Drug : 2-Deoxyglucose

CTRP1 Name : 2-deoxyglucose

Dataset : All
Synonyms :
Targets : HK2
Pathways : inhibitor of glycolysis via hexokinase

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
2-deoxyglucose GAMG CTRP1 0.2890 37.0080
2-deoxyglucose SF295 CTRP1 0.2890 37.0080
2-deoxyglucose HEC-108 CTRP1 0.2890 37.0080
2-deoxyglucose HEC-251 CTRP1 0.2890 37.0080
2-deoxyglucose HEC-265 CTRP1 0.2890 37.0080
2-deoxyglucose HEC-59 CTRP1 0.2890 37.0080
2-deoxyglucose HEC-6 CTRP1 0.2890 37.0080
2-deoxyglucose ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2890 37.0080
2-deoxyglucose KLE CTRP1 0.2890 37.0080
2-deoxyglucose MFE-319 CTRP1 0.2890 37.0080
2-deoxyglucose SNG-M CTRP1 0.2890 37.0080
2-deoxyglucose BL-70 CTRP1 0.2890 37.0080
2-deoxyglucose HT CTRP1 0.2890 37.0080
2-deoxyglucose KU812 CTRP1 0.2890 37.0080
2-deoxyglucose MC116 CTRP1 0.2890 37.0080
2-deoxyglucose P3HR-1 CTRP1 0.2890 37.0080
2-deoxyglucose VMRC-RCW CTRP1 0.2890 37.0080
2-deoxyglucose C2BBE1 CTRP1 0.2890 37.0080
2-deoxyglucose COLO205 CTRP1 0.2890 37.0080
2-deoxyglucose DLD-1 CTRP1 0.2890 37.0080
2-deoxyglucose GP2D CTRP1 0.2890 37.0080
2-deoxyglucose LS411N CTRP1 0.2890 37.0080
2-deoxyglucose LS513 CTRP1 0.2890 37.0080
2-deoxyglucose SK-CO-1 CTRP1 0.2890 37.0080
2-deoxyglucose SNU-C2A CTRP1 0.2890 37.0080
2-deoxyglucose SW403 CTRP1 0.2890 37.0080
2-deoxyglucose SW48 CTRP1 0.2890 37.0080
2-deoxyglucose JHH-6 CTRP1 0.2890 37.0080
2-deoxyglucose SNU-449 CTRP1 0.2890 37.0080
2-deoxyglucose A-549 CTRP1 0.2890 37.0080
2-deoxyglucose BEN CTRP1 0.2890 37.0080
2-deoxyglucose CALU-3 CTRP1 0.2890 37.0080
2-deoxyglucose CALU-6 CTRP1 0.2890 37.0080
2-deoxyglucose CHAGO-K-1 CTRP1 0.2890 37.0080
2-deoxyglucose COLO668 CTRP1 0.2890 37.0080
2-deoxyglucose COR-L279 CTRP1 0.2890 37.0080
2-deoxyglucose COR-L88 CTRP1 0.2890 37.0080
2-deoxyglucose DMS273 CTRP1 0.2890 37.0080
2-deoxyglucose DV-90 CTRP1 0.2890 37.0080
2-deoxyglucose EBC-1 CTRP1 0.2890 37.0080
2-deoxyglucose EPLC-272H CTRP1 0.2890 37.0080
2-deoxyglucose HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2890 37.0080
2-deoxyglucose HCC33 CTRP1 0.2890 37.0080
2-deoxyglucose HCC44 CTRP1 0.2890 37.0080
2-deoxyglucose HCC78 CTRP1 0.2890 37.0080
2-deoxyglucose KNS-62 CTRP1 0.2890 37.0080
2-deoxyglucose LC-1-SQ-SF CTRP1 0.2890 37.0080
2-deoxyglucose LCLC-103H CTRP1 0.2890 37.0080
2-deoxyglucose LCLC-97TM1 CTRP1 0.2890 37.0080
2-deoxyglucose LU-65 CTRP1 0.2890 37.0080
2-deoxyglucose LU-99 CTRP1 0.2890 37.0080
2-deoxyglucose LXF289 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1048 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1299 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1355 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1373 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1435 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1437 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1568 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1573 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1666 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1792 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1793 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1915 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1930 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1944 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H1975 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H2009 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H2029 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H2126 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H2286 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H23 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H2405 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H358 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H522 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H650 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H661 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H727 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H810 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H82 CTRP1 0.2890 37.0080
2-deoxyglucose RERF-LC-KJ CTRP1 0.2890 37.0080
2-deoxyglucose SHP-77 CTRP1 0.2890 37.0080
2-deoxyglucose VMRC-LCD CTRP1 0.2890 37.0080
2-deoxyglucose KYSE-140 CTRP1 0.2890 37.0080
2-deoxyglucose KYSE-410 CTRP1 0.2890 37.0080
2-deoxyglucose KYSE-450 CTRP1 0.2890 37.0080
2-deoxyglucose COV318 CTRP1 0.2890 37.0080
2-deoxyglucose EFO-21 CTRP1 0.2890 37.0080
2-deoxyglucose HEYA8 CTRP1 0.2890 37.0080
2-deoxyglucose JHOS-4 CTRP1 0.2890 37.0080
2-deoxyglucose OVMANA CTRP1 0.2890 37.0080
2-deoxyglucose SK-OV-3 CTRP1 0.2890 37.0080
2-deoxyglucose CAPAN-2 CTRP1 0.2890 37.0080
2-deoxyglucose CFPAC-1 CTRP1 0.2890 37.0080
2-deoxyglucose HPAC CTRP1 0.2890 37.0080
2-deoxyglucose HUP-T4 CTRP1 0.2890 37.0080
2-deoxyglucose KP-3 CTRP1 0.2890 37.0080
2-deoxyglucose PANC03.27 CTRP1 0.2890 37.0080
2-deoxyglucose PANC10.05 CTRP1 0.2890 37.0080
2-deoxyglucose PATU8902 CTRP1 0.2890 37.0080
2-deoxyglucose QGP-1 CTRP1 0.2890 37.0080
2-deoxyglucose SUIT-2 CTRP1 0.2890 37.0080
2-deoxyglucose MSTO-211H CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H2052 CTRP1 0.2890 37.0080
2-deoxyglucose NCI-H28 CTRP1 0.2890 37.0080
2-deoxyglucose MIAPACA-3 CTRP1 0.2890 37.0080
2-deoxyglucose COLO741 CTRP1 0.2890 37.0080
2-deoxyglucose G-361 CTRP1 0.2890 37.0080
2-deoxyglucose HS852.T CTRP1 0.2890 37.0080
2-deoxyglucose HS936.T CTRP1 0.2890 37.0080
2-deoxyglucose HS944.T CTRP1 0.2890 37.0080
2-deoxyglucose G-401 CTRP1 0.2890 37.0080
2-deoxyglucose FU97 CTRP1 0.2890 37.0080
2-deoxyglucose KE-97 CTRP1 0.2890 37.0080
2-deoxyglucose MKN7 CTRP1 0.2890 37.0080
2-deoxyglucose MKN74 CTRP1 0.2890 37.0080
2-deoxyglucose NUGC-4 CTRP1 0.2890 37.0080
2-deoxyglucose SH-10-TC CTRP1 0.2890 37.0080
2-deoxyglucose HSC-2 CTRP1 0.2890 37.0080
2-deoxyglucose 5637 CTRP1 0.2890 37.0080
2-deoxyglucose HT-1376 CTRP1 0.2890 37.0080
2-deoxyglucose KMBC-2 CTRP1 0.2890 37.0080
2-deoxyglucose RT-4 CTRP1 0.2890 37.0080
2-deoxyglucose UM-UC-3 CTRP1 0.2890 37.0080

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.