Drug : 6-Diazo-5-Oxo-L-Norleucine

CTRP1 Name : 6-diazo-5-oxo-L-norleucine

Dataset : All
Synonyms :
Targets : GLS
Pathways : inhibitor of glutaminase;inhibitor of glutamine-dependent biosynthetic pathways

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
6-diazo-5-oxo-L-norleucine MCF-7 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine GAMG CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LN-229 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SF295 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HEC-108 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HEC-151 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HEC-251 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HEC-265 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HEC-59 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HEC-6 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine JHUEM-2 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine KLE CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine MFE-319 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SNG-M CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine AMO1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine BL-70 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine EJM CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine GDM-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HT CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine KMS-11 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine KU812 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LP-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine MC116 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine MOLM-16 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NOMO-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NU-DUL-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OCI-AML-3 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OCI-LY10 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine P3HR-1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine PL21 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine RPMI-8226 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SKM-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SU-DHL-4 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SU-DHL-5 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine THP-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine U-937 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine WSU-DLCL2 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine RCC10RGB CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine VMRC-RCW CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine C2BBE1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine CL-34 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine CL-40 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COLO205 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine COLO320 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COLO678 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine CW-2 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine DLD-1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine GP2D CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HCT116 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HCT8 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HT115 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HT-29 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HT-55 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine KM12 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine LOVO CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine LS123 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine LS180 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine LS411N CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LS513 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine MDST8 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H508 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine RCM-1[HUMANESC] CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine RKO CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SK-CO-1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SNU-1040 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SNU-175 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SNU-61 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SNU-81 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SNU-C2A CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SNU-C4 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SNU-C5 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SW403 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SW48 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SW480 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SW620 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SW948 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HEP-G2 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine JHH-6 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SNU-398 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SNU-449 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine A-549 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine BEN CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine CAL-12T CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine CALU-3 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine CALU-6 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine CHAGO-K-1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine COLO668 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine COLO699 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COR-L23 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COR-L279 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine COR-L51 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COR-L88 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine DMS273 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine DV-90 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine EBC-1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine EPLC-272H CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HCC1195 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HCC1359 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HCC15 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HCC1833 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HCC2108 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HCC2935 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HCC33 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HCC4006 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HCC44 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HCC78 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HCC827 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine KNS-62 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LC-1-SQ-SF CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LCLC-103H CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LCLC-97TM1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LU-65 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LU-99 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine LXF289 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1048 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1105 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H1299 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1355 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1373 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1435 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1437 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1568 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1573 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1666 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1694 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H1755 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H1781 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H1792 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1793 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1836 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H1876 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H1915 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1930 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1944 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H1963 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H1975 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H2009 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H2023 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2029 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H2030 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2073 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2081 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2110 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2122 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2126 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H2141 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2172 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2286 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H23 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H2342 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H2405 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H3255 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H358 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H441 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H460 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H522 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H596 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine NCI-H650 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H661 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H727 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H810 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H82 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H841 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine RERF-LC-KJ CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SCLC-21H CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SHP-77 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SK-LU-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SQ-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine T3M-10 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine VMRC-LCD CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine KYSE-140 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine KYSE-410 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine KYSE-450 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine A2780 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine CAOV-3 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COV318 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine COV362 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COV434 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COV644 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine EFO-21 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine EFO-27 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine HEYA8 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine IGROV-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine JHOC-5 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine JHOM-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine JHOS-4 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine OAW42 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OV7 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OV-90 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OVCAR-4 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OVCAR-8 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OVK18 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OVKATE CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine OVMANA CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine RKN CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine RMG-I CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine RMUG-S CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SK-OV-3 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SNU-840 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine TYK-NU CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine CAPAN-2 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine CFPAC-1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HPAC CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HUP-T4 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine KP-3 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine PANC03.27 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine PANC10.05 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine PATU8902 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine QGP-1 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SUIT-2 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine MSTO-211H CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H2052 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NCI-H28 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine MIAPACA-3 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine A-375 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine COLO741 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine G-361 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HS852.T CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HS936.T CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HS944.T CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SK-MEL-1 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SK-MEL-28 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine SK-MEL-5 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine G-401 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HT-1080 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine AGS CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine FU97 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine KE-97 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine MKN7 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine MKN74 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine NUGC-4 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SH-10-TC CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HSC-2 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine SCC-9 CTRP1 1.0417 133.3300
6-diazo-5-oxo-L-norleucine 5637 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine HT-1376 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine KMBC-2 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine RT-4 CTRP1 0.2603 33.3330
6-diazo-5-oxo-L-norleucine UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.