Drug : Brd4770

CTRP1 Name : BRD4770
CTRP2 Name : QW-BI-011

Dataset : All
Synonyms :
Targets : EHMT2
Pathways : inhibitor of G9a histone methyltransferase

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BRD4770 U2OS CTRP2,CTRP1 0.0010 33.3330
BRD4770 MCF-7 CTRP2,CTRP1 0.0010 33.3330
BRD4770 GAMG CTRP1 0.2603 33.3330
BRD4770 LN-229 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HEC-108 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HEC-151 CTRP1 0.2604 33.3330
BRD4770 HEC-59 CTRP2,CTRP1 0.0010 33.3330
BRD4770 ISHIKAWA(HERAKLIO)02ER- CTRP2,CTRP1 0.0010 33.3330
BRD4770 JHUEM-2 CTRP2,CTRP1 0.0010 33.3330
BRD4770 KLE CTRP2,CTRP1 0.0010 33.3330
BRD4770 SNG-M CTRP1 0.2603 33.3330
BRD4770 AMO1 CTRP1 0.2604 33.3330
BRD4770 BL-70 CTRP1 0.2603 33.3330
BRD4770 EJM CTRP1 0.2604 33.3330
BRD4770 GDM-1 CTRP1 0.2604 33.3330
BRD4770 KMS-11 CTRP1 0.2604 33.3330
BRD4770 LP-1 CTRP1 0.2604 33.3330
BRD4770 MOLM-16 CTRP1 0.2604 33.3330
BRD4770 NOMO-1 CTRP1 0.2604 33.3330
BRD4770 NU-DUL-1 CTRP1 0.2604 33.3330
BRD4770 OCI-AML-3 CTRP1 0.2604 33.3330
BRD4770 OCI-LY10 CTRP1 0.2604 33.3330
BRD4770 PL21 CTRP1 0.2604 33.3330
BRD4770 RPMI-8226 CTRP1 0.2604 33.3330
BRD4770 SKM-1 CTRP1 0.2604 33.3330
BRD4770 SU-DHL-4 CTRP1 0.2604 33.3330
BRD4770 SU-DHL-5 CTRP1 0.2604 33.3330
BRD4770 THP-1 CTRP1 0.2604 33.3330
BRD4770 U-937 CTRP1 0.2604 33.3330
BRD4770 WSU-DLCL2 CTRP2,CTRP1 0.0010 33.3330
BRD4770 RCC10RGB CTRP1 0.2604 33.3330
BRD4770 CL-34 CTRP1 0.2604 33.3330
BRD4770 CL-40 CTRP1 0.2604 33.3330
BRD4770 COLO320 CTRP1 0.2604 16.6670
BRD4770 COLO678 CTRP1 0.2604 33.3330
BRD4770 CW-2 CTRP1 0.2604 33.3330
BRD4770 HCT116 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HCT8 CTRP1 0.2604 33.3330
BRD4770 HT115 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HT-29 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HT-55 CTRP1 0.2604 33.3330
BRD4770 KM12 CTRP1 0.2604 33.3330
BRD4770 LOVO CTRP1 0.2604 33.3330
BRD4770 LS123 CTRP1 0.2604 33.3330
BRD4770 LS180 CTRP2,CTRP1 0.0010 33.3330
BRD4770 MDST8 CTRP1 0.2604 33.3330
BRD4770 NCI-H508 CTRP1 0.2604 33.3330
BRD4770 RCM-1[HUMANESC] CTRP1 0.2604 33.3330
BRD4770 RKO CTRP1 0.2604 33.3330
BRD4770 SNU-1040 CTRP1 0.2604 33.3330
BRD4770 SNU-175 CTRP1 0.2604 33.3330
BRD4770 SNU-61 CTRP1 0.2604 33.3330
BRD4770 SNU-81 CTRP1 0.2604 33.3330
BRD4770 SNU-C4 CTRP1 0.2604 33.3330
BRD4770 SNU-C5 CTRP1 0.2604 33.3330
BRD4770 SW480 CTRP1 0.2604 33.3330
BRD4770 SW620 CTRP1 0.2604 33.3330
BRD4770 SW948 CTRP1 0.2604 33.3330
BRD4770 HEP-G2 CTRP1 0.2604 33.3330
BRD4770 JHH-6 CTRP1 0.2603 33.3330
BRD4770 SNU-398 CTRP1 0.2604 33.3330
BRD4770 SNU-449 CTRP1 0.2603 33.3330
BRD4770 CAL-12T CTRP2,CTRP1 0.0010 33.3330
BRD4770 COLO668 CTRP1 0.2603 33.3330
BRD4770 COLO699 CTRP2,CTRP1 0.0010 33.3330
BRD4770 COR-L23 CTRP1 0.2604 33.3330
BRD4770 COR-L51 CTRP1 0.2604 33.3330
BRD4770 HCC1195 CTRP1 0.2604 33.3330
BRD4770 HCC1359 CTRP1 0.2604 33.3330
BRD4770 HCC15 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HCC1833 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HCC2108 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HCC2935 CTRP1 0.2604 33.3330
BRD4770 HCC4006 CTRP1 0.2604 33.3330
BRD4770 HCC827 CTRP2,CTRP1 0.0010 33.3330
BRD4770 LXF289 CTRP1 0.2603 33.3330
BRD4770 NCI-H1105 CTRP1 0.2604 33.3330
BRD4770 NCI-H1435 CTRP1 0.2603 33.3330
BRD4770 NCI-H1694 CTRP1 0.2604 33.3330
BRD4770 NCI-H1755 CTRP1 0.2604 33.3330
BRD4770 NCI-H1781 CTRP1 0.2604 33.3330
BRD4770 NCI-H1836 CTRP1 0.2604 33.3330
BRD4770 NCI-H1876 CTRP1 0.2604 33.3330
BRD4770 NCI-H1915 CTRP1 0.2603 33.3330
BRD4770 NCI-H1930 CTRP1 0.2603 33.3330
BRD4770 NCI-H1963 CTRP1 0.2604 33.3330
BRD4770 NCI-H2009 CTRP2,CTRP1 0.0010 33.3330
BRD4770 NCI-H2023 CTRP1 0.2604 33.3330
BRD4770 NCI-H2030 CTRP2,CTRP1 0.0010 33.3330
BRD4770 NCI-H2073 CTRP1 0.2604 33.3330
BRD4770 NCI-H2081 CTRP1 0.2604 33.3330
BRD4770 NCI-H2110 CTRP1 0.2604 33.3330
BRD4770 NCI-H2122 CTRP1 0.2604 33.3330
BRD4770 NCI-H2141 CTRP1 0.2604 33.3330
BRD4770 NCI-H2172 CTRP1 0.2604 33.3330
BRD4770 NCI-H2286 CTRP1 0.2603 33.3330
BRD4770 NCI-H2342 CTRP1 0.2604 33.3330
BRD4770 NCI-H3255 CTRP1 0.2604 33.3330
BRD4770 NCI-H441 CTRP1 0.2604 33.3330
BRD4770 NCI-H460 CTRP2,CTRP1 0.0010 33.3330
BRD4770 NCI-H596 CTRP1 0.2604 33.3330
BRD4770 NCI-H841 CTRP1 0.2604 33.3330
BRD4770 RERF-LC-KJ CTRP1 0.2603 33.3330
BRD4770 SCLC-21H CTRP1 0.2604 33.3330
BRD4770 SK-LU-1 CTRP1 0.2604 33.3330
BRD4770 SQ-1 CTRP1 0.2604 33.3330
BRD4770 T3M-10 CTRP1 0.2604 33.3330
BRD4770 A2780 CTRP1 0.2604 33.3330
BRD4770 CAOV-3 CTRP1 0.2604 33.3330
BRD4770 COV318 CTRP1 0.2603 33.3330
BRD4770 COV362 CTRP1 0.2604 33.3330
BRD4770 COV434 CTRP1 0.2604 33.3330
BRD4770 COV644 CTRP1 0.2604 33.3330
BRD4770 EFO-27 CTRP1 0.2604 33.3330
BRD4770 IGROV-1 CTRP1 0.2604 33.3330
BRD4770 JHOC-5 CTRP2,CTRP1 0.0010 33.3330
BRD4770 JHOM-1 CTRP1 0.2604 33.3330
BRD4770 JHOS-4 CTRP1 0.2603 33.3330
BRD4770 OAW42 CTRP1 0.2604 33.3330
BRD4770 OV7 CTRP1 0.2604 33.3330
BRD4770 OV-90 CTRP1 0.2604 33.3330
BRD4770 OVCAR-4 CTRP1 0.2604 33.3330
BRD4770 OVCAR-8 CTRP1 0.2604 33.3330
BRD4770 OVK18 CTRP1 0.2604 33.3330
BRD4770 OVKATE CTRP1 0.2604 33.3330
BRD4770 OVMANA CTRP1 0.2603 33.3330
BRD4770 RKN CTRP1 0.2604 33.3330
BRD4770 RMG-I CTRP1 0.2604 33.3330
BRD4770 RMUG-S CTRP1 0.2604 33.3330
BRD4770 SNU-840 CTRP1 0.2604 33.3330
BRD4770 TYK-NU CTRP1 0.2604 33.3330
BRD4770 PATU8902 CTRP1 0.2603 33.3330
BRD4770 MIAPACA-3 CTRP1 0.2603 33.3330
BRD4770 A-375 CTRP2,CTRP1 0.0010 33.3330
BRD4770 HS852.T CTRP1 0.2603 33.3330
BRD4770 SK-MEL-1 CTRP2,CTRP1 0.0010 33.3330
BRD4770 SK-MEL-28 CTRP1 0.2604 33.3330
BRD4770 SK-MEL-5 CTRP1 0.2604 33.3330
BRD4770 HT-1080 CTRP1 0.2604 33.3330
BRD4770 AGS CTRP2,CTRP1 0.0010 33.3330
BRD4770 MKN74 CTRP1 0.2603 33.3330
BRD4770 SCC-9 CTRP1 0.2604 33.3330
BRD4770 CAS-1 CTRP2 0.0010 33.0000
BRD4770 KPL-1 CTRP2 0.0010 33.0000
BRD4770 MKN1 CTRP2 0.0010 33.0000
BRD4770 253J-BV CTRP2 0.0010 33.0000
BRD4770 BFTC-905 CTRP2 0.0010 33.0000
BRD4770 BFTC-909 CTRP2 0.0010 33.0000
BRD4770 CAL-120 CTRP2 0.0010 33.0000
BRD4770 CAL-29 CTRP2 0.0010 33.0000
BRD4770 CAL-62 CTRP2 0.0010 33.0000
BRD4770 HUCC-T1 CTRP2 0.0010 33.0000
BRD4770 NMC-G1 CTRP2 0.0010 33.0000
BRD4770 RPMI-7951 CTRP2 0.0010 33.0000
BRD4770 253J CTRP2 0.0010 33.0000
BRD4770 HDQ-P1 CTRP2 0.0010 33.0000
BRD4770 SNU-245 CTRP2 0.0010 33.0000
BRD4770 SNU-489 CTRP2 0.0010 33.0000
BRD4770 SNU-738 CTRP2 0.0010 33.0000
BRD4770 SNU-878 CTRP2 0.0010 33.0000
BRD4770 TUHR4TKB CTRP2 0.0010 33.0000
BRD4770 ACC-MESO-1 CTRP2 0.0010 33.0000
BRD4770 B-CPAP CTRP2 0.0010 33.0000
BRD4770 CGTH-W-1 CTRP2 0.0010 33.0000
BRD4770 COLO680N CTRP2 0.0010 33.0000
BRD4770 ECC12 CTRP2 0.0010 33.0000
BRD4770 HCC95 CTRP2 0.0010 33.0000
BRD4770 JMSU-1 CTRP2 0.0010 33.0000
BRD4770 RH41 CTRP2 0.0010 33.0000
BRD4770 23132-87 CTRP2 0.0010 33.0000
BRD4770 8305C CTRP2 0.0010 33.0000
BRD4770 BHY CTRP2 0.0010 33.0000
BRD4770 GSU CTRP2 0.0010 33.0000
BRD4770 JIMT-1 CTRP2 0.0010 33.0000
BRD4770 KMRC-20 CTRP2 0.0010 33.0000
BRD4770 OUMS-23 CTRP2 0.0010 33.0000
BRD4770 SNU-1076 CTRP2 0.0010 33.0000
BRD4770 SNU-1196 CTRP2 0.0010 33.0000
BRD4770 SNU-8 CTRP2 0.0010 33.0000
BRD4770 A-549 CTRP2 0.0010 33.0000
BRD4770 SNU-201 CTRP2 0.0010 33.0000
BRD4770 SUIT-2 CTRP2 0.0010 33.0000
BRD4770 SNU-1079 CTRP2 0.0010 33.0000
BRD4770 DEL CTRP2 0.0010 33.0000
BRD4770 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP2 0.0010 33.0000
BRD4770 KP-4 CTRP2 0.0010 33.0000
BRD4770 LU-99 CTRP2 0.0010 33.0000
BRD4770 NCI-H1155 CTRP2 0.0010 33.0000
BRD4770 NCI-H1581 CTRP2 0.0010 33.0000
BRD4770 NCI-H2106 CTRP2 0.0010 33.0000
BRD4770 NCI-H358 CTRP2 0.0010 33.0000
BRD4770 DLD-1 CTRP2 0.0010 33.0000
BRD4770 EM-2 CTRP2 0.0010 33.0000
BRD4770 JURL-MK1 CTRP2 0.0010 33.0000
BRD4770 P12-ICHIKAWA CTRP2 0.0010 33.0000
BRD4770 KE-37 CTRP2 0.0010 33.0000
BRD4770 KMS-21-BM CTRP2 0.0010 33.0000
BRD4770 LI-7 CTRP2 0.0010 33.0000
BRD4770 MOLM-13 CTRP2 0.0010 33.0000
BRD4770 NCI-H28 CTRP2 0.0010 33.0000
BRD4770 639V CTRP2 0.0010 33.0000
BRD4770 BXPC-3 CTRP2 0.0010 33.0000
BRD4770 CML-T1 CTRP2 0.0010 33.0000
BRD4770 GSS CTRP2 0.0010 33.0000
BRD4770 HCC366 CTRP2 0.0010 33.0000
BRD4770 KURAMOCHI CTRP2 0.0010 33.0000
BRD4770 LS411N CTRP2 0.0010 33.0000
BRD4770 LS513 CTRP2 0.0010 33.0000
BRD4770 ONCO-DG-1 CTRP2 0.0010 33.0000
BRD4770 ONS-76 CTRP2 0.0010 33.0000
BRD4770 SK-CO-1 CTRP2 0.0010 33.0000
BRD4770 SW48 CTRP2 0.0010 33.0000
BRD4770 VM-CUB-1 CTRP2 0.0010 33.0000
BRD4770 BEN CTRP2 0.0010 33.0000
BRD4770 CFPAC-1 CTRP2 0.0010 33.0000
BRD4770 HCC78 CTRP2 0.0010 33.0000
BRD4770 HT CTRP2 0.0010 33.0000
BRD4770 KU-19-19 CTRP2 0.0010 33.0000
BRD4770 NCI-H1299 CTRP2 0.0010 33.0000
BRD4770 NCI-H727 CTRP2 0.0010 33.0000
BRD4770 NCO2 CTRP2 0.0010 33.0000
BRD4770 OVTOKO CTRP2 0.0010 33.0000
BRD4770 P31-FUJ CTRP2 0.0010 33.0000
BRD4770 PEER CTRP2 0.0010 33.0000
BRD4770 RPMI-8402 CTRP2 0.0010 33.0000
BRD4770 SHP-77 CTRP2 0.0010 33.0000
BRD4770 SNU-1077 CTRP2 0.0010 33.0000
BRD4770 SNU-620 CTRP2 0.0010 33.0000
BRD4770 SU-DHL-1 CTRP2 0.0010 33.0000
BRD4770 COLO205 CTRP2 0.0010 33.0000
BRD4770 DOHH2 CTRP2 0.0010 17.0000
BRD4770 EHEB CTRP2 0.0010 17.0000
BRD4770 KI-JK CTRP2 0.0010 33.0000
BRD4770 KMM-1 CTRP2 0.0010 33.0000
BRD4770 LCLC-103H CTRP2 0.0010 33.0000
BRD4770 MKN45 CTRP2 0.0010 33.0000
BRD4770 NCI-H2405 CTRP2 0.0010 17.0000
BRD4770 NCI-H650 CTRP2 0.0010 33.0000
BRD4770 OS-RC-2 CTRP2 0.0010 33.0000
BRD4770 OVSAHO CTRP2 0.0010 33.0000
BRD4770 QGP-1 CTRP2 0.0010 17.0000
BRD4770 RL95-2 CTRP2 0.0010 33.0000
BRD4770 SNU-1041 CTRP2 0.0010 33.0000
BRD4770 SNU-1066 CTRP2 0.0010 33.0000
BRD4770 SW1353 CTRP2 0.0010 33.0000
BRD4770 SNU-213 CTRP2 0.0010 17.0000
BRD4770 8505C CTRP2 0.0010 17.0000
BRD4770 CALU-3 CTRP2 0.0010 17.0000
BRD4770 DAOY CTRP2 0.0010 17.0000
BRD4770 GB-1 CTRP2 0.0010 17.0000
BRD4770 HCC1171 CTRP2 0.0010 17.0000
BRD4770 HCC44 CTRP2 0.0010 17.0000
BRD4770 NCI-H211 CTRP2 0.0010 17.0000
BRD4770 RERF-LC-A1 CTRP2 0.0010 17.0000
BRD4770 SBC-5 CTRP2 0.0010 17.0000
BRD4770 SF126 CTRP2 0.0010 17.0000
BRD4770 SNU-119 CTRP2 0.0010 17.0000
BRD4770 SNU-182 CTRP2 0.0010 17.0000
BRD4770 TCCSUP CTRP2 0.0010 17.0000
BRD4770 CAMA-1 CTRP2 0.0010 17.0000
BRD4770 DETROIT562 CTRP2 0.0010 17.0000
BRD4770 HEC-1-B CTRP2 0.0010 17.0000
BRD4770 HEP3B2.1-7 CTRP2 0.0010 17.0000
BRD4770 HSC-3 CTRP2 0.0010 17.0000
BRD4770 SNU-1105 CTRP2 0.0010 17.0000
BRD4770 U-87MGATCC CTRP2 0.0010 17.0000
BRD4770 22RV1 CTRP2 0.0010 17.0000
BRD4770 769-P CTRP2 0.0010 17.0000
BRD4770 DOV13 CTRP2 0.0010 17.0000
BRD4770 ES2 CTRP2 0.0010 17.0000
BRD4770 HCC1806 CTRP2 0.0010 17.0000
BRD4770 HCC1954 CTRP2 0.0010 17.0000
BRD4770 HPAF-II CTRP2 0.0010 17.0000
BRD4770 KHM-1B CTRP2 0.0010 17.0000
BRD4770 OVISE CTRP2 0.0010 17.0000
BRD4770 JVM-3 CTRP2 0.0010 17.0000
BRD4770 SNU-C2A CTRP2 0.0010 17.0000
BRD4770 5637 CTRP2 0.0010 17.0000
BRD4770 DMS79 CTRP2 0.0010 17.0000
BRD4770 HCC1588 CTRP2 0.0010 17.0000
BRD4770 HCC2279 CTRP2 0.0010 17.0000
BRD4770 KE-97 CTRP2 0.0010 17.0000
BRD4770 KP-3 CTRP2 0.0010 17.0000
BRD4770 KU812 CTRP2 0.0010 17.0000
BRD4770 KYSE-140 CTRP2 0.0010 17.0000
BRD4770 NALM-6 CTRP2 0.0010 17.0000
BRD4770 NUGC-4 CTRP2 0.0010 17.0000
BRD4770 TT CTRP2 0.0010 17.0000
BRD4770 HMC-1-8 CTRP2 0.0010 17.0000
BRD4770 KYSE-180 CTRP2 0.0010 17.0000
BRD4770 MELHO CTRP2 0.0010 17.0000
BRD4770 MHH-ES-1 CTRP2 0.0010 17.0000
BRD4770 MOR-CPR CTRP2 0.0010 17.0000
BRD4770 HEC-251 CTRP2 0.0010 17.0000
BRD4770 HEC-265 CTRP2 0.0010 17.0000
BRD4770 HEC-6 CTRP2 0.0010 17.0000
BRD4770 HEL CTRP2 0.0010 8.3000
BRD4770 JURKAT CTRP2 0.0010 8.3000
BRD4770 JVM-2 CTRP2 0.0010 8.3000
BRD4770 KCL-22 CTRP2 0.0010 17.0000
BRD4770 KE-39 CTRP2 0.0010 17.0000
BRD4770 KM-H2 CTRP2 0.0010 8.3000
BRD4770 LAMA-84 CTRP2 0.0010 8.3000
BRD4770 SNU-719 CTRP2 0.0010 17.0000
BRD4770 KMS-26 CTRP2 0.0010 17.0000
BRD4770 KMS-27 CTRP2 0.0010 17.0000
BRD4770 NCI-H1838 CTRP2 0.0010 17.0000
BRD4770 NCI-H196 CTRP2 0.0010 17.0000
BRD4770 NCI-H292 CTRP2 0.0010 17.0000
BRD4770 HCC1937 CTRP2 0.0010 17.0000
BRD4770 HDLM-2 CTRP2 0.0010 17.0000
BRD4770 HUH-28 CTRP2 0.0010 17.0000
BRD4770 MV4-11 CTRP2 0.0010 17.0000
BRD4770 NCI-H526 CTRP2 0.0010 17.0000
BRD4770 NCI-H69 CTRP2 0.0010 17.0000
BRD4770 NCI-H929 CTRP2 0.0010 17.0000
BRD4770 NCI-N87 CTRP2 0.0010 17.0000
BRD4770 PF-382 CTRP2 0.0010 17.0000
BRD4770 SF295 CTRP2 0.0010 17.0000
BRD4770 SNU-1272 CTRP2 0.0010 17.0000
BRD4770 SNU-308 CTRP2 0.0010 17.0000
BRD4770 SNU-478 CTRP2 0.0010 17.0000
BRD4770 BHT-101 CTRP2 0.0010 17.0000
BRD4770 CAL-148 CTRP2 0.0010 17.0000
BRD4770 CAL-51 CTRP2 0.0010 17.0000
BRD4770 HCC1395 CTRP2 0.0010 17.0000
BRD4770 LN-18 CTRP2 0.0010 17.0000
BRD4770 NCI-H1734 CTRP2 0.0010 17.0000
BRD4770 NCI-H2291 CTRP2 0.0010 17.0000
BRD4770 RERF-LC-AD1 CTRP2 0.0010 17.0000
BRD4770 SNU-1214 CTRP2 0.0010 17.0000
BRD4770 SNU-46 CTRP2 0.0010 17.0000
BRD4770 SNU-466 CTRP2 0.0010 17.0000
BRD4770 SNU-5 CTRP2 0.0010 17.0000
BRD4770 SNU-668 CTRP2 0.0010 17.0000
BRD4770 SNU-899 CTRP2 0.0010 17.0000
BRD4770 TE-10 CTRP2 0.0010 17.0000
BRD4770 TE-9 CTRP2 0.0010 17.0000
BRD4770 YD-10B CTRP2 0.0010 17.0000
BRD4770 YD-15 CTRP2 0.0010 17.0000
BRD4770 YD-38 CTRP2 0.0010 17.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.