Drug : Brd-K13185470

CTRP2 Name : BRD-K13185470

Dataset : All
Synonyms :
Targets : MCL1
Pathways : stapled helical peptide targeting MCL1

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

:


Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BRD-K13185470 CAS-1 CTRP2 0.0020 66.0000
BRD-K13185470 KPL-1 CTRP2 0.0020 66.0000
BRD-K13185470 MKN1 CTRP2 0.0020 66.0000
BRD-K13185470 253J-BV CTRP2 0.0020 66.0000
BRD-K13185470 BFTC-905 CTRP2 0.0020 66.0000
BRD-K13185470 BFTC-909 CTRP2 0.0020 66.0000
BRD-K13185470 CAL-120 CTRP2 0.0020 66.0000
BRD-K13185470 CAL-29 CTRP2 0.0020 66.0000
BRD-K13185470 CAL-62 CTRP2 0.0020 66.0000
BRD-K13185470 HUCC-T1 CTRP2 0.0020 66.0000
BRD-K13185470 NMC-G1 CTRP2 0.0020 66.0000
BRD-K13185470 RPMI-7951 CTRP2 0.0020 66.0000
BRD-K13185470 253J CTRP2 0.0020 66.0000
BRD-K13185470 ALL-SIL CTRP2 0.0020 66.0000
BRD-K13185470 HDQ-P1 CTRP2 0.0020 66.0000
BRD-K13185470 SIMA CTRP2 0.0020 66.0000
BRD-K13185470 SNU-489 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-626 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-738 CTRP2 0.0020 66.0000
BRD-K13185470 TUHR4TKB CTRP2 0.0020 66.0000
BRD-K13185470 ACC-MESO-1 CTRP2 0.0020 66.0000
BRD-K13185470 B-CPAP CTRP2 0.0020 66.0000
BRD-K13185470 CGTH-W-1 CTRP2 0.0020 66.0000
BRD-K13185470 COLO680N CTRP2 0.0020 66.0000
BRD-K13185470 ECC12 CTRP2 0.0020 66.0000
BRD-K13185470 HCC95 CTRP2 0.0020 66.0000
BRD-K13185470 JMSU-1 CTRP2 0.0020 66.0000
BRD-K13185470 RH41 CTRP2 0.0020 66.0000
BRD-K13185470 WSU-DLCL2 CTRP2 0.0020 66.0000
BRD-K13185470 23132-87 CTRP2 0.0020 66.0000
BRD-K13185470 8305C CTRP2 0.0020 66.0000
BRD-K13185470 BHY CTRP2 0.0020 66.0000
BRD-K13185470 GSU CTRP2 0.0020 66.0000
BRD-K13185470 JIMT-1 CTRP2 0.0020 66.0000
BRD-K13185470 KMRC-20 CTRP2 0.0020 66.0000
BRD-K13185470 OUMS-23 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1076 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1196 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-8 CTRP2 0.0020 66.0000
BRD-K13185470 A-375 CTRP2 0.0020 66.0000
BRD-K13185470 A-549 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H2009 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-201 CTRP2 0.0020 66.0000
BRD-K13185470 SUIT-2 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1079 CTRP2 0.0020 66.0000
BRD-K13185470 DEL CTRP2 0.0020 66.0000
BRD-K13185470 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP2 0.0020 66.0000
BRD-K13185470 HCC15 CTRP2 0.0020 66.0000
BRD-K13185470 KP-4 CTRP2 0.0020 66.0000
BRD-K13185470 LU-99 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H1155 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H1581 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H2106 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H358 CTRP2 0.0020 66.0000
BRD-K13185470 DLD-1 CTRP2 0.0020 66.0000
BRD-K13185470 EM-2 CTRP2 0.0020 66.0000
BRD-K13185470 JURL-MK1 CTRP2 0.0020 66.0000
BRD-K13185470 P12-ICHIKAWA CTRP2 0.0020 66.0000
BRD-K13185470 KE-37 CTRP2 0.0020 66.0000
BRD-K13185470 KMS-21-BM CTRP2 0.0020 66.0000
BRD-K13185470 LI-7 CTRP2 0.0020 66.0000
BRD-K13185470 MHH-NB-11 CTRP2 0.0020 66.0000
BRD-K13185470 MOLM-13 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H1975 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H28 CTRP2 0.0020 66.0000
BRD-K13185470 639V CTRP2 0.0020 66.0000
BRD-K13185470 BXPC-3 CTRP2 0.0020 66.0000
BRD-K13185470 CML-T1 CTRP2 0.0020 66.0000
BRD-K13185470 GSS CTRP2 0.0020 66.0000
BRD-K13185470 HCC366 CTRP2 0.0020 66.0000
BRD-K13185470 KURAMOCHI CTRP2 0.0020 66.0000
BRD-K13185470 LS411N CTRP2 0.0020 66.0000
BRD-K13185470 LS513 CTRP2 0.0020 66.0000
BRD-K13185470 ONCO-DG-1 CTRP2 0.0020 66.0000
BRD-K13185470 ONS-76 CTRP2 0.0020 66.0000
BRD-K13185470 SK-CO-1 CTRP2 0.0020 66.0000
BRD-K13185470 SW48 CTRP2 0.0020 66.0000
BRD-K13185470 VM-CUB-1 CTRP2 0.0020 66.0000
BRD-K13185470 BEN CTRP2 0.0020 66.0000
BRD-K13185470 CFPAC-1 CTRP2 0.0020 66.0000
BRD-K13185470 HCC78 CTRP2 0.0020 66.0000
BRD-K13185470 HT CTRP2 0.0020 66.0000
BRD-K13185470 KU-19-19 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H1299 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H727 CTRP2 0.0020 66.0000
BRD-K13185470 OVTOKO CTRP2 0.0020 66.0000
BRD-K13185470 P31-FUJ CTRP2 0.0020 66.0000
BRD-K13185470 RPMI-8402 CTRP2 0.0020 66.0000
BRD-K13185470 SHP-77 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1077 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-620 CTRP2 0.0020 66.0000
BRD-K13185470 SU-DHL-1 CTRP2 0.0020 66.0000
BRD-K13185470 COLO205 CTRP2 0.0020 66.0000
BRD-K13185470 EHEB CTRP2 0.0020 66.0000
BRD-K13185470 KI-JK CTRP2 0.0020 66.0000
BRD-K13185470 KMM-1 CTRP2 0.0020 66.0000
BRD-K13185470 LCLC-103H CTRP2 0.0020 66.0000
BRD-K13185470 MKN45 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H2405 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H650 CTRP2 0.0020 66.0000
BRD-K13185470 OS-RC-2 CTRP2 0.0020 66.0000
BRD-K13185470 OVSAHO CTRP2 0.0020 66.0000
BRD-K13185470 QGP-1 CTRP2 0.0020 66.0000
BRD-K13185470 RL95-2 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1041 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1066 CTRP2 0.0020 66.0000
BRD-K13185470 SW1353 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-213 CTRP2 0.0020 66.0000
BRD-K13185470 8505C CTRP2 0.0020 66.0000
BRD-K13185470 CALU-3 CTRP2 0.0020 66.0000
BRD-K13185470 DAOY CTRP2 0.0020 66.0000
BRD-K13185470 GB-1 CTRP2 0.0020 66.0000
BRD-K13185470 HCC1171 CTRP2 0.0020 66.0000
BRD-K13185470 HCC44 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H211 CTRP2 0.0020 66.0000
BRD-K13185470 RERF-LC-A1 CTRP2 0.0020 66.0000
BRD-K13185470 SBC-5 CTRP2 0.0020 66.0000
BRD-K13185470 SF126 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-119 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-182 CTRP2 0.0020 66.0000
BRD-K13185470 TCCSUP CTRP2 0.0020 66.0000
BRD-K13185470 CAMA-1 CTRP2 0.0020 66.0000
BRD-K13185470 DETROIT562 CTRP2 0.0020 66.0000
BRD-K13185470 HEC-1-B CTRP2 0.0020 66.0000
BRD-K13185470 HEP3B2.1-7 CTRP2 0.0020 66.0000
BRD-K13185470 HSC-3 CTRP2 0.0020 66.0000
BRD-K13185470 MCF-7 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1105 CTRP2 0.0020 66.0000
BRD-K13185470 U-87MGATCC CTRP2 0.0020 66.0000
BRD-K13185470 22RV1 CTRP2 0.0020 66.0000
BRD-K13185470 769-P CTRP2 0.0020 66.0000
BRD-K13185470 COLO699 CTRP2 0.0020 66.0000
BRD-K13185470 DOV13 CTRP2 0.0020 66.0000
BRD-K13185470 ES2 CTRP2 0.0020 66.0000
BRD-K13185470 HCC1806 CTRP2 0.0020 66.0000
BRD-K13185470 HCC1954 CTRP2 0.0020 66.0000
BRD-K13185470 HPAF-II CTRP2 0.0020 66.0000
BRD-K13185470 KHM-1B CTRP2 0.0020 66.0000
BRD-K13185470 OVISE CTRP2 0.0020 66.0000
BRD-K13185470 JVM-3 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-C2A CTRP2 0.0020 66.0000
BRD-K13185470 U2OS CTRP2 0.0020 66.0000
BRD-K13185470 5637 CTRP2 0.0020 66.0000
BRD-K13185470 CAL-12T CTRP2 0.0020 66.0000
BRD-K13185470 DMS79 CTRP2 0.0020 66.0000
BRD-K13185470 HCC1588 CTRP2 0.0020 66.0000
BRD-K13185470 HCC1833 CTRP2 0.0020 66.0000
BRD-K13185470 HCC2279 CTRP2 0.0020 66.0000
BRD-K13185470 KE-97 CTRP2 0.0020 66.0000
BRD-K13185470 KP-3 CTRP2 0.0020 66.0000
BRD-K13185470 KU812 CTRP2 0.0020 66.0000
BRD-K13185470 KYSE-140 CTRP2 0.0020 66.0000
BRD-K13185470 NALM-6 CTRP2 0.0020 66.0000
BRD-K13185470 NUGC-4 CTRP2 0.0020 66.0000
BRD-K13185470 TT CTRP2 0.0020 66.0000
BRD-K13185470 AGS CTRP2 0.0020 66.0000
BRD-K13185470 HCT116 CTRP2 0.0020 66.0000
BRD-K13185470 HEC-108 CTRP2 0.0020 66.0000
BRD-K13185470 HEC-59 CTRP2 0.0020 66.0000
BRD-K13185470 HMC-1-8 CTRP2 0.0020 66.0000
BRD-K13185470 HT-29 CTRP2 0.0020 66.0000
BRD-K13185470 ISHIKAWA(HERAKLIO)02ER- CTRP2 0.0020 66.0000
BRD-K13185470 JHOC-5 CTRP2 0.0020 66.0000
BRD-K13185470 KYSE-180 CTRP2 0.0020 66.0000
BRD-K13185470 LS180 CTRP2 0.0020 66.0000
BRD-K13185470 MELHO CTRP2 0.0020 66.0000
BRD-K13185470 MHH-ES-1 CTRP2 0.0020 66.0000
BRD-K13185470 MOR-CPR CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H460 CTRP2 0.0020 66.0000
BRD-K13185470 HCC2108 CTRP2 0.0020 66.0000
BRD-K13185470 HCC827 CTRP2 0.0020 66.0000
BRD-K13185470 HEC-251 CTRP2 0.0020 66.0000
BRD-K13185470 HEC-265 CTRP2 0.0020 66.0000
BRD-K13185470 HEC-6 CTRP2 0.0020 66.0000
BRD-K13185470 HEL CTRP2 0.0020 66.0000
BRD-K13185470 JHUEM-2 CTRP2 0.0020 66.0000
BRD-K13185470 JURKAT CTRP2 0.0020 66.0000
BRD-K13185470 KCL-22 CTRP2 0.0020 66.0000
BRD-K13185470 KE-39 CTRP2 0.0020 66.0000
BRD-K13185470 KM-H2 CTRP2 0.0020 66.0000
BRD-K13185470 LAMA-84 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H2030 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-719 CTRP2 0.0020 66.0000
BRD-K13185470 HCC1569 CTRP2 0.0020 66.0000
BRD-K13185470 KLE CTRP2 0.0020 66.0000
BRD-K13185470 KMS-26 CTRP2 0.0020 66.0000
BRD-K13185470 KMS-27 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H1838 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H196 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H292 CTRP2 0.0020 66.0000
BRD-K13185470 SK-MEL-1 CTRP2 0.0020 66.0000
BRD-K13185470 HCC1937 CTRP2 0.0020 66.0000
BRD-K13185470 HDLM-2 CTRP2 0.0020 66.0000
BRD-K13185470 HUH-28 CTRP2 0.0020 66.0000
BRD-K13185470 MV4-11 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H526 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H69 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H929 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-N87 CTRP2 0.0020 66.0000
BRD-K13185470 PF-382 CTRP2 0.0020 66.0000
BRD-K13185470 SF295 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1272 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-308 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-478 CTRP2 0.0020 66.0000
BRD-K13185470 BHT-101 CTRP2 0.0020 66.0000
BRD-K13185470 CAL-148 CTRP2 0.0020 66.0000
BRD-K13185470 CAL-51 CTRP2 0.0020 66.0000
BRD-K13185470 HCC1395 CTRP2 0.0020 66.0000
BRD-K13185470 HT115 CTRP2 0.0020 66.0000
BRD-K13185470 LN-18 CTRP2 0.0020 66.0000
BRD-K13185470 LN-229 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H1734 CTRP2 0.0020 66.0000
BRD-K13185470 NCI-H2291 CTRP2 0.0020 66.0000
BRD-K13185470 RERF-LC-AD1 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-1214 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-46 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-466 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-5 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-668 CTRP2 0.0020 66.0000
BRD-K13185470 SNU-899 CTRP2 0.0020 66.0000
BRD-K13185470 TE-10 CTRP2 0.0020 66.0000
BRD-K13185470 TE-9 CTRP2 0.0020 66.0000
BRD-K13185470 YD-10B CTRP2 0.0020 66.0000
BRD-K13185470 YD-15 CTRP2 0.0020 66.0000
BRD-K13185470 YD-38 CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.