Drug : Rosiglitazone

CTRP1 Name : rosiglitazone

Dataset : All
Synonyms :
Targets : PPARG
Pathways : activator of PPAR?

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
rosiglitazone MCF-7 CTRP1 2.0833 266.6700
rosiglitazone GAMG CTRP1 0.2603 33.3330
rosiglitazone LN-229 CTRP1 2.0833 266.6700
rosiglitazone SF295 CTRP1 0.2603 33.3330
rosiglitazone HEC-108 CTRP1 0.2603 33.3330
rosiglitazone HEC-151 CTRP1 2.0833 266.6700
rosiglitazone HEC-251 CTRP1 0.2603 33.3330
rosiglitazone HEC-265 CTRP1 0.2603 33.3330
rosiglitazone HEC-59 CTRP1 0.2603 33.3330
rosiglitazone HEC-6 CTRP1 0.2603 33.3330
rosiglitazone ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
rosiglitazone JHUEM-2 CTRP1 2.0833 266.6700
rosiglitazone KLE CTRP1 0.2603 33.3330
rosiglitazone MFE-319 CTRP1 0.2603 33.3330
rosiglitazone SNG-M CTRP1 0.2603 33.3330
rosiglitazone AMO1 CTRP1 2.0833 266.6700
rosiglitazone BL-70 CTRP1 0.2603 33.3330
rosiglitazone EJM CTRP1 2.0833 266.6700
rosiglitazone GDM-1 CTRP1 2.0833 266.6700
rosiglitazone HT CTRP1 0.2603 33.3330
rosiglitazone KMS-11 CTRP1 2.0833 266.6700
rosiglitazone KU812 CTRP1 0.2603 33.3330
rosiglitazone LP-1 CTRP1 2.0833 266.6700
rosiglitazone MC116 CTRP1 0.2603 33.3330
rosiglitazone MOLM-16 CTRP1 2.0833 266.6700
rosiglitazone NOMO-1 CTRP1 2.0833 266.6700
rosiglitazone NU-DUL-1 CTRP1 2.0833 266.6700
rosiglitazone OCI-AML-3 CTRP1 2.0833 266.6700
rosiglitazone OCI-LY10 CTRP1 2.0833 266.6700
rosiglitazone P3HR-1 CTRP1 0.2603 33.3330
rosiglitazone PL21 CTRP1 2.0833 266.6700
rosiglitazone RPMI-8226 CTRP1 2.0833 266.6700
rosiglitazone SKM-1 CTRP1 2.0833 266.6700
rosiglitazone SU-DHL-4 CTRP1 2.0833 266.6700
rosiglitazone SU-DHL-5 CTRP1 2.0833 266.6700
rosiglitazone THP-1 CTRP1 2.0833 266.6700
rosiglitazone U-937 CTRP1 2.0833 266.6700
rosiglitazone WSU-DLCL2 CTRP1 2.0833 266.6700
rosiglitazone RCC10RGB CTRP1 2.0833 266.6700
rosiglitazone VMRC-RCW CTRP1 0.2603 33.3330
rosiglitazone C2BBE1 CTRP1 0.2603 33.3330
rosiglitazone CL-34 CTRP1 2.0833 266.6700
rosiglitazone CL-40 CTRP1 2.0833 266.6700
rosiglitazone COLO205 CTRP1 0.2603 33.3330
rosiglitazone COLO320 CTRP1 2.0833 266.6700
rosiglitazone COLO678 CTRP1 2.0833 266.6700
rosiglitazone CW-2 CTRP1 2.0833 266.6700
rosiglitazone DLD-1 CTRP1 0.2603 33.3330
rosiglitazone GP2D CTRP1 0.2603 33.3330
rosiglitazone HCT116 CTRP1 2.0833 266.6700
rosiglitazone HCT8 CTRP1 2.0833 266.6700
rosiglitazone HT115 CTRP1 2.0833 266.6700
rosiglitazone HT-29 CTRP1 2.0833 266.6700
rosiglitazone HT-55 CTRP1 2.0833 266.6700
rosiglitazone KM12 CTRP1 2.0833 266.6700
rosiglitazone LOVO CTRP1 2.0833 266.6700
rosiglitazone LS123 CTRP1 2.0833 266.6700
rosiglitazone LS180 CTRP1 2.0833 266.6700
rosiglitazone LS411N CTRP1 0.2603 33.3330
rosiglitazone LS513 CTRP1 0.2603 33.3330
rosiglitazone MDST8 CTRP1 2.0833 266.6700
rosiglitazone NCI-H508 CTRP1 2.0833 266.6700
rosiglitazone RCM-1[HUMANESC] CTRP1 2.0833 266.6700
rosiglitazone RKO CTRP1 2.0833 266.6700
rosiglitazone SK-CO-1 CTRP1 0.2603 33.3330
rosiglitazone SNU-1040 CTRP1 2.0833 266.6700
rosiglitazone SNU-175 CTRP1 2.0833 266.6700
rosiglitazone SNU-61 CTRP1 2.0833 266.6700
rosiglitazone SNU-81 CTRP1 2.0833 266.6700
rosiglitazone SNU-C2A CTRP1 0.2603 33.3330
rosiglitazone SNU-C4 CTRP1 2.0833 266.6700
rosiglitazone SNU-C5 CTRP1 2.0833 266.6700
rosiglitazone SW403 CTRP1 0.2603 33.3330
rosiglitazone SW48 CTRP1 0.2603 33.3330
rosiglitazone SW480 CTRP1 2.0833 266.6700
rosiglitazone SW620 CTRP1 2.0833 266.6700
rosiglitazone SW948 CTRP1 2.0833 266.6700
rosiglitazone HEP-G2 CTRP1 2.0833 266.6700
rosiglitazone JHH-6 CTRP1 0.2603 33.3330
rosiglitazone SNU-398 CTRP1 2.0833 266.6700
rosiglitazone SNU-449 CTRP1 0.2603 33.3330
rosiglitazone A-549 CTRP1 0.2603 33.3330
rosiglitazone BEN CTRP1 0.2603 33.3330
rosiglitazone CAL-12T CTRP1 2.0833 266.6700
rosiglitazone CALU-3 CTRP1 0.2603 33.3330
rosiglitazone CALU-6 CTRP1 0.2603 33.3330
rosiglitazone CHAGO-K-1 CTRP1 0.2603 33.3330
rosiglitazone COLO668 CTRP1 0.2603 33.3330
rosiglitazone COLO699 CTRP1 2.0833 266.6700
rosiglitazone COR-L23 CTRP1 2.0833 266.6700
rosiglitazone COR-L279 CTRP1 0.2603 33.3330
rosiglitazone COR-L51 CTRP1 2.0833 266.6700
rosiglitazone COR-L88 CTRP1 0.2603 33.3330
rosiglitazone DMS273 CTRP1 0.2603 33.3330
rosiglitazone DV-90 CTRP1 0.2603 33.3330
rosiglitazone EBC-1 CTRP1 0.2603 33.3330
rosiglitazone EPLC-272H CTRP1 0.2603 33.3330
rosiglitazone HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
rosiglitazone HCC1195 CTRP1 2.0833 266.6700
rosiglitazone HCC1359 CTRP1 2.0833 266.6700
rosiglitazone HCC15 CTRP1 2.0833 266.6700
rosiglitazone HCC1833 CTRP1 2.0833 266.6700
rosiglitazone HCC2108 CTRP1 2.0833 266.6700
rosiglitazone HCC2935 CTRP1 2.0833 266.6700
rosiglitazone HCC33 CTRP1 0.2603 33.3330
rosiglitazone HCC4006 CTRP1 2.0833 266.6700
rosiglitazone HCC44 CTRP1 0.2603 33.3330
rosiglitazone HCC78 CTRP1 0.2603 33.3330
rosiglitazone HCC827 CTRP1 2.0833 266.6700
rosiglitazone KNS-62 CTRP1 0.2603 33.3330
rosiglitazone LC-1-SQ-SF CTRP1 0.2603 33.3330
rosiglitazone LCLC-103H CTRP1 0.2603 33.3330
rosiglitazone LCLC-97TM1 CTRP1 0.2603 33.3330
rosiglitazone LU-65 CTRP1 0.2603 33.3330
rosiglitazone LU-99 CTRP1 0.2603 33.3330
rosiglitazone LXF289 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1048 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1105 CTRP1 2.0833 266.6700
rosiglitazone NCI-H1299 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1355 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1373 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1435 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1437 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1568 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1573 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1666 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1694 CTRP1 2.0833 266.6700
rosiglitazone NCI-H1755 CTRP1 2.0833 266.6700
rosiglitazone NCI-H1781 CTRP1 2.0833 266.6700
rosiglitazone NCI-H1792 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1793 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1836 CTRP1 2.0833 266.6700
rosiglitazone NCI-H1876 CTRP1 2.0833 266.6700
rosiglitazone NCI-H1915 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1930 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1944 CTRP1 0.2603 33.3330
rosiglitazone NCI-H1963 CTRP1 2.0833 266.6700
rosiglitazone NCI-H1975 CTRP1 0.2603 33.3330
rosiglitazone NCI-H2009 CTRP1 0.2603 33.3330
rosiglitazone NCI-H2023 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2029 CTRP1 0.2603 33.3330
rosiglitazone NCI-H2030 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2073 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2081 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2110 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2122 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2126 CTRP1 0.2603 33.3330
rosiglitazone NCI-H2141 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2172 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2286 CTRP1 0.2603 33.3330
rosiglitazone NCI-H23 CTRP1 0.2603 33.3330
rosiglitazone NCI-H2342 CTRP1 2.0833 266.6700
rosiglitazone NCI-H2405 CTRP1 0.2603 33.3330
rosiglitazone NCI-H3255 CTRP1 2.0833 266.6700
rosiglitazone NCI-H358 CTRP1 0.2603 33.3330
rosiglitazone NCI-H441 CTRP1 2.0833 266.6700
rosiglitazone NCI-H460 CTRP1 2.0833 266.6700
rosiglitazone NCI-H522 CTRP1 0.2603 33.3330
rosiglitazone NCI-H596 CTRP1 2.0833 266.6700
rosiglitazone NCI-H650 CTRP1 0.2603 33.3330
rosiglitazone NCI-H661 CTRP1 0.2603 33.3330
rosiglitazone NCI-H727 CTRP1 0.2603 33.3330
rosiglitazone NCI-H810 CTRP1 0.2603 33.3330
rosiglitazone NCI-H82 CTRP1 0.2603 33.3330
rosiglitazone NCI-H841 CTRP1 2.0833 266.6700
rosiglitazone RERF-LC-KJ CTRP1 0.2603 33.3330
rosiglitazone SCLC-21H CTRP1 2.0833 266.6700
rosiglitazone SHP-77 CTRP1 0.2603 33.3330
rosiglitazone SK-LU-1 CTRP1 2.0833 266.6700
rosiglitazone SQ-1 CTRP1 2.0833 266.6700
rosiglitazone T3M-10 CTRP1 2.0833 266.6700
rosiglitazone VMRC-LCD CTRP1 0.2603 33.3330
rosiglitazone KYSE-140 CTRP1 0.2603 33.3330
rosiglitazone KYSE-410 CTRP1 0.2603 33.3330
rosiglitazone KYSE-450 CTRP1 0.2603 33.3330
rosiglitazone A2780 CTRP1 2.0833 266.6700
rosiglitazone CAOV-3 CTRP1 2.0833 266.6700
rosiglitazone COV318 CTRP1 0.2603 33.3330
rosiglitazone COV362 CTRP1 2.0833 266.6700
rosiglitazone COV434 CTRP1 2.0833 266.6700
rosiglitazone COV644 CTRP1 2.0833 266.6700
rosiglitazone EFO-21 CTRP1 0.2603 33.3330
rosiglitazone EFO-27 CTRP1 2.0833 266.6700
rosiglitazone HEYA8 CTRP1 0.2603 33.3330
rosiglitazone IGROV-1 CTRP1 2.0833 266.6700
rosiglitazone JHOC-5 CTRP1 2.0833 266.6700
rosiglitazone JHOM-1 CTRP1 2.0833 266.6700
rosiglitazone JHOS-4 CTRP1 0.2603 33.3330
rosiglitazone OAW42 CTRP1 2.0833 266.6700
rosiglitazone OV7 CTRP1 2.0833 266.6700
rosiglitazone OV-90 CTRP1 2.0833 266.6700
rosiglitazone OVCAR-4 CTRP1 2.0833 266.6700
rosiglitazone OVCAR-8 CTRP1 2.0833 266.6700
rosiglitazone OVK18 CTRP1 2.0833 266.6700
rosiglitazone OVKATE CTRP1 2.0833 266.6700
rosiglitazone OVMANA CTRP1 0.2603 33.3330
rosiglitazone RKN CTRP1 2.0833 266.6700
rosiglitazone RMG-I CTRP1 2.0833 266.6700
rosiglitazone RMUG-S CTRP1 2.0833 266.6700
rosiglitazone SK-OV-3 CTRP1 0.2603 33.3330
rosiglitazone SNU-840 CTRP1 2.0833 266.6700
rosiglitazone TYK-NU CTRP1 2.0833 266.6700
rosiglitazone CAPAN-2 CTRP1 0.2603 33.3330
rosiglitazone CFPAC-1 CTRP1 0.2603 33.3330
rosiglitazone HPAC CTRP1 0.2603 33.3330
rosiglitazone HUP-T4 CTRP1 0.2603 33.3330
rosiglitazone KP-3 CTRP1 0.2603 33.3330
rosiglitazone PANC03.27 CTRP1 0.2603 33.3330
rosiglitazone PANC10.05 CTRP1 0.2603 33.3330
rosiglitazone PATU8902 CTRP1 0.2603 33.3330
rosiglitazone QGP-1 CTRP1 0.2603 33.3330
rosiglitazone SUIT-2 CTRP1 0.2603 33.3330
rosiglitazone MSTO-211H CTRP1 0.2603 33.3330
rosiglitazone NCI-H2052 CTRP1 0.2603 33.3330
rosiglitazone NCI-H28 CTRP1 0.2603 33.3330
rosiglitazone MIAPACA-3 CTRP1 0.2603 33.3330
rosiglitazone A-375 CTRP1 2.0833 266.6700
rosiglitazone COLO741 CTRP1 0.2603 33.3330
rosiglitazone G-361 CTRP1 0.2603 33.3330
rosiglitazone HS852.T CTRP1 0.2603 33.3330
rosiglitazone HS936.T CTRP1 0.2603 33.3330
rosiglitazone HS944.T CTRP1 0.2603 33.3330
rosiglitazone SK-MEL-1 CTRP1 2.0833 266.6700
rosiglitazone SK-MEL-28 CTRP1 2.0833 266.6700
rosiglitazone SK-MEL-5 CTRP1 2.0833 266.6700
rosiglitazone G-401 CTRP1 0.2603 33.3330
rosiglitazone HT-1080 CTRP1 2.0833 266.6700
rosiglitazone AGS CTRP1 2.0833 266.6700
rosiglitazone FU97 CTRP1 0.2603 33.3330
rosiglitazone KE-97 CTRP1 0.2603 33.3330
rosiglitazone MKN7 CTRP1 0.2603 33.3330
rosiglitazone MKN74 CTRP1 0.2603 33.3330
rosiglitazone NUGC-4 CTRP1 0.2603 33.3330
rosiglitazone SH-10-TC CTRP1 0.2603 33.3330
rosiglitazone HSC-2 CTRP1 0.2603 33.3330
rosiglitazone SCC-9 CTRP1 2.0833 266.6700
rosiglitazone 5637 CTRP1 0.2603 33.3330
rosiglitazone HT-1376 CTRP1 0.2603 33.3330
rosiglitazone KMBC-2 CTRP1 0.2603 33.3330
rosiglitazone RT-4 CTRP1 0.2603 33.3330
rosiglitazone UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.