Cellosaurus Index : CVCL_3001
Cellosaurus ID : KON
CCLE Name
: KON_UPPER_AERODIGESTIVE_TRACT
GDSC1 Name
, GDSC2 Name
: KON
Cancer Type : upper_aerodigestive_tract
Dataset : All
Click to show/hide information cards below or download all drug response information.
 Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.
Experimental information from All dataset, including cell line name, drug name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.
| Cellosaurus ID | Drug Name | Original Dataset(s) | Min Dose | Max Dose | Dose-response |
|---|---|---|---|---|---|
| KON | (5Z)-7-Oxozeaenol | GDSC1 | 0.0391 | 10.0000 |
|
| KON | 5-Fluorouracil | GDSC1,GDSC2 | 0.0200 | 32.0000 |
|
| KON | 965-D2 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | 993-D2 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | A-83-01 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | ABT737 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | ACY-1215 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Afatinib | GDSC1,GDSC2 | 0.0020 | 10.0000 |
|
| KON | Afuresertib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | AGI-5198 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | AGI-6780 | GDSC1,GDSC2 | 0.0020 | 10.0000 |
|
| KON | AGK-2 | GDSC2 | 0.0040 | 4.0000 |
|
| KON | AICA Ribonucleotide | GDSC1 | 7.8125 | 2000.0000 |
|
| KON | AKT inhibitor VIII | GDSC1 | 0.0100 | 10.2400 |
|
| KON | Alectinib | GDSC1 | 0.0200 | 5.1200 |
|
| KON | Alisertib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Alpelisib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | AMG-319 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Amuvatinib | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Apitolisib | GDSC1 | 0.0781 | 20.0000 |
|
| KON | AR-42 | GDSC1 | 0.0200 | 5.1200 |
|
| KON | Ara-G | GDSC1 | 0.0781 | 20.0000 |
|
| KON | ARRY-520 | GDSC1 | 0.0010 | 0.2560 |
|
| KON | AS601245 | GDSC1 | 0.0312 | 8.0000 |
|
| KON | AS605240 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | AST-1306 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | AT-7519 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | AT13148 | GDSC2 | 0.0080 | 8.0000 |
|
| KON | AT7867 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Avagacestat | GDSC1,GDSC2 | 0.0100 | 10.2400 |
|
| KON | Axitinib | GDSC1,GDSC2 | 0.0078 | 10.0000 |
|
| KON | AZ20 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | AZ6102 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | AZ960 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | AZD1208 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | AZD1332 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | AZD1480 | GDSC1 | 0.0098 | 2.5000 |
|
| KON | AZD2014 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | AZD3514 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | AZD3759 | GDSC2 | 0.0010 | 1.0000 |
|
| KON | AZD4547 | GDSC1,GDSC2 | 0.0039 | 10.0000 |
|
| KON | AZD4877 | GDSC1 | 0.0002 | 0.0390 |
|
| KON | AZD5363 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | AZD5438 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | AZD5582 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | AZD6094 | GDSC1 | 0.0098 | 2.5000 |
|
| KON | AZD6482 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | AZD6738 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | AZD7762 | GDSC1,GDSC2 | 0.0010 | 10.0000 |
|
| KON | AZD7969 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | AZD8055 | GDSC1 | 0.0078 | 2.0000 |
|
| KON | AZD8186 | GDSC1,GDSC2 | 0.0098 | 10.0000 |
|
| KON | AZD8835 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | AZD8931 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | BAM7 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | BAY ACCi | GDSC1 | 0.0391 | 10.0000 |
|
| KON | BAY AKT1 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | BAY-61-3606 | GDSC1 | 0.0312 | 8.0000 |
|
| KON | BAY-HDAC11_1 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | BAY-HDAC11_2 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | BAY-HDAC11_4 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | BAY-MPS-combo 2 (paclitaxel 1 uM) | GDSC1 | 0.0039 | 1.0000 |
|
| KON | BAY-MPS-combo-1 (paclitaxel 5 uM) | GDSC1 | 0.0039 | 1.0000 |
|
| KON | BAY-MPS1 | GDSC1 | 0.0117 | 3.0000 |
|
| KON | Belinostat | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Bexarotene | GDSC1 | 0.0312 | 8.0000 |
|
| KON | BI-2536 | GDSC2 | 0.0005 | 0.5000 |
|
| KON | BIBF-1120 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | BIBR-1532 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Bicalutamide | GDSC1,GDSC2 | 0.0040 | 10.0000 |
|
| KON | BIX02189 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Bleomycin | GDSC1 | 0.2500 | 64.0000 |
|
| KON | Bleomycin (10 uM) | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Bleomycin (50 uM) | GDSC1 | 0.1953 | 50.0000 |
|
| KON | BMS-345541 | GDSC1,GDSC2 | 0.0100 | 16.0000 |
|
| KON | BMS-536924 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | BMS-754807 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Bortezomib | GDSC2 | 0.0000 | 0.0200 |
|
| KON | Bosutinib | GDSC1,GDSC2 | 0.0020 | 2.0000 |
|
| KON | BPTES | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Brivanib, BMS-540215 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Bryostatin 1 | GDSC1 | 0.0000 | 0.0080 |
|
| KON | Buparlisib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | BX-912 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | BX795 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | C-75 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Cabozantinib | GDSC1 | 0.0200 | 5.1200 |
|
| KON | Camptothecin | GDSC2 | 0.0001 | 0.1000 |
|
| KON | CAP-232, TT-232, TLN-232 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Capivasertib | GDSC1 | 0.1172 | 30.0000 |
|
| KON | CAY10566 | GDSC1 | 0.0100 | 2.5600 |
|
| KON | CAY10603 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | CCT-018159 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | CCT007093 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | CCT245232 | GDSC1 | 0.0008 | 0.2000 |
|
| KON | CCT245467 | GDSC1 | 0.0008 | 0.2000 |
|
| KON | CD532 | GDSC1 | 0.0200 | 5.1200 |
|
| KON | Cediranib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Cetuximab | GDSC1 | 0.2570 | 65.8000 |
|
| KON | CHIR-99021 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | CI-1033 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | CI-1040 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Cisplatin | GDSC1 | 0.0117 | 10.0000 |
|
| KON | CP466722 | GDSC1 | 0.0625 | 16.0000 |
|
| KON | CP724714 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | CPI-613 | GDSC1 | 1.0000 | 256.0000 |
|
| KON | Crizotinib | GDSC2 | 0.0040 | 8.0000 |
|
| KON | CRT0105446 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | CRT0105950 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | CRT0160829 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | CUDC-101 | GDSC1 | 0.0200 | 5.1200 |
|
| KON | CX-5461 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Cyclophosphamide | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Cytarabine | GDSC1 | 0.0078 | 2.0000 |
|
| KON | CZC24832 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Dabrafenib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Dacinostat | GDSC1 | 0.0040 | 1.0240 |
|
| KON | Dactinomycin | GDSC2 | 0.0008 | 0.8000 |
|
| KON | Dactolisib | GDSC1,GDSC2 | 0.0003 | 0.2500 |
|
| KON | Daporinad | GDSC1,GDSC2 | 0.0010 | 1.0000 |
|
| KON | Dasatinib | GDSC2 | 0.0020 | 2.0000 |
|
| KON | Dinaciclib | GDSC2 | 0.0010 | 1.0000 |
|
| KON | DMOG | GDSC1 | 15.6250 | 4000.0000 |
|
| KON | Docetaxel | GDSC1,GDSC2 | 0.0000 | 0.0125 |
|
| KON | Doramapimod | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Doxorubicin | GDSC1 | 0.0040 | 5.0000 |
|
| KON | Dyrk1b_0191 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | eEF2K Inhibitor, A-484954 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | EHT-1864 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Elesclomol | GDSC1,GDSC2 | 0.0002 | 0.2000 |
|
| KON | Embelin | GDSC1 | 0.1250 | 32.0000 |
|
| KON | Entinostat | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Entospletinib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Enzastaurin | GDSC1 | 0.0781 | 20.0000 |
|
| KON | EphB4_9721 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Epirubicin | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Epothilone B | GDSC1 | 0.0001 | 0.0320 |
|
| KON | EPZ004777 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | EPZ5676 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Erlotinib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Etoposide | GDSC1 | 0.0625 | 16.0000 |
|
| KON | ETP-45835 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Fedratinib | GDSC1 | 0.0400 | 10.2400 |
|
| KON | FEN1_3940 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | FGFR_0939 | GDSC1 | 0.0098 | 2.5000 |
|
| KON | FGFR_3831 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | FH535 | GDSC1 | 0.1250 | 32.0000 |
|
| KON | Flavopiridol | GDSC1 | 0.0100 | 2.5600 |
|
| KON | FMK | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Foretinib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | FR-180204 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | FS106 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | FS112 | GDSC1 | 0.0195 | 5.0000 |
|
| KON | FTI-277 | GDSC1 | 0.0040 | 1.0240 |
|
| KON | FTY-720 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Fulvestrant | GDSC1,GDSC2 | 0.0010 | 10.0000 |
|
| KON | FY012 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | FY026 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | FY069 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | GDC0810 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Gefitinib | GDSC1,GDSC2 | 0.0020 | 2.0000 |
|
| KON | Gemcitabine | GDSC1,GDSC2 | 0.0002 | 10.0000 |
|
| KON | Genentech Cpd 10 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | GNE-317 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | GSK-J4 | GDSC1 | 0.1172 | 30.0000 |
|
| KON | GSK1059615 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | GSK1070916 | GDSC1 | 0.0100 | 2.5600 |
|
| KON | GSK1904529A | GDSC1,GDSC2 | 0.0040 | 5.0000 |
|
| KON | GSK2578215A | GDSC2 | 0.0100 | 10.0000 |
|
| KON | GSK2606414 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | GSK269962A | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | GSK343 | GDSC2 | 0.0010 | 1.0000 |
|
| KON | GSK429286A | GDSC1 | 0.0781 | 20.0000 |
|
| KON | GSK591 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | GSK650394 | GDSC1 | 0.0625 | 16.0000 |
|
| KON | GSK690693 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | GW-2580 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | GW441756 | GDSC1,GDSC2 | 0.0020 | 2.0000 |
|
| KON | HG6-64-1 | GDSC1 | 0.0200 | 5.1200 |
|
| KON | I-BET-762 | GDSC1,GDSC2 | 0.0100 | 20.0000 |
|
| KON | I-BET151 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | I-BRD9 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | I-CBP112 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | IAP_5620 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | IAP_7638 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Ibrutinib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | IC-87114 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | ICL1100013 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Idelalisib | GDSC1 | 0.0781 | 20.0000 |
|
| KON | IGFR_3801 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | IMD-0354 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | IOX2 | GDSC1,GDSC2 | 0.0004 | 0.5000 |
|
| KON | IPA-3 | GDSC1 | 0.1250 | 32.0000 |
|
| KON | Ipatasertib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Irinotecan | GDSC2 | 0.0050 | 5.0000 |
|
| KON | Ispinesib Mesylate | GDSC1 | 0.0005 | 0.1280 |
|
| KON | IWP-2 | GDSC2 | 0.0010 | 1.0000 |
|
| KON | JAK1_3715 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | JAK3_7406 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | JNJ38877605 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | JNK Inhibitor VIII | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | JNK-9L | GDSC1 | 0.0200 | 5.1200 |
|
| KON | JQ1 | GDSC1,GDSC2 | 0.0039 | 10.0000 |
|
| KON | JQ12 | GDSC1 | 0.0200 | 5.1200 |
|
| KON | JW-7-24-1 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | kb NB 142-70 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | KIN001-042 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | KIN001-236 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | KIN001-244 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | KIN001-260 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | KIN001-266 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | KIN001-270 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Kobe2602 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | KRAS (G12C) Inhibitor-12 | GDSC2 | 0.0200 | 20.0000 |
|
| KON | KU-55933 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | KU-60019 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Lapatinib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | LCL161 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | LDN-193189 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Leflunomide | GDSC2 | 0.1001 | 100.0000 |
|
| KON | Lenalidomide | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Lestaurtinib | GDSC1,GDSC2 | 0.0020 | 2.0000 |
|
| KON | LFM-A13 | GDSC1 | 0.0625 | 16.0000 |
|
| KON | LGK974 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | LIMK1 inhibitor BMS4 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Linifanib | GDSC1 | 0.0040 | 1.0240 |
|
| KON | Linsitinib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | LJI308 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Luminespib | GDSC1,GDSC2 | 0.0003 | 0.2560 |
|
| KON | LY2109761 | GDSC2 | 0.0050 | 5.0000 |
|
| KON | Masitinib | GDSC1 | 0.0781 | 20.0000 |
|
| KON | MCT1_6447 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | MCT4_1422 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | MetAP2 Inhibitor, A832234 | GDSC1 | 0.0100 | 2.5600 |
|
| KON | Methotrexate | GDSC1,GDSC2 | 0.0008 | 1.0000 |
|
| KON | MG-132 | GDSC2 | 0.0040 | 4.0000 |
|
| KON | Midostaurin | GDSC1 | 0.0020 | 0.5120 |
|
| KON | MIM1 | GDSC1 | 0.1562 | 40.0000 |
|
| KON | MIRA-1 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Mirin | GDSC1,GDSC2 | 0.1001 | 100.0000 |
|
| KON | Mitomycin-C | GDSC1 | 0.0625 | 16.0000 |
|
| KON | MK-1775 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | MK-2206 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | MK-8776 | GDSC2 | 0.0050 | 5.0000 |
|
| KON | ML323 | GDSC2 | 0.0200 | 20.0000 |
|
| KON | MN-64 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Motesanib | GDSC1,GDSC2 | 0.0078 | 10.0000 |
|
| KON | MPS-1-IN-1 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | N22899-6-C1 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | N23918-95-7 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | N24798-49-A1 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Navitoclax | GDSC1,GDSC2 | 0.0020 | 2.0000 |
|
| KON | NG-25 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Nilotinib | GDSC1,GDSC2 | 0.0078 | 10.0000 |
|
| KON | Niraparib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | NPK76-II-72-1 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | NSC-207895 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | NSC-87877 | GDSC1 | 0.0625 | 16.0000 |
|
| KON | NSC319726 | GDSC1 | 0.0010 | 0.2560 |
|
| KON | NU7441 | GDSC1,GDSC2 | 0.0078 | 10.0000 |
|
| KON | Nutlin-3a | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | NVP-ADW742 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | NVP-BHG712 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Obatoclax Mesylate | GDSC1 | 0.0625 | 16.0000 |
|
| KON | OF-1 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Olaparib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Omipalisib | GDSC1 | 0.0005 | 0.1280 |
|
| KON | OSI-027 | GDSC1,GDSC2 | 0.0100 | 20.0000 |
|
| KON | OSI-930 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Osimertinib | GDSC2 | 0.0010 | 1.0000 |
|
| KON | OSU-03012 | GDSC1 | 0.0625 | 16.0000 |
|
| KON | OTX015 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Oxaliplatin | GDSC2 | 0.0100 | 10.0000 |
|
| KON | P22077 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | PAC-1 | GDSC1 | 0.0100 | 2.5600 |
|
| KON | Paclitaxel | GDSC2 | 0.0001 | 0.1000 |
|
| KON | Palbociclib | GDSC1,GDSC2 | 0.0040 | 4.0000 |
|
| KON | Panobinostat | GDSC1 | 0.0040 | 1.0240 |
|
| KON | PARP_0108 | GDSC1 | 0.0098 | 2.5000 |
|
| KON | PARP_9482 | GDSC1 | 0.0098 | 2.5000 |
|
| KON | PARP_9495 | GDSC1 | 0.0098 | 2.5000 |
|
| KON | Pazopanib | GDSC1 | 0.0312 | 8.0000 |
|
| KON | PCI-34051 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | PD0325901 | GDSC1,GDSC2 | 0.0010 | 2.5000 |
|
| KON | PD173074 | GDSC1,GDSC2 | 0.0078 | 10.0000 |
|
| KON | Pelitinib | GDSC1 | 0.0098 | 2.5000 |
|
| KON | Pemetrexed | GDSC1 | 0.0100 | 2.5600 |
|
| KON | Pevonedistat | GDSC1,GDSC2 | 0.0039 | 10.0000 |
|
| KON | PF-00299804 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | PF-4708671 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | PF-562271 | GDSC1 | 0.0100 | 2.5600 |
|
| KON | PFI-1 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | PFI3 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | PHA-793887 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Phenformin | GDSC1 | 15.6250 | 4000.0000 |
|
| KON | PI-103 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | PI3Ka_4409 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Picolinici-acid | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Pictilisib | GDSC1,GDSC2 | 0.0040 | 4.0000 |
|
| KON | PIK-93 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Pilaralisib | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Piperlongumine | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | PLK_6522 | GDSC1 | 0.0024 | 0.6250 |
|
| KON | PLX-4720 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Ponatinib | GDSC1 | 0.0020 | 0.5120 |
|
| KON | PRIMA-1MET | GDSC2 | 0.0300 | 30.0000 |
|
| KON | PRT062607 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Pyridostatin | GDSC2 | 0.0100 | 10.0000 |
|
| KON | QL-X-138 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | QL-XI-92 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | QL-XII-47 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | QS11 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Quizartinib | GDSC1 | 0.0040 | 1.0240 |
|
| KON | RAF_9304 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Rapamycin | GDSC2 | 0.0001 | 0.1000 |
|
| KON | Refametinib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Ribociclib | GDSC2 | 0.0020 | 2.0000 |
|
| KON | RO-3306 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | rTRAIL | GDSC1 | 0.0004 | 0.1000 |
|
| KON | RU-SKI 43 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Rucaparib | GDSC1,GDSC2 | 0.0050 | 5.0000 |
|
| KON | Ruxolitinib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | RVX-208 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Sabutoclax | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Sapitinib | GDSC2 | 0.0050 | 5.0000 |
|
| KON | Savolitinib | GDSC2 | 0.0010 | 1.0000 |
|
| KON | SB216763 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | SB505124 | GDSC1,GDSC2 | 0.0100 | 20.0000 |
|
| KON | SB52334 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | SB590885 | GDSC1,GDSC2 | 0.0050 | 5.0000 |
|
| KON | SCH772984 | GDSC2 | 0.0050 | 5.0000 |
|
| KON | Selisistat | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Selumetinib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Sepantronium bromide | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Serdemetan | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | SGC0946 | GDSC1,GDSC2 | 0.0005 | 0.5000 |
|
| KON | Shikonin | GDSC1 | 0.0625 | 16.0000 |
|
| KON | SL0101 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | SN-38 | GDSC1,GDSC2 | 0.0002 | 10.0000 |
|
| KON | SNX-2112 | GDSC1 | 0.0100 | 2.5600 |
|
| KON | Sorafenib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Sphingosine Kinase 1 Inhibitor II | GDSC1 | 0.0100 | 2.5600 |
|
| KON | Staurosporine | GDSC2 | 0.0078 | 2.0000 |
|
| KON | STF-62247 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | SU11274 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | T0901317 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | TAK-715 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Talazoparib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Tamoxifen | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Tanespimycin | GDSC1,GDSC2 | 0.0010 | 1.0000 |
|
| KON | TANK_1366 | GDSC1 | 0.0098 | 2.5000 |
|
| KON | Taselisib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Telomerase Inhibitor IX | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Temozolomide | GDSC1,GDSC2 | 0.0300 | 30.0000 |
|
| KON | Temsirolimus | GDSC1,GDSC2 | 0.0008 | 1.0000 |
|
| KON | Tenovin-6 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Thapsigargin | GDSC1 | 0.0020 | 0.5120 |
|
| KON | THZ-2-102-1 | GDSC1 | 0.0098 | 2.5000 |
|
| KON | THZ-2-49 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Tipifarnib | GDSC1 | 0.0625 | 16.0000 |
|
| KON | Tivozanib | GDSC1 | 0.0005 | 0.1280 |
|
| KON | TL-1-85 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | TL-2-105 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Torin 2 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Tozasertib | GDSC2 | 0.0050 | 5.0000 |
|
| KON | TPCA-1 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Trametinib | GDSC1,GDSC2 | 0.0010 | 1.0000 |
|
| KON | Tretinoin | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Trichostatin A | GDSC1 | 0.0040 | 1.0240 |
|
| KON | TTK_3146 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | Tubastatin A | GDSC1 | 0.0781 | 20.0000 |
|
| KON | TW 37 | GDSC1 | 0.0195 | 5.0000 |
|
| KON | TWS119 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | Ulixertinib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | UNC0638 | GDSC1 | 0.0781 | 40.0000 |
|
| KON | UNC0642 | GDSC1 | 0.0020 | 0.5000 |
|
| KON | UNC1215 | GDSC1 | 0.0039 | 1.0000 |
|
| KON | Uprosertib | GDSC2 | 0.0100 | 10.0000 |
|
| KON | VE-822 | GDSC2 | 0.0050 | 5.0000 |
|
| KON | VE821 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Veliparib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Venetoclax | GDSC2 | 0.0010 | 1.0000 |
|
| KON | Venotoclax | GDSC1 | 0.0010 | 0.2560 |
|
| KON | Vinblastine | GDSC1 | 0.0004 | 0.1000 |
|
| KON | Vinorelbine | GDSC1,GDSC2 | 0.0001 | 0.1000 |
|
| KON | Vismodegib | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | VNLG-124 | GDSC1 | 0.0200 | 5.1200 |
|
| KON | Vorinostat | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | Voxtalisib | GDSC1 | 0.0781 | 20.0000 |
|
| KON | VX-11e | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | VX-702 | GDSC1 | 0.0078 | 2.0000 |
|
| KON | Wee1 Inhibitor | GDSC1,GDSC2 | 0.0078 | 10.0000 |
|
| KON | WEHI-539 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | WHI-P97 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | WIKI4 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | Wnt-C59 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | WYE-125132 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | WZ3105 | GDSC1 | 0.0050 | 1.2800 |
|
| KON | WZ4003 | GDSC2 | 0.0100 | 10.0000 |
|
| KON | XAV939 | GDSC1,GDSC2 | 0.0050 | 5.0000 |
|
| KON | XMD13-2 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | XMD14-99 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | XMD15-27 | GDSC1 | 0.0400 | 10.2400 |
|
| KON | Y-39983 | GDSC1 | 0.0781 | 20.0000 |
|
| KON | YK-4-279 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | YM201636 | GDSC1 | 0.0200 | 5.1200 |
|
| KON | Zibotentan | GDSC1 | 0.0781 | 20.0000 |
|
| KON | ZL049 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | ZL109 | GDSC1 | 0.0391 | 10.0000 |
|
| KON | ZM447439 | GDSC1,GDSC2 | 0.0100 | 10.0000 |
|
| KON | ZSTK474 | GDSC1 | 0.0200 | 5.1200 |
|