Drug : Gly-Gly-Palo

CTRP1 Name : Gly-Gly-PALO

Dataset : All
Synonyms :
Targets : OTC
Pathways : inhibitor of ornithine carbamoyltransferase

Information Cards

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Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
Gly-Gly-PALO U2OS CTRP1 2.0833 266.6700
Gly-Gly-PALO MCF-7 CTRP1 2.0833 266.6700
Gly-Gly-PALO GAMG CTRP1 0.2603 33.3330
Gly-Gly-PALO LN-229 CTRP1 2.0833 266.6700
Gly-Gly-PALO SF295 CTRP1 0.2603 33.3330
Gly-Gly-PALO HEC-108 CTRP1 0.2603 33.3330
Gly-Gly-PALO HEC-151 CTRP1 2.0833 266.6700
Gly-Gly-PALO HEC-251 CTRP1 0.2603 33.3330
Gly-Gly-PALO HEC-265 CTRP1 0.2603 33.3330
Gly-Gly-PALO HEC-59 CTRP1 0.2603 33.3330
Gly-Gly-PALO HEC-6 CTRP1 0.2603 33.3330
Gly-Gly-PALO ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
Gly-Gly-PALO JHUEM-2 CTRP1 2.0833 266.6700
Gly-Gly-PALO KLE CTRP1 0.2603 33.3330
Gly-Gly-PALO MFE-319 CTRP1 0.2603 33.3330
Gly-Gly-PALO SNG-M CTRP1 0.2603 33.3330
Gly-Gly-PALO AMO1 CTRP1 2.0833 266.6700
Gly-Gly-PALO BL-70 CTRP1 0.2603 33.3330
Gly-Gly-PALO EJM CTRP1 2.0833 266.6700
Gly-Gly-PALO GDM-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO HT CTRP1 0.2603 33.3330
Gly-Gly-PALO KMS-11 CTRP1 2.0833 266.6700
Gly-Gly-PALO KU812 CTRP1 0.2603 33.3330
Gly-Gly-PALO LP-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO MC116 CTRP1 0.2603 33.3330
Gly-Gly-PALO MOLM-16 CTRP1 2.0833 266.6700
Gly-Gly-PALO NOMO-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO NU-DUL-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO OCI-AML-3 CTRP1 2.0833 266.6700
Gly-Gly-PALO OCI-LY10 CTRP1 2.0833 266.6700
Gly-Gly-PALO P3HR-1 CTRP1 0.2603 33.3330
Gly-Gly-PALO PL21 CTRP1 2.0833 266.6700
Gly-Gly-PALO RPMI-8226 CTRP1 2.0833 266.6700
Gly-Gly-PALO SKM-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO SU-DHL-4 CTRP1 2.0833 266.6700
Gly-Gly-PALO SU-DHL-5 CTRP1 2.0833 266.6700
Gly-Gly-PALO THP-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO U-937 CTRP1 2.0833 266.6700
Gly-Gly-PALO WSU-DLCL2 CTRP1 2.0833 266.6700
Gly-Gly-PALO RCC10RGB CTRP1 2.0833 266.6700
Gly-Gly-PALO VMRC-RCW CTRP1 0.2603 33.3330
Gly-Gly-PALO C2BBE1 CTRP1 0.2603 33.3330
Gly-Gly-PALO CL-34 CTRP1 2.0833 266.6700
Gly-Gly-PALO CL-40 CTRP1 2.0833 266.6700
Gly-Gly-PALO COLO205 CTRP1 0.2603 33.3330
Gly-Gly-PALO COLO320 CTRP1 2.0833 266.6700
Gly-Gly-PALO COLO678 CTRP1 2.0833 266.6700
Gly-Gly-PALO CW-2 CTRP1 2.0833 266.6700
Gly-Gly-PALO DLD-1 CTRP1 0.2603 33.3330
Gly-Gly-PALO GP2D CTRP1 0.2603 33.3330
Gly-Gly-PALO HCT116 CTRP1 2.0833 266.6700
Gly-Gly-PALO HCT8 CTRP1 2.0833 266.6700
Gly-Gly-PALO HT115 CTRP1 2.0833 266.6700
Gly-Gly-PALO HT-29 CTRP1 2.0833 266.6700
Gly-Gly-PALO HT-55 CTRP1 2.0833 266.6700
Gly-Gly-PALO KM12 CTRP1 2.0833 266.6700
Gly-Gly-PALO LOVO CTRP1 2.0833 266.6700
Gly-Gly-PALO LS123 CTRP1 2.0833 266.6700
Gly-Gly-PALO LS180 CTRP1 2.0833 266.6700
Gly-Gly-PALO LS411N CTRP1 0.2603 33.3330
Gly-Gly-PALO LS513 CTRP1 0.2603 33.3330
Gly-Gly-PALO MDST8 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H508 CTRP1 2.0833 266.6700
Gly-Gly-PALO RCM-1[HUMANESC] CTRP1 2.0833 266.6700
Gly-Gly-PALO RKO CTRP1 2.0833 266.6700
Gly-Gly-PALO SK-CO-1 CTRP1 0.2603 33.3330
Gly-Gly-PALO SNU-1040 CTRP1 2.0833 266.6700
Gly-Gly-PALO SNU-175 CTRP1 2.0833 266.6700
Gly-Gly-PALO SNU-61 CTRP1 2.0833 266.6700
Gly-Gly-PALO SNU-81 CTRP1 2.0833 266.6700
Gly-Gly-PALO SNU-C2A CTRP1 0.2603 33.3330
Gly-Gly-PALO SNU-C4 CTRP1 2.0833 266.6700
Gly-Gly-PALO SNU-C5 CTRP1 2.0833 266.6700
Gly-Gly-PALO SW403 CTRP1 0.2603 33.3330
Gly-Gly-PALO SW48 CTRP1 0.2603 33.3330
Gly-Gly-PALO SW480 CTRP1 2.0833 266.6700
Gly-Gly-PALO SW620 CTRP1 2.0833 266.6700
Gly-Gly-PALO SW948 CTRP1 2.0833 266.6700
Gly-Gly-PALO HEP-G2 CTRP1 2.0833 266.6700
Gly-Gly-PALO JHH-6 CTRP1 0.2603 33.3330
Gly-Gly-PALO SNU-398 CTRP1 2.0833 266.6700
Gly-Gly-PALO SNU-449 CTRP1 0.2603 33.3330
Gly-Gly-PALO A-549 CTRP1 0.2603 33.3330
Gly-Gly-PALO BEN CTRP1 0.2603 33.3330
Gly-Gly-PALO CAL-12T CTRP1 2.0833 266.6700
Gly-Gly-PALO CALU-3 CTRP1 0.2603 33.3330
Gly-Gly-PALO CALU-6 CTRP1 0.2603 33.3330
Gly-Gly-PALO CHAGO-K-1 CTRP1 0.2603 33.3330
Gly-Gly-PALO COLO668 CTRP1 0.2603 33.3330
Gly-Gly-PALO COLO699 CTRP1 2.0833 266.6700
Gly-Gly-PALO COR-L23 CTRP1 2.0833 266.6700
Gly-Gly-PALO COR-L279 CTRP1 0.2603 33.3330
Gly-Gly-PALO COR-L51 CTRP1 2.0833 266.6700
Gly-Gly-PALO COR-L88 CTRP1 0.2603 33.3330
Gly-Gly-PALO DMS273 CTRP1 0.2603 33.3330
Gly-Gly-PALO DV-90 CTRP1 0.2603 33.3330
Gly-Gly-PALO EBC-1 CTRP1 0.2603 33.3330
Gly-Gly-PALO EPLC-272H CTRP1 0.2603 33.3330
Gly-Gly-PALO HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2603 33.3330
Gly-Gly-PALO HCC1195 CTRP1 2.0833 266.6700
Gly-Gly-PALO HCC1359 CTRP1 2.0833 266.6700
Gly-Gly-PALO HCC15 CTRP1 2.0833 266.6700
Gly-Gly-PALO HCC1833 CTRP1 2.0833 266.6700
Gly-Gly-PALO HCC2108 CTRP1 2.0833 266.6700
Gly-Gly-PALO HCC2935 CTRP1 2.0833 266.6700
Gly-Gly-PALO HCC33 CTRP1 0.2603 33.3330
Gly-Gly-PALO HCC4006 CTRP1 2.0833 266.6700
Gly-Gly-PALO HCC44 CTRP1 0.2603 33.3330
Gly-Gly-PALO HCC78 CTRP1 0.2603 33.3330
Gly-Gly-PALO HCC827 CTRP1 2.0833 266.6700
Gly-Gly-PALO KNS-62 CTRP1 0.2603 33.3330
Gly-Gly-PALO LC-1-SQ-SF CTRP1 0.2603 33.3330
Gly-Gly-PALO LCLC-103H CTRP1 0.2603 33.3330
Gly-Gly-PALO LCLC-97TM1 CTRP1 0.2603 33.3330
Gly-Gly-PALO LU-65 CTRP1 0.2603 33.3330
Gly-Gly-PALO LU-99 CTRP1 0.2603 33.3330
Gly-Gly-PALO LXF289 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1048 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1105 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H1299 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1355 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1373 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1435 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1437 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1568 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1573 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1666 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1694 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H1755 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H1781 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H1792 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1793 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1836 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H1876 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H1915 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1930 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1944 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H1963 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H1975 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H2009 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H2023 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2029 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H2030 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2073 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2081 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2110 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2122 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2126 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H2141 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2172 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2286 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H23 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H2342 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H2405 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H3255 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H358 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H441 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H460 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H522 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H596 CTRP1 2.0833 266.6700
Gly-Gly-PALO NCI-H650 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H661 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H727 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H810 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H82 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H841 CTRP1 2.0833 266.6700
Gly-Gly-PALO RERF-LC-KJ CTRP1 0.2603 33.3330
Gly-Gly-PALO SCLC-21H CTRP1 2.0833 266.6700
Gly-Gly-PALO SHP-77 CTRP1 0.2603 33.3330
Gly-Gly-PALO SK-LU-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO SQ-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO T3M-10 CTRP1 2.0833 266.6700
Gly-Gly-PALO VMRC-LCD CTRP1 0.2603 33.3330
Gly-Gly-PALO KYSE-140 CTRP1 0.2603 33.3330
Gly-Gly-PALO KYSE-410 CTRP1 0.2603 33.3330
Gly-Gly-PALO KYSE-450 CTRP1 0.2603 33.3330
Gly-Gly-PALO A2780 CTRP1 2.0833 266.6700
Gly-Gly-PALO CAOV-3 CTRP1 2.0833 266.6700
Gly-Gly-PALO COV318 CTRP1 0.2603 33.3330
Gly-Gly-PALO COV362 CTRP1 2.0833 266.6700
Gly-Gly-PALO COV434 CTRP1 2.0833 266.6700
Gly-Gly-PALO COV644 CTRP1 2.0833 266.6700
Gly-Gly-PALO EFO-21 CTRP1 0.2603 33.3330
Gly-Gly-PALO EFO-27 CTRP1 2.0833 266.6700
Gly-Gly-PALO HEYA8 CTRP1 0.2603 33.3330
Gly-Gly-PALO IGROV-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO JHOC-5 CTRP1 2.0833 266.6700
Gly-Gly-PALO JHOM-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO JHOS-4 CTRP1 0.2603 33.3330
Gly-Gly-PALO OAW42 CTRP1 2.0833 266.6700
Gly-Gly-PALO OV7 CTRP1 2.0833 266.6700
Gly-Gly-PALO OV-90 CTRP1 2.0833 266.6700
Gly-Gly-PALO OVCAR-4 CTRP1 2.0833 266.6700
Gly-Gly-PALO OVCAR-8 CTRP1 2.0833 266.6700
Gly-Gly-PALO OVK18 CTRP1 2.0833 266.6700
Gly-Gly-PALO OVKATE CTRP1 2.0833 266.6700
Gly-Gly-PALO OVMANA CTRP1 0.2603 33.3330
Gly-Gly-PALO RKN CTRP1 2.0833 266.6700
Gly-Gly-PALO RMG-I CTRP1 2.0833 266.6700
Gly-Gly-PALO RMUG-S CTRP1 2.0833 266.6700
Gly-Gly-PALO SK-OV-3 CTRP1 0.2603 33.3330
Gly-Gly-PALO SNU-840 CTRP1 2.0833 266.6700
Gly-Gly-PALO TYK-NU CTRP1 2.0833 266.6700
Gly-Gly-PALO CAPAN-2 CTRP1 0.2603 33.3330
Gly-Gly-PALO CFPAC-1 CTRP1 0.2603 33.3330
Gly-Gly-PALO HPAC CTRP1 0.2603 33.3330
Gly-Gly-PALO HUP-T4 CTRP1 0.2603 33.3330
Gly-Gly-PALO KP-3 CTRP1 0.2603 33.3330
Gly-Gly-PALO PANC03.27 CTRP1 0.2603 33.3330
Gly-Gly-PALO PANC10.05 CTRP1 0.2603 33.3330
Gly-Gly-PALO PATU8902 CTRP1 0.2603 33.3330
Gly-Gly-PALO QGP-1 CTRP1 0.2603 33.3330
Gly-Gly-PALO SUIT-2 CTRP1 0.2603 33.3330
Gly-Gly-PALO MSTO-211H CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H2052 CTRP1 0.2603 33.3330
Gly-Gly-PALO NCI-H28 CTRP1 0.2603 33.3330
Gly-Gly-PALO MIAPACA-3 CTRP1 0.2603 33.3330
Gly-Gly-PALO A-375 CTRP1 2.0833 266.6700
Gly-Gly-PALO COLO741 CTRP1 0.2603 33.3330
Gly-Gly-PALO G-361 CTRP1 0.2603 33.3330
Gly-Gly-PALO HS852.T CTRP1 0.2603 33.3330
Gly-Gly-PALO HS936.T CTRP1 0.2603 33.3330
Gly-Gly-PALO HS944.T CTRP1 0.2603 33.3330
Gly-Gly-PALO SK-MEL-1 CTRP1 2.0833 266.6700
Gly-Gly-PALO SK-MEL-28 CTRP1 2.0833 266.6700
Gly-Gly-PALO SK-MEL-5 CTRP1 2.0833 266.6700
Gly-Gly-PALO G-401 CTRP1 0.2603 33.3330
Gly-Gly-PALO HT-1080 CTRP1 2.0833 266.6700
Gly-Gly-PALO AGS CTRP1 2.0833 266.6700
Gly-Gly-PALO FU97 CTRP1 0.2603 33.3330
Gly-Gly-PALO KE-97 CTRP1 0.2603 33.3330
Gly-Gly-PALO MKN7 CTRP1 0.2603 33.3330
Gly-Gly-PALO MKN74 CTRP1 0.2603 33.3330
Gly-Gly-PALO NUGC-4 CTRP1 0.2603 33.3330
Gly-Gly-PALO SH-10-TC CTRP1 0.2603 33.3330
Gly-Gly-PALO HSC-2 CTRP1 0.2603 33.3330
Gly-Gly-PALO SCC-9 CTRP1 2.0833 266.6700
Gly-Gly-PALO 5637 CTRP1 0.2603 33.3330
Gly-Gly-PALO HT-1376 CTRP1 0.2603 33.3330
Gly-Gly-PALO KMBC-2 CTRP1 0.2603 33.3330
Gly-Gly-PALO RT-4 CTRP1 0.2603 33.3330
Gly-Gly-PALO UM-UC-3 CTRP1 0.2603 33.3330

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.