Drug : Brd-K86535717

CTRP2 Name : BRD-K86535717

Dataset : All
Synonyms :
Targets :
Pathways : product of diversity oriented synthesis

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BRD-K86535717 CAS-1 CTRP2 0.0020 66.0000
BRD-K86535717 KPL-1 CTRP2 0.0020 66.0000
BRD-K86535717 MKN1 CTRP2 0.0020 66.0000
BRD-K86535717 253J-BV CTRP2 0.0020 66.0000
BRD-K86535717 BFTC-905 CTRP2 0.0020 66.0000
BRD-K86535717 BFTC-909 CTRP2 0.0020 66.0000
BRD-K86535717 CAL-29 CTRP2 0.0020 66.0000
BRD-K86535717 CAL-62 CTRP2 0.0020 66.0000
BRD-K86535717 HUCC-T1 CTRP2 0.0020 66.0000
BRD-K86535717 NMC-G1 CTRP2 0.0020 66.0000
BRD-K86535717 RPMI-7951 CTRP2 0.0020 66.0000
BRD-K86535717 253J CTRP2 0.0020 66.0000
BRD-K86535717 HDQ-P1 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-489 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-626 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-738 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-878 CTRP2 0.0020 66.0000
BRD-K86535717 TUHR4TKB CTRP2 0.0020 66.0000
BRD-K86535717 ACC-MESO-1 CTRP2 0.0020 66.0000
BRD-K86535717 B-CPAP CTRP2 0.0020 66.0000
BRD-K86535717 CGTH-W-1 CTRP2 0.0020 66.0000
BRD-K86535717 COLO680N CTRP2 0.0020 66.0000
BRD-K86535717 ECC12 CTRP2 0.0020 66.0000
BRD-K86535717 HCC95 CTRP2 0.0020 66.0000
BRD-K86535717 JMSU-1 CTRP2 0.0020 66.0000
BRD-K86535717 RH41 CTRP2 0.0020 66.0000
BRD-K86535717 WSU-DLCL2 CTRP2 0.0020 66.0000
BRD-K86535717 23132-87 CTRP2 0.0020 66.0000
BRD-K86535717 8305C CTRP2 0.0020 66.0000
BRD-K86535717 BHY CTRP2 0.0020 66.0000
BRD-K86535717 GSU CTRP2 0.0020 66.0000
BRD-K86535717 JIMT-1 CTRP2 0.0020 66.0000
BRD-K86535717 KMRC-20 CTRP2 0.0020 66.0000
BRD-K86535717 OUMS-23 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1076 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1196 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-8 CTRP2 0.0020 66.0000
BRD-K86535717 A-375 CTRP2 0.0020 66.0000
BRD-K86535717 A-549 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H2009 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-201 CTRP2 0.0020 66.0000
BRD-K86535717 SUIT-2 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1079 CTRP2 0.0020 66.0000
BRD-K86535717 COLO741 CTRP2 0.0020 66.0000
BRD-K86535717 DEL CTRP2 0.0020 66.0000
BRD-K86535717 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP2 0.0020 66.0000
BRD-K86535717 HCC15 CTRP2 0.0020 66.0000
BRD-K86535717 KP-4 CTRP2 0.0020 66.0000
BRD-K86535717 LU-99 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H1155 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H1581 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H2106 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H358 CTRP2 0.0020 66.0000
BRD-K86535717 DLD-1 CTRP2 0.0020 66.0000
BRD-K86535717 EM-2 CTRP2 0.0020 66.0000
BRD-K86535717 JURL-MK1 CTRP2 0.0020 66.0000
BRD-K86535717 P12-ICHIKAWA CTRP2 0.0020 66.0000
BRD-K86535717 KE-37 CTRP2 0.0020 66.0000
BRD-K86535717 KMS-21-BM CTRP2 0.0020 66.0000
BRD-K86535717 LI-7 CTRP2 0.0020 66.0000
BRD-K86535717 MHH-NB-11 CTRP2 0.0020 66.0000
BRD-K86535717 MOLM-13 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H1975 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H28 CTRP2 0.0020 66.0000
BRD-K86535717 639V CTRP2 0.0020 66.0000
BRD-K86535717 BXPC-3 CTRP2 0.0020 66.0000
BRD-K86535717 CML-T1 CTRP2 0.0020 66.0000
BRD-K86535717 GSS CTRP2 0.0020 66.0000
BRD-K86535717 HCC366 CTRP2 0.0020 66.0000
BRD-K86535717 KURAMOCHI CTRP2 0.0020 66.0000
BRD-K86535717 LS411N CTRP2 0.0020 66.0000
BRD-K86535717 LS513 CTRP2 0.0020 66.0000
BRD-K86535717 ONCO-DG-1 CTRP2 0.0020 66.0000
BRD-K86535717 ONS-76 CTRP2 0.0020 66.0000
BRD-K86535717 SK-CO-1 CTRP2 0.0020 66.0000
BRD-K86535717 SW48 CTRP2 0.0020 66.0000
BRD-K86535717 VM-CUB-1 CTRP2 0.0020 66.0000
BRD-K86535717 BEN CTRP2 0.0020 66.0000
BRD-K86535717 CFPAC-1 CTRP2 0.0020 66.0000
BRD-K86535717 HCC78 CTRP2 0.0020 66.0000
BRD-K86535717 HT CTRP2 0.0020 66.0000
BRD-K86535717 KU-19-19 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H1299 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H727 CTRP2 0.0020 66.0000
BRD-K86535717 NCO2 CTRP2 0.0020 66.0000
BRD-K86535717 OVTOKO CTRP2 0.0020 66.0000
BRD-K86535717 P31-FUJ CTRP2 0.0020 66.0000
BRD-K86535717 PEER CTRP2 0.0020 66.0000
BRD-K86535717 RPMI-8402 CTRP2 0.0020 66.0000
BRD-K86535717 SHP-77 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1077 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-620 CTRP2 0.0020 66.0000
BRD-K86535717 SU-DHL-1 CTRP2 0.0020 66.0000
BRD-K86535717 COLO205 CTRP2 0.0020 66.0000
BRD-K86535717 EHEB CTRP2 0.0020 66.0000
BRD-K86535717 KI-JK CTRP2 0.0020 66.0000
BRD-K86535717 KMM-1 CTRP2 0.0020 66.0000
BRD-K86535717 LCLC-103H CTRP2 0.0020 66.0000
BRD-K86535717 MKN45 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H2405 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H650 CTRP2 0.0020 66.0000
BRD-K86535717 OS-RC-2 CTRP2 0.0020 66.0000
BRD-K86535717 OVSAHO CTRP2 0.0020 66.0000
BRD-K86535717 QGP-1 CTRP2 0.0020 66.0000
BRD-K86535717 RL95-2 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1041 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1066 CTRP2 0.0020 66.0000
BRD-K86535717 SW1353 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-213 CTRP2 0.0020 66.0000
BRD-K86535717 8505C CTRP2 0.0020 66.0000
BRD-K86535717 CALU-3 CTRP2 0.0020 66.0000
BRD-K86535717 DAOY CTRP2 0.0020 66.0000
BRD-K86535717 GB-1 CTRP2 0.0020 66.0000
BRD-K86535717 HCC1171 CTRP2 0.0020 66.0000
BRD-K86535717 HCC44 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H211 CTRP2 0.0020 66.0000
BRD-K86535717 RERF-LC-A1 CTRP2 0.0020 66.0000
BRD-K86535717 SBC-5 CTRP2 0.0020 66.0000
BRD-K86535717 SF126 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-119 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-182 CTRP2 0.0020 66.0000
BRD-K86535717 TCCSUP CTRP2 0.0020 66.0000
BRD-K86535717 CAMA-1 CTRP2 0.0020 66.0000
BRD-K86535717 DETROIT562 CTRP2 0.0020 66.0000
BRD-K86535717 HEC-1-B CTRP2 0.0020 66.0000
BRD-K86535717 HEP3B2.1-7 CTRP2 0.0020 66.0000
BRD-K86535717 HSC-3 CTRP2 0.0020 66.0000
BRD-K86535717 MCF-7 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1105 CTRP2 0.0020 66.0000
BRD-K86535717 U-87MGATCC CTRP2 0.0020 66.0000
BRD-K86535717 22RV1 CTRP2 0.0020 66.0000
BRD-K86535717 769-P CTRP2 0.0020 66.0000
BRD-K86535717 COLO699 CTRP2 0.0020 66.0000
BRD-K86535717 DOV13 CTRP2 0.0020 66.0000
BRD-K86535717 ES2 CTRP2 0.0020 66.0000
BRD-K86535717 HCC1806 CTRP2 0.0020 66.0000
BRD-K86535717 HCC1954 CTRP2 0.0020 66.0000
BRD-K86535717 HPAF-II CTRP2 0.0020 66.0000
BRD-K86535717 KHM-1B CTRP2 0.0020 66.0000
BRD-K86535717 OVISE CTRP2 0.0020 66.0000
BRD-K86535717 JVM-3 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-C2A CTRP2 0.0020 66.0000
BRD-K86535717 U2OS CTRP2 0.0020 66.0000
BRD-K86535717 5637 CTRP2 0.0020 66.0000
BRD-K86535717 CAL-12T CTRP2 0.0020 66.0000
BRD-K86535717 DMS79 CTRP2 0.0020 66.0000
BRD-K86535717 HCC1588 CTRP2 0.0020 66.0000
BRD-K86535717 HCC1833 CTRP2 0.0020 66.0000
BRD-K86535717 HCC2279 CTRP2 0.0020 66.0000
BRD-K86535717 KE-97 CTRP2 0.0020 66.0000
BRD-K86535717 KP-3 CTRP2 0.0020 66.0000
BRD-K86535717 KU812 CTRP2 0.0020 66.0000
BRD-K86535717 KYSE-140 CTRP2 0.0020 66.0000
BRD-K86535717 NALM-6 CTRP2 0.0020 66.0000
BRD-K86535717 NUGC-4 CTRP2 0.0020 66.0000
BRD-K86535717 TT CTRP2 0.0020 66.0000
BRD-K86535717 AGS CTRP2 0.0020 66.0000
BRD-K86535717 HCT116 CTRP2 0.0020 66.0000
BRD-K86535717 HEC-108 CTRP2 0.0020 66.0000
BRD-K86535717 HEC-59 CTRP2 0.0020 66.0000
BRD-K86535717 HMC-1-8 CTRP2 0.0020 66.0000
BRD-K86535717 HT-29 CTRP2 0.0020 66.0000
BRD-K86535717 ISHIKAWA(HERAKLIO)02ER- CTRP2 0.0020 66.0000
BRD-K86535717 JHOC-5 CTRP2 0.0020 66.0000
BRD-K86535717 KYSE-180 CTRP2 0.0020 66.0000
BRD-K86535717 LS180 CTRP2 0.0020 66.0000
BRD-K86535717 MELHO CTRP2 0.0020 66.0000
BRD-K86535717 MHH-ES-1 CTRP2 0.0020 66.0000
BRD-K86535717 MOR-CPR CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H460 CTRP2 0.0020 66.0000
BRD-K86535717 HCC2108 CTRP2 0.0020 66.0000
BRD-K86535717 HCC827 CTRP2 0.0020 66.0000
BRD-K86535717 HEC-251 CTRP2 0.0020 66.0000
BRD-K86535717 HEC-265 CTRP2 0.0020 66.0000
BRD-K86535717 HEC-6 CTRP2 0.0020 66.0000
BRD-K86535717 HEL CTRP2 0.0020 66.0000
BRD-K86535717 JHUEM-2 CTRP2 0.0020 66.0000
BRD-K86535717 JURKAT CTRP2 0.0020 66.0000
BRD-K86535717 JVM-2 CTRP2 0.0020 66.0000
BRD-K86535717 KCL-22 CTRP2 0.0020 66.0000
BRD-K86535717 KE-39 CTRP2 0.0020 66.0000
BRD-K86535717 KM-H2 CTRP2 0.0020 66.0000
BRD-K86535717 LAMA-84 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H2030 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-719 CTRP2 0.0020 66.0000
BRD-K86535717 KLE CTRP2 0.0020 66.0000
BRD-K86535717 KMS-26 CTRP2 0.0020 66.0000
BRD-K86535717 KMS-27 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H1838 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H196 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H292 CTRP2 0.0020 66.0000
BRD-K86535717 SK-MEL-1 CTRP2 0.0020 66.0000
BRD-K86535717 HCC1937 CTRP2 0.0020 66.0000
BRD-K86535717 HDLM-2 CTRP2 0.0020 66.0000
BRD-K86535717 HUH-28 CTRP2 0.0020 66.0000
BRD-K86535717 MV4-11 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H526 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H69 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H929 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-N87 CTRP2 0.0020 66.0000
BRD-K86535717 PF-382 CTRP2 0.0020 66.0000
BRD-K86535717 SF295 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1272 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-308 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-478 CTRP2 0.0020 66.0000
BRD-K86535717 BHT-101 CTRP2 0.0020 66.0000
BRD-K86535717 CAL-148 CTRP2 0.0020 66.0000
BRD-K86535717 CAL-51 CTRP2 0.0020 66.0000
BRD-K86535717 HCC1395 CTRP2 0.0020 66.0000
BRD-K86535717 HT115 CTRP2 0.0020 66.0000
BRD-K86535717 LN-18 CTRP2 0.0020 66.0000
BRD-K86535717 LN-229 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H1734 CTRP2 0.0020 66.0000
BRD-K86535717 NCI-H2291 CTRP2 0.0020 66.0000
BRD-K86535717 RERF-LC-AD1 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-1214 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-46 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-466 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-5 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-668 CTRP2 0.0020 66.0000
BRD-K86535717 SNU-899 CTRP2 0.0020 66.0000
BRD-K86535717 TE-10 CTRP2 0.0020 66.0000
BRD-K86535717 TE-9 CTRP2 0.0020 66.0000
BRD-K86535717 YD-10B CTRP2 0.0020 66.0000
BRD-K86535717 YD-15 CTRP2 0.0020 66.0000
BRD-K86535717 YD-38 CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.