Drug : Bms-641988

CTRP1 Name : BMS-641988

Dataset : All
Synonyms :
Targets : AR
Pathways : antagonist of androgen receptor

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BMS-641988 U2OS CTRP1 0.2891 37.0000
BMS-641988 MCF-7 CTRP1 0.2891 37.0000
BMS-641988 GAMG CTRP1 0.2890 37.0000
BMS-641988 LN-229 CTRP1 0.2891 37.0000
BMS-641988 SF295 CTRP1 0.2890 37.0000
BMS-641988 HEC-108 CTRP1 0.2890 37.0000
BMS-641988 HEC-151 CTRP1 0.2891 37.0000
BMS-641988 HEC-251 CTRP1 0.2890 37.0000
BMS-641988 HEC-265 CTRP1 0.2890 37.0000
BMS-641988 HEC-59 CTRP1 0.2890 37.0000
BMS-641988 HEC-6 CTRP1 0.2890 37.0000
BMS-641988 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2890 37.0000
BMS-641988 JHUEM-2 CTRP1 0.2891 37.0000
BMS-641988 KLE CTRP1 0.2890 37.0000
BMS-641988 MFE-319 CTRP1 0.2890 37.0000
BMS-641988 SNG-M CTRP1 0.2890 37.0000
BMS-641988 AMO1 CTRP1 0.2891 37.0000
BMS-641988 BL-70 CTRP1 0.2890 37.0000
BMS-641988 EJM CTRP1 0.2891 37.0000
BMS-641988 GDM-1 CTRP1 0.2891 37.0000
BMS-641988 HT CTRP1 0.2890 37.0000
BMS-641988 KMS-11 CTRP1 0.2891 37.0000
BMS-641988 KU812 CTRP1 0.2890 37.0000
BMS-641988 LP-1 CTRP1 0.2891 37.0000
BMS-641988 MC116 CTRP1 0.2890 37.0000
BMS-641988 MOLM-16 CTRP1 0.2891 37.0000
BMS-641988 NOMO-1 CTRP1 0.2891 37.0000
BMS-641988 NU-DUL-1 CTRP1 0.2891 37.0000
BMS-641988 OCI-AML-3 CTRP1 0.2891 37.0000
BMS-641988 OCI-LY10 CTRP1 0.2891 37.0000
BMS-641988 P3HR-1 CTRP1 0.2890 37.0000
BMS-641988 PL21 CTRP1 0.2891 37.0000
BMS-641988 RPMI-8226 CTRP1 0.2891 37.0000
BMS-641988 SKM-1 CTRP1 0.2891 37.0000
BMS-641988 SU-DHL-4 CTRP1 0.2891 37.0000
BMS-641988 SU-DHL-5 CTRP1 0.2891 37.0000
BMS-641988 THP-1 CTRP1 0.2891 37.0000
BMS-641988 U-937 CTRP1 0.2891 37.0000
BMS-641988 WSU-DLCL2 CTRP1 0.2891 37.0000
BMS-641988 RCC10RGB CTRP1 0.2891 37.0000
BMS-641988 VMRC-RCW CTRP1 0.2890 37.0000
BMS-641988 C2BBE1 CTRP1 0.2890 37.0000
BMS-641988 CL-34 CTRP1 0.2891 37.0000
BMS-641988 CL-40 CTRP1 0.2891 37.0000
BMS-641988 COLO205 CTRP1 0.2890 37.0000
BMS-641988 COLO320 CTRP1 0.2891 37.0000
BMS-641988 COLO678 CTRP1 0.2891 37.0000
BMS-641988 CW-2 CTRP1 0.2891 37.0000
BMS-641988 DLD-1 CTRP1 0.2890 37.0000
BMS-641988 GP2D CTRP1 0.2890 37.0000
BMS-641988 HCT116 CTRP1 0.2891 37.0000
BMS-641988 HCT8 CTRP1 0.2891 37.0000
BMS-641988 HT115 CTRP1 0.2891 37.0000
BMS-641988 HT-29 CTRP1 0.2891 37.0000
BMS-641988 HT-55 CTRP1 0.2891 37.0000
BMS-641988 KM12 CTRP1 0.2891 37.0000
BMS-641988 LOVO CTRP1 0.2891 37.0000
BMS-641988 LS123 CTRP1 0.2891 37.0000
BMS-641988 LS180 CTRP1 0.2891 37.0000
BMS-641988 LS411N CTRP1 0.2890 37.0000
BMS-641988 LS513 CTRP1 0.2890 37.0000
BMS-641988 MDST8 CTRP1 0.2891 37.0000
BMS-641988 NCI-H508 CTRP1 0.2891 37.0000
BMS-641988 RCM-1[HUMANESC] CTRP1 0.2891 37.0000
BMS-641988 RKO CTRP1 0.2891 37.0000
BMS-641988 SK-CO-1 CTRP1 0.2890 37.0000
BMS-641988 SNU-1040 CTRP1 0.2891 37.0000
BMS-641988 SNU-175 CTRP1 0.2891 37.0000
BMS-641988 SNU-61 CTRP1 0.2891 37.0000
BMS-641988 SNU-81 CTRP1 0.2891 37.0000
BMS-641988 SNU-C2A CTRP1 0.2890 37.0000
BMS-641988 SNU-C4 CTRP1 0.2891 37.0000
BMS-641988 SNU-C5 CTRP1 0.2891 37.0000
BMS-641988 SW403 CTRP1 0.2890 37.0000
BMS-641988 SW48 CTRP1 0.2890 37.0000
BMS-641988 SW480 CTRP1 0.2891 37.0000
BMS-641988 SW620 CTRP1 0.2891 37.0000
BMS-641988 SW948 CTRP1 0.2891 37.0000
BMS-641988 HEP-G2 CTRP1 0.2891 37.0000
BMS-641988 JHH-6 CTRP1 0.2890 37.0000
BMS-641988 SNU-398 CTRP1 0.2891 37.0000
BMS-641988 SNU-449 CTRP1 0.2890 37.0000
BMS-641988 A-549 CTRP1 0.2890 37.0000
BMS-641988 BEN CTRP1 0.2890 37.0000
BMS-641988 CAL-12T CTRP1 0.2891 37.0000
BMS-641988 CALU-3 CTRP1 0.2890 37.0000
BMS-641988 CALU-6 CTRP1 0.2890 37.0000
BMS-641988 CHAGO-K-1 CTRP1 0.2890 37.0000
BMS-641988 COLO668 CTRP1 0.2890 37.0000
BMS-641988 COLO699 CTRP1 0.2891 37.0000
BMS-641988 COR-L23 CTRP1 0.2891 37.0000
BMS-641988 COR-L279 CTRP1 0.2890 37.0000
BMS-641988 COR-L51 CTRP1 0.2891 37.0000
BMS-641988 COR-L88 CTRP1 0.2890 37.0000
BMS-641988 DMS273 CTRP1 0.2890 37.0000
BMS-641988 DV-90 CTRP1 0.2890 37.0000
BMS-641988 EBC-1 CTRP1 0.2890 37.0000
BMS-641988 EPLC-272H CTRP1 0.2890 37.0000
BMS-641988 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2890 37.0000
BMS-641988 HCC1195 CTRP1 0.2891 37.0000
BMS-641988 HCC1359 CTRP1 0.2891 37.0000
BMS-641988 HCC15 CTRP1 0.2891 37.0000
BMS-641988 HCC1833 CTRP1 0.2891 37.0000
BMS-641988 HCC2108 CTRP1 0.2891 37.0000
BMS-641988 HCC2935 CTRP1 0.2891 37.0000
BMS-641988 HCC33 CTRP1 0.2890 37.0000
BMS-641988 HCC4006 CTRP1 0.2891 37.0000
BMS-641988 HCC44 CTRP1 0.2890 37.0000
BMS-641988 HCC78 CTRP1 0.2890 37.0000
BMS-641988 HCC827 CTRP1 0.2891 37.0000
BMS-641988 KNS-62 CTRP1 0.2890 37.0000
BMS-641988 LC-1-SQ-SF CTRP1 0.2890 37.0000
BMS-641988 LCLC-103H CTRP1 0.2890 37.0000
BMS-641988 LCLC-97TM1 CTRP1 0.2890 37.0000
BMS-641988 LU-65 CTRP1 0.2890 37.0000
BMS-641988 LU-99 CTRP1 0.2890 37.0000
BMS-641988 LXF289 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1048 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1105 CTRP1 0.2891 37.0000
BMS-641988 NCI-H1299 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1355 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1373 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1435 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1437 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1568 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1573 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1666 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1694 CTRP1 0.2891 37.0000
BMS-641988 NCI-H1755 CTRP1 0.2891 37.0000
BMS-641988 NCI-H1781 CTRP1 0.2891 37.0000
BMS-641988 NCI-H1792 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1793 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1836 CTRP1 0.2891 37.0000
BMS-641988 NCI-H1876 CTRP1 0.2891 37.0000
BMS-641988 NCI-H1915 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1930 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1944 CTRP1 0.2890 37.0000
BMS-641988 NCI-H1963 CTRP1 0.2891 37.0000
BMS-641988 NCI-H1975 CTRP1 0.2890 37.0000
BMS-641988 NCI-H2009 CTRP1 0.2890 37.0000
BMS-641988 NCI-H2023 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2029 CTRP1 0.2890 37.0000
BMS-641988 NCI-H2030 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2073 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2081 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2110 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2122 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2126 CTRP1 0.2890 37.0000
BMS-641988 NCI-H2141 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2172 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2286 CTRP1 0.2890 37.0000
BMS-641988 NCI-H23 CTRP1 0.2890 37.0000
BMS-641988 NCI-H2342 CTRP1 0.2891 37.0000
BMS-641988 NCI-H2405 CTRP1 0.2890 37.0000
BMS-641988 NCI-H3255 CTRP1 0.2891 37.0000
BMS-641988 NCI-H358 CTRP1 0.2890 37.0000
BMS-641988 NCI-H441 CTRP1 0.2891 37.0000
BMS-641988 NCI-H460 CTRP1 0.2891 37.0000
BMS-641988 NCI-H522 CTRP1 0.2890 37.0000
BMS-641988 NCI-H596 CTRP1 0.2891 37.0000
BMS-641988 NCI-H650 CTRP1 0.2890 37.0000
BMS-641988 NCI-H661 CTRP1 0.2890 37.0000
BMS-641988 NCI-H727 CTRP1 0.2890 37.0000
BMS-641988 NCI-H810 CTRP1 0.2890 37.0000
BMS-641988 NCI-H82 CTRP1 0.2890 37.0000
BMS-641988 NCI-H841 CTRP1 0.2891 37.0000
BMS-641988 RERF-LC-KJ CTRP1 0.2890 37.0000
BMS-641988 SCLC-21H CTRP1 0.2891 37.0000
BMS-641988 SHP-77 CTRP1 0.2890 37.0000
BMS-641988 SK-LU-1 CTRP1 0.2891 37.0000
BMS-641988 SQ-1 CTRP1 0.2891 37.0000
BMS-641988 T3M-10 CTRP1 0.2891 37.0000
BMS-641988 VMRC-LCD CTRP1 0.2890 37.0000
BMS-641988 KYSE-140 CTRP1 0.2890 37.0000
BMS-641988 KYSE-410 CTRP1 0.2890 37.0000
BMS-641988 KYSE-450 CTRP1 0.2890 37.0000
BMS-641988 A2780 CTRP1 0.2891 37.0000
BMS-641988 CAOV-3 CTRP1 0.2891 37.0000
BMS-641988 COV318 CTRP1 0.2890 37.0000
BMS-641988 COV362 CTRP1 0.2891 37.0000
BMS-641988 COV434 CTRP1 0.2891 37.0000
BMS-641988 COV644 CTRP1 0.2891 37.0000
BMS-641988 EFO-21 CTRP1 0.2890 37.0000
BMS-641988 EFO-27 CTRP1 0.2891 37.0000
BMS-641988 HEYA8 CTRP1 0.2890 37.0000
BMS-641988 IGROV-1 CTRP1 0.2891 37.0000
BMS-641988 JHOC-5 CTRP1 0.2891 37.0000
BMS-641988 JHOM-1 CTRP1 0.2891 37.0000
BMS-641988 JHOS-4 CTRP1 0.2890 37.0000
BMS-641988 OAW42 CTRP1 0.2891 37.0000
BMS-641988 OV7 CTRP1 0.2891 37.0000
BMS-641988 OV-90 CTRP1 0.2891 37.0000
BMS-641988 OVCAR-4 CTRP1 0.2891 37.0000
BMS-641988 OVCAR-8 CTRP1 0.2891 37.0000
BMS-641988 OVK18 CTRP1 0.2891 37.0000
BMS-641988 OVKATE CTRP1 0.2891 37.0000
BMS-641988 OVMANA CTRP1 0.2890 37.0000
BMS-641988 RKN CTRP1 0.2891 37.0000
BMS-641988 RMG-I CTRP1 0.2891 37.0000
BMS-641988 RMUG-S CTRP1 0.2891 37.0000
BMS-641988 SK-OV-3 CTRP1 0.2890 37.0000
BMS-641988 SNU-840 CTRP1 0.2891 37.0000
BMS-641988 TYK-NU CTRP1 0.2891 37.0000
BMS-641988 CAPAN-2 CTRP1 0.2890 37.0000
BMS-641988 CFPAC-1 CTRP1 0.2890 37.0000
BMS-641988 HPAC CTRP1 0.2890 37.0000
BMS-641988 HUP-T4 CTRP1 0.2890 37.0000
BMS-641988 KP-3 CTRP1 0.2890 37.0000
BMS-641988 PANC03.27 CTRP1 0.2890 37.0000
BMS-641988 PANC10.05 CTRP1 0.2890 37.0000
BMS-641988 PATU8902 CTRP1 0.2890 37.0000
BMS-641988 QGP-1 CTRP1 0.2890 37.0000
BMS-641988 SUIT-2 CTRP1 0.2890 37.0000
BMS-641988 MSTO-211H CTRP1 0.2890 37.0000
BMS-641988 NCI-H2052 CTRP1 0.2890 37.0000
BMS-641988 NCI-H28 CTRP1 0.2890 37.0000
BMS-641988 MIAPACA-3 CTRP1 0.2890 37.0000
BMS-641988 A-375 CTRP1 0.2891 37.0000
BMS-641988 COLO741 CTRP1 0.2890 37.0000
BMS-641988 G-361 CTRP1 0.2890 37.0000
BMS-641988 HS852.T CTRP1 0.2890 37.0000
BMS-641988 HS936.T CTRP1 0.2890 37.0000
BMS-641988 HS944.T CTRP1 0.2890 37.0000
BMS-641988 SK-MEL-1 CTRP1 0.2891 37.0000
BMS-641988 SK-MEL-28 CTRP1 0.2891 37.0000
BMS-641988 SK-MEL-5 CTRP1 0.2891 37.0000
BMS-641988 G-401 CTRP1 0.2890 37.0000
BMS-641988 HT-1080 CTRP1 0.2891 37.0000
BMS-641988 AGS CTRP1 0.2891 37.0000
BMS-641988 FU97 CTRP1 0.2890 37.0000
BMS-641988 KE-97 CTRP1 0.2890 37.0000
BMS-641988 MKN7 CTRP1 0.2890 37.0000
BMS-641988 MKN74 CTRP1 0.2890 37.0000
BMS-641988 NUGC-4 CTRP1 0.2890 37.0000
BMS-641988 SH-10-TC CTRP1 0.2890 37.0000
BMS-641988 HSC-2 CTRP1 0.2890 37.0000
BMS-641988 SCC-9 CTRP1 0.2891 37.0000
BMS-641988 5637 CTRP1 0.2890 37.0000
BMS-641988 HT-1376 CTRP1 0.2890 37.0000
BMS-641988 KMBC-2 CTRP1 0.2890 37.0000
BMS-641988 RT-4 CTRP1 0.2890 37.0000
BMS-641988 UM-UC-3 CTRP1 0.2890 37.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.