Drug : Bml-259

CTRP1 Name : BML-259

Dataset : All
Synonyms :
Targets : CDK5;CDK2
Pathways : inhibitor of cyclin-dependent kinase 5 and cyclin-dependent kinase 2

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
BML-259 MCF-7 CTRP1 2.0833 266.6700
BML-259 GAMG CTRP1 0.2603 33.3330
BML-259 LN-229 CTRP1 2.0833 266.6700
BML-259 HEC-108 CTRP1 0.2603 33.3330
BML-259 HEC-151 CTRP1 2.0833 266.6700
BML-259 HEC-59 CTRP1 0.2603 33.3330
BML-259 ISHIKAWA(HERAKLIO)02ER- CTRP1 0.2603 33.3330
BML-259 JHUEM-2 CTRP1 2.0833 266.6700
BML-259 KLE CTRP1 0.2603 33.3330
BML-259 SNG-M CTRP1 0.2603 33.3330
BML-259 AMO1 CTRP1 2.0833 266.6700
BML-259 BL-70 CTRP1 0.2603 33.3330
BML-259 EJM CTRP1 2.0833 266.6700
BML-259 GDM-1 CTRP1 2.0833 266.6700
BML-259 KMS-11 CTRP1 2.0833 266.6700
BML-259 LP-1 CTRP1 2.0833 266.6700
BML-259 MOLM-16 CTRP1 2.0833 266.6700
BML-259 NOMO-1 CTRP1 2.0833 266.6700
BML-259 NU-DUL-1 CTRP1 2.0833 266.6700
BML-259 OCI-AML-3 CTRP1 2.0833 266.6700
BML-259 OCI-LY10 CTRP1 2.0833 266.6700
BML-259 PL21 CTRP1 2.0833 266.6700
BML-259 RPMI-8226 CTRP1 2.0833 266.6700
BML-259 SKM-1 CTRP1 2.0833 266.6700
BML-259 SU-DHL-4 CTRP1 2.0833 266.6700
BML-259 SU-DHL-5 CTRP1 2.0833 266.6700
BML-259 THP-1 CTRP1 2.0833 266.6700
BML-259 U-937 CTRP1 2.0833 266.6700
BML-259 WSU-DLCL2 CTRP1 2.0833 266.6700
BML-259 RCC10RGB CTRP1 2.0833 266.6700
BML-259 CL-34 CTRP1 2.0833 266.6700
BML-259 CL-40 CTRP1 2.0833 266.6700
BML-259 COLO320 CTRP1 2.0833 266.6700
BML-259 COLO678 CTRP1 2.0833 266.6700
BML-259 CW-2 CTRP1 2.0833 266.6700
BML-259 HCT116 CTRP1 2.0833 266.6700
BML-259 HCT8 CTRP1 2.0833 266.6700
BML-259 HT115 CTRP1 2.0833 266.6700
BML-259 HT-29 CTRP1 2.0833 266.6700
BML-259 HT-55 CTRP1 2.0833 266.6700
BML-259 KM12 CTRP1 2.0833 266.6700
BML-259 LOVO CTRP1 2.0833 266.6700
BML-259 LS123 CTRP1 2.0833 266.6700
BML-259 LS180 CTRP1 2.0833 266.6700
BML-259 MDST8 CTRP1 2.0833 266.6700
BML-259 NCI-H508 CTRP1 2.0833 266.6700
BML-259 RCM-1[HUMANESC] CTRP1 2.0833 266.6700
BML-259 RKO CTRP1 2.0833 266.6700
BML-259 SNU-1040 CTRP1 2.0833 266.6700
BML-259 SNU-175 CTRP1 2.0833 266.6700
BML-259 SNU-61 CTRP1 2.0833 266.6700
BML-259 SNU-81 CTRP1 2.0833 266.6700
BML-259 SNU-C4 CTRP1 2.0833 266.6700
BML-259 SNU-C5 CTRP1 2.0833 266.6700
BML-259 SW480 CTRP1 2.0833 266.6700
BML-259 SW620 CTRP1 2.0833 266.6700
BML-259 SW948 CTRP1 2.0833 266.6700
BML-259 HEP-G2 CTRP1 2.0833 266.6700
BML-259 JHH-6 CTRP1 0.2603 33.3330
BML-259 SNU-398 CTRP1 2.0833 266.6700
BML-259 SNU-449 CTRP1 0.2603 33.3330
BML-259 CAL-12T CTRP1 2.0833 266.6700
BML-259 COLO668 CTRP1 0.2603 33.3330
BML-259 COLO699 CTRP1 2.0833 266.6700
BML-259 COR-L23 CTRP1 2.0833 266.6700
BML-259 COR-L51 CTRP1 2.0833 266.6700
BML-259 HCC1195 CTRP1 2.0833 266.6700
BML-259 HCC1359 CTRP1 2.0833 266.6700
BML-259 HCC15 CTRP1 2.0833 266.6700
BML-259 HCC1833 CTRP1 2.0833 266.6700
BML-259 HCC2108 CTRP1 2.0833 266.6700
BML-259 HCC2935 CTRP1 2.0833 266.6700
BML-259 HCC4006 CTRP1 2.0833 266.6700
BML-259 HCC827 CTRP1 2.0833 266.6700
BML-259 LXF289 CTRP1 0.2603 33.3330
BML-259 NCI-H1105 CTRP1 2.0833 266.6700
BML-259 NCI-H1435 CTRP1 0.2603 33.3330
BML-259 NCI-H1694 CTRP1 2.0833 266.6700
BML-259 NCI-H1755 CTRP1 2.0833 266.6700
BML-259 NCI-H1781 CTRP1 2.0833 266.6700
BML-259 NCI-H1836 CTRP1 2.0833 266.6700
BML-259 NCI-H1876 CTRP1 2.0833 266.6700
BML-259 NCI-H1915 CTRP1 0.2603 33.3330
BML-259 NCI-H1930 CTRP1 0.2603 33.3330
BML-259 NCI-H1963 CTRP1 2.0833 266.6700
BML-259 NCI-H2023 CTRP1 2.0833 266.6700
BML-259 NCI-H2030 CTRP1 2.0833 266.6700
BML-259 NCI-H2073 CTRP1 2.0833 266.6700
BML-259 NCI-H2081 CTRP1 2.0833 266.6700
BML-259 NCI-H2110 CTRP1 2.0833 266.6700
BML-259 NCI-H2122 CTRP1 2.0833 266.6700
BML-259 NCI-H2141 CTRP1 2.0833 266.6700
BML-259 NCI-H2172 CTRP1 2.0833 266.6700
BML-259 NCI-H2286 CTRP1 0.2603 33.3330
BML-259 NCI-H2342 CTRP1 2.0833 266.6700
BML-259 NCI-H3255 CTRP1 2.0833 266.6700
BML-259 NCI-H441 CTRP1 2.0833 266.6700
BML-259 NCI-H460 CTRP1 2.0833 266.6700
BML-259 NCI-H596 CTRP1 2.0833 266.6700
BML-259 NCI-H841 CTRP1 2.0833 266.6700
BML-259 RERF-LC-KJ CTRP1 0.2603 33.3330
BML-259 SCLC-21H CTRP1 2.0833 266.6700
BML-259 SK-LU-1 CTRP1 2.0833 266.6700
BML-259 SQ-1 CTRP1 2.0833 266.6700
BML-259 T3M-10 CTRP1 2.0833 266.6700
BML-259 A2780 CTRP1 2.0833 266.6700
BML-259 CAOV-3 CTRP1 2.0833 266.6700
BML-259 COV318 CTRP1 0.2603 33.3330
BML-259 COV362 CTRP1 2.0833 266.6700
BML-259 COV434 CTRP1 2.0833 266.6700
BML-259 COV644 CTRP1 2.0833 266.6700
BML-259 EFO-27 CTRP1 2.0833 266.6700
BML-259 IGROV-1 CTRP1 2.0833 266.6700
BML-259 JHOC-5 CTRP1 2.0833 266.6700
BML-259 JHOM-1 CTRP1 2.0833 266.6700
BML-259 JHOS-4 CTRP1 0.2603 33.3330
BML-259 OAW42 CTRP1 2.0833 266.6700
BML-259 OV7 CTRP1 2.0833 266.6700
BML-259 OV-90 CTRP1 2.0833 266.6700
BML-259 OVCAR-4 CTRP1 2.0833 266.6700
BML-259 OVCAR-8 CTRP1 2.0833 266.6700
BML-259 OVK18 CTRP1 2.0833 266.6700
BML-259 OVKATE CTRP1 2.0833 266.6700
BML-259 OVMANA CTRP1 0.2603 33.3330
BML-259 RKN CTRP1 2.0833 266.6700
BML-259 RMG-I CTRP1 2.0833 266.6700
BML-259 RMUG-S CTRP1 2.0833 266.6700
BML-259 SNU-840 CTRP1 2.0833 266.6700
BML-259 TYK-NU CTRP1 2.0833 266.6700
BML-259 PATU8902 CTRP1 0.2603 33.3330
BML-259 MIAPACA-3 CTRP1 0.2603 33.3330
BML-259 A-375 CTRP1 2.0833 266.6700
BML-259 HS852.T CTRP1 0.2603 33.3330
BML-259 SK-MEL-1 CTRP1 2.0833 266.6700
BML-259 SK-MEL-28 CTRP1 2.0833 266.6700
BML-259 SK-MEL-5 CTRP1 2.0833 266.6700
BML-259 HT-1080 CTRP1 2.0833 266.6700
BML-259 AGS CTRP1 2.0833 266.6700
BML-259 MKN74 CTRP1 0.2603 33.3330
BML-259 SCC-9 CTRP1 2.0833 266.6700

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.