Drug : Cimetidine

CTRP2 Name : cimetidine

Dataset : All
Synonyms :
Targets : HRH2
Pathways : inhibitor of histidine receptor H2

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
cimetidine CAS-1 CTRP2 0.0081 130.0000
cimetidine KPL-1 CTRP2 0.0081 130.0000
cimetidine MKN1 CTRP2 0.0081 130.0000
cimetidine 253J-BV CTRP2 0.0081 270.0000
cimetidine BFTC-905 CTRP2 0.0081 270.0000
cimetidine BFTC-909 CTRP2 0.0081 270.0000
cimetidine CAL-120 CTRP2 0.0081 270.0000
cimetidine CAL-29 CTRP2 0.0081 270.0000
cimetidine CAL-62 CTRP2 0.0081 270.0000
cimetidine HUCC-T1 CTRP2 0.0081 270.0000
cimetidine NMC-G1 CTRP2 0.0081 270.0000
cimetidine RPMI-7951 CTRP2 0.0081 270.0000
cimetidine 253J CTRP2 0.0081 270.0000
cimetidine HDQ-P1 CTRP2 0.0081 270.0000
cimetidine SIMA CTRP2 0.0081 270.0000
cimetidine SNU-489 CTRP2 0.0081 270.0000
cimetidine SNU-626 CTRP2 0.0081 270.0000
cimetidine SNU-738 CTRP2 0.0081 270.0000
cimetidine SNU-878 CTRP2 0.0081 270.0000
cimetidine TUHR4TKB CTRP2 0.0081 270.0000
cimetidine ACC-MESO-1 CTRP2 0.0081 270.0000
cimetidine B-CPAP CTRP2 0.0081 270.0000
cimetidine CGTH-W-1 CTRP2 0.0081 270.0000
cimetidine COLO680N CTRP2 0.0081 270.0000
cimetidine ECC12 CTRP2 0.0081 270.0000
cimetidine HCC95 CTRP2 0.0081 270.0000
cimetidine JMSU-1 CTRP2 0.0081 270.0000
cimetidine RH41 CTRP2 0.0081 270.0000
cimetidine WSU-DLCL2 CTRP2 0.0081 270.0000
cimetidine 23132-87 CTRP2 0.0081 270.0000
cimetidine 8305C CTRP2 0.0081 270.0000
cimetidine BHY CTRP2 0.0081 270.0000
cimetidine GSU CTRP2 0.0081 270.0000
cimetidine JIMT-1 CTRP2 0.0081 270.0000
cimetidine KMRC-20 CTRP2 0.0081 270.0000
cimetidine OUMS-23 CTRP2 0.0081 270.0000
cimetidine SNU-1076 CTRP2 0.0081 270.0000
cimetidine SNU-1196 CTRP2 0.0081 270.0000
cimetidine SNU-8 CTRP2 0.0081 270.0000
cimetidine A-375 CTRP2 0.0081 270.0000
cimetidine A-549 CTRP2 0.0081 270.0000
cimetidine NCI-H2009 CTRP2 0.0081 270.0000
cimetidine SNU-201 CTRP2 0.0081 270.0000
cimetidine SUIT-2 CTRP2 0.0081 270.0000
cimetidine SNU-1079 CTRP2 0.0081 270.0000
cimetidine COLO741 CTRP2 0.0081 270.0000
cimetidine DEL CTRP2 0.0081 270.0000
cimetidine HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP2 0.0081 270.0000
cimetidine HCC15 CTRP2 0.0081 270.0000
cimetidine KP-4 CTRP2 0.0081 270.0000
cimetidine LU-99 CTRP2 0.0081 270.0000
cimetidine NCI-H1155 CTRP2 0.0081 270.0000
cimetidine NCI-H1581 CTRP2 0.0081 270.0000
cimetidine NCI-H2106 CTRP2 0.0081 270.0000
cimetidine NCI-H358 CTRP2 0.0081 270.0000
cimetidine DLD-1 CTRP2 0.0081 270.0000
cimetidine EM-2 CTRP2 0.0081 270.0000
cimetidine JURL-MK1 CTRP2 0.0081 270.0000
cimetidine P12-ICHIKAWA CTRP2 0.0081 270.0000
cimetidine KE-37 CTRP2 0.0081 270.0000
cimetidine KMS-21-BM CTRP2 0.0081 270.0000
cimetidine LI-7 CTRP2 0.0081 270.0000
cimetidine MHH-NB-11 CTRP2 0.0081 270.0000
cimetidine MOLM-13 CTRP2 0.0081 270.0000
cimetidine NCI-H1975 CTRP2 0.0081 270.0000
cimetidine NCI-H28 CTRP2 0.0081 270.0000
cimetidine 639V CTRP2 0.0081 270.0000
cimetidine BXPC-3 CTRP2 0.0081 270.0000
cimetidine CML-T1 CTRP2 0.0081 270.0000
cimetidine GSS CTRP2 0.0081 270.0000
cimetidine HCC366 CTRP2 0.0081 270.0000
cimetidine KURAMOCHI CTRP2 0.0081 270.0000
cimetidine LS411N CTRP2 0.0081 270.0000
cimetidine LS513 CTRP2 0.0081 270.0000
cimetidine ONCO-DG-1 CTRP2 0.0081 270.0000
cimetidine ONS-76 CTRP2 0.0081 270.0000
cimetidine SK-CO-1 CTRP2 0.0081 270.0000
cimetidine SW48 CTRP2 0.0081 270.0000
cimetidine VM-CUB-1 CTRP2 0.0081 270.0000
cimetidine BEN CTRP2 0.0081 270.0000
cimetidine CFPAC-1 CTRP2 0.0081 270.0000
cimetidine HCC78 CTRP2 0.0081 270.0000
cimetidine HT CTRP2 0.0081 270.0000
cimetidine KU-19-19 CTRP2 0.0081 270.0000
cimetidine NCI-H1299 CTRP2 0.0081 270.0000
cimetidine NCI-H727 CTRP2 0.0081 270.0000
cimetidine NCO2 CTRP2 0.0081 270.0000
cimetidine OVTOKO CTRP2 0.0081 270.0000
cimetidine P31-FUJ CTRP2 0.0081 270.0000
cimetidine PEER CTRP2 0.0081 270.0000
cimetidine RPMI-8402 CTRP2 0.0081 270.0000
cimetidine SHP-77 CTRP2 0.0081 270.0000
cimetidine SNU-1077 CTRP2 0.0081 270.0000
cimetidine SNU-620 CTRP2 0.0081 270.0000
cimetidine SU-DHL-1 CTRP2 0.0081 270.0000
cimetidine COLO205 CTRP2 0.0081 270.0000
cimetidine EHEB CTRP2 0.0081 270.0000
cimetidine KI-JK CTRP2 0.0081 270.0000
cimetidine KMM-1 CTRP2 0.0081 270.0000
cimetidine LCLC-103H CTRP2 0.0081 270.0000
cimetidine MKN45 CTRP2 0.0081 270.0000
cimetidine NCI-H2405 CTRP2 0.0081 270.0000
cimetidine NCI-H650 CTRP2 0.0081 270.0000
cimetidine OS-RC-2 CTRP2 0.0081 270.0000
cimetidine OVSAHO CTRP2 0.0081 270.0000
cimetidine QGP-1 CTRP2 0.0081 270.0000
cimetidine RL95-2 CTRP2 0.0081 270.0000
cimetidine SNU-1041 CTRP2 0.0081 270.0000
cimetidine SNU-1066 CTRP2 0.0081 270.0000
cimetidine SW1353 CTRP2 0.0081 270.0000
cimetidine SNU-213 CTRP2 0.0081 270.0000
cimetidine 8505C CTRP2 0.0081 270.0000
cimetidine CALU-3 CTRP2 0.0081 270.0000
cimetidine DAOY CTRP2 0.0081 270.0000
cimetidine GB-1 CTRP2 0.0081 270.0000
cimetidine HCC1171 CTRP2 0.0081 270.0000
cimetidine HCC44 CTRP2 0.0081 270.0000
cimetidine NCI-H211 CTRP2 0.0081 270.0000
cimetidine RERF-LC-A1 CTRP2 0.0081 270.0000
cimetidine SBC-5 CTRP2 0.0081 270.0000
cimetidine SF126 CTRP2 0.0081 270.0000
cimetidine SNU-119 CTRP2 0.0081 270.0000
cimetidine SNU-182 CTRP2 0.0081 270.0000
cimetidine TCCSUP CTRP2 0.0081 270.0000
cimetidine CAMA-1 CTRP2 0.0081 270.0000
cimetidine DETROIT562 CTRP2 0.0081 270.0000
cimetidine HEC-1-B CTRP2 0.0081 270.0000
cimetidine HEP3B2.1-7 CTRP2 0.0081 270.0000
cimetidine HSC-3 CTRP2 0.0081 270.0000
cimetidine MCF-7 CTRP2 0.0081 270.0000
cimetidine SNU-1105 CTRP2 0.0081 270.0000
cimetidine U-87MGATCC CTRP2 0.0081 270.0000
cimetidine 22RV1 CTRP2 0.0081 66.0000
cimetidine 769-P CTRP2 0.0081 270.0000
cimetidine COLO699 CTRP2 0.0081 270.0000
cimetidine DOV13 CTRP2 0.0081 270.0000
cimetidine ES2 CTRP2 0.0081 270.0000
cimetidine HCC1806 CTRP2 0.0081 270.0000
cimetidine HCC1954 CTRP2 0.0081 270.0000
cimetidine HPAF-II CTRP2 0.0081 66.0000
cimetidine KHM-1B CTRP2 0.0081 270.0000
cimetidine OVISE CTRP2 0.0081 270.0000
cimetidine JVM-3 CTRP2 0.0081 270.0000
cimetidine SNU-C2A CTRP2 0.0081 270.0000
cimetidine U2OS CTRP2 0.0081 130.0000
cimetidine 5637 CTRP2 0.0081 270.0000
cimetidine CAL-12T CTRP2 0.0081 270.0000
cimetidine HCC1588 CTRP2 0.0081 270.0000
cimetidine HCC1833 CTRP2 0.0081 270.0000
cimetidine HCC2279 CTRP2 0.0081 270.0000
cimetidine KE-97 CTRP2 0.0081 270.0000
cimetidine KP-3 CTRP2 0.0081 270.0000
cimetidine KU812 CTRP2 0.0081 270.0000
cimetidine KYSE-140 CTRP2 0.0081 270.0000
cimetidine NALM-6 CTRP2 0.0081 270.0000
cimetidine NUGC-4 CTRP2 0.0081 270.0000
cimetidine TT CTRP2 0.0081 270.0000
cimetidine AGS CTRP2 0.0081 270.0000
cimetidine HCT116 CTRP2 0.0081 270.0000
cimetidine HEC-108 CTRP2 0.0081 270.0000
cimetidine HEC-59 CTRP2 0.0081 270.0000
cimetidine HMC-1-8 CTRP2 0.0081 270.0000
cimetidine HT-29 CTRP2 0.0081 270.0000
cimetidine ISHIKAWA(HERAKLIO)02ER- CTRP2 0.0081 270.0000
cimetidine JHOC-5 CTRP2 0.0081 270.0000
cimetidine KYSE-180 CTRP2 0.0081 270.0000
cimetidine LS180 CTRP2 0.0081 270.0000
cimetidine MELHO CTRP2 0.0081 270.0000
cimetidine MHH-ES-1 CTRP2 0.0081 270.0000
cimetidine MOR-CPR CTRP2 0.0081 270.0000
cimetidine NCI-H460 CTRP2 0.0081 270.0000
cimetidine HCC2108 CTRP2 0.0081 270.0000
cimetidine HCC827 CTRP2 0.0081 270.0000
cimetidine HEC-251 CTRP2 0.0081 270.0000
cimetidine HEC-265 CTRP2 0.0081 270.0000
cimetidine HEC-6 CTRP2 0.0081 270.0000
cimetidine HEL CTRP2 0.0081 270.0000
cimetidine JHUEM-2 CTRP2 0.0081 270.0000
cimetidine JURKAT CTRP2 0.0081 270.0000
cimetidine JVM-2 CTRP2 0.0081 270.0000
cimetidine KCL-22 CTRP2 0.0081 270.0000
cimetidine KE-39 CTRP2 0.0081 270.0000
cimetidine KM-H2 CTRP2 0.0081 270.0000
cimetidine LAMA-84 CTRP2 0.0081 270.0000
cimetidine NCI-H2030 CTRP2 0.0081 270.0000
cimetidine SNU-719 CTRP2 0.0081 270.0000
cimetidine KLE CTRP2 0.0081 270.0000
cimetidine KMS-26 CTRP2 0.0081 270.0000
cimetidine KMS-27 CTRP2 0.0081 270.0000
cimetidine NCI-H1838 CTRP2 0.0081 270.0000
cimetidine NCI-H196 CTRP2 0.0081 270.0000
cimetidine NCI-H292 CTRP2 0.0081 270.0000
cimetidine SK-MEL-1 CTRP2 0.0081 270.0000
cimetidine HCC1937 CTRP2 0.0081 270.0000
cimetidine HDLM-2 CTRP2 0.0081 270.0000
cimetidine HUH-28 CTRP2 0.0081 270.0000
cimetidine MV4-11 CTRP2 0.0081 270.0000
cimetidine NCI-H526 CTRP2 0.0081 270.0000
cimetidine NCI-H69 CTRP2 0.0081 270.0000
cimetidine NCI-H929 CTRP2 0.0081 270.0000
cimetidine NCI-N87 CTRP2 0.0081 270.0000
cimetidine PF-382 CTRP2 0.0081 270.0000
cimetidine SF295 CTRP2 0.0081 270.0000
cimetidine SNU-1272 CTRP2 0.0081 270.0000
cimetidine SNU-308 CTRP2 0.0081 270.0000
cimetidine SNU-478 CTRP2 0.0081 270.0000
cimetidine BHT-101 CTRP2 0.0081 270.0000
cimetidine CAL-148 CTRP2 0.0081 270.0000
cimetidine CAL-51 CTRP2 0.0081 270.0000
cimetidine HCC1395 CTRP2 0.0081 270.0000
cimetidine HT115 CTRP2 0.0081 270.0000
cimetidine LN-18 CTRP2 0.0081 270.0000
cimetidine LN-229 CTRP2 0.0081 270.0000
cimetidine NCI-H1734 CTRP2 0.0081 270.0000
cimetidine NCI-H2291 CTRP2 0.0081 270.0000
cimetidine RERF-LC-AD1 CTRP2 0.0081 270.0000
cimetidine SNU-1214 CTRP2 0.0081 270.0000
cimetidine SNU-46 CTRP2 0.0081 270.0000
cimetidine SNU-466 CTRP2 0.0081 270.0000
cimetidine SNU-5 CTRP2 0.0081 270.0000
cimetidine SNU-668 CTRP2 0.0081 270.0000
cimetidine SNU-899 CTRP2 0.0081 270.0000
cimetidine TE-10 CTRP2 0.0081 270.0000
cimetidine TE-9 CTRP2 0.0081 270.0000
cimetidine YD-10B CTRP2 0.0081 270.0000
cimetidine YD-15 CTRP2 0.0081 270.0000
cimetidine YD-38 CTRP2 0.0081 270.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.