Drug : 4-Methylfasudil

CTRP1 Name : 4-methylfasudil

Dataset : All
Synonyms :
Targets : STK33;ROCK1
Pathways : inhibitor of kinases including STK33 and ROCK

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
4-methylfasudil U2OS CTRP1 1.0417 133.3300
4-methylfasudil MCF-7 CTRP1 1.0417 133.3300
4-methylfasudil GAMG CTRP1 0.2603 33.3330
4-methylfasudil LN-229 CTRP1 1.0417 133.3300
4-methylfasudil SF295 CTRP1 0.2603 33.3330
4-methylfasudil HEC-108 CTRP1 0.2603 33.3330
4-methylfasudil HEC-151 CTRP1 1.0417 133.3300
4-methylfasudil HEC-251 CTRP1 0.2603 33.3330
4-methylfasudil HEC-265 CTRP1 0.2603 33.3330
4-methylfasudil HEC-59 CTRP1 0.2603 33.3330
4-methylfasudil HEC-6 CTRP1 0.2603 33.3330
4-methylfasudil ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
4-methylfasudil JHUEM-2 CTRP1 1.0417 133.3300
4-methylfasudil KLE CTRP1 0.2603 33.3330
4-methylfasudil MFE-319 CTRP1 0.2603 33.3330
4-methylfasudil SNG-M CTRP1 0.2603 33.3330
4-methylfasudil AMO1 CTRP1 1.0417 133.3300
4-methylfasudil BL-70 CTRP1 0.2603 33.3330
4-methylfasudil EJM CTRP1 1.0417 133.3300
4-methylfasudil GDM-1 CTRP1 1.0417 133.3300
4-methylfasudil HT CTRP1 0.2603 33.3330
4-methylfasudil KMS-11 CTRP1 1.0417 133.3300
4-methylfasudil KU812 CTRP1 0.2603 33.3330
4-methylfasudil LP-1 CTRP1 1.0417 133.3300
4-methylfasudil MC116 CTRP1 0.2603 33.3330
4-methylfasudil MOLM-16 CTRP1 1.0417 133.3300
4-methylfasudil NOMO-1 CTRP1 1.0417 133.3300
4-methylfasudil NU-DUL-1 CTRP1 1.0417 133.3300
4-methylfasudil OCI-AML-3 CTRP1 1.0417 133.3300
4-methylfasudil OCI-LY10 CTRP1 1.0417 133.3300
4-methylfasudil P3HR-1 CTRP1 0.2603 33.3330
4-methylfasudil PL21 CTRP1 1.0417 133.3300
4-methylfasudil RPMI-8226 CTRP1 1.0417 133.3300
4-methylfasudil SKM-1 CTRP1 1.0417 133.3300
4-methylfasudil SU-DHL-4 CTRP1 1.0417 133.3300
4-methylfasudil SU-DHL-5 CTRP1 1.0417 133.3300
4-methylfasudil THP-1 CTRP1 1.0417 133.3300
4-methylfasudil U-937 CTRP1 1.0417 133.3300
4-methylfasudil WSU-DLCL2 CTRP1 1.0417 133.3300
4-methylfasudil RCC10RGB CTRP1 1.0417 133.3300
4-methylfasudil VMRC-RCW CTRP1 0.2603 33.3330
4-methylfasudil C2BBE1 CTRP1 0.2603 33.3330
4-methylfasudil CL-34 CTRP1 1.0417 133.3300
4-methylfasudil CL-40 CTRP1 1.0417 133.3300
4-methylfasudil COLO205 CTRP1 0.2603 33.3330
4-methylfasudil COLO320 CTRP1 1.0417 133.3300
4-methylfasudil COLO678 CTRP1 1.0417 133.3300
4-methylfasudil CW-2 CTRP1 1.0417 133.3300
4-methylfasudil DLD-1 CTRP1 0.2603 33.3330
4-methylfasudil GP2D CTRP1 0.2603 33.3330
4-methylfasudil HCT116 CTRP1 1.0417 133.3300
4-methylfasudil HCT8 CTRP1 1.0417 133.3300
4-methylfasudil HT115 CTRP1 1.0417 133.3300
4-methylfasudil HT-29 CTRP1 1.0417 133.3300
4-methylfasudil HT-55 CTRP1 1.0417 133.3300
4-methylfasudil KM12 CTRP1 1.0417 133.3300
4-methylfasudil LOVO CTRP1 1.0417 133.3300
4-methylfasudil LS123 CTRP1 1.0417 133.3300
4-methylfasudil LS180 CTRP1 1.0417 133.3300
4-methylfasudil LS411N CTRP1 0.2603 33.3330
4-methylfasudil LS513 CTRP1 0.2603 33.3330
4-methylfasudil MDST8 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H508 CTRP1 1.0417 133.3300
4-methylfasudil RCM-1[HUMANESC] CTRP1 1.0417 133.3300
4-methylfasudil RKO CTRP1 1.0417 133.3300
4-methylfasudil SK-CO-1 CTRP1 0.2603 33.3330
4-methylfasudil SNU-1040 CTRP1 1.0417 133.3300
4-methylfasudil SNU-175 CTRP1 1.0417 133.3300
4-methylfasudil SNU-61 CTRP1 1.0417 133.3300
4-methylfasudil SNU-81 CTRP1 1.0417 133.3300
4-methylfasudil SNU-C2A CTRP1 0.2603 33.3330
4-methylfasudil SNU-C4 CTRP1 1.0417 133.3300
4-methylfasudil SNU-C5 CTRP1 1.0417 133.3300
4-methylfasudil SW403 CTRP1 0.2603 33.3330
4-methylfasudil SW48 CTRP1 0.2603 33.3330
4-methylfasudil SW480 CTRP1 1.0417 133.3300
4-methylfasudil SW620 CTRP1 1.0417 133.3300
4-methylfasudil SW948 CTRP1 1.0417 133.3300
4-methylfasudil HEP-G2 CTRP1 1.0417 133.3300
4-methylfasudil JHH-6 CTRP1 0.2603 33.3330
4-methylfasudil SNU-398 CTRP1 1.0417 133.3300
4-methylfasudil SNU-449 CTRP1 0.2603 33.3330
4-methylfasudil A-549 CTRP1 0.2603 33.3330
4-methylfasudil BEN CTRP1 0.2603 33.3330
4-methylfasudil CAL-12T CTRP1 1.0417 133.3300
4-methylfasudil CALU-3 CTRP1 0.2603 33.3330
4-methylfasudil CALU-6 CTRP1 0.2603 33.3330
4-methylfasudil CHAGO-K-1 CTRP1 0.2603 33.3330
4-methylfasudil COLO668 CTRP1 0.2603 33.3330
4-methylfasudil COLO699 CTRP1 1.0417 133.3300
4-methylfasudil COR-L23 CTRP1 1.0417 133.3300
4-methylfasudil COR-L279 CTRP1 0.2603 33.3330
4-methylfasudil COR-L51 CTRP1 1.0417 133.3300
4-methylfasudil COR-L88 CTRP1 0.2603 33.3330
4-methylfasudil DMS273 CTRP1 0.2603 33.3330
4-methylfasudil DV-90 CTRP1 0.2603 33.3330
4-methylfasudil EBC-1 CTRP1 0.2603 33.3330
4-methylfasudil EPLC-272H CTRP1 0.2603 33.3330
4-methylfasudil HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
4-methylfasudil HCC1195 CTRP1 1.0417 133.3300
4-methylfasudil HCC1359 CTRP1 1.0417 133.3300
4-methylfasudil HCC15 CTRP1 1.0417 133.3300
4-methylfasudil HCC1833 CTRP1 1.0417 133.3300
4-methylfasudil HCC2108 CTRP1 1.0417 133.3300
4-methylfasudil HCC2935 CTRP1 1.0417 133.3300
4-methylfasudil HCC33 CTRP1 0.2603 33.3330
4-methylfasudil HCC4006 CTRP1 1.0417 133.3300
4-methylfasudil HCC44 CTRP1 0.2603 33.3330
4-methylfasudil HCC78 CTRP1 0.2603 33.3330
4-methylfasudil HCC827 CTRP1 1.0417 133.3300
4-methylfasudil KNS-62 CTRP1 0.2603 33.3330
4-methylfasudil LC-1-SQ-SF CTRP1 0.2603 33.3330
4-methylfasudil LCLC-103H CTRP1 0.2603 33.3330
4-methylfasudil LCLC-97TM1 CTRP1 0.2603 33.3330
4-methylfasudil LU-65 CTRP1 0.2603 33.3330
4-methylfasudil LU-99 CTRP1 0.2603 33.3330
4-methylfasudil LXF289 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1048 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1105 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H1299 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1355 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1373 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1435 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1437 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1568 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1573 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1666 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1694 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H1755 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H1781 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H1792 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1793 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1836 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H1876 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H1915 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1930 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1944 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H1963 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H1975 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H2009 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H2023 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2029 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H2030 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2073 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2081 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2110 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2122 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2126 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H2141 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2172 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2286 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H23 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H2342 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H2405 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H3255 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H358 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H441 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H460 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H522 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H596 CTRP1 1.0417 133.3300
4-methylfasudil NCI-H650 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H661 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H727 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H810 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H82 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H841 CTRP1 1.0417 133.3300
4-methylfasudil RERF-LC-KJ CTRP1 0.2603 33.3330
4-methylfasudil SCLC-21H CTRP1 1.0417 133.3300
4-methylfasudil SHP-77 CTRP1 0.2603 33.3330
4-methylfasudil SK-LU-1 CTRP1 1.0417 133.3300
4-methylfasudil SQ-1 CTRP1 1.0417 133.3300
4-methylfasudil T3M-10 CTRP1 1.0417 133.3300
4-methylfasudil VMRC-LCD CTRP1 0.2603 33.3330
4-methylfasudil KYSE-140 CTRP1 0.2603 33.3330
4-methylfasudil KYSE-410 CTRP1 0.2603 33.3330
4-methylfasudil KYSE-450 CTRP1 0.2603 33.3330
4-methylfasudil A2780 CTRP1 1.0417 133.3300
4-methylfasudil CAOV-3 CTRP1 1.0417 133.3300
4-methylfasudil COV318 CTRP1 0.2603 33.3330
4-methylfasudil COV362 CTRP1 1.0417 133.3300
4-methylfasudil COV434 CTRP1 1.0417 133.3300
4-methylfasudil COV644 CTRP1 1.0417 133.3300
4-methylfasudil EFO-21 CTRP1 0.2603 33.3330
4-methylfasudil EFO-27 CTRP1 1.0417 133.3300
4-methylfasudil HEYA8 CTRP1 0.2603 33.3330
4-methylfasudil IGROV-1 CTRP1 1.0417 133.3300
4-methylfasudil JHOC-5 CTRP1 1.0417 133.3300
4-methylfasudil JHOM-1 CTRP1 1.0417 133.3300
4-methylfasudil JHOS-4 CTRP1 0.2603 33.3330
4-methylfasudil OAW42 CTRP1 1.0417 133.3300
4-methylfasudil OV7 CTRP1 1.0417 133.3300
4-methylfasudil OV-90 CTRP1 1.0417 133.3300
4-methylfasudil OVCAR-4 CTRP1 1.0417 133.3300
4-methylfasudil OVCAR-8 CTRP1 1.0417 133.3300
4-methylfasudil OVK18 CTRP1 1.0417 133.3300
4-methylfasudil OVKATE CTRP1 1.0417 133.3300
4-methylfasudil OVMANA CTRP1 0.2603 33.3330
4-methylfasudil RKN CTRP1 1.0417 133.3300
4-methylfasudil RMG-I CTRP1 1.0417 133.3300
4-methylfasudil RMUG-S CTRP1 1.0417 133.3300
4-methylfasudil SK-OV-3 CTRP1 0.2603 33.3330
4-methylfasudil SNU-840 CTRP1 1.0417 133.3300
4-methylfasudil TYK-NU CTRP1 1.0417 133.3300
4-methylfasudil CAPAN-2 CTRP1 0.2603 33.3330
4-methylfasudil CFPAC-1 CTRP1 0.2603 33.3330
4-methylfasudil HPAC CTRP1 0.2603 33.3330
4-methylfasudil HUP-T4 CTRP1 0.2603 33.3330
4-methylfasudil KP-3 CTRP1 0.2603 33.3330
4-methylfasudil PANC03.27 CTRP1 0.2603 33.3330
4-methylfasudil PANC10.05 CTRP1 0.2603 33.3330
4-methylfasudil PATU8902 CTRP1 0.2603 33.3330
4-methylfasudil QGP-1 CTRP1 0.2603 33.3330
4-methylfasudil SUIT-2 CTRP1 0.2603 33.3330
4-methylfasudil MSTO-211H CTRP1 0.2603 33.3330
4-methylfasudil NCI-H2052 CTRP1 0.2603 33.3330
4-methylfasudil NCI-H28 CTRP1 0.2603 33.3330
4-methylfasudil MIAPACA-3 CTRP1 0.2603 33.3330
4-methylfasudil A-375 CTRP1 1.0417 133.3300
4-methylfasudil COLO741 CTRP1 0.2603 33.3330
4-methylfasudil G-361 CTRP1 0.2603 33.3330
4-methylfasudil HS852.T CTRP1 0.2603 33.3330
4-methylfasudil HS936.T CTRP1 0.2603 33.3330
4-methylfasudil HS944.T CTRP1 0.2603 33.3330
4-methylfasudil SK-MEL-1 CTRP1 1.0417 133.3300
4-methylfasudil SK-MEL-28 CTRP1 1.0417 133.3300
4-methylfasudil SK-MEL-5 CTRP1 1.0417 133.3300
4-methylfasudil G-401 CTRP1 0.2603 33.3330
4-methylfasudil HT-1080 CTRP1 1.0417 133.3300
4-methylfasudil AGS CTRP1 1.0417 133.3300
4-methylfasudil FU97 CTRP1 0.2603 33.3330
4-methylfasudil KE-97 CTRP1 0.2603 33.3330
4-methylfasudil MKN7 CTRP1 0.2603 33.3330
4-methylfasudil MKN74 CTRP1 0.2603 33.3330
4-methylfasudil NUGC-4 CTRP1 0.2603 33.3330
4-methylfasudil SH-10-TC CTRP1 0.2603 33.3330
4-methylfasudil HSC-2 CTRP1 0.2603 33.3330
4-methylfasudil SCC-9 CTRP1 1.0417 133.3300
4-methylfasudil 5637 CTRP1 0.2603 33.3330
4-methylfasudil HT-1376 CTRP1 0.2603 33.3330
4-methylfasudil KMBC-2 CTRP1 0.2603 33.3330
4-methylfasudil RT-4 CTRP1 0.2603 33.3330
4-methylfasudil UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.