Drug : Glibenclamide

CTRP1 Name : glibenclamide

Dataset : All
Synonyms :
Targets : KCNJ8;KCNJ11;CFTR
Pathways : inhibitor of ATP-dependent K+ channel (Kir6, KATP) and CFTR Cl- channel

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
glibenclamide U2OS CTRP1 0.2604 33.3330
glibenclamide MCF-7 CTRP1 0.2604 33.3330
glibenclamide GAMG CTRP1 0.2603 33.3330
glibenclamide LN-229 CTRP1 0.2604 33.3330
glibenclamide SF295 CTRP1 0.2603 33.3330
glibenclamide HEC-108 CTRP1 0.2603 33.3330
glibenclamide HEC-151 CTRP1 0.2604 33.3330
glibenclamide HEC-251 CTRP1 0.2603 33.3330
glibenclamide HEC-265 CTRP1 0.2603 33.3330
glibenclamide HEC-59 CTRP1 0.2603 33.3330
glibenclamide HEC-6 CTRP1 0.2603 33.3330
glibenclamide ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
glibenclamide JHUEM-2 CTRP1 0.2604 33.3330
glibenclamide KLE CTRP1 0.2603 33.3330
glibenclamide MFE-319 CTRP1 0.2603 33.3330
glibenclamide SNG-M CTRP1 0.2603 33.3330
glibenclamide AMO1 CTRP1 0.2604 33.3330
glibenclamide BL-70 CTRP1 0.2603 33.3330
glibenclamide EJM CTRP1 0.2604 33.3330
glibenclamide GDM-1 CTRP1 0.2604 33.3330
glibenclamide HT CTRP1 0.2603 33.3330
glibenclamide KMS-11 CTRP1 0.2604 33.3330
glibenclamide KU812 CTRP1 0.2603 33.3330
glibenclamide LP-1 CTRP1 0.2604 33.3330
glibenclamide MC116 CTRP1 0.2603 33.3330
glibenclamide MOLM-16 CTRP1 0.2604 33.3330
glibenclamide NOMO-1 CTRP1 0.2604 33.3330
glibenclamide NU-DUL-1 CTRP1 0.2604 33.3330
glibenclamide OCI-AML-3 CTRP1 0.2604 33.3330
glibenclamide OCI-LY10 CTRP1 0.2604 33.3330
glibenclamide P3HR-1 CTRP1 0.2603 33.3330
glibenclamide PL21 CTRP1 0.2604 33.3330
glibenclamide RPMI-8226 CTRP1 0.2604 33.3330
glibenclamide SKM-1 CTRP1 0.2604 33.3330
glibenclamide SU-DHL-4 CTRP1 0.2604 33.3330
glibenclamide SU-DHL-5 CTRP1 0.2604 33.3330
glibenclamide THP-1 CTRP1 0.2604 33.3330
glibenclamide U-937 CTRP1 0.2604 33.3330
glibenclamide WSU-DLCL2 CTRP1 0.2604 33.3330
glibenclamide RCC10RGB CTRP1 0.2604 33.3330
glibenclamide VMRC-RCW CTRP1 0.2603 33.3330
glibenclamide C2BBE1 CTRP1 0.2603 33.3330
glibenclamide CL-34 CTRP1 0.2604 33.3330
glibenclamide CL-40 CTRP1 0.2604 33.3330
glibenclamide COLO205 CTRP1 0.2603 33.3330
glibenclamide COLO320 CTRP1 0.2604 33.3330
glibenclamide COLO678 CTRP1 0.2604 33.3330
glibenclamide CW-2 CTRP1 0.2604 33.3330
glibenclamide DLD-1 CTRP1 0.2603 33.3330
glibenclamide GP2D CTRP1 0.2603 33.3330
glibenclamide HCT116 CTRP1 0.2604 33.3330
glibenclamide HCT8 CTRP1 0.2604 33.3330
glibenclamide HT115 CTRP1 0.2604 33.3330
glibenclamide HT-29 CTRP1 0.2604 33.3330
glibenclamide HT-55 CTRP1 0.2604 33.3330
glibenclamide KM12 CTRP1 0.2604 33.3330
glibenclamide LOVO CTRP1 0.2604 33.3330
glibenclamide LS123 CTRP1 0.2604 33.3330
glibenclamide LS180 CTRP1 0.2604 33.3330
glibenclamide LS411N CTRP1 0.2603 33.3330
glibenclamide LS513 CTRP1 0.2603 33.3330
glibenclamide MDST8 CTRP1 0.2604 33.3330
glibenclamide NCI-H508 CTRP1 0.2604 33.3330
glibenclamide RCM-1[HUMANESC] CTRP1 0.2604 33.3330
glibenclamide RKO CTRP1 0.2604 33.3330
glibenclamide SK-CO-1 CTRP1 0.2603 33.3330
glibenclamide SNU-1040 CTRP1 0.2604 33.3330
glibenclamide SNU-175 CTRP1 0.2604 33.3330
glibenclamide SNU-61 CTRP1 0.2604 33.3330
glibenclamide SNU-81 CTRP1 0.2604 33.3330
glibenclamide SNU-C2A CTRP1 0.2603 33.3330
glibenclamide SNU-C4 CTRP1 0.2604 33.3330
glibenclamide SNU-C5 CTRP1 0.2604 33.3330
glibenclamide SW403 CTRP1 0.2603 33.3330
glibenclamide SW48 CTRP1 0.2603 33.3330
glibenclamide SW480 CTRP1 0.2604 33.3330
glibenclamide SW620 CTRP1 0.2604 33.3330
glibenclamide SW948 CTRP1 0.2604 33.3330
glibenclamide HEP-G2 CTRP1 0.2604 33.3330
glibenclamide JHH-6 CTRP1 0.2603 33.3330
glibenclamide SNU-398 CTRP1 0.2604 33.3330
glibenclamide SNU-449 CTRP1 0.2603 33.3330
glibenclamide A-549 CTRP1 0.2603 33.3330
glibenclamide BEN CTRP1 0.2603 33.3330
glibenclamide CAL-12T CTRP1 0.2604 33.3330
glibenclamide CALU-3 CTRP1 0.2603 33.3330
glibenclamide CALU-6 CTRP1 0.2603 33.3330
glibenclamide CHAGO-K-1 CTRP1 0.2603 33.3330
glibenclamide COLO668 CTRP1 0.2603 33.3330
glibenclamide COLO699 CTRP1 0.2604 33.3330
glibenclamide COR-L23 CTRP1 0.2604 33.3330
glibenclamide COR-L279 CTRP1 0.2603 33.3330
glibenclamide COR-L51 CTRP1 0.2604 33.3330
glibenclamide COR-L88 CTRP1 0.2603 33.3330
glibenclamide DMS273 CTRP1 0.2603 33.3330
glibenclamide DV-90 CTRP1 0.2603 33.3330
glibenclamide EBC-1 CTRP1 0.2603 33.3330
glibenclamide EPLC-272H CTRP1 0.2603 33.3330
glibenclamide HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
glibenclamide HCC1195 CTRP1 0.2604 33.3330
glibenclamide HCC1359 CTRP1 0.2604 33.3330
glibenclamide HCC15 CTRP1 0.2604 33.3330
glibenclamide HCC1833 CTRP1 0.2604 33.3330
glibenclamide HCC2108 CTRP1 0.2604 33.3330
glibenclamide HCC2935 CTRP1 0.2604 33.3330
glibenclamide HCC33 CTRP1 0.2603 33.3330
glibenclamide HCC4006 CTRP1 0.2604 33.3330
glibenclamide HCC44 CTRP1 0.2603 33.3330
glibenclamide HCC78 CTRP1 0.2603 33.3330
glibenclamide HCC827 CTRP1 0.2604 33.3330
glibenclamide KNS-62 CTRP1 0.2603 33.3330
glibenclamide LC-1-SQ-SF CTRP1 0.2603 33.3330
glibenclamide LCLC-103H CTRP1 0.2603 33.3330
glibenclamide LCLC-97TM1 CTRP1 0.2603 33.3330
glibenclamide LU-65 CTRP1 0.2603 33.3330
glibenclamide LU-99 CTRP1 0.2603 33.3330
glibenclamide LXF289 CTRP1 0.2603 33.3330
glibenclamide NCI-H1048 CTRP1 0.2603 33.3330
glibenclamide NCI-H1105 CTRP1 0.2604 33.3330
glibenclamide NCI-H1299 CTRP1 0.2603 33.3330
glibenclamide NCI-H1355 CTRP1 0.2603 33.3330
glibenclamide NCI-H1373 CTRP1 0.2603 33.3330
glibenclamide NCI-H1435 CTRP1 0.2603 33.3330
glibenclamide NCI-H1437 CTRP1 0.2603 33.3330
glibenclamide NCI-H1568 CTRP1 0.2603 33.3330
glibenclamide NCI-H1573 CTRP1 0.2603 33.3330
glibenclamide NCI-H1666 CTRP1 0.2603 33.3330
glibenclamide NCI-H1694 CTRP1 0.2604 33.3330
glibenclamide NCI-H1755 CTRP1 0.2604 33.3330
glibenclamide NCI-H1781 CTRP1 0.2604 33.3330
glibenclamide NCI-H1792 CTRP1 0.2603 33.3330
glibenclamide NCI-H1793 CTRP1 0.2603 33.3330
glibenclamide NCI-H1836 CTRP1 0.2604 33.3330
glibenclamide NCI-H1876 CTRP1 0.2604 33.3330
glibenclamide NCI-H1915 CTRP1 0.2603 33.3330
glibenclamide NCI-H1930 CTRP1 0.2603 33.3330
glibenclamide NCI-H1944 CTRP1 0.2603 33.3330
glibenclamide NCI-H1963 CTRP1 0.2604 33.3330
glibenclamide NCI-H1975 CTRP1 0.2603 33.3330
glibenclamide NCI-H2009 CTRP1 0.2603 33.3330
glibenclamide NCI-H2023 CTRP1 0.2604 33.3330
glibenclamide NCI-H2029 CTRP1 0.2603 33.3330
glibenclamide NCI-H2030 CTRP1 0.2604 33.3330
glibenclamide NCI-H2073 CTRP1 0.2604 33.3330
glibenclamide NCI-H2081 CTRP1 0.2604 33.3330
glibenclamide NCI-H2110 CTRP1 0.2604 33.3330
glibenclamide NCI-H2122 CTRP1 0.2604 33.3330
glibenclamide NCI-H2126 CTRP1 0.2603 33.3330
glibenclamide NCI-H2141 CTRP1 0.2604 33.3330
glibenclamide NCI-H2172 CTRP1 0.2604 33.3330
glibenclamide NCI-H2286 CTRP1 0.2603 33.3330
glibenclamide NCI-H23 CTRP1 0.2603 33.3330
glibenclamide NCI-H2342 CTRP1 0.2604 33.3330
glibenclamide NCI-H2405 CTRP1 0.2603 33.3330
glibenclamide NCI-H3255 CTRP1 0.2604 33.3330
glibenclamide NCI-H358 CTRP1 0.2603 33.3330
glibenclamide NCI-H441 CTRP1 0.2604 33.3330
glibenclamide NCI-H460 CTRP1 0.2604 33.3330
glibenclamide NCI-H522 CTRP1 0.2603 33.3330
glibenclamide NCI-H596 CTRP1 0.2604 33.3330
glibenclamide NCI-H650 CTRP1 0.2603 33.3330
glibenclamide NCI-H661 CTRP1 0.2603 33.3330
glibenclamide NCI-H727 CTRP1 0.2603 33.3330
glibenclamide NCI-H810 CTRP1 0.2603 33.3330
glibenclamide NCI-H82 CTRP1 0.2603 33.3330
glibenclamide NCI-H841 CTRP1 0.2604 33.3330
glibenclamide RERF-LC-KJ CTRP1 0.2603 33.3330
glibenclamide SCLC-21H CTRP1 0.2604 33.3330
glibenclamide SHP-77 CTRP1 0.2603 33.3330
glibenclamide SK-LU-1 CTRP1 0.2604 33.3330
glibenclamide SQ-1 CTRP1 0.2604 33.3330
glibenclamide T3M-10 CTRP1 0.2604 33.3330
glibenclamide VMRC-LCD CTRP1 0.2603 33.3330
glibenclamide KYSE-140 CTRP1 0.2603 33.3330
glibenclamide KYSE-410 CTRP1 0.2603 33.3330
glibenclamide KYSE-450 CTRP1 0.2603 33.3330
glibenclamide A2780 CTRP1 0.2604 33.3330
glibenclamide CAOV-3 CTRP1 0.2604 33.3330
glibenclamide COV318 CTRP1 0.2603 33.3330
glibenclamide COV362 CTRP1 0.2604 33.3330
glibenclamide COV434 CTRP1 0.2604 33.3330
glibenclamide COV644 CTRP1 0.2604 33.3330
glibenclamide EFO-21 CTRP1 0.2603 33.3330
glibenclamide EFO-27 CTRP1 0.2604 33.3330
glibenclamide HEYA8 CTRP1 0.2603 33.3330
glibenclamide IGROV-1 CTRP1 0.2604 33.3330
glibenclamide JHOC-5 CTRP1 0.2604 33.3330
glibenclamide JHOM-1 CTRP1 0.2604 33.3330
glibenclamide JHOS-4 CTRP1 0.2603 33.3330
glibenclamide OAW42 CTRP1 0.2604 33.3330
glibenclamide OV7 CTRP1 0.2604 33.3330
glibenclamide OV-90 CTRP1 0.2604 33.3330
glibenclamide OVCAR-4 CTRP1 0.2604 33.3330
glibenclamide OVCAR-8 CTRP1 0.2604 33.3330
glibenclamide OVK18 CTRP1 0.2604 33.3330
glibenclamide OVKATE CTRP1 0.2604 33.3330
glibenclamide OVMANA CTRP1 0.2603 33.3330
glibenclamide RKN CTRP1 0.2604 33.3330
glibenclamide RMG-I CTRP1 0.2604 33.3330
glibenclamide RMUG-S CTRP1 0.2604 33.3330
glibenclamide SK-OV-3 CTRP1 0.2603 33.3330
glibenclamide SNU-840 CTRP1 0.2604 33.3330
glibenclamide TYK-NU CTRP1 0.2604 33.3330
glibenclamide CAPAN-2 CTRP1 0.2603 33.3330
glibenclamide CFPAC-1 CTRP1 0.2603 33.3330
glibenclamide HPAC CTRP1 0.2603 33.3330
glibenclamide HUP-T4 CTRP1 0.2603 33.3330
glibenclamide KP-3 CTRP1 0.2603 33.3330
glibenclamide PANC03.27 CTRP1 0.2603 33.3330
glibenclamide PANC10.05 CTRP1 0.2603 33.3330
glibenclamide PATU8902 CTRP1 0.2603 33.3330
glibenclamide QGP-1 CTRP1 0.2603 33.3330
glibenclamide SUIT-2 CTRP1 0.2603 33.3330
glibenclamide MSTO-211H CTRP1 0.2603 33.3330
glibenclamide NCI-H2052 CTRP1 0.2603 33.3330
glibenclamide NCI-H28 CTRP1 0.2603 33.3330
glibenclamide MIAPACA-3 CTRP1 0.2603 33.3330
glibenclamide A-375 CTRP1 0.2604 33.3330
glibenclamide COLO741 CTRP1 0.2603 33.3330
glibenclamide G-361 CTRP1 0.2603 33.3330
glibenclamide HS852.T CTRP1 0.2603 33.3330
glibenclamide HS936.T CTRP1 0.2603 33.3330
glibenclamide HS944.T CTRP1 0.2603 33.3330
glibenclamide SK-MEL-1 CTRP1 0.2604 33.3330
glibenclamide SK-MEL-28 CTRP1 0.2604 33.3330
glibenclamide SK-MEL-5 CTRP1 0.2604 33.3330
glibenclamide G-401 CTRP1 0.2603 33.3330
glibenclamide HT-1080 CTRP1 0.2604 33.3330
glibenclamide AGS CTRP1 0.2604 33.3330
glibenclamide FU97 CTRP1 0.2603 33.3330
glibenclamide KE-97 CTRP1 0.2603 33.3330
glibenclamide MKN7 CTRP1 0.2603 33.3330
glibenclamide MKN74 CTRP1 0.2603 33.3330
glibenclamide NUGC-4 CTRP1 0.2603 33.3330
glibenclamide SH-10-TC CTRP1 0.2603 33.3330
glibenclamide HSC-2 CTRP1 0.2603 33.3330
glibenclamide SCC-9 CTRP1 0.2604 33.3330
glibenclamide 5637 CTRP1 0.2603 33.3330
glibenclamide HT-1376 CTRP1 0.2603 33.3330
glibenclamide KMBC-2 CTRP1 0.2603 33.3330
glibenclamide RT-4 CTRP1 0.2603 33.3330
glibenclamide UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.