Drug : Afuresertib

GDSC1 Name , GDSC2 Name : Afuresertib

Dataset : All
Synonyms :
Targets : AKT1, AKT2, AKT3
Pathways : PI3K/MTOR signaling

Information Cards

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Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
Afuresertib PC-14 GDSC2 0.0100 10.0000
Afuresertib A-549 GDSC2 0.0100 10.0000
Afuresertib A-375 GDSC2 0.0100 10.0000
Afuresertib DEL GDSC2 0.0100 10.0000
Afuresertib EW-13 GDSC2 0.0100 10.0000
Afuresertib MHH-ES-1 GDSC2 0.0100 10.0000
Afuresertib C32[HUMANMELANOMA] GDSC2 0.0100 10.0000
Afuresertib U2OS GDSC2 0.0100 10.0000
Afuresertib TC-71 GDSC2 0.0100 10.0000
Afuresertib DIFI GDSC2 0.0100 10.0000
Afuresertib RKO GDSC2 0.0100 10.0000
Afuresertib NCI-H747 GDSC2 0.0100 10.0000
Afuresertib CL-11 GDSC2 0.0100 10.0000
Afuresertib COLO320HSR GDSC2 0.0100 10.0000
Afuresertib SW620 GDSC2 0.0100 10.0000
Afuresertib HT-29 GDSC2 0.0100 10.0000
Afuresertib HCT15 GDSC2 0.0100 10.0000
Afuresertib SNU-C2B GDSC2 0.0100 10.0000
Afuresertib MFM-223 GDSC2 0.0100 10.0000
Afuresertib SR GDSC2 0.0100 10.0000
Afuresertib SKM-1 GDSC2 0.0100 10.0000
Afuresertib CCK-81 GDSC2 0.0100 10.0000
Afuresertib COLO205 GDSC2 0.0100 10.0000
Afuresertib SK-CO-1 GDSC2 0.0100 10.0000
Afuresertib LS411N GDSC2 0.0100 10.0000
Afuresertib LS123 GDSC2 0.0100 10.0000
Afuresertib LS1034 GDSC2 0.0100 10.0000
Afuresertib HCC2998 GDSC2 0.0100 10.0000
Afuresertib NCI-H929 GDSC2 0.0100 10.0000
Afuresertib CP66-MEL GDSC2 0.0100 10.0000
Afuresertib KU812 GDSC2 0.0100 10.0000
Afuresertib VAL GDSC2 0.0100 10.0000
Afuresertib RF-48 GDSC2 0.0100 10.0000
Afuresertib L-540 GDSC2 0.0100 10.0000
Afuresertib DB GDSC2 0.0100 10.0000
Afuresertib MDST8 GDSC2 0.0100 10.0000
Afuresertib HT-55 GDSC2 0.0100 10.0000
Afuresertib CA9-22 GDSC2 0.0100 10.0000
Afuresertib DOK GDSC2 0.0100 10.0000
Afuresertib KM12 GDSC2 0.0100 10.0000
Afuresertib CAR-1 GDSC2 0.0100 10.0000
Afuresertib HT115 GDSC2 0.0100 10.0000
Afuresertib GP5D GDSC2 0.0100 10.0000
Afuresertib CW-2 GDSC2 0.0100 10.0000
Afuresertib HUTU80 GDSC2 0.0100 10.0000
Afuresertib HCT116 GDSC2 0.0100 10.0000
Afuresertib SNU-C5 GDSC2 0.0100 10.0000
Afuresertib SW48 GDSC2 0.0100 10.0000
Afuresertib C2BBE1 GDSC2 0.0100 10.0000
Afuresertib EM-2 GDSC2 0.0100 10.0000
Afuresertib KCL-22 GDSC2 0.0100 10.0000
Afuresertib BICR10 GDSC2 0.0100 10.0000
Afuresertib CS-1[HUMANCHONDROSARCOMA] GDSC2 0.0100 10.0000
Afuresertib SKN GDSC2 0.0100 10.0000
Afuresertib PEO1 GDSC2 0.0100 10.0000
Afuresertib TE-12 GDSC2 0.0100 10.0000
Afuresertib LP-1 GDSC2 0.0100 10.0000
Afuresertib HSC-3 GDSC2 0.0100 10.0000
Afuresertib PCI-04B GDSC2 0.0100 10.0000
Afuresertib SNU-407 GDSC2 0.0100 10.0000
Afuresertib OACP4C GDSC2 0.0100 10.0000
Afuresertib SK-GT-4 GDSC2 0.0100 10.0000
Afuresertib NCI-H841 GDSC2 0.0100 10.0000
Afuresertib SNU-175 GDSC2 0.0100 10.0000
Afuresertib COLO678 GDSC2 0.0100 10.0000
Afuresertib T84 GDSC2 0.0100 10.0000
Afuresertib NCI-H2135 GDSC2 0.0100 10.0000
Afuresertib ABC-1 GDSC2 0.0100 10.0000
Afuresertib SK-MEL-5 GDSC2 0.0100 10.0000
Afuresertib A-427 GDSC2 0.0100 10.0000
Afuresertib RCM-1[HUMANESC] GDSC2 0.0100 10.0000
Afuresertib LOVO GDSC2 0.0100 10.0000
Afuresertib LS180 GDSC2 0.0100 10.0000
Afuresertib NCI-H1876 GDSC2 0.0100 10.0000
Afuresertib OVK18 GDSC2 0.0100 10.0000
Afuresertib MRK-NU-1 GDSC2 0.0100 10.0000
Afuresertib NCC010 GDSC2 0.0100 10.0000
Afuresertib RKN GDSC2 0.0100 10.0000
Afuresertib SW1417 GDSC2 0.0100 10.0000
Afuresertib 5637 GDSC2 0.0100 10.0000
Afuresertib 697 GDSC2 0.0100 10.0000
Afuresertib OSC-20 GDSC2 0.0100 10.0000
Afuresertib 8505C GDSC2 0.0100 10.0000
Afuresertib 786-O GDSC2 0.0100 10.0000
Afuresertib 647V GDSC2 0.0100 10.0000
Afuresertib 42-MG-BA GDSC2 0.0100 10.0000
Afuresertib SW837 GDSC2 0.0100 10.0000
Afuresertib A101D GDSC2 0.0100 10.0000
Afuresertib VMRC-RCZ GDSC2 0.0100 10.0000
Afuresertib 639V GDSC2 0.0100 10.0000
Afuresertib B-CPAP GDSC2 0.0100 10.0000
Afuresertib A-172 GDSC2 0.0100 10.0000
Afuresertib 8-MG-BA GDSC2 0.0100 10.0000
Afuresertib BHT-101 GDSC2 0.0100 10.0000
Afuresertib H-EMC-SS GDSC2 0.0100 10.0000
Afuresertib A2058 GDSC2 0.0100 10.0000
Afuresertib SW1116 GDSC2 0.0100 10.0000
Afuresertib BPH-1 GDSC2 0.0100 10.0000
Afuresertib JIYOYE GDSC2 0.0100 10.0000
Afuresertib SUIT-2 GDSC2 0.0100 10.0000
Afuresertib UACC-257 GDSC2 0.0100 10.0000
Afuresertib 23132-87 GDSC2 0.0100 10.0000
Afuresertib WM793 GDSC2 0.0100 10.0000
Afuresertib BFTC-909 GDSC2 0.0100 10.0000
Afuresertib SW948 GDSC2 0.0100 10.0000
Afuresertib PANC02.03 GDSC2 0.0100 10.0000
Afuresertib AGS GDSC2 0.0100 10.0000
Afuresertib QGP-1 GDSC2 0.0100 10.0000
Afuresertib NCI-H345 GDSC2 0.0100 10.0000
Afuresertib RERF-LC-KJ GDSC2 0.0100 10.0000
Afuresertib CHP-134 GDSC2 0.0100 10.0000
Afuresertib SU.86.86 GDSC2 0.0100 10.0000
Afuresertib C-4-I GDSC2 0.0100 10.0000
Afuresertib BT-474 GDSC2 0.0100 10.0000
Afuresertib CAL-120 GDSC2 0.0100 10.0000
Afuresertib HCC1806 GDSC2 0.0100 10.0000
Afuresertib EW-18 GDSC2 0.0100 10.0000
Afuresertib SK-N-BE(2)-M17 GDSC2 0.0100 10.0000
Afuresertib A3-KAWAKAMI GDSC2 0.0100 10.0000
Afuresertib GOTO GDSC2 0.0100 10.0000
Afuresertib G-402 GDSC2 0.0100 10.0000
Afuresertib HEP-G2-C3A GDSC2 0.0100 10.0000
Afuresertib CADO-ES1 GDSC2 0.0100 10.0000
Afuresertib FADU GDSC2 0.0100 10.0000
Afuresertib BALL-1 GDSC2 0.0100 10.0000
Afuresertib NCI-H2227 GDSC2 0.0100 10.0000
Afuresertib BT-549 GDSC2 0.0100 10.0000
Afuresertib SIHA GDSC2 0.0100 10.0000
Afuresertib SNU-81 GDSC2 0.0100 10.0000
Afuresertib BB49-HNC GDSC2 0.0100 10.0000
Afuresertib ZR-75-30 GDSC2 0.0100 10.0000
Afuresertib HC-1 GDSC2 0.0100 10.0000
Afuresertib TK[HUMANB-CELLLYMPHOMA] GDSC2 0.0100 10.0000
Afuresertib EVSA-T GDSC2 0.0100 10.0000
Afuresertib NEC8 GDSC2 0.0100 10.0000
Afuresertib SF268 GDSC2 0.0100 10.0000
Afuresertib PATU8902 GDSC2 0.0100 10.0000
Afuresertib HEY GDSC2 0.0100 10.0000
Afuresertib NCI-H1781 GDSC2 0.0100 10.0000
Afuresertib DAN-G GDSC2 0.0100 10.0000
Afuresertib HCC78 GDSC2 0.0100 10.0000
Afuresertib NUGC-3 GDSC2 0.0100 10.0000
Afuresertib KYSE-410 GDSC2 0.0100 10.0000
Afuresertib CAL-27 GDSC2 0.0100 10.0000
Afuresertib ASH-3 GDSC2 0.0100 10.0000
Afuresertib TE-4 GDSC2 0.0100 10.0000
Afuresertib NCI-H661 GDSC2 0.0100 10.0000
Afuresertib VA-ES-BJ GDSC2 0.0100 10.0000
Afuresertib CAL-51 GDSC2 0.0100 10.0000
Afuresertib CAL-33 GDSC2 0.0100 10.0000
Afuresertib DAOY GDSC2 0.0100 10.0000
Afuresertib DETROIT562 GDSC2 0.0100 10.0000
Afuresertib AN3-CA GDSC2 0.0100 10.0000
Afuresertib EBC-1 GDSC2 0.0100 10.0000
Afuresertib EC-GI-10 GDSC2 0.0100 10.0000
Afuresertib CALU-6 GDSC2 0.0100 10.0000
Afuresertib ES-2 GDSC2 0.0100 10.0000
Afuresertib ES4 GDSC2 0.0100 10.0000
Afuresertib CHP-212 GDSC2 0.0100 10.0000
Afuresertib ETK-1 GDSC2 0.0100 10.0000
Afuresertib COLO829 GDSC2 0.0100 10.0000
Afuresertib COR-L23 GDSC2 0.0100 10.0000
Afuresertib GCT GDSC2 0.0100 10.0000
Afuresertib NCI-H2373 GDSC2 0.0100 10.0000
Afuresertib NCI-H2369 GDSC2 0.0100 10.0000
Afuresertib RD GDSC2 0.0100 10.0000
Afuresertib RC-K8 GDSC2 0.0100 10.0000
Afuresertib CAL-78 GDSC2 0.0100 10.0000
Afuresertib EW-1 GDSC2 0.0100 10.0000
Afuresertib CAL-29 GDSC2 0.0100 10.0000
Afuresertib OE19 GDSC2 0.0100 10.0000
Afuresertib JURKAT GDSC2 0.0100 10.0000
Afuresertib PL4 GDSC2 0.0100 10.0000
Afuresertib OVTOKO GDSC2 0.0100 10.0000
Afuresertib NH-12 GDSC2 0.0100 10.0000
Afuresertib A-498 GDSC2 0.0100 10.0000
Afuresertib IGROV-1 GDSC2 0.0100 10.0000
Afuresertib ASPC-1 GDSC2 0.0100 10.0000
Afuresertib RH30 GDSC2 0.0100 10.0000
Afuresertib G-401 GDSC2 0.0100 10.0000
Afuresertib HUH-1 GDSC2 0.0100 10.0000
Afuresertib ALL-PO GDSC2 0.0100 10.0000
Afuresertib COLO792 GDSC2 0.0100 10.0000
Afuresertib EPLC-272H GDSC2 0.0100 10.0000
Afuresertib ESO-51 GDSC2 0.0100 10.0000
Afuresertib CFPAC-1 GDSC2 0.0100 10.0000
Afuresertib RAJI GDSC2 0.0100 10.0000
Afuresertib DAUDI GDSC2 0.0100 10.0000
Afuresertib NCI-H2591 GDSC2 0.0100 10.0000
Afuresertib ARH-77 GDSC2 0.0100 10.0000
Afuresertib ME-180 GDSC2 0.0100 10.0000
Afuresertib CA46 GDSC2 0.0100 10.0000
Afuresertib ALL-SIL GDSC2 0.0100 10.0000
Afuresertib GRANTA-519 GDSC2 0.0100 10.0000
Afuresertib DBTRG-05MG GDSC2 0.0100 10.0000
Afuresertib LXF289 GDSC2 0.0100 10.0000
Afuresertib NCI-H513 GDSC2 0.0100 10.0000
Afuresertib GB-1 GDSC2 0.0100 10.0000
Afuresertib DK-MG GDSC2 0.0100 10.0000
Afuresertib GI-ME-N GDSC2 0.0100 10.0000
Afuresertib AU565 GDSC2 0.0100 10.0000
Afuresertib G-361 GDSC2 0.0100 10.0000
Afuresertib EW-16 GDSC2 0.0100 10.0000
Afuresertib LN-18 GDSC2 0.0100 10.0000
Afuresertib SNU-61 GDSC2 0.0100 10.0000
Afuresertib AM-38 GDSC2 0.0100 10.0000
Afuresertib DMS53 GDSC2 0.0100 10.0000
Afuresertib NB(TU)1 GDSC2 0.0100 10.0000
Afuresertib HELA GDSC2 0.0100 10.0000
Afuresertib NCI-H1623 GDSC2 0.0100 10.0000
Afuresertib SW1463 GDSC2 0.0100 10.0000
Afuresertib NCI-H2122 GDSC2 0.0100 10.0000
Afuresertib LN-405 GDSC2 0.0100 10.0000
Afuresertib NCI-H2228 GDSC2 0.0100 10.0000
Afuresertib MOLT-16 GDSC2 0.0100 10.0000
Afuresertib SNU-C1 GDSC2 0.0100 10.0000
Afuresertib P12-ICHIKAWA GDSC2 0.0100 10.0000
Afuresertib SK-MM-2 GDSC2 0.0100 10.0000
Afuresertib NCI-H1563 GDSC2 0.0100 10.0000
Afuresertib GA-10 GDSC2 0.0100 10.0000
Afuresertib CESS GDSC2 0.0100 10.0000
Afuresertib HTC-C3 GDSC2 0.0100 10.0000
Afuresertib KMRC-20 GDSC2 0.0100 10.0000
Afuresertib HT-1080 GDSC2 0.0100 10.0000
Afuresertib HT-3 GDSC2 0.0100 10.0000
Afuresertib EJM GDSC2 0.0100 10.0000
Afuresertib HCC15 GDSC2 0.0100 10.0000
Afuresertib KP-1N GDSC2 0.0100 10.0000
Afuresertib JHH-1 GDSC2 0.0100 10.0000
Afuresertib HOP-62 GDSC2 0.0100 10.0000
Afuresertib KM-H2 GDSC2 0.0100 10.0000
Afuresertib KOPN-8 GDSC2 0.0100 10.0000
Afuresertib JJN-3 GDSC2 0.0100 10.0000
Afuresertib A-204 GDSC2 0.0100 10.0000
Afuresertib JIMT-1 GDSC2 0.0100 10.0000
Afuresertib ATN-1 GDSC2 0.0100 10.0000
Afuresertib DG-75 GDSC2 0.0100 10.0000
Afuresertib OCI-M1 GDSC2 0.0100 10.0000
Afuresertib KYSE-520 GDSC2 0.0100 10.0000
Afuresertib HUP-T4 GDSC2 0.0100 10.0000
Afuresertib KMOE-2 GDSC2 0.0100 10.0000
Afuresertib JSC-1 GDSC2 0.0100 10.0000
Afuresertib EFM-192A GDSC2 0.0100 10.0000
Afuresertib RT-4 GDSC2 0.0100 10.0000
Afuresertib KYSE-50 GDSC2 0.0100 10.0000
Afuresertib U-251MG GDSC2 0.0100 10.0000
Afuresertib IGR-1 GDSC2 0.0100 10.0000
Afuresertib FTC-133 GDSC2 0.0100 10.0000
Afuresertib CAS-1 GDSC2 0.0100 10.0000
Afuresertib HEC-1 GDSC2 0.0100 10.0000
Afuresertib MFE-296 GDSC2 0.0100 10.0000
Afuresertib M14 GDSC2 0.0100 10.0000
Afuresertib MM1.S GDSC2 0.0100 10.0000
Afuresertib HT-144 GDSC2 0.0100 10.0000
Afuresertib LB996-RCC GDSC2 0.0100 10.0000
Afuresertib IMR-5 GDSC2 0.0100 10.0000
Afuresertib HUO9 GDSC2 0.0100 10.0000
Afuresertib OV56 GDSC2 0.0100 10.0000
Afuresertib NCI-H446 GDSC2 0.0100 10.0000
Afuresertib OAW28 GDSC2 0.0100 10.0000
Afuresertib OVCAR-4 GDSC2 0.0100 10.0000
Afuresertib SK-N-DZ GDSC2 0.0100 10.0000
Afuresertib NCI-H2405 GDSC2 0.0100 10.0000
Afuresertib SW872 GDSC2 0.0100 10.0000
Afuresertib SW1573 GDSC2 0.0100 10.0000
Afuresertib RL95-2 GDSC2 0.0100 10.0000
Afuresertib TCCSUP GDSC2 0.0100 10.0000
Afuresertib SK-ES-1 GDSC2 0.0100 10.0000
Afuresertib TT2609-C02 GDSC2 0.0100 10.0000
Afuresertib WM35 GDSC2 0.0100 10.0000
Afuresertib SU-DHL-8 GDSC2 0.0100 10.0000
Afuresertib RCC10RGB GDSC2 0.0100 10.0000
Afuresertib SISO GDSC2 0.0100 10.0000
Afuresertib UMC-11 GDSC2 0.0100 10.0000
Afuresertib SK-MG-1 GDSC2 0.0100 10.0000
Afuresertib SKN-3 GDSC2 0.0100 10.0000
Afuresertib LNCAPCLONEFGC GDSC2 0.0100 10.0000
Afuresertib NCI-H1944 GDSC2 0.0100 10.0000
Afuresertib SW780 GDSC2 0.0100 10.0000
Afuresertib OVCA420 GDSC2 0.0100 10.0000
Afuresertib OAW42 GDSC2 0.0100 10.0000
Afuresertib WM278 GDSC2 0.0100 10.0000
Afuresertib OACM5.1C GDSC2 0.0100 10.0000
Afuresertib KARPAS-231 GDSC2 0.0100 10.0000
Afuresertib A-704 GDSC2 0.0100 10.0000
Afuresertib JHH-6 GDSC2 0.0100 10.0000
Afuresertib MHH-CALL-2 GDSC2 0.0100 10.0000
Afuresertib JHH-4 GDSC2 0.0100 10.0000
Afuresertib ESO-26 GDSC2 0.0100 10.0000
Afuresertib OE21 GDSC2 0.0100 10.0000
Afuresertib NCI-H1693 GDSC2 0.0100 10.0000
Afuresertib HCC1187 GDSC2 0.0100 10.0000
Afuresertib HSC-4 GDSC2 0.0100 10.0000
Afuresertib LU-99A GDSC2 0.0100 10.0000
Afuresertib MOLP-8 GDSC2 0.0100 10.0000
Afuresertib MHH-PREB-1 GDSC2 0.0100 10.0000
Afuresertib MOLT-13 GDSC2 0.0100 10.0000
Afuresertib MDA-MB-231 GDSC2 0.0100 10.0000
Afuresertib NCI-H2722 GDSC2 0.0100 10.0000
Afuresertib OS-RC-2 GDSC2 0.0100 10.0000
Afuresertib OVCAR-3 GDSC2 0.0100 10.0000
Afuresertib KY821 GDSC2 0.0100 10.0000
Afuresertib HS445 GDSC2 0.0100 10.0000
Afuresertib SNU-1 GDSC2 0.0100 10.0000
Afuresertib HCC1143 GDSC2 0.0100 10.0000
Afuresertib NCI-H1650 GDSC2 0.0100 10.0000
Afuresertib NCI-H1048 GDSC2 0.0100 10.0000
Afuresertib HS746.T GDSC2 0.0100 10.0000
Afuresertib KARPAS-45 GDSC2 0.0100 10.0000
Afuresertib YAPC GDSC2 0.0100 10.0000
Afuresertib SUP-M2 GDSC2 0.0100 10.0000
Afuresertib SCC-3 GDSC2 0.0100 10.0000
Afuresertib P32-ISH GDSC2 0.0100 10.0000
Afuresertib RERF-LC-SQ1 GDSC2 0.0100 10.0000
Afuresertib MSTO-211H GDSC2 0.0100 10.0000
Afuresertib MOLM-13 GDSC2 0.0100 10.0000
Afuresertib MFE-319 GDSC2 0.0100 10.0000
Afuresertib LN-229 GDSC2 0.0100 10.0000
Afuresertib J82 GDSC2 0.0100 10.0000
Afuresertib IA-LM GDSC2 0.0100 10.0000
Afuresertib OVISE GDSC2 0.0100 10.0000
Afuresertib HCC827 GDSC2 0.0100 10.0000
Afuresertib HCC2157 GDSC2 0.0100 10.0000
Afuresertib NCI-H1155 GDSC2 0.0100 10.0000
Afuresertib BT-20 GDSC2 0.0100 10.0000
Afuresertib COLO824 GDSC2 0.0100 10.0000
Afuresertib DU4475 GDSC2 0.0100 10.0000
Afuresertib HOP-92 GDSC2 0.0100 10.0000
Afuresertib HUP-T3 GDSC2 0.0100 10.0000
Afuresertib KG-1 GDSC2 0.0100 10.0000
Afuresertib MELJUSO GDSC2 0.0100 10.0000
Afuresertib MES-SA GDSC2 0.0100 10.0000
Afuresertib NCI-H1568 GDSC2 0.0100 10.0000
Afuresertib OVCAR-8 GDSC2 0.0100 10.0000
Afuresertib P30-OHK GDSC2 0.0100 10.0000
Afuresertib SW756 GDSC2 0.0100 10.0000
Afuresertib A2780 GDSC2 0.0100 10.0000
Afuresertib BECKER GDSC2 0.0100 10.0000
Afuresertib ES7 GDSC2 0.0100 10.0000
Afuresertib A-253 GDSC2 0.0100 10.0000
Afuresertib NCI-H716 GDSC2 0.0100 10.0000
Afuresertib HCC1428 GDSC2 0.0100 10.0000
Afuresertib HGC-27 GDSC2 0.0100 10.0000
Afuresertib KASUMI-1 GDSC2 0.0100 10.0000
Afuresertib HUH-7 GDSC2 0.0100 10.0000
Afuresertib HUO-3N1 GDSC2 0.0100 10.0000
Afuresertib NCI-H196 GDSC2 0.0100 10.0000
Afuresertib NCI-H2141 GDSC2 0.0100 10.0000
Afuresertib BL-41 GDSC2 0.0100 10.0000
Afuresertib CAL-39 GDSC2 0.0100 10.0000
Afuresertib EW-3 GDSC2 0.0100 10.0000
Afuresertib HPAC GDSC2 0.0100 10.0000
Afuresertib IM95 GDSC2 0.0100 10.0000
Afuresertib NCI-H1694 GDSC2 0.0100 10.0000
Afuresertib NCI-H2170 GDSC2 0.0100 10.0000
Afuresertib NOS-1[HUMANOSTEOSARCOMA] GDSC2 0.0100 10.0000
Afuresertib RERF-GC-1B GDSC2 0.0100 10.0000
Afuresertib TE-6 GDSC2 0.0100 10.0000
Afuresertib TYK-NU GDSC2 0.0100 10.0000
Afuresertib CHL-1 GDSC2 0.0100 10.0000
Afuresertib HCC1954 GDSC2 0.0100 10.0000
Afuresertib NCI-H1975 GDSC2 0.0100 10.0000
Afuresertib NCI-H2052 GDSC2 0.0100 10.0000
Afuresertib NCI-H322M GDSC2 0.0100 10.0000
Afuresertib NCI-H596 GDSC2 0.0100 10.0000
Afuresertib RH1 GDSC2 0.0100 10.0000
Afuresertib A-673 GDSC2 0.0100 10.0000
Afuresertib BXPC-3 GDSC2 0.0100 10.0000
Afuresertib KE-37 GDSC2 0.0100 10.0000
Afuresertib PC-3 GDSC2 0.0100 10.0000
Afuresertib SCC-15 GDSC2 0.0100 10.0000
Afuresertib UPCI-SCC-090 GDSC2 0.0100 10.0000
Afuresertib PWR-1E GDSC2 0.0100 10.0000
Afuresertib SAT[HUMANHNSCC] GDSC2 0.0100 10.0000
Afuresertib SIMA GDSC2 0.0100 10.0000
Afuresertib TE-1 GDSC2 0.0100 10.0000
Afuresertib LCLC-97TM1 GDSC2 0.0100 10.0000
Afuresertib LOU-NH91 GDSC2 0.0100 10.0000
Afuresertib NCI-H1092 GDSC2 0.0100 10.0000
Afuresertib NCI-H720 GDSC2 0.0100 10.0000
Afuresertib KYSE-180 GDSC2 0.0100 10.0000
Afuresertib LC-1-SQ GDSC2 0.0100 10.0000
Afuresertib 769-P GDSC2 0.0100 10.0000
Afuresertib HT-1197 GDSC2 0.0100 10.0000
Afuresertib KLE GDSC2 0.0100 10.0000
Afuresertib L-428 GDSC2 0.0100 10.0000
Afuresertib SNU-5 GDSC2 0.0100 10.0000
Afuresertib PATU8988T GDSC2 0.0100 10.0000
Afuresertib PFSK-1 GDSC2 0.0100 10.0000
Afuresertib RPMI-7951 GDSC2 0.0100 10.0000
Afuresertib SK-GT-2 GDSC2 0.0100 10.0000
Afuresertib SUP-HD1 GDSC2 0.0100 10.0000
Afuresertib 22RV1 GDSC2 0.0100 10.0000
Afuresertib 8305C GDSC2 0.0100 10.0000
Afuresertib ACHN GDSC2 0.0100 10.0000
Afuresertib CAPAN-2 GDSC2 0.0100 10.0000
Afuresertib CASKI GDSC2 0.0100 10.0000
Afuresertib FLO-1 GDSC2 0.0100 10.0000
Afuresertib GR-ST GDSC2 0.0100 10.0000
Afuresertib KALS-1 GDSC2 0.0100 10.0000
Afuresertib KARPAS-422 GDSC2 0.0100 10.0000
Afuresertib KELLY GDSC2 0.0100 10.0000
Afuresertib KP-2 GDSC2 0.0100 10.0000
Afuresertib KP-3 GDSC2 0.0100 10.0000
Afuresertib LB771-HNC GDSC2 0.0100 10.0000
Afuresertib PANC08.13 GDSC2 0.0100 10.0000
Afuresertib SK-HEP-1 GDSC2 0.0100 10.0000
Afuresertib SN12C GDSC2 0.0100 10.0000
Afuresertib T-47D GDSC2 0.0100 10.0000
Afuresertib TGBC24TKB GDSC2 0.0100 10.0000
Afuresertib TOV-112D GDSC2 0.0100 10.0000
Afuresertib TUR GDSC2 0.0100 10.0000
Afuresertib U-118MG GDSC2 0.0100 10.0000
Afuresertib U-87MGATCC GDSC2 0.0100 10.0000
Afuresertib NCI-H1963 GDSC2 0.0100 10.0000
Afuresertib NCI-H209 GDSC2 0.0100 10.0000
Afuresertib NCI-H250 GDSC2 0.0100 10.0000
Afuresertib NUGC-4 GDSC2 0.0100 10.0000
Afuresertib SBC-5 GDSC2 0.0100 10.0000
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Afuresertib D-247MG GDSC2 0.0100 10.0000
Afuresertib SF295 GDSC2 0.0100 10.0000
Afuresertib K2[HUMANMELANOMA] GDSC2 0.0100 10.0000
Afuresertib JAR GDSC2 0.0100 10.0000
Afuresertib ML-1[HUMANLEUKEMIA] GDSC2 0.0100 10.0000
Afuresertib JM1 GDSC2 0.0100 10.0000
Afuresertib RERF-LC-MS GDSC2 0.0100 10.0000
Afuresertib RCH-ACV GDSC2 0.0100 10.0000
Afuresertib A-388 GDSC2 0.0100 10.0000
Afuresertib NMC-G1 GDSC2 0.0100 10.0000
Afuresertib BHY GDSC2 0.0100 10.0000
Afuresertib SK-MEL-30 GDSC2 0.0100 10.0000
Afuresertib SW962 GDSC2 0.0100 10.0000
Afuresertib PCI-15A GDSC2 0.0100 10.0000
Afuresertib OMC-1[HUMANCERVICALCARCINOMA] GDSC2 0.0100 10.0000
Afuresertib NCI-H1437 GDSC2 0.0100 10.0000
Afuresertib THP-1 GDSC2 0.0100 10.0000
Afuresertib TE-10 GDSC2 0.0100 10.0000
Afuresertib OV17R GDSC2 0.0100 10.0000
Afuresertib MZ-MEL-2 GDSC2 0.0100 10.0000
Afuresertib LU-134-A GDSC2 0.0100 10.0000
Afuresertib NCI-H1770 GDSC2 0.0100 10.0000
Afuresertib MY-M12 GDSC2 0.0100 10.0000
Afuresertib KMS-11 GDSC2 0.0100 10.0000
Afuresertib CP50-MEL-B GDSC2 0.0100 10.0000
Afuresertib NB4 GDSC2 0.0100 10.0000
Afuresertib BB30-HNC GDSC2 0.0100 10.0000
Afuresertib SW156 GDSC2 0.0100 10.0000
Afuresertib YKG-1 GDSC2 0.0100 10.0000
Afuresertib LA-N-6 GDSC2 0.0100 10.0000
Afuresertib KTCTL-26A GDSC2 0.0100 10.0000
Afuresertib BC-3 GDSC2 0.0100 10.0000
Afuresertib SNB-75 GDSC2 0.0100 10.0000
Afuresertib VMRC-MELG GDSC2 0.0100 10.0000
Afuresertib MELHO GDSC2 0.0100 10.0000
Afuresertib NCI-H146 GDSC2 0.0100 10.0000
Afuresertib VMRC-RCW GDSC2 0.0100 10.0000
Afuresertib KP-N-YS GDSC2 0.0100 10.0000
Afuresertib HCC33 GDSC2 0.0100 10.0000
Afuresertib TE441.T GDSC2 0.0100 10.0000
Afuresertib EW-12 GDSC2 0.0100 10.0000
Afuresertib CAOV-3 GDSC2 0.0100 10.0000
Afuresertib RVH-421 GDSC2 0.0100 10.0000
Afuresertib NCI-H647 GDSC2 0.0100 10.0000
Afuresertib CRO-AP2 GDSC2 0.0100 10.0000
Afuresertib A-431 GDSC2 0.0100 10.0000
Afuresertib CHSA0011 GDSC2 0.0100 10.0000
Afuresertib NCI-H2172 GDSC2 0.0100 10.0000
Afuresertib PCI-06A GDSC2 0.0100 10.0000
Afuresertib D-245MG GDSC2 0.0100 10.0000
Afuresertib SK-MEL-3 GDSC2 0.0100 10.0000
Afuresertib NCI-H2081 GDSC2 0.0100 10.0000
Afuresertib HS940.T GDSC2 0.0100 10.0000
Afuresertib KTCTL-140 GDSC2 0.0100 10.0000
Afuresertib D-566MG GDSC2 0.0100 10.0000
Afuresertib SBC-1 GDSC2 0.0100 10.0000
Afuresertib OCI-LY19 GDSC2 0.0100 10.0000
Afuresertib MZ-MEL-7 GDSC2 0.0100 10.0000
Afuresertib HS683 GDSC2 0.0100 10.0000
Afuresertib SF126 GDSC2 0.0100 10.0000
Afuresertib D-336MG GDSC2 0.0100 10.0000
Afuresertib STS-0421 GDSC2 0.0100 10.0000
Afuresertib PL-21 GDSC2 0.0100 10.0000
Afuresertib MOLM-16 GDSC2 0.0100 10.0000
Afuresertib NCI-H2110 GDSC2 0.0100 10.0000
Afuresertib ONDA11 GDSC2 0.0100 10.0000
Afuresertib TMK-1 GDSC2 0.0100 10.0000
Afuresertib KTCTL-13 GDSC2 0.0100 10.0000
Afuresertib LC-2-AD GDSC2 0.0100 10.0000
Afuresertib SK-MEL-28 GDSC2 0.0100 10.0000
Afuresertib KTCTL-1M GDSC2 0.0100 10.0000
Afuresertib OVCA433 GDSC2 0.0100 10.0000
Afuresertib SW954 GDSC2 0.0100 10.0000
Afuresertib LB373-MEL-D GDSC2 0.0100 10.0000
Afuresertib JHU-029 GDSC2 0.0100 10.0000
Afuresertib NCI-H460 GDSC2 0.0100 10.0000
Afuresertib NCI-H838 GDSC2 0.0100 10.0000
Afuresertib UO-31 GDSC2 0.0100 10.0000
Afuresertib NCI-H1105 GDSC2 0.0100 10.0000
Afuresertib SK-N-MC-IXC GDSC2 0.0100 10.0000
Afuresertib JHOS-3 GDSC2 0.0100 10.0000
Afuresertib TE-11 GDSC2 0.0100 10.0000
Afuresertib NCC021 GDSC2 0.0100 10.0000
Afuresertib NU-DUL-1 GDSC2 0.0100 10.0000
Afuresertib SU-DHL-16 GDSC2 0.0100 10.0000
Afuresertib EMC-BAC-1 GDSC2 0.0100 10.0000
Afuresertib OCI-LY7 GDSC2 0.0100 10.0000
Afuresertib SU-DHL-4 GDSC2 0.0100 10.0000
Afuresertib SIG-M5 GDSC2 0.0100 10.0000
Afuresertib LB2518-MEL GDSC2 0.0100 10.0000
Afuresertib COLO783 GDSC2 0.0100 10.0000
Afuresertib COR-L303 GDSC2 0.0100 10.0000
Afuresertib CHP-126 GDSC2 0.0100 10.0000
Afuresertib SNU-283 GDSC2 0.0100 10.0000
Afuresertib CHSA0108 GDSC2 0.0100 10.0000
Afuresertib NCI-H748 GDSC2 0.0100 10.0000
Afuresertib ROS-50 GDSC2 0.0100 10.0000
Afuresertib MHH-NB-11 GDSC2 0.0100 10.0000
Afuresertib UWB1.289 GDSC2 0.0100 10.0000
Afuresertib BICR31 GDSC2 0.0100 10.0000
Afuresertib LB647-SCLC GDSC2 0.0100 10.0000
Afuresertib NCI-H2291 GDSC2 0.0100 10.0000
Afuresertib NCI-H740 GDSC2 0.0100 10.0000
Afuresertib COR-L321 GDSC2 0.0100 10.0000
Afuresertib NCI-H1436 GDSC2 0.0100 10.0000
Afuresertib MHH-CALL-4 GDSC2 0.0100 10.0000
Afuresertib IST-SL1 GDSC2 0.0100 10.0000
Afuresertib SCC-25 GDSC2 0.0100 10.0000
Afuresertib NCI-H1734 GDSC2 0.0100 10.0000
Afuresertib U-CH2 GDSC2 0.0100 10.0000
Afuresertib NCI-H2444 GDSC2 0.0100 10.0000
Afuresertib YMB-1-E GDSC2 0.0100 10.0000
Afuresertib KP-N-RT-BM-1 GDSC2 0.0100 10.0000
Afuresertib SJNB-6 GDSC2 0.0100 10.0000
Afuresertib BONNA-12 GDSC2 0.0100 10.0000
Afuresertib NCI-H510A GDSC2 0.0100 10.0000
Afuresertib NCI-H2171 GDSC2 0.0100 10.0000
Afuresertib NCI-H1836 GDSC2 0.0100 10.0000
Afuresertib NCI-H2196 GDSC2 0.0100 10.0000
Afuresertib NCI-H660 GDSC2 0.0100 10.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.