Drug : Losartan

CTRP1 Name : losartan

Dataset : All
Synonyms :
Targets : AGTR2
Pathways : inhibitor of angiotensin II receptor

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
losartan U2OS CTRP1 4.1667 533.3300
losartan MCF-7 CTRP1 4.1667 533.3300
losartan GAMG CTRP1 0.2603 33.3330
losartan LN-229 CTRP1 4.1667 533.3300
losartan SF295 CTRP1 0.2603 33.3330
losartan HEC-108 CTRP1 0.2603 33.3330
losartan HEC-151 CTRP1 4.1667 533.3300
losartan HEC-251 CTRP1 0.2603 33.3330
losartan HEC-265 CTRP1 0.2603 33.3330
losartan HEC-59 CTRP1 0.2603 33.3330
losartan HEC-6 CTRP1 0.2603 33.3330
losartan ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
losartan JHUEM-2 CTRP1 4.1667 533.3300
losartan KLE CTRP1 0.2603 33.3330
losartan MFE-319 CTRP1 0.2603 33.3330
losartan SNG-M CTRP1 0.2603 33.3330
losartan AMO1 CTRP1 4.1667 533.3300
losartan BL-70 CTRP1 0.2603 33.3330
losartan EJM CTRP1 4.1667 533.3300
losartan GDM-1 CTRP1 4.1667 533.3300
losartan HT CTRP1 0.2603 33.3330
losartan KMS-11 CTRP1 4.1667 533.3300
losartan KU812 CTRP1 0.2603 33.3330
losartan LP-1 CTRP1 4.1667 533.3300
losartan MC116 CTRP1 0.2603 33.3330
losartan MOLM-16 CTRP1 4.1667 533.3300
losartan NOMO-1 CTRP1 4.1667 533.3300
losartan NU-DUL-1 CTRP1 4.1667 533.3300
losartan OCI-AML-3 CTRP1 4.1667 533.3300
losartan OCI-LY10 CTRP1 4.1667 533.3300
losartan P3HR-1 CTRP1 0.2603 33.3330
losartan PL21 CTRP1 4.1667 533.3300
losartan RPMI-8226 CTRP1 4.1667 533.3300
losartan SKM-1 CTRP1 4.1667 533.3300
losartan SU-DHL-4 CTRP1 4.1667 533.3300
losartan SU-DHL-5 CTRP1 4.1667 533.3300
losartan THP-1 CTRP1 4.1667 533.3300
losartan U-937 CTRP1 4.1667 533.3300
losartan WSU-DLCL2 CTRP1 4.1667 533.3300
losartan RCC10RGB CTRP1 4.1667 533.3300
losartan VMRC-RCW CTRP1 0.2603 33.3330
losartan C2BBE1 CTRP1 0.2603 33.3330
losartan CL-34 CTRP1 4.1667 533.3300
losartan CL-40 CTRP1 4.1667 533.3300
losartan COLO205 CTRP1 0.2603 33.3330
losartan COLO320 CTRP1 4.1667 533.3300
losartan COLO678 CTRP1 4.1667 533.3300
losartan CW-2 CTRP1 4.1667 533.3300
losartan DLD-1 CTRP1 0.2603 33.3330
losartan GP2D CTRP1 0.2603 33.3330
losartan HCT116 CTRP1 4.1667 533.3300
losartan HCT8 CTRP1 4.1667 533.3300
losartan HT115 CTRP1 4.1667 533.3300
losartan HT-29 CTRP1 4.1667 533.3300
losartan HT-55 CTRP1 4.1667 533.3300
losartan KM12 CTRP1 4.1667 533.3300
losartan LOVO CTRP1 4.1667 533.3300
losartan LS123 CTRP1 4.1667 533.3300
losartan LS180 CTRP1 4.1667 533.3300
losartan LS411N CTRP1 0.2603 33.3330
losartan LS513 CTRP1 0.2603 33.3330
losartan MDST8 CTRP1 4.1667 533.3300
losartan NCI-H508 CTRP1 4.1667 533.3300
losartan RCM-1[HUMANESC] CTRP1 4.1667 533.3300
losartan RKO CTRP1 4.1667 533.3300
losartan SK-CO-1 CTRP1 0.2603 33.3330
losartan SNU-1040 CTRP1 4.1667 533.3300
losartan SNU-175 CTRP1 4.1667 533.3300
losartan SNU-61 CTRP1 4.1667 533.3300
losartan SNU-81 CTRP1 4.1667 533.3300
losartan SNU-C2A CTRP1 0.2603 33.3330
losartan SNU-C4 CTRP1 4.1667 533.3300
losartan SNU-C5 CTRP1 4.1667 533.3300
losartan SW403 CTRP1 0.2603 33.3330
losartan SW48 CTRP1 0.2603 33.3330
losartan SW480 CTRP1 4.1667 533.3300
losartan SW620 CTRP1 4.1667 533.3300
losartan SW948 CTRP1 4.1667 533.3300
losartan HEP-G2 CTRP1 4.1667 533.3300
losartan JHH-6 CTRP1 0.2603 33.3330
losartan SNU-398 CTRP1 4.1667 533.3300
losartan SNU-449 CTRP1 0.2603 33.3330
losartan A-549 CTRP1 0.2603 33.3330
losartan BEN CTRP1 0.2603 33.3330
losartan CAL-12T CTRP1 4.1667 533.3300
losartan CALU-3 CTRP1 0.2603 33.3330
losartan CALU-6 CTRP1 0.2603 33.3330
losartan CHAGO-K-1 CTRP1 0.2603 33.3330
losartan COLO668 CTRP1 0.2603 33.3330
losartan COLO699 CTRP1 4.1667 533.3300
losartan COR-L23 CTRP1 4.1667 533.3300
losartan COR-L279 CTRP1 0.2603 33.3330
losartan COR-L51 CTRP1 4.1667 533.3300
losartan COR-L88 CTRP1 0.2603 33.3330
losartan DMS273 CTRP1 0.2603 33.3330
losartan DV-90 CTRP1 0.2603 33.3330
losartan EBC-1 CTRP1 0.2603 33.3330
losartan EPLC-272H CTRP1 0.2603 33.3330
losartan HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
losartan HCC1195 CTRP1 4.1667 533.3300
losartan HCC1359 CTRP1 4.1667 533.3300
losartan HCC15 CTRP1 4.1667 533.3300
losartan HCC1833 CTRP1 4.1667 533.3300
losartan HCC2108 CTRP1 4.1667 533.3300
losartan HCC2935 CTRP1 4.1667 533.3300
losartan HCC33 CTRP1 0.2603 33.3330
losartan HCC4006 CTRP1 4.1667 533.3300
losartan HCC44 CTRP1 0.2603 33.3330
losartan HCC78 CTRP1 0.2603 33.3330
losartan HCC827 CTRP1 4.1667 533.3300
losartan KNS-62 CTRP1 0.2603 33.3330
losartan LC-1-SQ-SF CTRP1 0.2603 33.3330
losartan LCLC-103H CTRP1 0.2603 33.3330
losartan LCLC-97TM1 CTRP1 0.2603 33.3330
losartan LU-65 CTRP1 0.2603 33.3330
losartan LU-99 CTRP1 0.2603 33.3330
losartan LXF289 CTRP1 0.2603 33.3330
losartan NCI-H1048 CTRP1 0.2603 33.3330
losartan NCI-H1105 CTRP1 4.1667 533.3300
losartan NCI-H1299 CTRP1 0.2603 33.3330
losartan NCI-H1355 CTRP1 0.2603 33.3330
losartan NCI-H1373 CTRP1 0.2603 33.3330
losartan NCI-H1435 CTRP1 0.2603 33.3330
losartan NCI-H1437 CTRP1 0.2603 33.3330
losartan NCI-H1568 CTRP1 0.2603 33.3330
losartan NCI-H1573 CTRP1 0.2603 33.3330
losartan NCI-H1666 CTRP1 0.2603 33.3330
losartan NCI-H1694 CTRP1 4.1667 533.3300
losartan NCI-H1755 CTRP1 4.1667 533.3300
losartan NCI-H1781 CTRP1 4.1667 533.3300
losartan NCI-H1792 CTRP1 0.2603 33.3330
losartan NCI-H1793 CTRP1 0.2603 33.3330
losartan NCI-H1836 CTRP1 4.1667 533.3300
losartan NCI-H1876 CTRP1 4.1667 533.3300
losartan NCI-H1915 CTRP1 0.2603 33.3330
losartan NCI-H1930 CTRP1 0.2603 33.3330
losartan NCI-H1944 CTRP1 0.2603 33.3330
losartan NCI-H1963 CTRP1 4.1667 533.3300
losartan NCI-H1975 CTRP1 0.2603 33.3330
losartan NCI-H2009 CTRP1 0.2603 33.3330
losartan NCI-H2023 CTRP1 4.1667 533.3300
losartan NCI-H2029 CTRP1 0.2603 33.3330
losartan NCI-H2030 CTRP1 4.1667 533.3300
losartan NCI-H2073 CTRP1 4.1667 533.3300
losartan NCI-H2081 CTRP1 4.1667 533.3300
losartan NCI-H2110 CTRP1 4.1667 533.3300
losartan NCI-H2122 CTRP1 4.1667 533.3300
losartan NCI-H2126 CTRP1 0.2603 33.3330
losartan NCI-H2141 CTRP1 4.1667 533.3300
losartan NCI-H2172 CTRP1 4.1667 533.3300
losartan NCI-H2286 CTRP1 0.2603 33.3330
losartan NCI-H23 CTRP1 0.2603 33.3330
losartan NCI-H2342 CTRP1 4.1667 533.3300
losartan NCI-H2405 CTRP1 0.2603 33.3330
losartan NCI-H3255 CTRP1 4.1667 533.3300
losartan NCI-H358 CTRP1 0.2603 33.3330
losartan NCI-H441 CTRP1 4.1667 533.3300
losartan NCI-H460 CTRP1 4.1667 533.3300
losartan NCI-H522 CTRP1 0.2603 33.3330
losartan NCI-H596 CTRP1 4.1667 533.3300
losartan NCI-H650 CTRP1 0.2603 33.3330
losartan NCI-H661 CTRP1 0.2603 33.3330
losartan NCI-H727 CTRP1 0.2603 33.3330
losartan NCI-H810 CTRP1 0.2603 33.3330
losartan NCI-H82 CTRP1 0.2603 33.3330
losartan NCI-H841 CTRP1 4.1667 533.3300
losartan RERF-LC-KJ CTRP1 0.2603 33.3330
losartan SCLC-21H CTRP1 4.1667 533.3300
losartan SHP-77 CTRP1 0.2603 33.3330
losartan SK-LU-1 CTRP1 4.1667 533.3300
losartan SQ-1 CTRP1 4.1667 533.3300
losartan T3M-10 CTRP1 4.1667 533.3300
losartan VMRC-LCD CTRP1 0.2603 33.3330
losartan KYSE-140 CTRP1 0.2603 33.3330
losartan KYSE-410 CTRP1 0.2603 33.3330
losartan KYSE-450 CTRP1 0.2603 33.3330
losartan A2780 CTRP1 4.1667 533.3300
losartan CAOV-3 CTRP1 4.1667 533.3300
losartan COV318 CTRP1 0.2603 33.3330
losartan COV362 CTRP1 4.1667 533.3300
losartan COV434 CTRP1 4.1667 533.3300
losartan COV644 CTRP1 4.1667 533.3300
losartan EFO-21 CTRP1 0.2603 33.3330
losartan EFO-27 CTRP1 4.1667 533.3300
losartan HEYA8 CTRP1 0.2603 33.3330
losartan IGROV-1 CTRP1 4.1667 533.3300
losartan JHOC-5 CTRP1 4.1667 533.3300
losartan JHOM-1 CTRP1 4.1667 533.3300
losartan JHOS-4 CTRP1 0.2603 33.3330
losartan OAW42 CTRP1 4.1667 533.3300
losartan OV7 CTRP1 4.1667 533.3300
losartan OV-90 CTRP1 4.1667 533.3300
losartan OVCAR-4 CTRP1 4.1667 533.3300
losartan OVCAR-8 CTRP1 4.1667 533.3300
losartan OVK18 CTRP1 4.1667 533.3300
losartan OVKATE CTRP1 4.1667 533.3300
losartan OVMANA CTRP1 0.2603 33.3330
losartan RKN CTRP1 4.1667 533.3300
losartan RMG-I CTRP1 4.1667 533.3300
losartan RMUG-S CTRP1 4.1667 533.3300
losartan SK-OV-3 CTRP1 0.2603 33.3330
losartan SNU-840 CTRP1 4.1667 533.3300
losartan TYK-NU CTRP1 4.1667 533.3300
losartan CAPAN-2 CTRP1 0.2603 33.3330
losartan CFPAC-1 CTRP1 0.2603 33.3330
losartan HPAC CTRP1 0.2603 33.3330
losartan HUP-T4 CTRP1 0.2603 33.3330
losartan KP-3 CTRP1 0.2603 33.3330
losartan PANC03.27 CTRP1 0.2603 33.3330
losartan PANC10.05 CTRP1 0.2603 33.3330
losartan PATU8902 CTRP1 0.2603 33.3330
losartan QGP-1 CTRP1 0.2603 33.3330
losartan SUIT-2 CTRP1 0.2603 33.3330
losartan MSTO-211H CTRP1 0.2603 33.3330
losartan NCI-H2052 CTRP1 0.2603 33.3330
losartan NCI-H28 CTRP1 0.2603 33.3330
losartan MIAPACA-3 CTRP1 0.2603 33.3330
losartan A-375 CTRP1 4.1667 533.3300
losartan COLO741 CTRP1 0.2603 33.3330
losartan G-361 CTRP1 0.2603 33.3330
losartan HS852.T CTRP1 0.2603 33.3330
losartan HS936.T CTRP1 0.2603 33.3330
losartan HS944.T CTRP1 0.2603 33.3330
losartan SK-MEL-1 CTRP1 4.1667 533.3300
losartan SK-MEL-28 CTRP1 4.1667 533.3300
losartan SK-MEL-5 CTRP1 4.1667 533.3300
losartan G-401 CTRP1 0.2603 33.3330
losartan HT-1080 CTRP1 4.1667 533.3300
losartan AGS CTRP1 4.1667 533.3300
losartan FU97 CTRP1 0.2603 33.3330
losartan KE-97 CTRP1 0.2603 33.3330
losartan MKN7 CTRP1 0.2603 33.3330
losartan MKN74 CTRP1 0.2603 33.3330
losartan NUGC-4 CTRP1 0.2603 33.3330
losartan SH-10-TC CTRP1 0.2603 33.3330
losartan HSC-2 CTRP1 0.2603 33.3330
losartan SCC-9 CTRP1 4.1667 533.3300
losartan 5637 CTRP1 0.2603 33.3330
losartan HT-1376 CTRP1 0.2603 33.3330
losartan KMBC-2 CTRP1 0.2603 33.3330
losartan RT-4 CTRP1 0.2603 33.3330
losartan UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.