Drug : Dalcetrapib

CTRP1 Name : dalcetrapib

Dataset : All
Synonyms :
Targets : CETP
Pathways : inhibitor of cholesteryl ester transfer protein

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
dalcetrapib U2OS CTRP1 2.0687 264.8000
dalcetrapib MCF-7 CTRP1 2.0687 264.8000
dalcetrapib GAMG CTRP1 0.2587 33.1000
dalcetrapib LN-229 CTRP1 2.0687 264.8000
dalcetrapib SF295 CTRP1 0.2587 33.1000
dalcetrapib HEC-108 CTRP1 0.2587 33.1000
dalcetrapib HEC-151 CTRP1 2.0687 264.8000
dalcetrapib HEC-251 CTRP1 0.2587 33.1000
dalcetrapib HEC-265 CTRP1 0.2587 33.1000
dalcetrapib HEC-59 CTRP1 0.2587 33.1000
dalcetrapib HEC-6 CTRP1 0.2587 33.1000
dalcetrapib ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2587 33.1000
dalcetrapib JHUEM-2 CTRP1 2.0687 264.8000
dalcetrapib KLE CTRP1 0.2587 33.1000
dalcetrapib MFE-319 CTRP1 0.2587 33.1000
dalcetrapib SNG-M CTRP1 0.2587 33.1000
dalcetrapib AMO1 CTRP1 2.0687 264.8000
dalcetrapib BL-70 CTRP1 0.2587 33.1000
dalcetrapib EJM CTRP1 2.0687 264.8000
dalcetrapib GDM-1 CTRP1 2.0687 264.8000
dalcetrapib HT CTRP1 0.2587 33.1000
dalcetrapib KMS-11 CTRP1 2.0687 264.8000
dalcetrapib KU812 CTRP1 0.2587 33.1000
dalcetrapib LP-1 CTRP1 2.0687 264.8000
dalcetrapib MC116 CTRP1 0.2587 33.1000
dalcetrapib MOLM-16 CTRP1 2.0687 264.8000
dalcetrapib NOMO-1 CTRP1 2.0687 264.8000
dalcetrapib NU-DUL-1 CTRP1 2.0687 264.8000
dalcetrapib OCI-AML-3 CTRP1 2.0687 264.8000
dalcetrapib OCI-LY10 CTRP1 2.0687 264.8000
dalcetrapib P3HR-1 CTRP1 0.2587 33.1000
dalcetrapib PL21 CTRP1 2.0687 264.8000
dalcetrapib RPMI-8226 CTRP1 2.0687 264.8000
dalcetrapib SKM-1 CTRP1 2.0687 264.8000
dalcetrapib SU-DHL-4 CTRP1 2.0687 264.8000
dalcetrapib SU-DHL-5 CTRP1 2.0687 264.8000
dalcetrapib THP-1 CTRP1 2.0687 264.8000
dalcetrapib U-937 CTRP1 2.0687 264.8000
dalcetrapib WSU-DLCL2 CTRP1 2.0687 264.8000
dalcetrapib RCC10RGB CTRP1 2.0687 264.8000
dalcetrapib VMRC-RCW CTRP1 0.2587 33.1000
dalcetrapib C2BBE1 CTRP1 0.2587 33.1000
dalcetrapib CL-34 CTRP1 2.0687 264.8000
dalcetrapib CL-40 CTRP1 2.0687 264.8000
dalcetrapib COLO205 CTRP1 0.2587 33.1000
dalcetrapib COLO320 CTRP1 2.0687 264.8000
dalcetrapib COLO678 CTRP1 2.0687 264.8000
dalcetrapib CW-2 CTRP1 2.0687 264.8000
dalcetrapib DLD-1 CTRP1 0.2587 33.1000
dalcetrapib GP2D CTRP1 0.2587 33.1000
dalcetrapib HCT116 CTRP1 2.0687 264.8000
dalcetrapib HCT8 CTRP1 2.0687 264.8000
dalcetrapib HT115 CTRP1 2.0687 264.8000
dalcetrapib HT-29 CTRP1 2.0687 264.8000
dalcetrapib HT-55 CTRP1 2.0687 264.8000
dalcetrapib KM12 CTRP1 2.0687 264.8000
dalcetrapib LOVO CTRP1 2.0687 264.8000
dalcetrapib LS123 CTRP1 2.0687 264.8000
dalcetrapib LS180 CTRP1 2.0687 264.8000
dalcetrapib LS411N CTRP1 0.2587 33.1000
dalcetrapib LS513 CTRP1 0.2587 33.1000
dalcetrapib MDST8 CTRP1 2.0687 264.8000
dalcetrapib NCI-H508 CTRP1 2.0687 264.8000
dalcetrapib RCM-1[HUMANESC] CTRP1 2.0687 264.8000
dalcetrapib RKO CTRP1 2.0687 264.8000
dalcetrapib SK-CO-1 CTRP1 0.2587 33.1000
dalcetrapib SNU-1040 CTRP1 2.0687 264.8000
dalcetrapib SNU-175 CTRP1 2.0687 264.8000
dalcetrapib SNU-61 CTRP1 2.0687 264.8000
dalcetrapib SNU-81 CTRP1 2.0687 264.8000
dalcetrapib SNU-C2A CTRP1 0.2587 33.1000
dalcetrapib SNU-C4 CTRP1 2.0687 264.8000
dalcetrapib SNU-C5 CTRP1 2.0687 264.8000
dalcetrapib SW403 CTRP1 0.2587 33.1000
dalcetrapib SW48 CTRP1 0.2587 33.1000
dalcetrapib SW480 CTRP1 2.0687 264.8000
dalcetrapib SW620 CTRP1 2.0687 264.8000
dalcetrapib SW948 CTRP1 2.0687 264.8000
dalcetrapib HEP-G2 CTRP1 2.0687 264.8000
dalcetrapib JHH-6 CTRP1 0.2587 33.1000
dalcetrapib SNU-398 CTRP1 2.0687 264.8000
dalcetrapib SNU-449 CTRP1 0.2587 33.1000
dalcetrapib A-549 CTRP1 0.2587 33.1000
dalcetrapib BEN CTRP1 0.2587 33.1000
dalcetrapib CAL-12T CTRP1 2.0687 264.8000
dalcetrapib CALU-3 CTRP1 0.2587 33.1000
dalcetrapib CALU-6 CTRP1 0.2587 33.1000
dalcetrapib CHAGO-K-1 CTRP1 0.2587 33.1000
dalcetrapib COLO668 CTRP1 0.2587 33.1000
dalcetrapib COLO699 CTRP1 2.0687 264.8000
dalcetrapib COR-L23 CTRP1 2.0687 264.8000
dalcetrapib COR-L279 CTRP1 0.2587 33.1000
dalcetrapib COR-L51 CTRP1 2.0687 264.8000
dalcetrapib COR-L88 CTRP1 0.2587 33.1000
dalcetrapib DMS273 CTRP1 0.2587 33.1000
dalcetrapib DV-90 CTRP1 0.2587 33.1000
dalcetrapib EBC-1 CTRP1 0.2587 33.1000
dalcetrapib EPLC-272H CTRP1 0.2587 33.1000
dalcetrapib HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2587 33.1000
dalcetrapib HCC1195 CTRP1 2.0687 264.8000
dalcetrapib HCC1359 CTRP1 2.0687 264.8000
dalcetrapib HCC15 CTRP1 2.0687 264.8000
dalcetrapib HCC1833 CTRP1 2.0687 264.8000
dalcetrapib HCC2108 CTRP1 2.0687 264.8000
dalcetrapib HCC2935 CTRP1 2.0687 264.8000
dalcetrapib HCC33 CTRP1 0.2587 33.1000
dalcetrapib HCC4006 CTRP1 2.0687 264.8000
dalcetrapib HCC44 CTRP1 0.2587 33.1000
dalcetrapib HCC78 CTRP1 0.2587 33.1000
dalcetrapib HCC827 CTRP1 2.0687 264.8000
dalcetrapib KNS-62 CTRP1 0.2587 33.1000
dalcetrapib LC-1-SQ-SF CTRP1 0.2587 33.1000
dalcetrapib LCLC-103H CTRP1 0.2587 33.1000
dalcetrapib LCLC-97TM1 CTRP1 0.2587 33.1000
dalcetrapib LU-65 CTRP1 0.2587 33.1000
dalcetrapib LU-99 CTRP1 0.2587 33.1000
dalcetrapib LXF289 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1048 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1105 CTRP1 2.0687 264.8000
dalcetrapib NCI-H1299 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1355 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1373 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1435 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1437 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1568 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1573 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1666 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1694 CTRP1 2.0687 264.8000
dalcetrapib NCI-H1755 CTRP1 2.0687 264.8000
dalcetrapib NCI-H1781 CTRP1 2.0687 264.8000
dalcetrapib NCI-H1792 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1793 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1836 CTRP1 2.0687 264.8000
dalcetrapib NCI-H1876 CTRP1 2.0687 264.8000
dalcetrapib NCI-H1915 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1930 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1944 CTRP1 0.2587 33.1000
dalcetrapib NCI-H1963 CTRP1 2.0687 264.8000
dalcetrapib NCI-H1975 CTRP1 0.2587 33.1000
dalcetrapib NCI-H2009 CTRP1 0.2587 33.1000
dalcetrapib NCI-H2023 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2029 CTRP1 0.2587 33.1000
dalcetrapib NCI-H2030 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2073 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2081 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2110 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2122 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2126 CTRP1 0.2587 33.1000
dalcetrapib NCI-H2141 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2172 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2286 CTRP1 0.2587 33.1000
dalcetrapib NCI-H23 CTRP1 0.2587 33.1000
dalcetrapib NCI-H2342 CTRP1 2.0687 264.8000
dalcetrapib NCI-H2405 CTRP1 0.2587 33.1000
dalcetrapib NCI-H3255 CTRP1 2.0687 264.8000
dalcetrapib NCI-H358 CTRP1 0.2587 33.1000
dalcetrapib NCI-H441 CTRP1 2.0687 264.8000
dalcetrapib NCI-H460 CTRP1 2.0687 264.8000
dalcetrapib NCI-H522 CTRP1 0.2587 33.1000
dalcetrapib NCI-H596 CTRP1 2.0687 264.8000
dalcetrapib NCI-H650 CTRP1 0.2587 33.1000
dalcetrapib NCI-H661 CTRP1 0.2587 33.1000
dalcetrapib NCI-H727 CTRP1 0.2587 33.1000
dalcetrapib NCI-H810 CTRP1 0.2587 33.1000
dalcetrapib NCI-H82 CTRP1 0.2587 33.1000
dalcetrapib NCI-H841 CTRP1 2.0687 264.8000
dalcetrapib RERF-LC-KJ CTRP1 0.2587 33.1000
dalcetrapib SCLC-21H CTRP1 2.0687 264.8000
dalcetrapib SHP-77 CTRP1 0.2587 33.1000
dalcetrapib SK-LU-1 CTRP1 2.0687 264.8000
dalcetrapib SQ-1 CTRP1 2.0687 264.8000
dalcetrapib T3M-10 CTRP1 2.0687 264.8000
dalcetrapib VMRC-LCD CTRP1 0.2587 33.1000
dalcetrapib KYSE-140 CTRP1 0.2587 33.1000
dalcetrapib KYSE-410 CTRP1 0.2587 33.1000
dalcetrapib KYSE-450 CTRP1 0.2587 33.1000
dalcetrapib A2780 CTRP1 2.0687 264.8000
dalcetrapib CAOV-3 CTRP1 2.0687 264.8000
dalcetrapib COV318 CTRP1 0.2587 33.1000
dalcetrapib COV362 CTRP1 2.0687 264.8000
dalcetrapib COV434 CTRP1 2.0687 264.8000
dalcetrapib COV644 CTRP1 2.0687 264.8000
dalcetrapib EFO-21 CTRP1 0.2587 33.1000
dalcetrapib EFO-27 CTRP1 2.0687 264.8000
dalcetrapib HEYA8 CTRP1 0.2587 33.1000
dalcetrapib IGROV-1 CTRP1 2.0687 264.8000
dalcetrapib JHOC-5 CTRP1 2.0687 264.8000
dalcetrapib JHOM-1 CTRP1 2.0687 264.8000
dalcetrapib JHOS-4 CTRP1 0.2587 33.1000
dalcetrapib OAW42 CTRP1 2.0687 264.8000
dalcetrapib OV7 CTRP1 2.0687 264.8000
dalcetrapib OV-90 CTRP1 2.0687 264.8000
dalcetrapib OVCAR-4 CTRP1 2.0687 264.8000
dalcetrapib OVCAR-8 CTRP1 2.0687 264.8000
dalcetrapib OVK18 CTRP1 2.0687 264.8000
dalcetrapib OVKATE CTRP1 2.0687 264.8000
dalcetrapib OVMANA CTRP1 0.2587 33.1000
dalcetrapib RKN CTRP1 2.0687 264.8000
dalcetrapib RMG-I CTRP1 2.0687 264.8000
dalcetrapib RMUG-S CTRP1 2.0687 264.8000
dalcetrapib SK-OV-3 CTRP1 0.2587 33.1000
dalcetrapib SNU-840 CTRP1 2.0687 264.8000
dalcetrapib TYK-NU CTRP1 2.0687 264.8000
dalcetrapib CAPAN-2 CTRP1 0.2587 33.1000
dalcetrapib CFPAC-1 CTRP1 0.2587 33.1000
dalcetrapib HPAC CTRP1 0.2587 33.1000
dalcetrapib HUP-T4 CTRP1 0.2587 33.1000
dalcetrapib KP-3 CTRP1 0.2587 33.1000
dalcetrapib PANC03.27 CTRP1 0.2587 33.1000
dalcetrapib PANC10.05 CTRP1 0.2587 33.1000
dalcetrapib PATU8902 CTRP1 0.2587 33.1000
dalcetrapib QGP-1 CTRP1 0.2587 33.1000
dalcetrapib SUIT-2 CTRP1 0.2587 33.1000
dalcetrapib MSTO-211H CTRP1 0.2587 33.1000
dalcetrapib NCI-H2052 CTRP1 0.2587 33.1000
dalcetrapib NCI-H28 CTRP1 0.2587 33.1000
dalcetrapib MIAPACA-3 CTRP1 0.2587 33.1000
dalcetrapib A-375 CTRP1 2.0687 264.8000
dalcetrapib COLO741 CTRP1 0.2587 33.1000
dalcetrapib G-361 CTRP1 0.2587 33.1000
dalcetrapib HS852.T CTRP1 0.2587 33.1000
dalcetrapib HS936.T CTRP1 0.2587 33.1000
dalcetrapib HS944.T CTRP1 0.2587 33.1000
dalcetrapib SK-MEL-1 CTRP1 2.0687 264.8000
dalcetrapib SK-MEL-28 CTRP1 2.0687 264.8000
dalcetrapib SK-MEL-5 CTRP1 2.0687 264.8000
dalcetrapib G-401 CTRP1 0.2587 33.1000
dalcetrapib HT-1080 CTRP1 2.0687 264.8000
dalcetrapib AGS CTRP1 2.0687 264.8000
dalcetrapib FU97 CTRP1 0.2587 33.1000
dalcetrapib KE-97 CTRP1 0.2587 33.1000
dalcetrapib MKN7 CTRP1 0.2587 33.1000
dalcetrapib MKN74 CTRP1 0.2587 33.1000
dalcetrapib NUGC-4 CTRP1 0.2587 33.1000
dalcetrapib SH-10-TC CTRP1 0.2587 33.1000
dalcetrapib HSC-2 CTRP1 0.2587 33.1000
dalcetrapib SCC-9 CTRP1 2.0687 264.8000
dalcetrapib 5637 CTRP1 0.2587 33.1000
dalcetrapib HT-1376 CTRP1 0.2587 33.1000
dalcetrapib KMBC-2 CTRP1 0.2587 33.1000
dalcetrapib RT-4 CTRP1 0.2587 33.1000
dalcetrapib UM-UC-3 CTRP1 0.2587 33.1000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.