Drug : Racemic-2,4-Dideoxy-Dc-45-A2

CTRP1 Name : racemic-2,4-dideoxy-DC-45-A2

Dataset : All
Synonyms :
Targets :
Pathways : trioxacarcin natural product analog

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
racemic-2,4-dideoxy-DC-45-A2 GAMG CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 SF295 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HEC-108 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 HEC-251 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HEC-265 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HEC-59 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 HEC-6 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 KLE CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 MFE-319 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 SNG-M CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 BL-70 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 HT CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 KU812 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 MC116 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 P3HR-1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 VMRC-RCW CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 C2BBE1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 COLO205 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 DLD-1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 GP2D CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 LS411N CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 LS513 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 SK-CO-1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 SNU-C2A CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 SW403 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 SW48 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 JHH-6 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 SNU-449 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 A-549 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 BEN CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 CALU-3 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 CALU-6 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 CHAGO-K-1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 COLO668 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 COR-L279 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 COR-L88 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 DMS273 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 DV-90 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 EBC-1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 EPLC-272H CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HARA[HUMANSQUAMOUSCELLLUNGCARCINOMA] CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HCC33 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HCC44 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HCC78 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 KNS-62 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 LC-1-SQ-SF CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 LCLC-103H CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 LCLC-97TM1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 LU-65 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 LU-99 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 LXF289 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1048 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1299 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1355 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1373 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1435 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1437 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1568 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1573 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1666 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1792 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1793 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1915 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1930 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1944 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H1975 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H2009 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H2029 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H2126 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H2286 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H23 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H2405 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H358 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H522 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H650 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H661 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H727 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H810 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H82 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 RERF-LC-KJ CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 SHP-77 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 VMRC-LCD CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 KYSE-140 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 KYSE-410 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 KYSE-450 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 COV318 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 EFO-21 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HEYA8 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 JHOS-4 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 OVMANA CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 SK-OV-3 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 CAPAN-2 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 CFPAC-1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HPAC CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HUP-T4 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 KP-3 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 PANC03.27 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 PANC10.05 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 PATU8902 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 QGP-1 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 SUIT-2 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 MSTO-211H CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H2052 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 NCI-H28 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 MIAPACA-3 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 COLO741 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 G-361 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HS852.T CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 HS936.T CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HS944.T CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 G-401 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 FU97 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 KE-97 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 MKN7 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 MKN74 CTRP1 0.0030 37.0000
racemic-2,4-dideoxy-DC-45-A2 NUGC-4 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 SH-10-TC CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HSC-2 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 5637 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 HT-1376 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 KMBC-2 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 RT-4 CTRP1 0.2890 37.0000
racemic-2,4-dideoxy-DC-45-A2 UM-UC-3 CTRP1 0.2890 37.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.