Drug : Ml312

CTRP2 Name : ML312

Dataset : All
Synonyms :
Targets : SCARB1
Pathways : inhibitor of scavenger receptor class B, member 1 (SCARB1)-mediated lipid uptake

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

:


Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
ML312 CAS-1 CTRP2 0.0020 66.0000
ML312 KPL-1 CTRP2 0.0020 66.0000
ML312 MKN1 CTRP2 0.0020 66.0000
ML312 BFTC-909 CTRP2 0.0020 66.0000
ML312 CAL-120 CTRP2 0.0020 66.0000
ML312 CAL-29 CTRP2 0.0020 66.0000
ML312 HUCC-T1 CTRP2 0.0020 66.0000
ML312 NMC-G1 CTRP2 0.0020 66.0000
ML312 RPMI-7951 CTRP2 0.0020 66.0000
ML312 253J CTRP2 0.0020 66.0000
ML312 ALL-SIL CTRP2 0.0020 66.0000
ML312 HDQ-P1 CTRP2 0.0020 66.0000
ML312 SNU-489 CTRP2 0.0020 66.0000
ML312 SNU-626 CTRP2 0.0020 66.0000
ML312 SNU-738 CTRP2 0.0020 66.0000
ML312 SNU-878 CTRP2 0.0020 66.0000
ML312 TUHR4TKB CTRP2 0.0020 66.0000
ML312 ACC-MESO-1 CTRP2 0.0020 66.0000
ML312 B-CPAP CTRP2 0.0020 66.0000
ML312 CGTH-W-1 CTRP2 0.0020 66.0000
ML312 COLO680N CTRP2 0.0020 66.0000
ML312 ECC12 CTRP2 0.0020 66.0000
ML312 HCC95 CTRP2 0.0020 66.0000
ML312 JMSU-1 CTRP2 0.0020 66.0000
ML312 RH41 CTRP2 0.0020 66.0000
ML312 WSU-DLCL2 CTRP2 0.0020 66.0000
ML312 23132-87 CTRP2 0.0020 66.0000
ML312 8305C CTRP2 0.0020 66.0000
ML312 BHY CTRP2 0.0020 66.0000
ML312 GSU CTRP2 0.0020 66.0000
ML312 JIMT-1 CTRP2 0.0020 66.0000
ML312 KMRC-20 CTRP2 0.0020 66.0000
ML312 OUMS-23 CTRP2 0.0020 66.0000
ML312 SNU-1076 CTRP2 0.0020 66.0000
ML312 SNU-1196 CTRP2 0.0020 66.0000
ML312 SNU-8 CTRP2 0.0020 66.0000
ML312 A-375 CTRP2 0.0020 66.0000
ML312 A-549 CTRP2 0.0020 66.0000
ML312 NCI-H2009 CTRP2 0.0020 66.0000
ML312 SNU-201 CTRP2 0.0020 66.0000
ML312 SUIT-2 CTRP2 0.0020 66.0000
ML312 SNU-1079 CTRP2 0.0020 66.0000
ML312 COLO741 CTRP2 0.0020 66.0000
ML312 DEL CTRP2 0.0020 66.0000
ML312 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP2 0.0020 66.0000
ML312 HCC15 CTRP2 0.0020 66.0000
ML312 KP-4 CTRP2 0.0020 66.0000
ML312 LU-99 CTRP2 0.0020 66.0000
ML312 NCI-H1155 CTRP2 0.0020 66.0000
ML312 NCI-H1581 CTRP2 0.0020 66.0000
ML312 NCI-H2106 CTRP2 0.0020 66.0000
ML312 NCI-H358 CTRP2 0.0020 66.0000
ML312 DLD-1 CTRP2 0.0020 66.0000
ML312 EM-2 CTRP2 0.0020 66.0000
ML312 JURL-MK1 CTRP2 0.0020 66.0000
ML312 P12-ICHIKAWA CTRP2 0.0020 66.0000
ML312 KE-37 CTRP2 0.0020 66.0000
ML312 KMS-21-BM CTRP2 0.0020 66.0000
ML312 LI-7 CTRP2 0.0020 66.0000
ML312 MOLM-13 CTRP2 0.0020 66.0000
ML312 NCI-H1975 CTRP2 0.0020 66.0000
ML312 NCI-H28 CTRP2 0.0020 66.0000
ML312 639V CTRP2 0.0020 66.0000
ML312 BXPC-3 CTRP2 0.0020 66.0000
ML312 CML-T1 CTRP2 0.0020 66.0000
ML312 GSS CTRP2 0.0020 66.0000
ML312 HCC366 CTRP2 0.0020 66.0000
ML312 KURAMOCHI CTRP2 0.0020 66.0000
ML312 LS411N CTRP2 0.0020 66.0000
ML312 LS513 CTRP2 0.0020 66.0000
ML312 ONCO-DG-1 CTRP2 0.0020 66.0000
ML312 ONS-76 CTRP2 0.0020 66.0000
ML312 SK-CO-1 CTRP2 0.0020 66.0000
ML312 SW48 CTRP2 0.0020 66.0000
ML312 VM-CUB-1 CTRP2 0.0020 66.0000
ML312 BEN CTRP2 0.0020 66.0000
ML312 CFPAC-1 CTRP2 0.0020 66.0000
ML312 HCC78 CTRP2 0.0020 66.0000
ML312 HT CTRP2 0.0020 66.0000
ML312 KU-19-19 CTRP2 0.0020 66.0000
ML312 NCI-H1299 CTRP2 0.0020 66.0000
ML312 NCI-H727 CTRP2 0.0020 66.0000
ML312 NCO2 CTRP2 0.0020 66.0000
ML312 OVTOKO CTRP2 0.0020 66.0000
ML312 P31-FUJ CTRP2 0.0020 66.0000
ML312 PEER CTRP2 0.0020 66.0000
ML312 RPMI-8402 CTRP2 0.0020 66.0000
ML312 SHP-77 CTRP2 0.0020 66.0000
ML312 SNU-1077 CTRP2 0.0020 66.0000
ML312 SNU-620 CTRP2 0.0020 66.0000
ML312 SU-DHL-1 CTRP2 0.0020 66.0000
ML312 COLO205 CTRP2 0.0020 66.0000
ML312 EHEB CTRP2 0.0020 66.0000
ML312 KI-JK CTRP2 0.0020 66.0000
ML312 KMM-1 CTRP2 0.0020 66.0000
ML312 LCLC-103H CTRP2 0.0020 66.0000
ML312 MKN45 CTRP2 0.0020 66.0000
ML312 NCI-H2405 CTRP2 0.0020 66.0000
ML312 NCI-H650 CTRP2 0.0020 66.0000
ML312 OS-RC-2 CTRP2 0.0020 66.0000
ML312 OVSAHO CTRP2 0.0020 66.0000
ML312 QGP-1 CTRP2 0.0020 66.0000
ML312 RL95-2 CTRP2 0.0020 66.0000
ML312 SNU-1041 CTRP2 0.0020 66.0000
ML312 SNU-1066 CTRP2 0.0020 66.0000
ML312 SW1353 CTRP2 0.0020 66.0000
ML312 SNU-213 CTRP2 0.0020 66.0000
ML312 8505C CTRP2 0.0020 66.0000
ML312 CALU-3 CTRP2 0.0020 66.0000
ML312 DAOY CTRP2 0.0020 66.0000
ML312 GB-1 CTRP2 0.0020 66.0000
ML312 HCC1171 CTRP2 0.0020 66.0000
ML312 HCC44 CTRP2 0.0020 66.0000
ML312 NCI-H211 CTRP2 0.0020 66.0000
ML312 RERF-LC-A1 CTRP2 0.0020 66.0000
ML312 SBC-5 CTRP2 0.0020 66.0000
ML312 SF126 CTRP2 0.0020 66.0000
ML312 SNU-119 CTRP2 0.0020 66.0000
ML312 SNU-182 CTRP2 0.0020 66.0000
ML312 TCCSUP CTRP2 0.0020 66.0000
ML312 CAMA-1 CTRP2 0.0020 66.0000
ML312 DETROIT562 CTRP2 0.0020 66.0000
ML312 HEC-1-B CTRP2 0.0020 66.0000
ML312 HEP3B2.1-7 CTRP2 0.0020 66.0000
ML312 HSC-3 CTRP2 0.0020 66.0000
ML312 MCF-7 CTRP2 0.0020 66.0000
ML312 SNU-1105 CTRP2 0.0020 66.0000
ML312 U-87MGATCC CTRP2 0.0020 66.0000
ML312 22RV1 CTRP2 0.0020 66.0000
ML312 769-P CTRP2 0.0020 66.0000
ML312 COLO699 CTRP2 0.0020 66.0000
ML312 DOV13 CTRP2 0.0020 66.0000
ML312 ES2 CTRP2 0.0020 66.0000
ML312 HCC1806 CTRP2 0.0020 66.0000
ML312 HCC1954 CTRP2 0.0020 66.0000
ML312 HPAF-II CTRP2 0.0020 66.0000
ML312 KHM-1B CTRP2 0.0020 66.0000
ML312 OVISE CTRP2 0.0020 66.0000
ML312 JVM-3 CTRP2 0.0020 66.0000
ML312 SNU-C2A CTRP2 0.0020 66.0000
ML312 U2OS CTRP2 0.0020 66.0000
ML312 5637 CTRP2 0.0020 66.0000
ML312 CAL-12T CTRP2 0.0020 66.0000
ML312 HCC1588 CTRP2 0.0020 66.0000
ML312 HCC1833 CTRP2 0.0020 66.0000
ML312 HCC2279 CTRP2 0.0020 66.0000
ML312 KE-97 CTRP2 0.0020 66.0000
ML312 KP-3 CTRP2 0.0020 66.0000
ML312 KU812 CTRP2 0.0020 66.0000
ML312 KYSE-140 CTRP2 0.0020 66.0000
ML312 NALM-6 CTRP2 0.0020 66.0000
ML312 NUGC-4 CTRP2 0.0020 66.0000
ML312 TT CTRP2 0.0020 66.0000
ML312 AGS CTRP2 0.0020 66.0000
ML312 HCT116 CTRP2 0.0020 66.0000
ML312 HEC-108 CTRP2 0.0020 66.0000
ML312 HEC-59 CTRP2 0.0020 66.0000
ML312 HMC-1-8 CTRP2 0.0020 66.0000
ML312 HT-29 CTRP2 0.0020 66.0000
ML312 ISHIKAWA(HERAKLIO)02ER- CTRP2 0.0020 66.0000
ML312 JHOC-5 CTRP2 0.0020 66.0000
ML312 KYSE-180 CTRP2 0.0020 66.0000
ML312 LS180 CTRP2 0.0020 66.0000
ML312 MELHO CTRP2 0.0020 66.0000
ML312 MHH-ES-1 CTRP2 0.0020 66.0000
ML312 MOR-CPR CTRP2 0.0020 66.0000
ML312 NCI-H460 CTRP2 0.0020 66.0000
ML312 HCC2108 CTRP2 0.0020 66.0000
ML312 HCC827 CTRP2 0.0020 66.0000
ML312 HEC-251 CTRP2 0.0020 66.0000
ML312 HEC-265 CTRP2 0.0020 66.0000
ML312 HEC-6 CTRP2 0.0020 66.0000
ML312 HEL CTRP2 0.0020 66.0000
ML312 JHUEM-2 CTRP2 0.0020 66.0000
ML312 JURKAT CTRP2 0.0020 66.0000
ML312 KCL-22 CTRP2 0.0020 66.0000
ML312 KE-39 CTRP2 0.0020 66.0000
ML312 KM-H2 CTRP2 0.0020 66.0000
ML312 LAMA-84 CTRP2 0.0020 66.0000
ML312 NCI-H2030 CTRP2 0.0020 66.0000
ML312 SNU-719 CTRP2 0.0020 66.0000
ML312 HCC1569 CTRP2 0.0020 66.0000
ML312 KMS-26 CTRP2 0.0020 66.0000
ML312 NCI-H1838 CTRP2 0.0020 66.0000
ML312 NCI-H196 CTRP2 0.0020 66.0000
ML312 NCI-H292 CTRP2 0.0020 66.0000
ML312 HCC1937 CTRP2 0.0020 66.0000
ML312 HUH-28 CTRP2 0.0020 66.0000
ML312 NCI-H526 CTRP2 0.0020 66.0000
ML312 NCI-H69 CTRP2 0.0020 66.0000
ML312 NCI-H929 CTRP2 0.0020 66.0000
ML312 PF-382 CTRP2 0.0020 66.0000
ML312 SF295 CTRP2 0.0020 66.0000
ML312 SNU-1272 CTRP2 0.0020 66.0000
ML312 SNU-308 CTRP2 0.0020 66.0000
ML312 SNU-478 CTRP2 0.0020 66.0000
ML312 BHT-101 CTRP2 0.0020 66.0000
ML312 CAL-148 CTRP2 0.0020 66.0000
ML312 CAL-51 CTRP2 0.0020 66.0000
ML312 HCC1395 CTRP2 0.0020 66.0000
ML312 HT115 CTRP2 0.0020 66.0000
ML312 LN-18 CTRP2 0.0020 66.0000
ML312 LN-229 CTRP2 0.0020 66.0000
ML312 NCI-H1734 CTRP2 0.0020 66.0000
ML312 NCI-H2291 CTRP2 0.0020 66.0000
ML312 RERF-LC-AD1 CTRP2 0.0020 66.0000
ML312 SNU-1214 CTRP2 0.0020 66.0000
ML312 SNU-46 CTRP2 0.0020 66.0000
ML312 SNU-668 CTRP2 0.0020 66.0000
ML312 SNU-899 CTRP2 0.0020 66.0000
ML312 TE-10 CTRP2 0.0020 66.0000
ML312 TE-9 CTRP2 0.0020 66.0000
ML312 YD-15 CTRP2 0.0020 66.0000
ML312 YD-38 CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.