Drug : Abt-751

CTRP1 Name : ABT-751

Dataset : All
Synonyms :
Targets : TUBB
Pathways : inhibitor of beta-tubulin

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

:


Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
ABT-751 U2OS CTRP1 0.2604 33.3330
ABT-751 MCF-7 CTRP1 0.2604 33.3330
ABT-751 GAMG CTRP1 0.2603 33.3330
ABT-751 LN-229 CTRP1 0.2604 33.3330
ABT-751 SF295 CTRP1 0.2603 33.3330
ABT-751 HEC-108 CTRP1 0.2603 33.3330
ABT-751 HEC-151 CTRP1 0.2604 33.3330
ABT-751 HEC-251 CTRP1 0.2603 33.3330
ABT-751 HEC-265 CTRP1 0.2603 33.3330
ABT-751 HEC-59 CTRP1 0.2603 33.3330
ABT-751 HEC-6 CTRP1 0.2603 33.3330
ABT-751 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
ABT-751 JHUEM-2 CTRP1 0.2604 33.3330
ABT-751 KLE CTRP1 0.2603 33.3330
ABT-751 MFE-319 CTRP1 0.2603 33.3330
ABT-751 SNG-M CTRP1 0.2603 33.3330
ABT-751 AMO1 CTRP1 0.2604 33.3330
ABT-751 BL-70 CTRP1 0.2603 33.3330
ABT-751 EJM CTRP1 0.2604 33.3330
ABT-751 GDM-1 CTRP1 0.2604 33.3330
ABT-751 HT CTRP1 0.2603 33.3330
ABT-751 KMS-11 CTRP1 0.2604 33.3330
ABT-751 KU812 CTRP1 0.2603 33.3330
ABT-751 LP-1 CTRP1 0.2604 33.3330
ABT-751 MC116 CTRP1 0.2603 33.3330
ABT-751 MOLM-16 CTRP1 0.2604 33.3330
ABT-751 NOMO-1 CTRP1 0.2604 33.3330
ABT-751 NU-DUL-1 CTRP1 0.2604 33.3330
ABT-751 OCI-AML-3 CTRP1 0.2604 33.3330
ABT-751 OCI-LY10 CTRP1 0.2604 33.3330
ABT-751 P3HR-1 CTRP1 0.2603 33.3330
ABT-751 PL21 CTRP1 0.2604 33.3330
ABT-751 RPMI-8226 CTRP1 0.2604 33.3330
ABT-751 SKM-1 CTRP1 0.2604 33.3330
ABT-751 SU-DHL-4 CTRP1 0.2604 33.3330
ABT-751 SU-DHL-5 CTRP1 0.2604 33.3330
ABT-751 THP-1 CTRP1 0.2604 33.3330
ABT-751 U-937 CTRP1 0.2604 33.3330
ABT-751 WSU-DLCL2 CTRP1 0.2604 33.3330
ABT-751 RCC10RGB CTRP1 0.2604 33.3330
ABT-751 VMRC-RCW CTRP1 0.2603 33.3330
ABT-751 CL-34 CTRP1 0.2604 33.3330
ABT-751 CL-40 CTRP1 0.2604 33.3330
ABT-751 COLO320 CTRP1 0.2604 33.3330
ABT-751 COLO678 CTRP1 0.2604 33.3330
ABT-751 CW-2 CTRP1 0.2604 33.3330
ABT-751 HCT116 CTRP1 0.2604 33.3330
ABT-751 HCT8 CTRP1 0.2604 33.3330
ABT-751 HT115 CTRP1 0.2604 33.3330
ABT-751 HT-29 CTRP1 0.2604 33.3330
ABT-751 HT-55 CTRP1 0.2604 33.3330
ABT-751 KM12 CTRP1 0.2604 33.3330
ABT-751 LOVO CTRP1 0.2604 33.3330
ABT-751 LS123 CTRP1 0.2604 33.3330
ABT-751 LS180 CTRP1 0.2604 33.3330
ABT-751 MDST8 CTRP1 0.2604 33.3330
ABT-751 NCI-H508 CTRP1 0.2604 33.3330
ABT-751 RCM-1[HUMANESC] CTRP1 0.2604 33.3330
ABT-751 RKO CTRP1 0.2604 33.3330
ABT-751 SNU-1040 CTRP1 0.2604 33.3330
ABT-751 SNU-175 CTRP1 0.2604 33.3330
ABT-751 SNU-61 CTRP1 0.2604 33.3330
ABT-751 SNU-81 CTRP1 0.2604 33.3330
ABT-751 SNU-C2A CTRP1 0.2603 33.3330
ABT-751 SNU-C4 CTRP1 0.2604 33.3330
ABT-751 SNU-C5 CTRP1 0.2604 33.3330
ABT-751 SW403 CTRP1 0.2603 33.3330
ABT-751 SW480 CTRP1 0.2604 33.3330
ABT-751 SW620 CTRP1 0.2604 33.3330
ABT-751 SW948 CTRP1 0.2604 33.3330
ABT-751 HEP-G2 CTRP1 0.2604 33.3330
ABT-751 JHH-6 CTRP1 0.2603 33.3330
ABT-751 SNU-398 CTRP1 0.2604 33.3330
ABT-751 SNU-449 CTRP1 0.2603 33.3330
ABT-751 A-549 CTRP1 0.2603 33.3330
ABT-751 BEN CTRP1 0.2603 33.3330
ABT-751 CAL-12T CTRP1 0.2604 33.3330
ABT-751 CALU-3 CTRP1 0.2603 33.3330
ABT-751 CALU-6 CTRP1 0.2603 33.3330
ABT-751 CHAGO-K-1 CTRP1 0.2603 33.3330
ABT-751 COLO668 CTRP1 0.2603 33.3330
ABT-751 COLO699 CTRP1 0.2604 33.3330
ABT-751 COR-L23 CTRP1 0.2604 33.3330
ABT-751 COR-L279 CTRP1 0.2603 33.3330
ABT-751 COR-L51 CTRP1 0.2604 33.3330
ABT-751 COR-L88 CTRP1 0.2603 33.3330
ABT-751 DMS273 CTRP1 0.2603 33.3330
ABT-751 DV-90 CTRP1 0.2603 33.3330
ABT-751 EPLC-272H CTRP1 0.2603 33.3330
ABT-751 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
ABT-751 HCC1195 CTRP1 0.2604 33.3330
ABT-751 HCC1359 CTRP1 0.2604 33.3330
ABT-751 HCC15 CTRP1 0.2604 33.3330
ABT-751 HCC1833 CTRP1 0.2604 33.3330
ABT-751 HCC2108 CTRP1 0.2604 33.3330
ABT-751 HCC2935 CTRP1 0.2604 33.3330
ABT-751 HCC33 CTRP1 0.2603 33.3330
ABT-751 HCC4006 CTRP1 0.2604 33.3330
ABT-751 HCC44 CTRP1 0.2603 33.3330
ABT-751 HCC827 CTRP1 0.2604 33.3330
ABT-751 KNS-62 CTRP1 0.2603 33.3330
ABT-751 LC-1-SQ-SF CTRP1 0.2603 33.3330
ABT-751 LCLC-103H CTRP1 0.2603 33.3330
ABT-751 LCLC-97TM1 CTRP1 0.2603 33.3330
ABT-751 LU-65 CTRP1 0.2603 33.3330
ABT-751 LXF289 CTRP1 0.2603 33.3330
ABT-751 NCI-H1048 CTRP1 0.2603 33.3330
ABT-751 NCI-H1105 CTRP1 0.2604 33.3330
ABT-751 NCI-H1299 CTRP1 0.2603 33.3330
ABT-751 NCI-H1355 CTRP1 0.2603 33.3330
ABT-751 NCI-H1435 CTRP1 0.2603 33.3330
ABT-751 NCI-H1437 CTRP1 0.2603 33.3330
ABT-751 NCI-H1568 CTRP1 0.2603 33.3330
ABT-751 NCI-H1573 CTRP1 0.2603 33.3330
ABT-751 NCI-H1666 CTRP1 0.2603 33.3330
ABT-751 NCI-H1694 CTRP1 0.2604 33.3330
ABT-751 NCI-H1755 CTRP1 0.2604 33.3330
ABT-751 NCI-H1781 CTRP1 0.2604 33.3330
ABT-751 NCI-H1792 CTRP1 0.2603 33.3330
ABT-751 NCI-H1836 CTRP1 0.2604 33.3330
ABT-751 NCI-H1876 CTRP1 0.2604 33.3330
ABT-751 NCI-H1915 CTRP1 0.2603 33.3330
ABT-751 NCI-H1930 CTRP1 0.2603 33.3330
ABT-751 NCI-H1944 CTRP1 0.2603 33.3330
ABT-751 NCI-H1963 CTRP1 0.2604 33.3330
ABT-751 NCI-H1975 CTRP1 0.2603 33.3330
ABT-751 NCI-H2009 CTRP1 0.2603 33.3330
ABT-751 NCI-H2023 CTRP1 0.2604 33.3330
ABT-751 NCI-H2029 CTRP1 0.2603 33.3330
ABT-751 NCI-H2030 CTRP1 0.2604 33.3330
ABT-751 NCI-H2073 CTRP1 0.2604 33.3330
ABT-751 NCI-H2081 CTRP1 0.2604 33.3330
ABT-751 NCI-H2110 CTRP1 0.2604 33.3330
ABT-751 NCI-H2122 CTRP1 0.2604 33.3330
ABT-751 NCI-H2126 CTRP1 0.2603 33.3330
ABT-751 NCI-H2141 CTRP1 0.2604 33.3330
ABT-751 NCI-H2172 CTRP1 0.2604 33.3330
ABT-751 NCI-H2286 CTRP1 0.2603 33.3330
ABT-751 NCI-H23 CTRP1 0.2603 33.3330
ABT-751 NCI-H2342 CTRP1 0.2604 33.3330
ABT-751 NCI-H2405 CTRP1 0.2603 33.3330
ABT-751 NCI-H3255 CTRP1 0.2604 33.3330
ABT-751 NCI-H441 CTRP1 0.2604 33.3330
ABT-751 NCI-H460 CTRP1 0.2604 33.3330
ABT-751 NCI-H596 CTRP1 0.2604 33.3330
ABT-751 NCI-H650 CTRP1 0.2603 33.3330
ABT-751 NCI-H661 CTRP1 0.2603 33.3330
ABT-751 NCI-H727 CTRP1 0.2603 33.3330
ABT-751 NCI-H810 CTRP1 0.2603 33.3330
ABT-751 NCI-H82 CTRP1 0.2603 33.3330
ABT-751 NCI-H841 CTRP1 0.2604 33.3330
ABT-751 RERF-LC-KJ CTRP1 0.2603 33.3330
ABT-751 SCLC-21H CTRP1 0.2604 33.3330
ABT-751 SHP-77 CTRP1 0.2603 33.3330
ABT-751 SK-LU-1 CTRP1 0.2604 33.3330
ABT-751 SQ-1 CTRP1 0.2604 33.3330
ABT-751 T3M-10 CTRP1 0.2604 33.3330
ABT-751 VMRC-LCD CTRP1 0.2603 33.3330
ABT-751 KYSE-140 CTRP1 0.2603 33.3330
ABT-751 KYSE-410 CTRP1 0.2603 33.3330
ABT-751 KYSE-450 CTRP1 0.2603 33.3330
ABT-751 A2780 CTRP1 0.2604 33.3330
ABT-751 CAOV-3 CTRP1 0.2604 33.3330
ABT-751 COV318 CTRP1 0.2603 33.3330
ABT-751 COV362 CTRP1 0.2604 33.3330
ABT-751 COV434 CTRP1 0.2604 33.3330
ABT-751 COV644 CTRP1 0.2604 33.3330
ABT-751 EFO-21 CTRP1 0.2603 33.3330
ABT-751 EFO-27 CTRP1 0.2604 33.3330
ABT-751 HEYA8 CTRP1 0.2603 33.3330
ABT-751 IGROV-1 CTRP1 0.2604 33.3330
ABT-751 JHOC-5 CTRP1 0.2604 33.3330
ABT-751 JHOM-1 CTRP1 0.2604 33.3330
ABT-751 JHOS-4 CTRP1 0.2603 33.3330
ABT-751 OAW42 CTRP1 0.2604 33.3330
ABT-751 OV7 CTRP1 0.2604 33.3330
ABT-751 OV-90 CTRP1 0.2604 33.3330
ABT-751 OVCAR-4 CTRP1 0.2604 33.3330
ABT-751 OVCAR-8 CTRP1 0.2604 33.3330
ABT-751 OVK18 CTRP1 0.2604 33.3330
ABT-751 OVKATE CTRP1 0.2604 33.3330
ABT-751 OVMANA CTRP1 0.2603 33.3330
ABT-751 RKN CTRP1 0.2604 33.3330
ABT-751 RMG-I CTRP1 0.2604 33.3330
ABT-751 RMUG-S CTRP1 0.2604 33.3330
ABT-751 SK-OV-3 CTRP1 0.2603 33.3330
ABT-751 SNU-840 CTRP1 0.2604 33.3330
ABT-751 TYK-NU CTRP1 0.2604 33.3330
ABT-751 CAPAN-2 CTRP1 0.2603 33.3330
ABT-751 HUP-T4 CTRP1 0.2603 33.3330
ABT-751 KP-3 CTRP1 0.2603 33.3330
ABT-751 PANC03.27 CTRP1 0.2603 33.3330
ABT-751 PATU8902 CTRP1 0.2603 33.3330
ABT-751 QGP-1 CTRP1 0.2603 33.3330
ABT-751 SUIT-2 CTRP1 0.2603 33.3330
ABT-751 MSTO-211H CTRP1 0.2603 33.3330
ABT-751 NCI-H2052 CTRP1 0.2603 33.3330
ABT-751 NCI-H28 CTRP1 0.2603 33.3330
ABT-751 MIAPACA-3 CTRP1 0.2603 33.3330
ABT-751 A-375 CTRP1 0.2604 33.3330
ABT-751 G-361 CTRP1 0.2603 33.3330
ABT-751 HS852.T CTRP1 0.2603 33.3330
ABT-751 HS936.T CTRP1 0.2603 33.3330
ABT-751 HS944.T CTRP1 0.2603 33.3330
ABT-751 SK-MEL-1 CTRP1 0.2604 33.3330
ABT-751 SK-MEL-28 CTRP1 0.2604 33.3330
ABT-751 SK-MEL-5 CTRP1 0.2604 33.3330
ABT-751 G-401 CTRP1 0.2603 33.3330
ABT-751 HT-1080 CTRP1 0.2604 33.3330
ABT-751 AGS CTRP1 0.2604 33.3330
ABT-751 FU97 CTRP1 0.2603 33.3330
ABT-751 KE-97 CTRP1 0.2603 33.3330
ABT-751 MKN7 CTRP1 0.2603 33.3330
ABT-751 MKN74 CTRP1 0.2603 33.3330
ABT-751 NUGC-4 CTRP1 0.2603 33.3330
ABT-751 SH-10-TC CTRP1 0.2603 33.3330
ABT-751 HSC-2 CTRP1 0.2603 33.3330
ABT-751 SCC-9 CTRP1 0.2604 33.3330
ABT-751 5637 CTRP1 0.2603 33.3330
ABT-751 HT-1376 CTRP1 0.2603 33.3330
ABT-751 KMBC-2 CTRP1 0.2603 33.3330
ABT-751 RT-4 CTRP1 0.2603 33.3330
ABT-751 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.