone B CHAGO-K-1 CTRP1 0.2603 33.3330
cytosporone B COLO668 CTRP1 0.2603 33.3330
cytosporone B COLO699 CTRP1 0.2604 33.3330
cytosporone B COR-L23 CTRP1 0.2604 33.3330
cytosporone B COR-L279 CTRP1 0.2603 33.3330
cytosporone B COR-L51 CTRP1 0.2604 33.3330
cytosporone B COR-L88 CTRP1 0.2603 33.3330
cytosporone B DMS273 CTRP1 0.2603 33.3330
cytosporone B DV-90 CTRP1 0.2603 33.3330
cytosporone B EBC-1 CTRP1 0.2603 33.3330
cytosporone B EPLC-272H CTRP1 0.2603 33.3330
cytosporone B HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
cytosporone B HCC1195 CTRP1 0.2604 33.3330
cytosporone B HCC1359 CTRP1 0.2604 33.3330
cytosporone B HCC15 CTRP1 0.2604 33.3330
cytosporone B HCC1833 CTRP1 0.2604 33.3330
cytosporone B HCC2108 CTRP1 0.2604 33.3330
cytosporone B HCC2935 CTRP1 0.2604 33.3330
cytosporone B HCC33 CTRP1 0.2603 33.3330
cytosporone B HCC4006 CTRP1 0.2604 33.3330
cytosporone B HCC44 CTRP1 0.2603 33.3330
cytosporone B HCC78 CTRP1 0.2603 33.3330
cytosporone B HCC827 CTRP1 0.2604 33.3330
cytosporone B KNS-62 CTRP1 0.2603 33.3330
cytosporone B LC-1-SQ-SF CTRP1 0.2603 33.3330
cytosporone B LCLC-103H CTRP1 0.2603 33.3330
cytosporone B LCLC-97TM1 CTRP1 0.2603 33.3330
cytosporone B LU-65 CTRP1 0.2603 33.3330
cytosporone B LU-99 CTRP1 0.2603 33.3330
cytosporone B LXF289 CTRP1 0.2603 33.3330
cytosporone B NCI-H1048 CTRP1 0.2603 33.3330
cytosporone B NCI-H1105 CTRP1 0.2604 33.3330
cytosporone B NCI-H1299 CTRP1 0.2603 33.3330
cytosporone B NCI-H1355 CTRP1 0.2603 33.3330
cytosporone B NCI-H1373 CTRP1 0.2603 33.3330
cytosporone B NCI-H1435 CTRP1 0.2603 33.3330
cytosporone B NCI-H1437 CTRP1 0.2603 33.3330
cytosporone B NCI-H1568 CTRP1 0.2603 33.3330
cytosporone B NCI-H1573 CTRP1 0.2603 33.3330
cytosporone B NCI-H1666 CTRP1 0.2603 33.3330
cytosporone B NCI-H1694 CTRP1 0.2604 33.3330
cytosporone B NCI-H1755 CTRP1 0.2604 33.3330
cytosporone B NCI-H1781 CTRP1 0.2604 33.3330
cytosporone B NCI-H1792 CTRP1 0.2603 33.3330
cytosporone B NCI-H1793 CTRP1 0.2603 33.3330
cytosporone B NCI-H1836 CTRP1 0.2604 33.3330
cytosporone B NCI-H1876 CTRP1 0.2604 33.3330
cytosporone B NCI-H1915 CTRP1 0.2603 33.3330
cytosporone B NCI-H1930 CTRP1 0.2603 33.3330
cytosporone B NCI-H1944 CTRP1 0.2603 33.3330
cytosporone B NCI-H1963 CTRP1 0.2604 33.3330
cytosporone B NCI-H1975 CTRP1 0.2603 33.3330
cytosporone B NCI-H2009 CTRP1 0.2603 33.3330
cytosporone B NCI-H2023 CTRP1 0.2604 33.3330
cytosporone B NCI-H2029 CTRP1 0.2603 33.3330
cytosporone B NCI-H2030 CTRP1 0.2604 33.3330
cytosporone B NCI-H2073 CTRP1 0.2604 33.3330
cytosporone B NCI-H2081 CTRP1 0.2604 33.3330
cytosporone B NCI-H2110 CTRP1 0.2604 33.3330
cytosporone B NCI-H2122 CTRP1 0.2604 33.3330
cytosporone B NCI-H2126 CTRP1 0.2603 33.3330
cytosporone B NCI-H2141 CTRP1 0.2604 33.3330
cytosporone B NCI-H2172 CTRP1 0.2604 33.3330
cytosporone B NCI-H2286 CTRP1 0.2603 33.3330
cytosporone B NCI-H23 CTRP1 0.2603 33.3330
cytosporone B NCI-H2342 CTRP1 0.2604 33.3330
cytosporone B NCI-H2405 CTRP1 0.2603 33.3330
cytosporone B NCI-H3255 CTRP1 0.2604 33.3330
cytosporone B NCI-H358 CTRP1 0.2603 33.3330
cytosporone B NCI-H441 CTRP1 0.2604 33.3330
cytosporone B NCI-H460 CTRP1 0.2604 33.3330
cytosporone B NCI-H522 CTRP1 0.2603 33.3330
cytosporone B NCI-H596 CTRP1 0.2604 33.3330
cytosporone B NCI-H650 CTRP1 0.2603 33.3330
cytosporone B NCI-H661 CTRP1 0.2603 33.3330
cytosporone B NCI-H727 CTRP1 0.2603 33.3330
cytosporone B NCI-H810 CTRP1 0.2603 33.3330
cytosporone B NCI-H82 CTRP1 0.2603 33.3330
cytosporone B NCI-H841 CTRP1 0.2604 33.3330
cytosporone B RERF-LC-KJ CTRP1 0.2603 33.3330
cytosporone B SCLC-21H CTRP1 0.2604 33.3330
cytosporone B SHP-77 CTRP1 0.2603 33.3330
cytosporone B SK-LU-1 CTRP1 0.2604 33.3330
cytosporone B SQ-1 CTRP1 0.2604 33.3330
cytosporone B T3M-10 CTRP1 0.2604 33.3330
cytosporone B VMRC-LCD CTRP1 0.2603 33.3330
cytosporone B KYSE-140 CTRP1 0.2603 33.3330
cytosporone B KYSE-410 CTRP1 0.2603 33.3330
cytosporone B KYSE-450 CTRP1 0.2603 33.3330
cytosporone B A2780 CTRP1 0.2604 33.3330
cytosporone B CAOV-3 CTRP1 0.2604 33.3330
cytosporone B COV318 CTRP1 0.2603 33.3330
cytosporone B COV362 CTRP1 0.2604 33.3330
cytosporone B COV434 CTRP1 0.2604 33.3330
cytosporone B COV644 CTRP1 0.2604 33.3330
cytosporone B EFO-21 CTRP1 0.2603 33.3330
cytosporone B EFO-27 CTRP1 0.2604 33.3330
cytosporone B HEYA8 CTRP1 0.2603 33.3330
cytosporone B IGROV-1 CTRP1 0.2604 33.3330
cytosporone B JHOC-5 CTRP1 0.2604 33.3330
cytosporone B JHOM-1 CTRP1 0.2604 33.3330
cytosporone B JHOS-4 CTRP1 0.2603 33.3330
cytosporone B OAW42 CTRP1 0.2604 33.3330
cytosporone B OV7 CTRP1 0.2604 33.3330
cytosporone B OV-90 CTRP1 0.2604 33.3330
cytosporone B OVCAR-4 CTRP1 0.2604 33.3330
cytosporone B OVCAR-8 CTRP1 0.2604 33.3330
cytosporone B OVK18 CTRP1 0.2604 33.3330
cytosporone B OVKATE CTRP1 0.2604 33.3330
cytosporone B OVMANA CTRP1 0.2603 33.3330
cytosporone B RKN CTRP1 0.2604 33.3330
cytosporone B RMG-I CTRP1 0.2604 33.3330
cytosporone B RMUG-S CTRP1 0.2604 33.3330
cytosporone B SK-OV-3 CTRP1 0.2603 33.3330
cytosporone B SNU-840 CTRP1 0.2604 33.3330
cytosporone B TYK-NU CTRP1 0.2604 33.3330
cytosporone B CAPAN-2 CTRP1 0.2603 33.3330
cytosporone B CFPAC-1 CTRP1 0.2603 33.3330
cytosporone B HPAC CTRP1 0.2603 33.3330
cytosporone B HUP-T4 CTRP1 0.2603 33.3330
cytosporone B KP-3 CTRP1 0.2603 33.3330
cytosporone B PANC03.27 CTRP1 0.2603 33.3330
cytosporone B PANC10.05 CTRP1 0.2603 33.3330
cytosporone B PATU8902 CTRP1 0.2603 33.3330
cytosporone B QGP-1 CTRP1 0.2603 33.3330
cytosporone B SUIT-2 CTRP1 0.2603 33.3330
cytosporone B MSTO-211H CTRP1 0.2603 33.3330
cytosporone B NCI-H2052 CTRP1 0.2603 33.3330
cytosporone B NCI-H28 CTRP1 0.2603 33.3330
cytosporone B MIAPACA-3 CTRP1 0.2603 33.3330
cytosporone B A-375 CTRP1 0.2604 33.3330
cytosporone B COLO741 CTRP1 0.2603 33.3330
cytosporone B G-361 CTRP1 0.2603 33.3330
cytosporone B HS852.T CTRP1 0.2603 33.3330
cytosporone B HS936.T CTRP1 0.2603 33.3330
cytosporone B HS944.T CTRP1 0.2603 33.3330
cytosporone B SK-MEL-1 CTRP1 0.2604 33.3330
cytosporone B SK-MEL-28 CTRP1 0.2604 33.3330
cytosporone B SK-MEL-5 CTRP1 0.2604 33.3330
cytosporone B G-401 CTRP1 0.2603 33.3330
cytosporone B HT-1080 CTRP1 0.2604 33.3330
cytosporone B AGS CTRP1 0.2604 33.3330
cytosporone B FU97 CTRP1 0.2603 33.3330
cytosporone B KE-97 CTRP1 0.2603 33.3330
cytosporone B MKN7 CTRP1 0.2603 33.3330
cytosporone B MKN74 CTRP1 0.2603 33.3330
cytosporone B NUGC-4 CTRP1 0.2603 33.3330
cytosporone B SH-10-TC CTRP1 0.2603 33.3330
cytosporone B HSC-2 CTRP1 0.2603 33.3330
cytosporone B SCC-9 CTRP1 0.2604 33.3330
cytosporone B 5637 CTRP1 0.2603 33.3330
cytosporone B HT-1376 CTRP1 0.2603 33.3330
cytosporone B KMBC-2 CTRP1 0.2603 33.3330
cytosporone B RT-4 CTRP1 0.2603 33.3330
cytosporone B UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.