Drug : Wt-161

CTRP1 Name : WT-161

Dataset : All
Synonyms :
Targets : HDAC6
Pathways : inhibitor of HDAC6;inhibitor of tubulin deacetylation

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
WT-161 U2OS CTRP1 0.2604 33.3330
WT-161 MCF-7 CTRP1 0.2604 33.3330
WT-161 GAMG CTRP1 0.2603 33.3330
WT-161 LN-229 CTRP1 0.2604 33.3330
WT-161 SF295 CTRP1 0.2603 33.3330
WT-161 HEC-108 CTRP1 0.2603 33.3330
WT-161 HEC-151 CTRP1 0.2604 33.3330
WT-161 HEC-251 CTRP1 0.2603 33.3330
WT-161 HEC-265 CTRP1 0.2603 33.3330
WT-161 HEC-59 CTRP1 0.2603 33.3330
WT-161 HEC-6 CTRP1 0.2603 33.3330
WT-161 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
WT-161 JHUEM-2 CTRP1 0.2604 33.3330
WT-161 KLE CTRP1 0.2603 33.3330
WT-161 MFE-319 CTRP1 0.2603 33.3330
WT-161 SNG-M CTRP1 0.2603 33.3330
WT-161 AMO1 CTRP1 0.2604 33.3330
WT-161 BL-70 CTRP1 0.2603 33.3330
WT-161 EJM CTRP1 0.2604 33.3330
WT-161 GDM-1 CTRP1 0.2604 33.3330
WT-161 HT CTRP1 0.2603 33.3330
WT-161 KMS-11 CTRP1 0.2604 33.3330
WT-161 KU812 CTRP1 0.2603 33.3330
WT-161 LP-1 CTRP1 0.2604 33.3330
WT-161 MC116 CTRP1 0.2603 33.3330
WT-161 MOLM-16 CTRP1 0.2604 33.3330
WT-161 NOMO-1 CTRP1 0.2604 33.3330
WT-161 NU-DUL-1 CTRP1 0.2604 33.3330
WT-161 OCI-AML-3 CTRP1 0.2604 33.3330
WT-161 OCI-LY10 CTRP1 0.2604 33.3330
WT-161 P3HR-1 CTRP1 0.2603 33.3330
WT-161 PL21 CTRP1 0.2604 33.3330
WT-161 RPMI-8226 CTRP1 0.2604 33.3330
WT-161 SKM-1 CTRP1 0.2604 33.3330
WT-161 SU-DHL-4 CTRP1 0.2604 33.3330
WT-161 SU-DHL-5 CTRP1 0.2604 33.3330
WT-161 THP-1 CTRP1 0.2604 33.3330
WT-161 U-937 CTRP1 0.2604 33.3330
WT-161 WSU-DLCL2 CTRP1 0.2604 33.3330
WT-161 RCC10RGB CTRP1 0.2604 33.3330
WT-161 VMRC-RCW CTRP1 0.2603 33.3330
WT-161 C2BBE1 CTRP1 0.2603 33.3330
WT-161 CL-34 CTRP1 0.2604 33.3330
WT-161 CL-40 CTRP1 0.2604 33.3330
WT-161 COLO205 CTRP1 0.2603 33.3330
WT-161 COLO320 CTRP1 0.2604 33.3330
WT-161 COLO678 CTRP1 0.2604 33.3330
WT-161 CW-2 CTRP1 0.2604 33.3330
WT-161 DLD-1 CTRP1 0.2603 33.3330
WT-161 GP2D CTRP1 0.2603 33.3330
WT-161 HCT116 CTRP1 0.2604 33.3330
WT-161 HCT8 CTRP1 0.2604 33.3330
WT-161 HT115 CTRP1 0.2604 33.3330
WT-161 HT-29 CTRP1 0.2604 33.3330
WT-161 HT-55 CTRP1 0.2604 33.3330
WT-161 KM12 CTRP1 0.2604 33.3330
WT-161 LOVO CTRP1 0.2604 33.3330
WT-161 LS123 CTRP1 0.2604 33.3330
WT-161 LS180 CTRP1 0.2604 33.3330
WT-161 LS411N CTRP1 0.2603 33.3330
WT-161 LS513 CTRP1 0.2603 33.3330
WT-161 MDST8 CTRP1 0.2604 33.3330
WT-161 NCI-H508 CTRP1 0.2604 33.3330
WT-161 RCM-1[HUMANESC] CTRP1 0.2604 33.3330
WT-161 RKO CTRP1 0.2604 33.3330
WT-161 SK-CO-1 CTRP1 0.2603 33.3330
WT-161 SNU-1040 CTRP1 0.2604 33.3330
WT-161 SNU-175 CTRP1 0.2604 33.3330
WT-161 SNU-61 CTRP1 0.2604 33.3330
WT-161 SNU-81 CTRP1 0.2604 33.3330
WT-161 SNU-C2A CTRP1 0.2603 33.3330
WT-161 SNU-C4 CTRP1 0.2604 33.3330
WT-161 SNU-C5 CTRP1 0.2604 33.3330
WT-161 SW403 CTRP1 0.2603 33.3330
WT-161 SW48 CTRP1 0.2603 33.3330
WT-161 SW480 CTRP1 0.2604 33.3330
WT-161 SW620 CTRP1 0.2604 33.3330
WT-161 SW948 CTRP1 0.2604 33.3330
WT-161 HEP-G2 CTRP1 0.2604 33.3330
WT-161 JHH-6 CTRP1 0.2603 33.3330
WT-161 SNU-398 CTRP1 0.2604 33.3330
WT-161 SNU-449 CTRP1 0.2603 33.3330
WT-161 A-549 CTRP1 0.2603 33.3330
WT-161 BEN CTRP1 0.2603 33.3330
WT-161 CAL-12T CTRP1 0.2604 33.3330
WT-161 CALU-3 CTRP1 0.2603 33.3330
WT-161 CALU-6 CTRP1 0.2603 33.3330
WT-161 CHAGO-K-1 CTRP1 0.2603 33.3330
WT-161 COLO668 CTRP1 0.2603 33.3330
WT-161 COLO699 CTRP1 0.2604 33.3330
WT-161 COR-L23 CTRP1 0.2604 33.3330
WT-161 COR-L279 CTRP1 0.2603 33.3330
WT-161 COR-L51 CTRP1 0.2604 33.3330
WT-161 COR-L88 CTRP1 0.2603 33.3330
WT-161 DMS273 CTRP1 0.2603 33.3330
WT-161 DV-90 CTRP1 0.2603 33.3330
WT-161 EBC-1 CTRP1 0.2603 33.3330
WT-161 EPLC-272H CTRP1 0.2603 33.3330
WT-161 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
WT-161 HCC1195 CTRP1 0.2604 33.3330
WT-161 HCC1359 CTRP1 0.2604 33.3330
WT-161 HCC15 CTRP1 0.2604 33.3330
WT-161 HCC1833 CTRP1 0.2604 33.3330
WT-161 HCC2108 CTRP1 0.2604 33.3330
WT-161 HCC2935 CTRP1 0.2604 33.3330
WT-161 HCC33 CTRP1 0.2603 33.3330
WT-161 HCC4006 CTRP1 0.2604 33.3330
WT-161 HCC44 CTRP1 0.2603 33.3330
WT-161 HCC78 CTRP1 0.2603 33.3330
WT-161 HCC827 CTRP1 0.2604 33.3330
WT-161 KNS-62 CTRP1 0.2603 33.3330
WT-161 LC-1-SQ-SF CTRP1 0.2603 33.3330
WT-161 LCLC-103H CTRP1 0.2603 33.3330
WT-161 LCLC-97TM1 CTRP1 0.2603 33.3330
WT-161 LU-65 CTRP1 0.2603 33.3330
WT-161 LU-99 CTRP1 0.2603 33.3330
WT-161 LXF289 CTRP1 0.2603 33.3330
WT-161 NCI-H1048 CTRP1 0.2603 33.3330
WT-161 NCI-H1105 CTRP1 0.2604 33.3330
WT-161 NCI-H1299 CTRP1 0.2603 33.3330
WT-161 NCI-H1355 CTRP1 0.2603 33.3330
WT-161 NCI-H1373 CTRP1 0.2603 33.3330
WT-161 NCI-H1435 CTRP1 0.2603 33.3330
WT-161 NCI-H1437 CTRP1 0.2603 33.3330
WT-161 NCI-H1568 CTRP1 0.2603 33.3330
WT-161 NCI-H1573 CTRP1 0.2603 33.3330
WT-161 NCI-H1666 CTRP1 0.2603 33.3330
WT-161 NCI-H1694 CTRP1 0.2604 33.3330
WT-161 NCI-H1755 CTRP1 0.2604 33.3330
WT-161 NCI-H1781 CTRP1 0.2604 33.3330
WT-161 NCI-H1792 CTRP1 0.2603 33.3330
WT-161 NCI-H1793 CTRP1 0.2603 33.3330
WT-161 NCI-H1836 CTRP1 0.2604 33.3330
WT-161 NCI-H1876 CTRP1 0.2604 33.3330
WT-161 NCI-H1915 CTRP1 0.2603 33.3330
WT-161 NCI-H1930 CTRP1 0.2603 33.3330
WT-161 NCI-H1944 CTRP1 0.2603 33.3330
WT-161 NCI-H1963 CTRP1 0.2604 33.3330
WT-161 NCI-H1975 CTRP1 0.2603 33.3330
WT-161 NCI-H2009 CTRP1 0.2603 33.3330
WT-161 NCI-H2023 CTRP1 0.2604 33.3330
WT-161 NCI-H2029 CTRP1 0.2603 33.3330
WT-161 NCI-H2030 CTRP1 0.2604 33.3330
WT-161 NCI-H2073 CTRP1 0.2604 33.3330
WT-161 NCI-H2081 CTRP1 0.2604 33.3330
WT-161 NCI-H2110 CTRP1 0.2604 33.3330
WT-161 NCI-H2122 CTRP1 0.2604 33.3330
WT-161 NCI-H2126 CTRP1 0.2603 33.3330
WT-161 NCI-H2141 CTRP1 0.2604 33.3330
WT-161 NCI-H2172 CTRP1 0.2604 33.3330
WT-161 NCI-H2286 CTRP1 0.2603 33.3330
WT-161 NCI-H23 CTRP1 0.2603 33.3330
WT-161 NCI-H2342 CTRP1 0.2604 33.3330
WT-161 NCI-H2405 CTRP1 0.2603 33.3330
WT-161 NCI-H3255 CTRP1 0.2604 33.3330
WT-161 NCI-H358 CTRP1 0.2603 33.3330
WT-161 NCI-H441 CTRP1 0.2604 33.3330
WT-161 NCI-H460 CTRP1 0.2604 33.3330
WT-161 NCI-H522 CTRP1 0.2603 33.3330
WT-161 NCI-H596 CTRP1 0.2604 33.3330
WT-161 NCI-H650 CTRP1 0.2603 33.3330
WT-161 NCI-H661 CTRP1 0.2603 33.3330
WT-161 NCI-H727 CTRP1 0.2603 33.3330
WT-161 NCI-H810 CTRP1 0.2603 33.3330
WT-161 NCI-H82 CTRP1 0.2603 33.3330
WT-161 NCI-H841 CTRP1 0.2604 33.3330
WT-161 RERF-LC-KJ CTRP1 0.2603 33.3330
WT-161 SCLC-21H CTRP1 0.2604 33.3330
WT-161 SHP-77 CTRP1 0.2603 33.3330
WT-161 SK-LU-1 CTRP1 0.2604 33.3330
WT-161 SQ-1 CTRP1 0.2604 33.3330
WT-161 T3M-10 CTRP1 0.2604 33.3330
WT-161 VMRC-LCD CTRP1 0.2603 33.3330
WT-161 KYSE-140 CTRP1 0.2603 33.3330
WT-161 KYSE-410 CTRP1 0.2603 33.3330
WT-161 KYSE-450 CTRP1 0.2603 33.3330
WT-161 A2780 CTRP1 0.2604 33.3330
WT-161 CAOV-3 CTRP1 0.2604 33.3330
WT-161 COV318 CTRP1 0.2603 33.3330
WT-161 COV362 CTRP1 0.2604 33.3330
WT-161 COV434 CTRP1 0.2604 33.3330
WT-161 COV644 CTRP1 0.2604 33.3330
WT-161 EFO-21 CTRP1 0.2603 33.3330
WT-161 EFO-27 CTRP1 0.2604 33.3330
WT-161 HEYA8 CTRP1 0.2603 33.3330
WT-161 IGROV-1 CTRP1 0.2604 33.3330
WT-161 JHOC-5 CTRP1 0.2604 33.3330
WT-161 JHOM-1 CTRP1 0.2604 33.3330
WT-161 JHOS-4 CTRP1 0.2603 33.3330
WT-161 OAW42 CTRP1 0.2604 33.3330
WT-161 OV7 CTRP1 0.2604 33.3330
WT-161 OV-90 CTRP1 0.2604 33.3330
WT-161 OVCAR-4 CTRP1 0.2604 33.3330
WT-161 OVCAR-8 CTRP1 0.2604 33.3330
WT-161 OVK18 CTRP1 0.2604 33.3330
WT-161 OVKATE CTRP1 0.2604 33.3330
WT-161 OVMANA CTRP1 0.2603 33.3330
WT-161 RKN CTRP1 0.2604 33.3330
WT-161 RMG-I CTRP1 0.2604 33.3330
WT-161 RMUG-S CTRP1 0.2604 33.3330
WT-161 SK-OV-3 CTRP1 0.2603 33.3330
WT-161 SNU-840 CTRP1 0.2604 33.3330
WT-161 TYK-NU CTRP1 0.2604 33.3330
WT-161 CAPAN-2 CTRP1 0.2603 33.3330
WT-161 CFPAC-1 CTRP1 0.2603 33.3330
WT-161 HPAC CTRP1 0.2603 33.3330
WT-161 HUP-T4 CTRP1 0.2603 33.3330
WT-161 KP-3 CTRP1 0.2603 33.3330
WT-161 PANC03.27 CTRP1 0.2603 33.3330
WT-161 PANC10.05 CTRP1 0.2603 33.3330
WT-161 PATU8902 CTRP1 0.2603 33.3330
WT-161 QGP-1 CTRP1 0.2603 33.3330
WT-161 SUIT-2 CTRP1 0.2603 33.3330
WT-161 MSTO-211H CTRP1 0.2603 33.3330
WT-161 NCI-H2052 CTRP1 0.2603 33.3330
WT-161 NCI-H28 CTRP1 0.2603 33.3330
WT-161 MIAPACA-3 CTRP1 0.2603 33.3330
WT-161 A-375 CTRP1 0.2604 33.3330
WT-161 COLO741 CTRP1 0.2603 33.3330
WT-161 G-361 CTRP1 0.2603 33.3330
WT-161 HS852.T CTRP1 0.2603 33.3330
WT-161 HS936.T CTRP1 0.2603 33.3330
WT-161 HS944.T CTRP1 0.2603 33.3330
WT-161 SK-MEL-1 CTRP1 0.2604 33.3330
WT-161 SK-MEL-28 CTRP1 0.2604 33.3330
WT-161 SK-MEL-5 CTRP1 0.2604 33.3330
WT-161 G-401 CTRP1 0.2603 33.3330
WT-161 HT-1080 CTRP1 0.2604 33.3330
WT-161 AGS CTRP1 0.2604 33.3330
WT-161 FU97 CTRP1 0.2603 33.3330
WT-161 KE-97 CTRP1 0.2603 33.3330
WT-161 MKN7 CTRP1 0.2603 33.3330
WT-161 MKN74 CTRP1 0.2603 33.3330
WT-161 NUGC-4 CTRP1 0.2603 33.3330
WT-161 SH-10-TC CTRP1 0.2603 33.3330
WT-161 HSC-2 CTRP1 0.2603 33.3330
WT-161 SCC-9 CTRP1 0.2604 33.3330
WT-161 5637 CTRP1 0.2603 33.3330
WT-161 HT-1376 CTRP1 0.2603 33.3330
WT-161 KMBC-2 CTRP1 0.2603 33.3330
WT-161 RT-4 CTRP1 0.2603 33.3330
WT-161 UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.