Drug : Dl-Tboa

CTRP1 Name : DL-TBOA

Dataset : All
Synonyms :
Targets : SLC1A3;SLC1A2;SLC1A1;SLC1A6;SLC1A7
Pathways : inhibitor of excitatory amino acid transporters (EAAT1-5)

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
DL-TBOA U2OS CTRP1 4.1667 533.3300
DL-TBOA MCF-7 CTRP1 4.1667 533.3300
DL-TBOA GAMG CTRP1 0.2603 33.3330
DL-TBOA LN-229 CTRP1 4.1667 533.3300
DL-TBOA SF295 CTRP1 0.2603 33.3330
DL-TBOA HEC-108 CTRP1 0.2603 33.3330
DL-TBOA HEC-151 CTRP1 4.1667 533.3300
DL-TBOA HEC-251 CTRP1 0.2603 33.3330
DL-TBOA HEC-265 CTRP1 0.2603 33.3330
DL-TBOA HEC-59 CTRP1 0.2603 33.3330
DL-TBOA HEC-6 CTRP1 0.2603 33.3330
DL-TBOA ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
DL-TBOA JHUEM-2 CTRP1 4.1667 533.3300
DL-TBOA KLE CTRP1 0.2603 33.3330
DL-TBOA MFE-319 CTRP1 0.2603 33.3330
DL-TBOA SNG-M CTRP1 0.2603 33.3330
DL-TBOA AMO1 CTRP1 4.1667 533.3300
DL-TBOA BL-70 CTRP1 0.2603 33.3330
DL-TBOA EJM CTRP1 4.1667 533.3300
DL-TBOA GDM-1 CTRP1 4.1667 533.3300
DL-TBOA HT CTRP1 0.2603 33.3330
DL-TBOA KMS-11 CTRP1 4.1667 533.3300
DL-TBOA KU812 CTRP1 0.2603 33.3330
DL-TBOA LP-1 CTRP1 4.1667 533.3300
DL-TBOA MC116 CTRP1 0.2603 33.3330
DL-TBOA MOLM-16 CTRP1 4.1667 533.3300
DL-TBOA NOMO-1 CTRP1 4.1667 533.3300
DL-TBOA NU-DUL-1 CTRP1 4.1667 533.3300
DL-TBOA OCI-AML-3 CTRP1 4.1667 533.3300
DL-TBOA OCI-LY10 CTRP1 4.1667 533.3300
DL-TBOA P3HR-1 CTRP1 0.2603 33.3330
DL-TBOA PL21 CTRP1 4.1667 533.3300
DL-TBOA RPMI-8226 CTRP1 4.1667 533.3300
DL-TBOA SKM-1 CTRP1 4.1667 533.3300
DL-TBOA SU-DHL-4 CTRP1 4.1667 533.3300
DL-TBOA SU-DHL-5 CTRP1 4.1667 533.3300
DL-TBOA THP-1 CTRP1 4.1667 533.3300
DL-TBOA U-937 CTRP1 4.1667 533.3300
DL-TBOA WSU-DLCL2 CTRP1 4.1667 533.3300
DL-TBOA RCC10RGB CTRP1 4.1667 533.3300
DL-TBOA VMRC-RCW CTRP1 0.2603 33.3330
DL-TBOA C2BBE1 CTRP1 0.2603 33.3330
DL-TBOA CL-34 CTRP1 4.1667 533.3300
DL-TBOA CL-40 CTRP1 4.1667 533.3300
DL-TBOA COLO205 CTRP1 0.2603 33.3330
DL-TBOA COLO320 CTRP1 4.1667 533.3300
DL-TBOA COLO678 CTRP1 4.1667 533.3300
DL-TBOA CW-2 CTRP1 4.1667 533.3300
DL-TBOA DLD-1 CTRP1 0.2603 33.3330
DL-TBOA GP2D CTRP1 0.2603 33.3330
DL-TBOA HCT116 CTRP1 4.1667 533.3300
DL-TBOA HCT8 CTRP1 4.1667 533.3300
DL-TBOA HT115 CTRP1 4.1667 533.3300
DL-TBOA HT-29 CTRP1 4.1667 533.3300
DL-TBOA HT-55 CTRP1 4.1667 533.3300
DL-TBOA KM12 CTRP1 4.1667 533.3300
DL-TBOA LOVO CTRP1 4.1667 533.3300
DL-TBOA LS123 CTRP1 4.1667 533.3300
DL-TBOA LS180 CTRP1 4.1667 533.3300
DL-TBOA LS411N CTRP1 0.2603 33.3330
DL-TBOA LS513 CTRP1 0.2603 33.3330
DL-TBOA MDST8 CTRP1 4.1667 533.3300
DL-TBOA NCI-H508 CTRP1 4.1667 533.3300
DL-TBOA RCM-1[HUMANESC] CTRP1 4.1667 533.3300
DL-TBOA RKO CTRP1 4.1667 533.3300
DL-TBOA SK-CO-1 CTRP1 0.2603 33.3330
DL-TBOA SNU-1040 CTRP1 4.1667 533.3300
DL-TBOA SNU-175 CTRP1 4.1667 533.3300
DL-TBOA SNU-61 CTRP1 4.1667 533.3300
DL-TBOA SNU-81 CTRP1 4.1667 533.3300
DL-TBOA SNU-C2A CTRP1 0.2603 33.3330
DL-TBOA SNU-C4 CTRP1 4.1667 533.3300
DL-TBOA SNU-C5 CTRP1 4.1667 533.3300
DL-TBOA SW403 CTRP1 0.2603 33.3330
DL-TBOA SW48 CTRP1 0.2603 33.3330
DL-TBOA SW480 CTRP1 4.1667 533.3300
DL-TBOA SW620 CTRP1 4.1667 533.3300
DL-TBOA SW948 CTRP1 4.1667 533.3300
DL-TBOA HEP-G2 CTRP1 4.1667 533.3300
DL-TBOA JHH-6 CTRP1 0.2603 33.3330
DL-TBOA SNU-398 CTRP1 4.1667 533.3300
DL-TBOA SNU-449 CTRP1 0.2603 33.3330
DL-TBOA A-549 CTRP1 0.2603 33.3330
DL-TBOA BEN CTRP1 0.2603 33.3330
DL-TBOA CAL-12T CTRP1 4.1667 533.3300
DL-TBOA CALU-3 CTRP1 0.2603 33.3330
DL-TBOA CALU-6 CTRP1 0.2603 33.3330
DL-TBOA CHAGO-K-1 CTRP1 0.2603 33.3330
DL-TBOA COLO668 CTRP1 0.2603 33.3330
DL-TBOA COLO699 CTRP1 4.1667 533.3300
DL-TBOA COR-L23 CTRP1 4.1667 533.3300
DL-TBOA COR-L279 CTRP1 0.2603 33.3330
DL-TBOA COR-L51 CTRP1 4.1667 533.3300
DL-TBOA COR-L88 CTRP1 0.2603 33.3330
DL-TBOA DMS273 CTRP1 0.2603 33.3330
DL-TBOA DV-90 CTRP1 0.2603 33.3330
DL-TBOA EBC-1 CTRP1 0.2603 33.3330
DL-TBOA EPLC-272H CTRP1 0.2603 33.3330
DL-TBOA HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
DL-TBOA HCC1195 CTRP1 4.1667 533.3300
DL-TBOA HCC1359 CTRP1 4.1667 533.3300
DL-TBOA HCC15 CTRP1 4.1667 533.3300
DL-TBOA HCC1833 CTRP1 4.1667 533.3300
DL-TBOA HCC2108 CTRP1 4.1667 533.3300
DL-TBOA HCC2935 CTRP1 4.1667 533.3300
DL-TBOA HCC33 CTRP1 0.2603 33.3330
DL-TBOA HCC4006 CTRP1 4.1667 533.3300
DL-TBOA HCC44 CTRP1 0.2603 33.3330
DL-TBOA HCC78 CTRP1 0.2603 33.3330
DL-TBOA HCC827 CTRP1 4.1667 533.3300
DL-TBOA KNS-62 CTRP1 0.2603 33.3330
DL-TBOA LC-1-SQ-SF CTRP1 0.2603 33.3330
DL-TBOA LCLC-103H CTRP1 0.2603 33.3330
DL-TBOA LCLC-97TM1 CTRP1 0.2603 33.3330
DL-TBOA LU-65 CTRP1 0.2603 33.3330
DL-TBOA LU-99 CTRP1 0.2603 33.3330
DL-TBOA LXF289 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1048 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1105 CTRP1 4.1667 533.3300
DL-TBOA NCI-H1299 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1355 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1373 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1435 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1437 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1568 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1573 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1666 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1694 CTRP1 4.1667 533.3300
DL-TBOA NCI-H1755 CTRP1 4.1667 533.3300
DL-TBOA NCI-H1781 CTRP1 4.1667 533.3300
DL-TBOA NCI-H1792 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1793 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1836 CTRP1 4.1667 533.3300
DL-TBOA NCI-H1876 CTRP1 4.1667 533.3300
DL-TBOA NCI-H1915 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1930 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1944 CTRP1 0.2603 33.3330
DL-TBOA NCI-H1963 CTRP1 4.1667 533.3300
DL-TBOA NCI-H1975 CTRP1 0.2603 33.3330
DL-TBOA NCI-H2009 CTRP1 0.2603 33.3330
DL-TBOA NCI-H2023 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2029 CTRP1 0.2603 33.3330
DL-TBOA NCI-H2030 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2073 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2081 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2110 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2122 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2126 CTRP1 0.2603 33.3330
DL-TBOA NCI-H2141 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2172 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2286 CTRP1 0.2603 33.3330
DL-TBOA NCI-H23 CTRP1 0.2603 33.3330
DL-TBOA NCI-H2342 CTRP1 4.1667 533.3300
DL-TBOA NCI-H2405 CTRP1 0.2603 33.3330
DL-TBOA NCI-H3255 CTRP1 4.1667 533.3300
DL-TBOA NCI-H358 CTRP1 0.2603 33.3330
DL-TBOA NCI-H441 CTRP1 4.1667 533.3300
DL-TBOA NCI-H460 CTRP1 4.1667 533.3300
DL-TBOA NCI-H522 CTRP1 0.2603 33.3330
DL-TBOA NCI-H596 CTRP1 4.1667 533.3300
DL-TBOA NCI-H650 CTRP1 0.2603 33.3330
DL-TBOA NCI-H661 CTRP1 0.2603 33.3330
DL-TBOA NCI-H727 CTRP1 0.2603 33.3330
DL-TBOA NCI-H810 CTRP1 0.2603 33.3330
DL-TBOA NCI-H82 CTRP1 0.2603 33.3330
DL-TBOA NCI-H841 CTRP1 4.1667 533.3300
DL-TBOA RERF-LC-KJ CTRP1 0.2603 33.3330
DL-TBOA SCLC-21H CTRP1 4.1667 533.3300
DL-TBOA SHP-77 CTRP1 0.2603 33.3330
DL-TBOA SK-LU-1 CTRP1 4.1667 533.3300
DL-TBOA SQ-1 CTRP1 4.1667 533.3300
DL-TBOA T3M-10 CTRP1 4.1667 533.3300
DL-TBOA VMRC-LCD CTRP1 0.2603 33.3330
DL-TBOA KYSE-140 CTRP1 0.2603 33.3330
DL-TBOA KYSE-410 CTRP1 0.2603 33.3330
DL-TBOA KYSE-450 CTRP1 0.2603 33.3330
DL-TBOA A2780 CTRP1 4.1667 533.3300
DL-TBOA CAOV-3 CTRP1 4.1667 533.3300
DL-TBOA COV318 CTRP1 0.2603 33.3330
DL-TBOA COV362 CTRP1 4.1667 533.3300
DL-TBOA COV434 CTRP1 4.1667 533.3300
DL-TBOA COV644 CTRP1 4.1667 533.3300
DL-TBOA EFO-21 CTRP1 0.2603 33.3330
DL-TBOA EFO-27 CTRP1 4.1667 533.3300
DL-TBOA HEYA8 CTRP1 0.2603 33.3330
DL-TBOA IGROV-1 CTRP1 4.1667 533.3300
DL-TBOA JHOC-5 CTRP1 4.1667 533.3300
DL-TBOA JHOM-1 CTRP1 4.1667 533.3300
DL-TBOA JHOS-4 CTRP1 0.2603 33.3330
DL-TBOA OAW42 CTRP1 4.1667 533.3300
DL-TBOA OV7 CTRP1 4.1667 533.3300
DL-TBOA OV-90 CTRP1 4.1667 533.3300
DL-TBOA OVCAR-4 CTRP1 4.1667 533.3300
DL-TBOA OVCAR-8 CTRP1 4.1667 533.3300
DL-TBOA OVK18 CTRP1 4.1667 533.3300
DL-TBOA OVKATE CTRP1 4.1667 533.3300
DL-TBOA OVMANA CTRP1 0.2603 33.3330
DL-TBOA RKN CTRP1 4.1667 533.3300
DL-TBOA RMG-I CTRP1 4.1667 533.3300
DL-TBOA RMUG-S CTRP1 4.1667 533.3300
DL-TBOA SK-OV-3 CTRP1 0.2603 33.3330
DL-TBOA SNU-840 CTRP1 4.1667 533.3300
DL-TBOA TYK-NU CTRP1 4.1667 533.3300
DL-TBOA CAPAN-2 CTRP1 0.2603 33.3330
DL-TBOA CFPAC-1 CTRP1 0.2603 33.3330
DL-TBOA HPAC CTRP1 0.2603 33.3330
DL-TBOA HUP-T4 CTRP1 0.2603 33.3330
DL-TBOA KP-3 CTRP1 0.2603 33.3330
DL-TBOA PANC03.27 CTRP1 0.2603 33.3330
DL-TBOA PANC10.05 CTRP1 0.2603 33.3330
DL-TBOA PATU8902 CTRP1 0.2603 33.3330
DL-TBOA QGP-1 CTRP1 0.2603 33.3330
DL-TBOA SUIT-2 CTRP1 0.2603 33.3330
DL-TBOA MSTO-211H CTRP1 0.2603 33.3330
DL-TBOA NCI-H2052 CTRP1 0.2603 33.3330
DL-TBOA NCI-H28 CTRP1 0.2603 33.3330
DL-TBOA MIAPACA-3 CTRP1 0.2603 33.3330
DL-TBOA A-375 CTRP1 4.1667 533.3300
DL-TBOA COLO741 CTRP1 0.2603 33.3330
DL-TBOA G-361 CTRP1 0.2603 33.3330
DL-TBOA HS852.T CTRP1 0.2603 33.3330
DL-TBOA HS936.T CTRP1 0.2603 33.3330
DL-TBOA HS944.T CTRP1 0.2603 33.3330
DL-TBOA SK-MEL-1 CTRP1 4.1667 533.3300
DL-TBOA SK-MEL-28 CTRP1 4.1667 533.3300
DL-TBOA SK-MEL-5 CTRP1 4.1667 533.3300
DL-TBOA G-401 CTRP1 0.2603 33.3330
DL-TBOA HT-1080 CTRP1 4.1667 533.3300
DL-TBOA AGS CTRP1 4.1667 533.3300
DL-TBOA FU97 CTRP1 0.2603 33.3330
DL-TBOA KE-97 CTRP1 0.2603 33.3330
DL-TBOA MKN7 CTRP1 0.2603 33.3330
DL-TBOA MKN74 CTRP1 0.2603 33.3330
DL-TBOA NUGC-4 CTRP1 0.2603 33.3330
DL-TBOA SH-10-TC CTRP1 0.2603 33.3330
DL-TBOA HSC-2 CTRP1 0.2603 33.3330
DL-TBOA SCC-9 CTRP1 4.1667 533.3300
DL-TBOA 5637 CTRP1 0.2603 33.3330
DL-TBOA HT-1376 CTRP1 0.2603 33.3330
DL-TBOA KMBC-2 CTRP1 0.2603 33.3330
DL-TBOA RT-4 CTRP1 0.2603 33.3330
DL-TBOA UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.