Drug : 3-Chloro-L-Alanine

CTRP1 Name : 3-chloro-L-alanine

Dataset : All
Synonyms :
Targets : GPT
Pathways : inhibitor of alanine transaminase (ALT1)

Information Cards

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Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
3-chloro-L-alanine U2OS CTRP1 0.0163 2.0833
3-chloro-L-alanine MCF-7 CTRP1 0.0163 2.0833
3-chloro-L-alanine GAMG CTRP1 0.2603 33.3330
3-chloro-L-alanine LN-229 CTRP1 0.0163 2.0833
3-chloro-L-alanine SF295 CTRP1 0.2603 33.3330
3-chloro-L-alanine HEC-108 CTRP1 0.2603 33.3330
3-chloro-L-alanine HEC-151 CTRP1 0.0163 2.0833
3-chloro-L-alanine HEC-251 CTRP1 0.2603 33.3330
3-chloro-L-alanine HEC-265 CTRP1 0.2603 33.3330
3-chloro-L-alanine HEC-59 CTRP1 0.2603 33.3330
3-chloro-L-alanine HEC-6 CTRP1 0.2603 33.3330
3-chloro-L-alanine ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
3-chloro-L-alanine JHUEM-2 CTRP1 0.0163 2.0833
3-chloro-L-alanine KLE CTRP1 0.2603 33.3330
3-chloro-L-alanine MFE-319 CTRP1 0.2603 33.3330
3-chloro-L-alanine SNG-M CTRP1 0.2603 33.3330
3-chloro-L-alanine AMO1 CTRP1 0.0163 2.0833
3-chloro-L-alanine BL-70 CTRP1 0.2603 33.3330
3-chloro-L-alanine EJM CTRP1 0.0163 2.0833
3-chloro-L-alanine GDM-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine HT CTRP1 0.2603 33.3330
3-chloro-L-alanine KMS-11 CTRP1 0.0163 2.0833
3-chloro-L-alanine KU812 CTRP1 0.2603 33.3330
3-chloro-L-alanine LP-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine MC116 CTRP1 0.2603 33.3330
3-chloro-L-alanine MOLM-16 CTRP1 0.0163 2.0833
3-chloro-L-alanine NOMO-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine NU-DUL-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine OCI-AML-3 CTRP1 0.0163 2.0833
3-chloro-L-alanine OCI-LY10 CTRP1 0.0163 2.0833
3-chloro-L-alanine P3HR-1 CTRP1 0.2603 33.3330
3-chloro-L-alanine PL21 CTRP1 0.0163 2.0833
3-chloro-L-alanine RPMI-8226 CTRP1 0.0163 2.0833
3-chloro-L-alanine SKM-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine SU-DHL-4 CTRP1 0.0163 2.0833
3-chloro-L-alanine SU-DHL-5 CTRP1 0.0163 2.0833
3-chloro-L-alanine THP-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine U-937 CTRP1 0.0163 2.0833
3-chloro-L-alanine WSU-DLCL2 CTRP1 0.0163 2.0833
3-chloro-L-alanine RCC10RGB CTRP1 0.0163 2.0833
3-chloro-L-alanine VMRC-RCW CTRP1 0.2603 33.3330
3-chloro-L-alanine C2BBE1 CTRP1 0.2603 33.3330
3-chloro-L-alanine CL-34 CTRP1 0.0163 2.0833
3-chloro-L-alanine CL-40 CTRP1 0.0163 2.0833
3-chloro-L-alanine COLO205 CTRP1 0.2603 33.3330
3-chloro-L-alanine COLO320 CTRP1 0.0163 2.0833
3-chloro-L-alanine COLO678 CTRP1 0.0163 2.0833
3-chloro-L-alanine CW-2 CTRP1 0.0163 2.0833
3-chloro-L-alanine DLD-1 CTRP1 0.2603 33.3330
3-chloro-L-alanine GP2D CTRP1 0.2603 33.3330
3-chloro-L-alanine HCT116 CTRP1 0.0163 2.0833
3-chloro-L-alanine HCT8 CTRP1 0.0163 2.0833
3-chloro-L-alanine HT115 CTRP1 0.0163 2.0833
3-chloro-L-alanine HT-29 CTRP1 0.0163 2.0833
3-chloro-L-alanine HT-55 CTRP1 0.0163 2.0833
3-chloro-L-alanine KM12 CTRP1 0.0163 2.0833
3-chloro-L-alanine LOVO CTRP1 0.0163 2.0833
3-chloro-L-alanine LS123 CTRP1 0.0163 2.0833
3-chloro-L-alanine LS180 CTRP1 0.0163 2.0833
3-chloro-L-alanine LS411N CTRP1 0.2603 33.3330
3-chloro-L-alanine LS513 CTRP1 0.2603 33.3330
3-chloro-L-alanine MDST8 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H508 CTRP1 0.0163 2.0833
3-chloro-L-alanine RCM-1[HUMANESC] CTRP1 0.0163 2.0833
3-chloro-L-alanine RKO CTRP1 0.0163 2.0833
3-chloro-L-alanine SK-CO-1 CTRP1 0.2603 33.3330
3-chloro-L-alanine SNU-1040 CTRP1 0.0163 2.0833
3-chloro-L-alanine SNU-175 CTRP1 0.0163 2.0833
3-chloro-L-alanine SNU-61 CTRP1 0.0163 2.0833
3-chloro-L-alanine SNU-81 CTRP1 0.0163 2.0833
3-chloro-L-alanine SNU-C2A CTRP1 0.2603 33.3330
3-chloro-L-alanine SNU-C4 CTRP1 0.0163 2.0833
3-chloro-L-alanine SNU-C5 CTRP1 0.0163 2.0833
3-chloro-L-alanine SW403 CTRP1 0.2603 33.3330
3-chloro-L-alanine SW48 CTRP1 0.2603 33.3330
3-chloro-L-alanine SW480 CTRP1 0.0163 2.0833
3-chloro-L-alanine SW620 CTRP1 0.0163 2.0833
3-chloro-L-alanine SW948 CTRP1 0.0163 2.0833
3-chloro-L-alanine HEP-G2 CTRP1 0.0163 2.0833
3-chloro-L-alanine JHH-6 CTRP1 0.2603 33.3330
3-chloro-L-alanine SNU-398 CTRP1 0.0163 2.0833
3-chloro-L-alanine SNU-449 CTRP1 0.2603 33.3330
3-chloro-L-alanine A-549 CTRP1 0.2603 33.3330
3-chloro-L-alanine BEN CTRP1 0.2603 33.3330
3-chloro-L-alanine CAL-12T CTRP1 0.0163 2.0833
3-chloro-L-alanine CALU-3 CTRP1 0.2603 33.3330
3-chloro-L-alanine CALU-6 CTRP1 0.2603 33.3330
3-chloro-L-alanine CHAGO-K-1 CTRP1 0.2603 33.3330
3-chloro-L-alanine COLO668 CTRP1 0.2603 33.3330
3-chloro-L-alanine COLO699 CTRP1 0.0163 2.0833
3-chloro-L-alanine COR-L23 CTRP1 0.0163 2.0833
3-chloro-L-alanine COR-L279 CTRP1 0.2603 33.3330
3-chloro-L-alanine COR-L51 CTRP1 0.0163 2.0833
3-chloro-L-alanine COR-L88 CTRP1 0.2603 33.3330
3-chloro-L-alanine DMS273 CTRP1 0.2603 33.3330
3-chloro-L-alanine DV-90 CTRP1 0.2603 33.3330
3-chloro-L-alanine EBC-1 CTRP1 0.2603 33.3330
3-chloro-L-alanine EPLC-272H CTRP1 0.2603 33.3330
3-chloro-L-alanine HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
3-chloro-L-alanine HCC1195 CTRP1 0.0163 2.0833
3-chloro-L-alanine HCC1359 CTRP1 0.0163 2.0833
3-chloro-L-alanine HCC15 CTRP1 0.0163 2.0833
3-chloro-L-alanine HCC1833 CTRP1 0.0163 2.0833
3-chloro-L-alanine HCC2108 CTRP1 0.0163 2.0833
3-chloro-L-alanine HCC2935 CTRP1 0.0163 2.0833
3-chloro-L-alanine HCC33 CTRP1 0.2603 33.3330
3-chloro-L-alanine HCC4006 CTRP1 0.0163 2.0833
3-chloro-L-alanine HCC44 CTRP1 0.2603 33.3330
3-chloro-L-alanine HCC78 CTRP1 0.2603 33.3330
3-chloro-L-alanine HCC827 CTRP1 0.0163 2.0833
3-chloro-L-alanine KNS-62 CTRP1 0.2603 33.3330
3-chloro-L-alanine LC-1-SQ-SF CTRP1 0.2603 33.3330
3-chloro-L-alanine LCLC-103H CTRP1 0.2603 33.3330
3-chloro-L-alanine LCLC-97TM1 CTRP1 0.2603 33.3330
3-chloro-L-alanine LU-65 CTRP1 0.2603 33.3330
3-chloro-L-alanine LU-99 CTRP1 0.2603 33.3330
3-chloro-L-alanine LXF289 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1048 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1105 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H1299 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1355 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1373 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1435 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1437 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1568 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1573 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1666 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1694 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H1755 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H1781 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H1792 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1793 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1836 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H1876 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H1915 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1930 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1944 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H1963 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H1975 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H2009 CTRP1 0.0163 33.3330
3-chloro-L-alanine NCI-H2023 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2029 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H2030 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2073 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2081 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2110 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2122 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2126 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H2141 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2172 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2286 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H23 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H2342 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H2405 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H3255 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H358 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H441 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H460 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H522 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H596 CTRP1 0.0163 2.0833
3-chloro-L-alanine NCI-H650 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H661 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H727 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H810 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H82 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H841 CTRP1 0.0163 2.0833
3-chloro-L-alanine RERF-LC-KJ CTRP1 0.2603 33.3330
3-chloro-L-alanine SCLC-21H CTRP1 0.0163 2.0833
3-chloro-L-alanine SHP-77 CTRP1 0.2603 33.3330
3-chloro-L-alanine SK-LU-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine SQ-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine T3M-10 CTRP1 0.0163 2.0833
3-chloro-L-alanine VMRC-LCD CTRP1 0.2603 33.3330
3-chloro-L-alanine KYSE-140 CTRP1 0.2603 33.3330
3-chloro-L-alanine KYSE-410 CTRP1 0.2603 33.3330
3-chloro-L-alanine KYSE-450 CTRP1 0.2603 33.3330
3-chloro-L-alanine A2780 CTRP1 0.0163 2.0833
3-chloro-L-alanine CAOV-3 CTRP1 0.0163 2.0833
3-chloro-L-alanine COV318 CTRP1 0.2603 33.3330
3-chloro-L-alanine COV362 CTRP1 0.0163 2.0833
3-chloro-L-alanine COV434 CTRP1 0.0163 2.0833
3-chloro-L-alanine COV644 CTRP1 0.0163 2.0833
3-chloro-L-alanine EFO-21 CTRP1 0.2603 33.3330
3-chloro-L-alanine EFO-27 CTRP1 0.0163 2.0833
3-chloro-L-alanine HEYA8 CTRP1 0.2603 33.3330
3-chloro-L-alanine IGROV-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine JHOC-5 CTRP1 0.0163 2.0833
3-chloro-L-alanine JHOM-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine JHOS-4 CTRP1 0.2603 33.3330
3-chloro-L-alanine OAW42 CTRP1 0.0163 2.0833
3-chloro-L-alanine OV7 CTRP1 0.0163 2.0833
3-chloro-L-alanine OV-90 CTRP1 0.0163 2.0833
3-chloro-L-alanine OVCAR-4 CTRP1 0.0163 2.0833
3-chloro-L-alanine OVCAR-8 CTRP1 0.0163 2.0833
3-chloro-L-alanine OVK18 CTRP1 0.0163 2.0833
3-chloro-L-alanine OVKATE CTRP1 0.0163 2.0833
3-chloro-L-alanine OVMANA CTRP1 0.2603 33.3330
3-chloro-L-alanine RKN CTRP1 0.0163 2.0833
3-chloro-L-alanine RMG-I CTRP1 0.0163 2.0833
3-chloro-L-alanine RMUG-S CTRP1 0.0163 2.0833
3-chloro-L-alanine SK-OV-3 CTRP1 0.2603 33.3330
3-chloro-L-alanine SNU-840 CTRP1 0.0163 2.0833
3-chloro-L-alanine TYK-NU CTRP1 0.0163 2.0833
3-chloro-L-alanine CAPAN-2 CTRP1 0.2603 33.3330
3-chloro-L-alanine CFPAC-1 CTRP1 0.2603 33.3330
3-chloro-L-alanine HPAC CTRP1 0.2603 33.3330
3-chloro-L-alanine HUP-T4 CTRP1 0.2603 33.3330
3-chloro-L-alanine KP-3 CTRP1 0.2603 33.3330
3-chloro-L-alanine PANC03.27 CTRP1 0.2603 33.3330
3-chloro-L-alanine PANC10.05 CTRP1 0.2603 33.3330
3-chloro-L-alanine PATU8902 CTRP1 0.2603 33.3330
3-chloro-L-alanine QGP-1 CTRP1 0.2603 33.3330
3-chloro-L-alanine SUIT-2 CTRP1 0.2603 33.3330
3-chloro-L-alanine MSTO-211H CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H2052 CTRP1 0.2603 33.3330
3-chloro-L-alanine NCI-H28 CTRP1 0.2603 33.3330
3-chloro-L-alanine MIAPACA-3 CTRP1 0.2603 33.3330
3-chloro-L-alanine A-375 CTRP1 0.0163 2.0833
3-chloro-L-alanine COLO741 CTRP1 0.2603 33.3330
3-chloro-L-alanine G-361 CTRP1 0.2603 33.3330
3-chloro-L-alanine HS852.T CTRP1 0.2603 33.3330
3-chloro-L-alanine HS936.T CTRP1 0.2603 33.3330
3-chloro-L-alanine HS944.T CTRP1 0.2603 33.3330
3-chloro-L-alanine SK-MEL-1 CTRP1 0.0163 2.0833
3-chloro-L-alanine SK-MEL-28 CTRP1 0.0163 2.0833
3-chloro-L-alanine SK-MEL-5 CTRP1 0.0163 2.0833
3-chloro-L-alanine G-401 CTRP1 0.2603 33.3330
3-chloro-L-alanine HT-1080 CTRP1 0.0163 2.0833
3-chloro-L-alanine AGS CTRP1 0.0163 2.0833
3-chloro-L-alanine FU97 CTRP1 0.2603 33.3330
3-chloro-L-alanine KE-97 CTRP1 0.2603 33.3330
3-chloro-L-alanine MKN7 CTRP1 0.2603 33.3330
3-chloro-L-alanine MKN74 CTRP1 0.2603 33.3330
3-chloro-L-alanine NUGC-4 CTRP1 0.2603 33.3330
3-chloro-L-alanine SH-10-TC CTRP1 0.2603 33.3330
3-chloro-L-alanine HSC-2 CTRP1 0.2603 33.3330
3-chloro-L-alanine SCC-9 CTRP1 0.0163 2.0833
3-chloro-L-alanine 5637 CTRP1 0.2603 33.3330
3-chloro-L-alanine HT-1376 CTRP1 0.2603 33.3330
3-chloro-L-alanine KMBC-2 CTRP1 0.2603 33.3330
3-chloro-L-alanine RT-4 CTRP1 0.2603 33.3330
3-chloro-L-alanine UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.