Drug : Pf-3758309

CTRP2 Name : PF-3758309

Dataset : All
Synonyms :
Targets : PAK4
Pathways : inhibitor of serine/threonine p21-activating kinase 4

Information Cards

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Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
PF-3758309 C2BBE1 CTRP2 0.0020 66.0000
PF-3758309 CHAGO-K-1 CTRP2 0.0020 66.0000
PF-3758309 COLO668 CTRP2 0.0020 66.0000
PF-3758309 COV362 CTRP2 0.0020 66.0000
PF-3758309 DV-90 CTRP2 0.0020 66.0000
PF-3758309 EFO-27 CTRP2 0.0020 66.0000
PF-3758309 HD-MY-Z CTRP2 0.0020 66.0000
PF-3758309 NCI-H2170 CTRP2 0.0020 66.0000
PF-3758309 NCI-H647 CTRP2 0.0020 66.0000
PF-3758309 NCI-H810 CTRP2 0.0020 66.0000
PF-3758309 OCI-AML-3 CTRP2 0.0020 66.0000
PF-3758309 PATU8988S CTRP2 0.0020 66.0000
PF-3758309 MIAPACA-3 CTRP2 0.0020 66.0000
PF-3758309 TE-5 CTRP2 0.0020 66.0000
PF-3758309 UACC-257 CTRP2 0.0020 66.0000
PF-3758309 UACC-62 CTRP2 0.0020 66.0000
PF-3758309 BICR6 CTRP2 0.0020 66.0000
PF-3758309 BT145 CTRP2 0.0020 66.0000
PF-3758309 BT179 CTRP2 0.0020 66.0000
PF-3758309 EC-GI-10 CTRP2 0.0020 66.0000
PF-3758309 EFO-21 CTRP2 0.0020 66.0000
PF-3758309 FTC-133 CTRP2 0.0020 66.0000
PF-3758309 JHUEM-3 CTRP2 0.0020 66.0000
PF-3758309 LK2 CTRP2 0.0020 66.0000
PF-3758309 LNCAPCLONEFGC CTRP2 0.0020 66.0000
PF-3758309 LS1034 CTRP2 0.0020 66.0000
PF-3758309 MKN7 CTRP2 0.0020 66.0000
PF-3758309 HCC1428 CTRP2 0.0020 66.0000
PF-3758309 NCI-H2029 CTRP2 0.0020 66.0000
PF-3758309 OE21 CTRP2 0.0020 66.0000
PF-3758309 MKN74 CTRP2 0.0020 66.0000
PF-3758309 SH-10-TC CTRP2 0.0020 66.0000
PF-3758309 SNU-449 CTRP2 0.0020 66.0000
PF-3758309 T3M-10 CTRP2 0.0020 66.0000
PF-3758309 BT112 CTRP2 0.0020 66.0000
PF-3758309 BT164 CTRP2 0.0020 66.0000
PF-3758309 CCF-STTG1 CTRP2 0.0020 66.0000
PF-3758309 COLO800 CTRP2 0.0020 66.0000
PF-3758309 DK-MG CTRP2 0.0020 66.0000
PF-3758309 GP2D CTRP2 0.0020 66.0000
PF-3758309 NCI-H1869 CTRP2 0.0020 66.0000
PF-3758309 HCC38 CTRP2 0.0020 66.0000
PF-3758309 IA-LM CTRP2 0.0020 66.0000
PF-3758309 JHOM-1 CTRP2 0.0020 66.0000
PF-3758309 JHUEM-7 CTRP2 0.0020 66.0000
PF-3758309 JL-1 CTRP2 0.0020 66.0000
PF-3758309 KYSE-450 CTRP2 0.0020 66.0000
PF-3758309 LC-1-SQ-SF CTRP2 0.0020 66.0000
PF-3758309 RCM-1[HUMANESC] CTRP2 0.0020 66.0000
PF-3758309 SNU-685 CTRP2 0.0020 66.0000
PF-3758309 VMRC-LCD CTRP2 0.0020 66.0000
PF-3758309 BT224 CTRP2 0.0020 33.0000
PF-3758309 BT-549 CTRP2 0.0020 66.0000
PF-3758309 HELA CTRP2 0.0020 66.0000
PF-3758309 HCC202 CTRP2 0.0020 33.0000
PF-3758309 H-STS CTRP2 0.0020 33.0000
PF-3758309 K029AX CTRP2 0.0020 33.0000
PF-3758309 KYSE-520 CTRP2 0.0020 66.0000
PF-3758309 LOX-IMVI CTRP2 0.0020 66.0000
PF-3758309 NCI-H1623 CTRP2 0.0020 66.0000
PF-3758309 NCI-H716 CTRP2 0.0020 33.0000
PF-3758309 OE19 CTRP2 0.0020 33.0000
PF-3758309 OE33 CTRP2 0.0020 33.0000
PF-3758309 N2A-PK1 CTRP2 0.0020 33.0000
PF-3758309 PK-45H CTRP2 0.0020 33.0000
PF-3758309 P-STS CTRP2 0.0020 66.0000
PF-3758309 RERF-LC-AD2 CTRP2 0.0020 66.0000
PF-3758309 U-CH1 CTRP2 0.0020 66.0000
PF-3758309 697 CTRP2 0.0020 66.0000
PF-3758309 A3-KAWAKAMI CTRP2 0.0020 66.0000
PF-3758309 BL-41 CTRP2 0.0020 66.0000
PF-3758309 CA46 CTRP2 0.0020 66.0000
PF-3758309 COR-L279 CTRP2 0.0020 66.0000
PF-3758309 COR-L47 CTRP2 0.0020 66.0000
PF-3758309 COR-L51 CTRP2 0.0020 66.0000
PF-3758309 DU4475 CTRP2 0.0020 66.0000
PF-3758309 EB1 CTRP2 0.0020 66.0000
PF-3758309 EOL-1 CTRP2 0.0020 66.0000
PF-3758309 GA-10 CTRP2 0.0020 66.0000
PF-3758309 MOLT-3 CTRP2 0.0020 66.0000
PF-3758309 NAMALWA CTRP2 0.0020 66.0000
PF-3758309 OPM-2 CTRP2 0.0020 66.0000
PF-3758309 PFEIFFER CTRP2 0.0020 66.0000
PF-3758309 SCLC-21H CTRP2 0.0020 66.0000
PF-3758309 SUP-M2 CTRP2 0.0020 66.0000
PF-3758309 TOLEDO CTRP2 0.0020 66.0000
PF-3758309 COLO829 CTRP2 0.0020 66.0000
PF-3758309 DAN-G CTRP2 0.0020 66.0000
PF-3758309 EJM CTRP2 0.0020 66.0000
PF-3758309 GRANTA-519 CTRP2 0.0020 66.0000
PF-3758309 HCC1500 CTRP2 0.0020 66.0000
PF-3758309 IGR-1 CTRP2 0.0020 66.0000
PF-3758309 NCI-H841 CTRP2 0.0020 66.0000
PF-3758309 OCI-LY10 CTRP2 0.0020 66.0000
PF-3758309 OCI-LY19 CTRP2 0.0020 66.0000
PF-3758309 OCI-LY3 CTRP2 0.0020 66.0000
PF-3758309 U-118MG CTRP2 0.0020 66.0000
PF-3758309 COR-L88 CTRP2 0.0020 66.0000
PF-3758309 LU-65 CTRP2 0.0020 66.0000
PF-3758309 NCI-H2081 CTRP2 0.0020 66.0000
PF-3758309 NCI-H2141 CTRP2 0.0020 66.0000
PF-3758309 A-172 CTRP2 0.0020 66.0000
PF-3758309 COV644 CTRP2 0.0020 66.0000
PF-3758309 IM95 CTRP2 0.0020 66.0000
PF-3758309 J82 CTRP2 0.0020 66.0000
PF-3758309 NCI-H23 CTRP2 0.0020 66.0000
PF-3758309 RD CTRP2 0.0020 66.0000
PF-3758309 SK-UT-1 CTRP2 0.0020 66.0000
PF-3758309 T98G CTRP2 0.0020 66.0000
PF-3758309 BECKER CTRP2 0.0020 66.0000
PF-3758309 HS578T CTRP2 0.0020 66.0000
PF-3758309 HS611.T CTRP2 0.0020 66.0000
PF-3758309 JHH-4 CTRP2 0.0020 66.0000
PF-3758309 KARPAS-422 CTRP2 0.0020 66.0000
PF-3758309 KMRC-1 CTRP2 0.0020 66.0000
PF-3758309 LP-1 CTRP2 0.0020 66.0000
PF-3758309 MDA-MB-468 CTRP2 0.0020 66.0000
PF-3758309 SH4 CTRP2 0.0020 33.0000
PF-3758309 SK-HEP-1 CTRP2 0.0020 66.0000
PF-3758309 SUP-HD1 CTRP2 0.0020 66.0000
PF-3758309 AN3-CA CTRP2 0.0020 66.0000
PF-3758309 ACHN CTRP2 0.0020 66.0000
PF-3758309 CMK CTRP2 0.0020 66.0000
PF-3758309 EN CTRP2 0.0020 66.0000
PF-3758309 KASUMI-1 CTRP2 0.0020 66.0000
PF-3758309 NCI-H2342 CTRP2 0.0020 66.0000
PF-3758309 OV-90 CTRP2 0.0020 66.0000
PF-3758309 RERF-LC-MS CTRP2 0.0020 66.0000
PF-3758309 RPMI-6666 CTRP2 0.0020 66.0000
PF-3758309 SK-N-MC CTRP2 0.0020 66.0000
PF-3758309 A-253 CTRP2 0.0020 66.0000
PF-3758309 BC-3C CTRP2 0.0020 66.0000
PF-3758309 C32[HUMANMELANOMA] CTRP2 0.0020 66.0000
PF-3758309 CAL-85-1 CTRP2 0.0020 66.0000
PF-3758309 COLO684 CTRP2 0.0020 66.0000
PF-3758309 HS746.T CTRP2 0.0020 66.0000
PF-3758309 HSC-2 CTRP2 0.0020 66.0000
PF-3758309 HT-144 CTRP2 0.0020 66.0000
PF-3758309 VMRC-RCZ CTRP2 0.0020 66.0000
PF-3758309 MES-SA CTRP2 0.0020 66.0000
PF-3758309 NCI-H1105 CTRP2 0.0020 66.0000
PF-3758309 NCI-H322 CTRP2 0.0020 66.0000
PF-3758309 OAW42 CTRP2 0.0020 66.0000
PF-3758309 PSN1 CTRP2 0.0020 66.0000
PF-3758309 T24 CTRP2 0.0020 66.0000
PF-3758309 TE441.T CTRP2 0.0020 66.0000
PF-3758309 TT2609-C02 CTRP2 0.0020 66.0000
PF-3758309 CAKI-1 CTRP2 0.0020 66.0000
PF-3758309 COR-L105 CTRP2 0.0020 66.0000
PF-3758309 DMS273 CTRP2 0.0020 66.0000
PF-3758309 ESS-1 CTRP2 0.0020 66.0000
PF-3758309 G-402 CTRP2 0.0020 66.0000
PF-3758309 HOS CTRP2 0.0020 66.0000
PF-3758309 HS294T CTRP2 0.0020 66.0000
PF-3758309 JHH-6 CTRP2 0.0020 66.0000
PF-3758309 MFE-319 CTRP2 0.0020 66.0000
PF-3758309 MOLP-8 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1339 CTRP2 0.0020 66.0000
PF-3758309 OV7 CTRP2 0.0020 66.0000
PF-3758309 PANC03.27 CTRP2 0.0020 66.0000
PF-3758309 PLC-PRF-5 CTRP2 0.0020 66.0000
PF-3758309 SCC-9 CTRP2 0.0020 66.0000
PF-3758309 SK-LMS-1 CTRP2 0.0020 66.0000
PF-3758309 SK-MEL-2 CTRP2 0.0020 66.0000
PF-3758309 JHH-2 CTRP2 0.0020 66.0000
PF-3758309 HLF CTRP2 0.0020 66.0000
PF-3758309 JHH-1 CTRP2 0.0020 66.0000
PF-3758309 OAW28 CTRP2 0.0020 66.0000
PF-3758309 OV56 CTRP2 0.0020 66.0000
PF-3758309 PANC02.03 CTRP2 0.0020 66.0000
PF-3758309 SNU-475 CTRP2 0.0020 66.0000
PF-3758309 TOV-21G CTRP2 0.0020 66.0000
PF-3758309 647V CTRP2 0.0020 66.0000
PF-3758309 8-MG-BA CTRP2 0.0020 66.0000
PF-3758309 A101D CTRP2 0.0020 66.0000
PF-3758309 A2058 CTRP2 0.0020 66.0000
PF-3758309 ASPC-1 CTRP2 0.0020 66.0000
PF-3758309 CAKI-2 CTRP2 0.0020 66.0000
PF-3758309 CAL-27 CTRP2 0.0020 66.0000
PF-3758309 COLO792 CTRP2 0.0020 66.0000
PF-3758309 FTC-238 CTRP2 0.0020 66.0000
PF-3758309 GMS-10 CTRP2 0.0020 66.0000
PF-3758309 GOS-3 CTRP2 0.0020 66.0000
PF-3758309 HMCB CTRP2 0.0020 66.0000
PF-3758309 HUH-1 CTRP2 0.0020 66.0000
PF-3758309 IGR-39 CTRP2 0.0020 66.0000
PF-3758309 IST-MES1 CTRP2 0.0020 66.0000
PF-3758309 M059K CTRP2 0.0020 66.0000
PF-3758309 PATU8988T CTRP2 0.0020 66.0000
PF-3758309 SCABER CTRP2 0.0020 66.0000
PF-3758309 SK-N-SH CTRP2 0.0020 66.0000
PF-3758309 TM-31 CTRP2 0.0020 66.0000
PF-3758309 YH-13 CTRP2 0.0020 66.0000
PF-3758309 A-673 CTRP2 0.0020 66.0000
PF-3758309 DU145 CTRP2 0.0020 66.0000
PF-3758309 FADU CTRP2 0.0020 66.0000
PF-3758309 HCC4006 CTRP2 0.0020 66.0000
PF-3758309 HS683 CTRP2 0.0020 66.0000
PF-3758309 HS729.T CTRP2 0.0020 66.0000
PF-3758309 HT-1080 CTRP2 0.0020 66.0000
PF-3758309 JHH-5 CTRP2 0.0020 66.0000
PF-3758309 JHUEM-1 CTRP2 0.0020 66.0000
PF-3758309 MEWO CTRP2 0.0020 66.0000
PF-3758309 MIAPACA-2 CTRP2 0.0020 66.0000
PF-3758309 NCC-STC-K140 CTRP2 0.0020 66.0000
PF-3758309 SK-MES-1 CTRP2 0.0020 66.0000
PF-3758309 SK-N-DZ CTRP2 0.0020 66.0000
PF-3758309 SW579 CTRP2 0.0020 66.0000
PF-3758309 WM115 CTRP2 0.0020 66.0000
PF-3758309 WM266-4 CTRP2 0.0020 66.0000
PF-3758309 BT-20 CTRP2 0.0020 66.0000
PF-3758309 CAL-54 CTRP2 0.0020 66.0000
PF-3758309 CAPAN-1 CTRP2 0.0020 66.0000
PF-3758309 CHP-212 CTRP2 0.0020 66.0000
PF-3758309 HS895.T CTRP2 0.0020 66.0000
PF-3758309 KATOIII CTRP2 0.0020 66.0000
PF-3758309 KMRC-2 CTRP2 0.0020 66.0000
PF-3758309 KNS-42 CTRP2 0.0020 66.0000
PF-3758309 MPP89 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1693 CTRP2 0.0020 66.0000
PF-3758309 PANC04.03 CTRP2 0.0020 66.0000
PF-3758309 PE-CA-PJ49 CTRP2 0.0020 66.0000
PF-3758309 SK-MEL-24 CTRP2 0.0020 66.0000
PF-3758309 SK-N-AS CTRP2 0.0020 66.0000
PF-3758309 TE617.T CTRP2 0.0020 66.0000
PF-3758309 YKG-1 CTRP2 0.0020 66.0000
PF-3758309 BCP-1 CTRP2 0.0020 66.0000
PF-3758309 BL-70 CTRP2 0.0020 66.0000
PF-3758309 COR-L95 CTRP2 0.0020 66.0000
PF-3758309 D283MED CTRP2 0.0020 66.0000
PF-3758309 HL-60 CTRP2 0.0020 66.0000
PF-3758309 HUP-T3 CTRP2 0.0020 66.0000
PF-3758309 IMR-32 CTRP2 0.0020 66.0000
PF-3758309 KO52 CTRP2 0.0020 66.0000
PF-3758309 MEC1 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1092 CTRP2 0.0020 66.0000
PF-3758309 NCI-H2171 CTRP2 0.0020 66.0000
PF-3758309 NCI-H2196 CTRP2 0.0020 66.0000
PF-3758309 NH-6 CTRP2 0.0020 66.0000
PF-3758309 OCI-M1 CTRP2 0.0020 66.0000
PF-3758309 SIG-M5 CTRP2 0.0020 66.0000
PF-3758309 TF-1 CTRP2 0.0020 66.0000
PF-3758309 UACC-812 CTRP2 0.0020 66.0000
PF-3758309 786-O CTRP2 0.0020 66.0000
PF-3758309 A4-FUKUDA CTRP2 0.0020 66.0000
PF-3758309 HCT15 CTRP2 0.0020 66.0000
PF-3758309 HEL92.1.7 CTRP2 0.0020 66.0000
PF-3758309 HUNS1 CTRP2 0.0020 66.0000
PF-3758309 JHOS-2 CTRP2 0.0020 66.0000
PF-3758309 K-562 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1341 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1568 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1703 CTRP2 0.0020 66.0000
PF-3758309 NCI-H838 CTRP2 0.0020 66.0000
PF-3758309 SK-N-FI CTRP2 0.0020 66.0000
PF-3758309 TE-11 CTRP2 0.0020 66.0000
PF-3758309 DAUDI CTRP2 0.0020 66.0000
PF-3758309 HH[HUMANLYMPHOMA] CTRP2 0.0020 66.0000
PF-3758309 HT-1197 CTRP2 0.0020 66.0000
PF-3758309 LUDLU-1 CTRP2 0.0020 66.0000
PF-3758309 NCI-H146 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1915 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1944 CTRP2 0.0020 66.0000
PF-3758309 NCI-H520 CTRP2 0.0020 66.0000
PF-3758309 NCI-H522 CTRP2 0.0020 66.0000
PF-3758309 PE-CA-PJ41(CLONED2) CTRP2 0.0020 66.0000
PF-3758309 PE-CA-PJ15 CTRP2 0.0020 66.0000
PF-3758309 RVH-421 CTRP2 0.0020 66.0000
PF-3758309 SET-2 CTRP2 0.0020 66.0000
PF-3758309 SNU-16 CTRP2 0.0020 66.0000
PF-3758309 TOV-112D CTRP2 0.0020 66.0000
PF-3758309 DB CTRP2 0.0020 66.0000
PF-3758309 HCC1419 CTRP2 0.0020 66.0000
PF-3758309 HCC-56 CTRP2 0.0020 66.0000
PF-3758309 HS839.T CTRP2 0.0020 66.0000
PF-3758309 NCI-H2110 CTRP2 0.0020 66.0000
PF-3758309 PE-CA-PJ34(CLONEC12) CTRP2 0.0020 66.0000
PF-3758309 SNU-387 CTRP2 0.0020 66.0000
PF-3758309 SNU-503 CTRP2 0.0020 66.0000
PF-3758309 SNU-869 CTRP2 0.0020 66.0000
PF-3758309 SNU-C1 CTRP2 0.0020 66.0000
PF-3758309 SW1990 CTRP2 0.0020 66.0000
PF-3758309 SW948 CTRP2 0.0020 66.0000
PF-3758309 TE15 CTRP2 0.0020 66.0000
PF-3758309 UM-UC-1 CTRP2 0.0020 66.0000
PF-3758309 WM88 CTRP2 0.0020 66.0000
PF-3758309 WM983B CTRP2 0.0020 66.0000
PF-3758309 ZR-75-30 CTRP2 0.0020 66.0000
PF-3758309 CI-1 CTRP2 0.0020 66.0000
PF-3758309 CJM[HUMANMELANOMA] CTRP2 0.0020 66.0000
PF-3758309 HUG1-N CTRP2 0.0020 66.0000
PF-3758309 JEKO-1 CTRP2 0.0020 66.0000
PF-3758309 JM1 CTRP2 0.0020 66.0000
PF-3758309 KP-2 CTRP2 0.0020 66.0000
PF-3758309 LMSU CTRP2 0.0020 66.0000
PF-3758309 MG-63 CTRP2 0.0020 66.0000
PF-3758309 MINO CTRP2 0.0020 66.0000
PF-3758309 MJ CTRP2 0.0020 66.0000
PF-3758309 MOTN-1 CTRP2 0.0020 66.0000
PF-3758309 RL CTRP2 0.0020 66.0000
PF-3758309 SK-MEL-3 CTRP2 0.0020 66.0000
PF-3758309 SNU-1 CTRP2 0.0020 66.0000
PF-3758309 ST486 CTRP2 0.0020 66.0000
PF-3758309 SUP-B15 CTRP2 0.0020 66.0000
PF-3758309 TC71 CTRP2 0.0020 66.0000
PF-3758309 BICR18 CTRP2 0.0020 66.0000
PF-3758309 BICR22 CTRP2 0.0020 66.0000
PF-3758309 BICR31 CTRP2 0.0020 66.0000
PF-3758309 COLO678 CTRP2 0.0020 66.0000
PF-3758309 EFM-192A CTRP2 0.0020 66.0000
PF-3758309 G-401 CTRP2 0.0020 66.0000
PF-3758309 HS888.LU CTRP2 0.0020 66.0000
PF-3758309 KP-N-YN CTRP2 0.0020 66.0000
PF-3758309 NCI-H1395 CTRP2 0.0020 66.0000
PF-3758309 SNU-423 CTRP2 0.0020 66.0000
PF-3758309 SW1417 CTRP2 0.0020 66.0000
PF-3758309 SW1783 CTRP2 0.0020 66.0000
PF-3758309 VCAP CTRP2 0.0020 66.0000
PF-3758309 KE-39 CTRP2 0.0020 66.0000
PF-3758309 DMS454 CTRP2 0.0020 66.0000
PF-3758309 GCT CTRP2 0.0020 66.0000
PF-3758309 HCC2935 CTRP2 0.0020 66.0000
PF-3758309 HOP-62 CTRP2 0.0020 66.0000
PF-3758309 NCI-H747 CTRP2 0.0020 66.0000
PF-3758309 OVCAR-5 CTRP2 0.0020 66.0000
PF-3758309 SF268 CTRP2 0.0020 66.0000
PF-3758309 SF539 CTRP2 0.0020 66.0000
PF-3758309 TUHR14TKB CTRP2 0.5200 66.0000
PF-3758309 U-251MG CTRP2 0.0020 66.0000
PF-3758309 DMS53 CTRP2 0.0020 66.0000
PF-3758309 HEC-1-A CTRP2 0.0020 66.0000
PF-3758309 IGR-37 CTRP2 0.0020 66.0000
PF-3758309 KNS-62 CTRP2 0.0020 66.0000
PF-3758309 MDA-MB-157 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1563 CTRP2 0.0020 66.0000
PF-3758309 OC314 CTRP2 0.0020 66.0000
PF-3758309 UO-31 CTRP2 0.0020 66.0000
PF-3758309 BICR56 CTRP2 0.0020 66.0000
PF-3758309 CAL-33 CTRP2 0.0020 66.0000
PF-3758309 CALU-1 CTRP2 0.0020 66.0000
PF-3758309 CAPAN-2 CTRP2 0.0020 66.0000
PF-3758309 DMS114 CTRP2 0.0020 66.0000
PF-3758309 EKVX CTRP2 0.0020 66.0000
PF-3758309 HCC1438 CTRP2 0.0020 66.0000
PF-3758309 HCT8 CTRP2 0.0020 66.0000
PF-3758309 HOP-92 CTRP2 0.0020 66.0000
PF-3758309 KYM-1 CTRP2 0.0020 66.0000
PF-3758309 KYSE-30 CTRP2 0.0020 66.0000
PF-3758309 KYSE-510 CTRP2 0.0020 66.0000
PF-3758309 L-428 CTRP2 0.0020 66.0000
PF-3758309 MDA-MB-361 CTRP2 0.0020 66.0000
PF-3758309 MFE-296 CTRP2 0.0020 66.0000
PF-3758309 NU-DHL-1 CTRP2 0.0020 66.0000
PF-3758309 SNB-75 CTRP2 0.0020 66.0000
PF-3758309 SNU-216 CTRP2 0.0020 66.0000
PF-3758309 BICR16 CTRP2 0.0020 66.0000
PF-3758309 F-36P CTRP2 0.0020 66.0000
PF-3758309 JJN-3 CTRP2 0.0020 66.0000
PF-3758309 KASUMI-2 CTRP2 0.0020 66.0000
PF-3758309 KG-1-C CTRP2 0.0020 66.0000
PF-3758309 KMS-20 CTRP2 0.0020 66.0000
PF-3758309 KYSE-150 CTRP2 0.0020 66.0000
PF-3758309 OCI-AML-5 CTRP2 0.0020 66.0000
PF-3758309 PANC08.13 CTRP2 0.0020 66.0000
PF-3758309 SNU-601 CTRP2 0.0020 66.0000
PF-3758309 SNU-C4 CTRP2 0.0020 66.0000
PF-3758309 T-47D CTRP2 0.0020 66.0000
PF-3758309 T84 CTRP2 0.0020 66.0000
PF-3758309 TE-14 CTRP2 0.0020 66.0000
PF-3758309 U266B1 CTRP2 0.0020 66.0000
PF-3758309 42-MG-BA CTRP2 0.0020 66.0000
PF-3758309 BT139 CTRP2 0.0020 66.0000
PF-3758309 BT159 CTRP2 0.0020 66.0000
PF-3758309 BT228 CTRP2 0.0020 66.0000
PF-3758309 BT231 CTRP2 0.0020 66.0000
PF-3758309 BT239 CTRP2 0.0020 66.0000
PF-3758309 BT-474 CTRP2 0.0020 66.0000
PF-3758309 COV434 CTRP2 0.0020 66.0000
PF-3758309 DND-41 CTRP2 0.0020 66.0000
PF-3758309 G-292CLONEA141B1 CTRP2 0.0020 66.0000
PF-3758309 HCC2218 CTRP2 0.0020 66.0000
PF-3758309 HS766T CTRP2 0.0020 66.0000
PF-3758309 KMRC-3 CTRP2 0.0020 66.0000
PF-3758309 M-07E CTRP2 0.0020 66.0000
PF-3758309 NCI-H1651 CTRP2 0.0020 66.0000
PF-3758309 SK-BR-3 CTRP2 0.0020 66.0000
PF-3758309 SNU-1033 CTRP2 0.0020 66.0000
PF-3758309 A-204 CTRP2 0.0020 66.0000
PF-3758309 AML-193 CTRP2 0.0020 66.0000
PF-3758309 HGC-27 CTRP2 0.0020 66.0000
PF-3758309 HS578BST CTRP2 0.0020 66.0000
PF-3758309 MALME-3M CTRP2 0.0020 66.0000
PF-3758309 HS934.T CTRP2 0.0020 66.0000
PF-3758309 HS688(A).T CTRP2 0.0020 66.0000
PF-3758309 HUT78 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1793 CTRP2 0.0020 66.0000
PF-3758309 SCC-4 CTRP2 0.0020 66.0000
PF-3758309 SK-ES-1 CTRP2 0.0020 66.0000
PF-3758309 HS888.T CTRP2 0.0020 66.0000
PF-3758309 MDA-MB-453 CTRP2 0.0020 66.0000
PF-3758309 NCI-H660 CTRP2 0.0020 66.0000
PF-3758309 SAOS-2 CTRP2 0.0020 66.0000
PF-3758309 U-BLC1 CTRP2 0.0020 66.0000
PF-3758309 BT248 CTRP2 0.0020 66.0000
PF-3758309 NCI-H1694 CTRP2 0.0020 66.0000
PF-3758309 SEM CTRP2 0.0020 66.0000
PF-3758309 HS822.T CTRP2 0.0020 66.0000
PF-3758309 HS940.T CTRP2 0.0020 66.0000
PF-3758309 KMBC-2 CTRP2 0.0020 66.0000
PF-3758309 RCC10RGB CTRP2 0.0020 66.0000
PF-3758309 SK-N-BE(2) CTRP2 0.0020 66.0000
PF-3758309 AU565 CTRP2 0.0020 66.0000
PF-3758309 COLO320 CTRP2 0.0020 66.0000
PF-3758309 MDA-MB-415 CTRP2 0.0020 66.0000
PF-3758309 PANC10.05 CTRP2 0.0020 66.0000
PF-3758309 BT131 CTRP2 0.0020 66.0000
PF-3758309 BT147 CTRP2 0.0020 66.0000
PF-3758309 BT172 CTRP2 0.0020 66.0000
PF-3758309 BT216 CTRP2 0.0020 66.0000
PF-3758309 BT232 CTRP2 0.0020 66.0000
PF-3758309 BT245 CTRP2 0.0020 66.0000
PF-3758309 BT271 CTRP2 0.0020 66.0000
PF-3758309 BT286 CTRP2 0.0020 66.0000
PF-3758309 BT320 CTRP2 0.0020 66.0000
PF-3758309 BT328 CTRP2 0.0020 66.0000
PF-3758309 BT330 CTRP2 0.0020 66.0000
PF-3758309 BT333 CTRP2 0.0020 66.0000
PF-3758309 BT340 CTRP2 0.0020 66.0000
PF-3758309 BT359 CTRP2 0.0020 66.0000
PF-3758309 BT416 CTRP2 0.0020 66.0000
PF-3758309 BT422 CTRP2 0.0020 66.0000
PF-3758309 BT440 CTRP2 0.0020 66.0000
PF-3758309 BT444 CTRP2 0.0020 66.0000
PF-3758309 BT482 CTRP2 0.0020 66.0000
PF-3758309 BT498 CTRP2 0.0020 66.0000
PF-3758309 BT504 CTRP2 0.0020 66.0000
PF-3758309 2004 CTRP2 0.0020 66.0000
PF-3758309 ASKA-SS CTRP2 0.0020 66.0000
PF-3758309 BT-12 CTRP2 0.0020 66.0000
PF-3758309 BT-16 CTRP2 0.0020 66.0000
PF-3758309 SW982 CTRP2 0.0020 66.0000
PF-3758309 SYO-1 CTRP2 0.0020 66.0000
PF-3758309 TM87-16 CTRP2 0.0020 66.0000
PF-3758309 TTC-709 CTRP2 0.0020 66.0000
PF-3758309 YAMATO-SS CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.