Drug : Ml101

CTRP1 Name : ML101

Dataset : All
Synonyms :
Targets : XIAP;BIRC2;BIRC3
Pathways : antagonist of IAP family of anti-apoptotic proteins

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
ML101 MCF-7 CTRP1 2.0833 266.6700
ML101 GAMG CTRP1 0.2890 37.0000
ML101 LN-229 CTRP1 2.0833 266.6700
ML101 SF295 CTRP1 0.2890 37.0000
ML101 HEC-108 CTRP1 0.2890 37.0000
ML101 HEC-151 CTRP1 2.0833 266.6700
ML101 HEC-251 CTRP1 0.2890 37.0000
ML101 HEC-265 CTRP1 0.2890 37.0000
ML101 HEC-59 CTRP1 0.2890 37.0000
ML101 HEC-6 CTRP1 0.2890 37.0000
ML101 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2890 37.0000
ML101 JHUEM-2 CTRP1 2.0833 266.6700
ML101 KLE CTRP1 0.2890 37.0000
ML101 MFE-319 CTRP1 0.2890 37.0000
ML101 SNG-M CTRP1 0.2890 37.0000
ML101 AMO1 CTRP1 2.0833 266.6700
ML101 BL-70 CTRP1 0.2890 37.0000
ML101 EJM CTRP1 2.0833 266.6700
ML101 GDM-1 CTRP1 2.0833 266.6700
ML101 HT CTRP1 0.2890 37.0000
ML101 KMS-11 CTRP1 2.0833 266.6700
ML101 KU812 CTRP1 0.2890 37.0000
ML101 LP-1 CTRP1 2.0833 266.6700
ML101 MC116 CTRP1 0.2890 37.0000
ML101 MOLM-16 CTRP1 2.0833 266.6700
ML101 NOMO-1 CTRP1 2.0833 266.6700
ML101 NU-DUL-1 CTRP1 2.0833 266.6700
ML101 OCI-AML-3 CTRP1 2.0833 266.6700
ML101 OCI-LY10 CTRP1 2.0833 266.6700
ML101 P3HR-1 CTRP1 0.2890 37.0000
ML101 PL21 CTRP1 2.0833 266.6700
ML101 RPMI-8226 CTRP1 2.0833 266.6700
ML101 SKM-1 CTRP1 2.0833 266.6700
ML101 SU-DHL-4 CTRP1 2.0833 266.6700
ML101 SU-DHL-5 CTRP1 2.0833 266.6700
ML101 THP-1 CTRP1 2.0833 266.6700
ML101 U-937 CTRP1 2.0833 266.6700
ML101 WSU-DLCL2 CTRP1 2.0833 266.6700
ML101 RCC10RGB CTRP1 2.0833 266.6700
ML101 VMRC-RCW CTRP1 0.2890 37.0000
ML101 CL-34 CTRP1 2.0833 266.6700
ML101 CL-40 CTRP1 2.0833 266.6700
ML101 COLO320 CTRP1 2.0833 266.6700
ML101 COLO678 CTRP1 2.0833 266.6700
ML101 CW-2 CTRP1 2.0833 266.6700
ML101 HCT116 CTRP1 2.0833 266.6700
ML101 HCT8 CTRP1 2.0833 266.6700
ML101 HT115 CTRP1 2.0833 266.6700
ML101 HT-29 CTRP1 2.0833 266.6700
ML101 HT-55 CTRP1 2.0833 266.6700
ML101 KM12 CTRP1 2.0833 266.6700
ML101 LOVO CTRP1 2.0833 266.6700
ML101 LS123 CTRP1 2.0833 266.6700
ML101 LS180 CTRP1 2.0833 266.6700
ML101 MDST8 CTRP1 2.0833 266.6700
ML101 NCI-H508 CTRP1 2.0833 266.6700
ML101 RCM-1[HUMANESC] CTRP1 2.0833 266.6700
ML101 RKO CTRP1 2.0833 266.6700
ML101 SNU-1040 CTRP1 2.0833 266.6700
ML101 SNU-175 CTRP1 2.0833 266.6700
ML101 SNU-61 CTRP1 2.0833 266.6700
ML101 SNU-81 CTRP1 2.0833 266.6700
ML101 SNU-C2A CTRP1 0.2890 37.0000
ML101 SNU-C4 CTRP1 2.0833 266.6700
ML101 SNU-C5 CTRP1 2.0833 266.6700
ML101 SW403 CTRP1 0.2890 37.0000
ML101 SW480 CTRP1 2.0833 266.6700
ML101 SW620 CTRP1 2.0833 266.6700
ML101 SW948 CTRP1 2.0833 266.6700
ML101 HEP-G2 CTRP1 2.0833 266.6700
ML101 JHH-6 CTRP1 0.2890 37.0000
ML101 SNU-398 CTRP1 2.0833 266.6700
ML101 SNU-449 CTRP1 0.2890 37.0000
ML101 A-549 CTRP1 0.2890 37.0000
ML101 BEN CTRP1 0.2890 37.0000
ML101 CAL-12T CTRP1 2.0833 266.6700
ML101 CALU-3 CTRP1 0.2890 37.0000
ML101 CALU-6 CTRP1 0.2890 37.0000
ML101 CHAGO-K-1 CTRP1 0.2890 37.0000
ML101 COLO668 CTRP1 0.2890 37.0000
ML101 COLO699 CTRP1 2.0833 266.6700
ML101 COR-L23 CTRP1 2.0833 266.6700
ML101 COR-L279 CTRP1 0.2890 37.0000
ML101 COR-L51 CTRP1 2.0833 266.6700
ML101 COR-L88 CTRP1 0.2890 37.0000
ML101 DMS273 CTRP1 0.2890 37.0000
ML101 DV-90 CTRP1 0.2890 37.0000
ML101 EPLC-272H CTRP1 0.2890 37.0000
ML101 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2890 37.0000
ML101 HCC1195 CTRP1 2.0833 266.6700
ML101 HCC1359 CTRP1 2.0833 266.6700
ML101 HCC15 CTRP1 2.0833 266.6700
ML101 HCC1833 CTRP1 2.0833 266.6700
ML101 HCC2108 CTRP1 2.0833 266.6700
ML101 HCC2935 CTRP1 2.0833 266.6700
ML101 HCC33 CTRP1 0.2890 37.0000
ML101 HCC4006 CTRP1 2.0833 266.6700
ML101 HCC44 CTRP1 0.2890 37.0000
ML101 HCC827 CTRP1 2.0833 266.6700
ML101 KNS-62 CTRP1 0.2890 37.0000
ML101 LC-1-SQ-SF CTRP1 0.2890 37.0000
ML101 LCLC-103H CTRP1 0.2890 37.0000
ML101 LCLC-97TM1 CTRP1 0.2890 37.0000
ML101 LU-65 CTRP1 0.2890 37.0000
ML101 LXF289 CTRP1 0.2890 37.0000
ML101 NCI-H1048 CTRP1 0.2890 37.0000
ML101 NCI-H1105 CTRP1 2.0833 266.6700
ML101 NCI-H1299 CTRP1 0.2890 37.0000
ML101 NCI-H1355 CTRP1 0.2890 37.0000
ML101 NCI-H1435 CTRP1 0.2890 37.0000
ML101 NCI-H1437 CTRP1 0.2890 37.0000
ML101 NCI-H1568 CTRP1 0.2890 37.0000
ML101 NCI-H1573 CTRP1 0.2890 37.0000
ML101 NCI-H1666 CTRP1 0.2890 37.0000
ML101 NCI-H1694 CTRP1 2.0833 266.6700
ML101 NCI-H1755 CTRP1 2.0833 266.6700
ML101 NCI-H1781 CTRP1 2.0833 266.6700
ML101 NCI-H1792 CTRP1 0.2890 37.0000
ML101 NCI-H1836 CTRP1 2.0833 266.6700
ML101 NCI-H1876 CTRP1 2.0833 266.6700
ML101 NCI-H1915 CTRP1 0.2890 37.0000
ML101 NCI-H1930 CTRP1 0.2890 37.0000
ML101 NCI-H1944 CTRP1 0.2890 37.0000
ML101 NCI-H1963 CTRP1 2.0833 266.6700
ML101 NCI-H1975 CTRP1 0.2890 37.0000
ML101 NCI-H2009 CTRP1 0.2890 37.0000
ML101 NCI-H2023 CTRP1 2.0833 266.6700
ML101 NCI-H2029 CTRP1 0.2890 37.0000
ML101 NCI-H2030 CTRP1 2.0833 266.6700
ML101 NCI-H2073 CTRP1 2.0833 266.6700
ML101 NCI-H2081 CTRP1 2.0833 266.6700
ML101 NCI-H2110 CTRP1 2.0833 266.6700
ML101 NCI-H2122 CTRP1 2.0833 266.6700
ML101 NCI-H2126 CTRP1 0.2890 37.0000
ML101 NCI-H2141 CTRP1 2.0833 266.6700
ML101 NCI-H2172 CTRP1 2.0833 266.6700
ML101 NCI-H2286 CTRP1 0.2890 37.0000
ML101 NCI-H23 CTRP1 0.2890 37.0000
ML101 NCI-H2342 CTRP1 2.0833 266.6700
ML101 NCI-H2405 CTRP1 0.2890 37.0000
ML101 NCI-H3255 CTRP1 2.0833 266.6700
ML101 NCI-H441 CTRP1 2.0833 266.6700
ML101 NCI-H460 CTRP1 2.0833 266.6700
ML101 NCI-H596 CTRP1 2.0833 266.6700
ML101 NCI-H650 CTRP1 0.2890 37.0000
ML101 NCI-H661 CTRP1 0.2890 37.0000
ML101 NCI-H727 CTRP1 0.2890 37.0000
ML101 NCI-H810 CTRP1 0.2890 37.0000
ML101 NCI-H82 CTRP1 0.2890 37.0000
ML101 NCI-H841 CTRP1 2.0833 266.6700
ML101 RERF-LC-KJ CTRP1 0.2890 37.0000
ML101 SCLC-21H CTRP1 2.0833 266.6700
ML101 SHP-77 CTRP1 0.2890 37.0000
ML101 SK-LU-1 CTRP1 2.0833 266.6700
ML101 SQ-1 CTRP1 2.0833 266.6700
ML101 T3M-10 CTRP1 2.0833 266.6700
ML101 VMRC-LCD CTRP1 0.2890 37.0000
ML101 KYSE-140 CTRP1 0.2890 37.0000
ML101 KYSE-410 CTRP1 0.2890 37.0000
ML101 KYSE-450 CTRP1 0.2890 37.0000
ML101 A2780 CTRP1 2.0833 266.6700
ML101 CAOV-3 CTRP1 2.0833 266.6700
ML101 COV318 CTRP1 0.2890 37.0000
ML101 COV362 CTRP1 2.0833 266.6700
ML101 COV434 CTRP1 2.0833 266.6700
ML101 COV644 CTRP1 2.0833 266.6700
ML101 EFO-21 CTRP1 0.2890 37.0000
ML101 EFO-27 CTRP1 2.0833 266.6700
ML101 HEYA8 CTRP1 0.2890 37.0000
ML101 IGROV-1 CTRP1 2.0833 266.6700
ML101 JHOC-5 CTRP1 2.0833 266.6700
ML101 JHOM-1 CTRP1 2.0833 266.6700
ML101 JHOS-4 CTRP1 0.2890 37.0000
ML101 OAW42 CTRP1 2.0833 266.6700
ML101 OV7 CTRP1 2.0833 266.6700
ML101 OV-90 CTRP1 2.0833 266.6700
ML101 OVCAR-4 CTRP1 2.0833 266.6700
ML101 OVCAR-8 CTRP1 2.0833 266.6700
ML101 OVK18 CTRP1 2.0833 266.6700
ML101 OVKATE CTRP1 2.0833 266.6700
ML101 OVMANA CTRP1 0.2890 37.0000
ML101 RKN CTRP1 2.0833 266.6700
ML101 RMG-I CTRP1 2.0833 266.6700
ML101 RMUG-S CTRP1 2.0833 266.6700
ML101 SK-OV-3 CTRP1 0.2890 37.0000
ML101 SNU-840 CTRP1 2.0833 266.6700
ML101 TYK-NU CTRP1 2.0833 266.6700
ML101 CAPAN-2 CTRP1 0.2890 37.0000
ML101 HUP-T4 CTRP1 0.2890 37.0000
ML101 KP-3 CTRP1 0.2890 37.0000
ML101 PANC03.27 CTRP1 0.2890 37.0000
ML101 PATU8902 CTRP1 0.2890 37.0000
ML101 QGP-1 CTRP1 0.2890 37.0000
ML101 SUIT-2 CTRP1 0.2890 37.0000
ML101 MSTO-211H CTRP1 0.2890 37.0000
ML101 NCI-H2052 CTRP1 0.2890 37.0000
ML101 NCI-H28 CTRP1 0.2890 37.0000
ML101 MIAPACA-3 CTRP1 0.2890 37.0000
ML101 A-375 CTRP1 2.0833 266.6700
ML101 G-361 CTRP1 0.2890 37.0000
ML101 HS852.T CTRP1 0.2890 37.0000
ML101 HS936.T CTRP1 0.2890 37.0000
ML101 HS944.T CTRP1 0.2890 37.0000
ML101 SK-MEL-1 CTRP1 2.0833 266.6700
ML101 SK-MEL-28 CTRP1 2.0833 266.6700
ML101 SK-MEL-5 CTRP1 2.0833 266.6700
ML101 G-401 CTRP1 0.2890 37.0000
ML101 HT-1080 CTRP1 2.0833 266.6700
ML101 AGS CTRP1 2.0833 266.6700
ML101 FU97 CTRP1 0.2890 37.0000
ML101 KE-97 CTRP1 0.2890 37.0000
ML101 MKN7 CTRP1 0.2890 37.0000
ML101 MKN74 CTRP1 0.2890 37.0000
ML101 NUGC-4 CTRP1 0.2890 37.0000
ML101 SH-10-TC CTRP1 0.2890 37.0000
ML101 HSC-2 CTRP1 0.2890 37.0000
ML101 SCC-9 CTRP1 2.0833 266.6700
ML101 5637 CTRP1 0.2890 37.0000
ML101 HT-1376 CTRP1 0.2890 37.0000
ML101 KMBC-2 CTRP1 0.2890 37.0000
ML101 RT-4 CTRP1 0.2890 37.0000
ML101 UM-UC-3 CTRP1 0.2890 37.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.