Drug : Mln2480

CTRP2 Name : MLN2480

Dataset : All
Synonyms :
Targets : ARAF;BRAF;RAF1
Pathways : inhibitor of RAF kinases

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
MLN2480 C2BBE1 CTRP2 0.0020 66.0000
MLN2480 CHAGO-K-1 CTRP2 0.0020 66.0000
MLN2480 COLO668 CTRP2 0.0020 66.0000
MLN2480 COV362 CTRP2 0.0020 66.0000
MLN2480 DV-90 CTRP2 0.0020 66.0000
MLN2480 EFO-27 CTRP2 0.0020 66.0000
MLN2480 HD-MY-Z CTRP2 0.0020 66.0000
MLN2480 NCI-H2170 CTRP2 0.0020 66.0000
MLN2480 NCI-H647 CTRP2 0.0020 66.0000
MLN2480 NCI-H810 CTRP2 0.0020 66.0000
MLN2480 OCI-AML-3 CTRP2 0.0020 66.0000
MLN2480 PATU8988S CTRP2 0.0020 66.0000
MLN2480 MIAPACA-3 CTRP2 0.0020 66.0000
MLN2480 TE-5 CTRP2 0.0020 66.0000
MLN2480 UACC-257 CTRP2 0.0020 66.0000
MLN2480 UACC-62 CTRP2 0.0020 66.0000
MLN2480 BICR6 CTRP2 0.0020 66.0000
MLN2480 BT145 CTRP2 0.0020 66.0000
MLN2480 BT179 CTRP2 0.0020 66.0000
MLN2480 EC-GI-10 CTRP2 0.0020 66.0000
MLN2480 EFO-21 CTRP2 0.0020 66.0000
MLN2480 FTC-133 CTRP2 0.0020 66.0000
MLN2480 JHUEM-3 CTRP2 0.0020 66.0000
MLN2480 LK2 CTRP2 0.0020 66.0000
MLN2480 LNCAPCLONEFGC CTRP2 0.0020 66.0000
MLN2480 LS1034 CTRP2 0.0020 66.0000
MLN2480 MKN7 CTRP2 0.0020 66.0000
MLN2480 HCC1428 CTRP2 0.0020 66.0000
MLN2480 NCI-H2029 CTRP2 0.0020 66.0000
MLN2480 OE21 CTRP2 0.0020 66.0000
MLN2480 MKN74 CTRP2 0.0020 66.0000
MLN2480 SH-10-TC CTRP2 0.0020 66.0000
MLN2480 SNU-449 CTRP2 0.0020 66.0000
MLN2480 T3M-10 CTRP2 0.0020 66.0000
MLN2480 BT112 CTRP2 0.0020 66.0000
MLN2480 BT164 CTRP2 0.0020 66.0000
MLN2480 CCF-STTG1 CTRP2 0.0020 66.0000
MLN2480 COLO800 CTRP2 0.0020 66.0000
MLN2480 DK-MG CTRP2 0.0020 66.0000
MLN2480 GP2D CTRP2 0.0020 66.0000
MLN2480 NCI-H1869 CTRP2 0.0020 66.0000
MLN2480 HCC38 CTRP2 0.0020 66.0000
MLN2480 IA-LM CTRP2 0.0020 66.0000
MLN2480 JHOM-1 CTRP2 0.0020 66.0000
MLN2480 JHUEM-7 CTRP2 0.0020 66.0000
MLN2480 JL-1 CTRP2 0.0020 66.0000
MLN2480 KYSE-450 CTRP2 0.0020 66.0000
MLN2480 LC-1-SQ-SF CTRP2 0.0020 66.0000
MLN2480 RCM-1[HUMANESC] CTRP2 0.0020 66.0000
MLN2480 SNU-685 CTRP2 0.0020 66.0000
MLN2480 VMRC-LCD CTRP2 0.0020 66.0000
MLN2480 BT224 CTRP2 0.0020 66.0000
MLN2480 BT-549 CTRP2 0.0020 66.0000
MLN2480 HELA CTRP2 0.0020 66.0000
MLN2480 HCC202 CTRP2 0.0020 66.0000
MLN2480 H-STS CTRP2 0.0020 66.0000
MLN2480 K029AX CTRP2 0.0020 66.0000
MLN2480 KYSE-520 CTRP2 0.0020 66.0000
MLN2480 LOX-IMVI CTRP2 0.0020 66.0000
MLN2480 NCI-H1623 CTRP2 0.0020 66.0000
MLN2480 NCI-H716 CTRP2 0.0020 66.0000
MLN2480 OE19 CTRP2 0.0020 66.0000
MLN2480 OE33 CTRP2 0.0020 66.0000
MLN2480 N2A-PK1 CTRP2 0.0020 66.0000
MLN2480 PK-45H CTRP2 0.0020 66.0000
MLN2480 P-STS CTRP2 0.0020 66.0000
MLN2480 RERF-LC-AD2 CTRP2 0.0020 66.0000
MLN2480 U-CH1 CTRP2 0.0020 66.0000
MLN2480 697 CTRP2 0.0020 66.0000
MLN2480 A3-KAWAKAMI CTRP2 0.0020 66.0000
MLN2480 BL-41 CTRP2 0.0020 66.0000
MLN2480 CA46 CTRP2 0.0020 66.0000
MLN2480 COR-L51 CTRP2 0.0020 66.0000
MLN2480 DU4475 CTRP2 0.0020 66.0000
MLN2480 EB1 CTRP2 0.0020 66.0000
MLN2480 EOL-1 CTRP2 0.0020 66.0000
MLN2480 GA-10 CTRP2 0.0020 66.0000
MLN2480 MOLT-3 CTRP2 0.0020 66.0000
MLN2480 NAMALWA CTRP2 0.0020 66.0000
MLN2480 OPM-2 CTRP2 0.0020 66.0000
MLN2480 PFEIFFER CTRP2 0.0020 66.0000
MLN2480 SUP-M2 CTRP2 0.0020 66.0000
MLN2480 TOLEDO CTRP2 0.0020 66.0000
MLN2480 COLO829 CTRP2 0.0020 66.0000
MLN2480 DAN-G CTRP2 0.0020 66.0000
MLN2480 EJM CTRP2 0.0020 66.0000
MLN2480 GRANTA-519 CTRP2 0.0020 66.0000
MLN2480 HCC1500 CTRP2 0.0020 66.0000
MLN2480 IGR-1 CTRP2 0.0020 66.0000
MLN2480 NCI-H841 CTRP2 0.0020 66.0000
MLN2480 OCI-LY10 CTRP2 0.0020 66.0000
MLN2480 OCI-LY19 CTRP2 0.0020 66.0000
MLN2480 OCI-LY3 CTRP2 0.0020 66.0000
MLN2480 U-118MG CTRP2 0.0020 66.0000
MLN2480 LU-65 CTRP2 0.0020 66.0000
MLN2480 NCI-H2081 CTRP2 0.0020 66.0000
MLN2480 NCI-H2141 CTRP2 0.0020 66.0000
MLN2480 A-172 CTRP2 0.0020 66.0000
MLN2480 COV644 CTRP2 0.0020 66.0000
MLN2480 IM95 CTRP2 0.0020 66.0000
MLN2480 J82 CTRP2 0.0020 66.0000
MLN2480 NCI-H23 CTRP2 0.0020 66.0000
MLN2480 RD CTRP2 0.0020 66.0000
MLN2480 SK-UT-1 CTRP2 0.0020 66.0000
MLN2480 T98G CTRP2 0.0020 66.0000
MLN2480 BECKER CTRP2 0.0020 66.0000
MLN2480 HS578T CTRP2 0.0020 66.0000
MLN2480 HS611.T CTRP2 0.0020 66.0000
MLN2480 JHH-4 CTRP2 0.0020 66.0000
MLN2480 KARPAS-422 CTRP2 0.0020 66.0000
MLN2480 KMRC-1 CTRP2 0.0020 66.0000
MLN2480 LP-1 CTRP2 0.0020 66.0000
MLN2480 MDA-MB-468 CTRP2 0.0020 66.0000
MLN2480 SH4 CTRP2 0.0020 66.0000
MLN2480 SK-HEP-1 CTRP2 0.0020 66.0000
MLN2480 SUP-HD1 CTRP2 0.0020 66.0000
MLN2480 AN3-CA CTRP2 0.0020 66.0000
MLN2480 ACHN CTRP2 0.0020 66.0000
MLN2480 CMK CTRP2 0.0020 66.0000
MLN2480 EN CTRP2 0.0020 66.0000
MLN2480 KASUMI-1 CTRP2 0.0020 66.0000
MLN2480 NCI-H2342 CTRP2 0.0020 66.0000
MLN2480 OV-90 CTRP2 0.0020 66.0000
MLN2480 RERF-LC-MS CTRP2 0.0020 66.0000
MLN2480 RPMI-6666 CTRP2 0.0020 66.0000
MLN2480 SK-N-MC CTRP2 0.0020 66.0000
MLN2480 A-253 CTRP2 0.0041 33.0000
MLN2480 BC-3C CTRP2 0.0041 33.0000
MLN2480 C32[HUMANMELANOMA] CTRP2 0.0041 33.0000
MLN2480 CAL-85-1 CTRP2 0.0041 33.0000
MLN2480 COLO684 CTRP2 0.0041 33.0000
MLN2480 HS746.T CTRP2 0.0041 33.0000
MLN2480 HSC-2 CTRP2 0.0041 33.0000
MLN2480 HT-144 CTRP2 0.0041 33.0000
MLN2480 VMRC-RCZ CTRP2 0.0041 33.0000
MLN2480 MES-SA CTRP2 0.0041 33.0000
MLN2480 NCI-H1105 CTRP2 0.0041 33.0000
MLN2480 NCI-H322 CTRP2 0.0041 33.0000
MLN2480 OAW42 CTRP2 0.0041 33.0000
MLN2480 PSN1 CTRP2 0.0041 33.0000
MLN2480 T24 CTRP2 0.0041 33.0000
MLN2480 TE441.T CTRP2 0.0041 33.0000
MLN2480 TT2609-C02 CTRP2 0.0041 33.0000
MLN2480 CAKI-1 CTRP2 0.0041 33.0000
MLN2480 COR-L105 CTRP2 0.0041 33.0000
MLN2480 DMS273 CTRP2 0.0041 33.0000
MLN2480 ESS-1 CTRP2 0.0041 33.0000
MLN2480 G-402 CTRP2 0.0041 33.0000
MLN2480 HOS CTRP2 0.0041 33.0000
MLN2480 HS294T CTRP2 0.0041 33.0000
MLN2480 JHH-6 CTRP2 0.0041 33.0000
MLN2480 MFE-319 CTRP2 0.0041 33.0000
MLN2480 MOLP-8 CTRP2 0.0041 33.0000
MLN2480 NCI-H1339 CTRP2 0.0041 33.0000
MLN2480 OV7 CTRP2 0.0041 33.0000
MLN2480 PANC03.27 CTRP2 0.0041 33.0000
MLN2480 PLC-PRF-5 CTRP2 0.0041 33.0000
MLN2480 SCC-9 CTRP2 0.0041 33.0000
MLN2480 SK-LMS-1 CTRP2 0.0041 33.0000
MLN2480 SK-MEL-2 CTRP2 0.0041 33.0000
MLN2480 JHH-2 CTRP2 0.0041 33.0000
MLN2480 A-498 CTRP2 0.0041 33.0000
MLN2480 HLF CTRP2 0.0041 33.0000
MLN2480 JHH-1 CTRP2 0.0041 33.0000
MLN2480 OAW28 CTRP2 0.0041 33.0000
MLN2480 OV56 CTRP2 0.0041 33.0000
MLN2480 PANC02.03 CTRP2 0.0041 33.0000
MLN2480 SNU-475 CTRP2 0.0041 33.0000
MLN2480 TOV-21G CTRP2 0.0041 33.0000
MLN2480 647V CTRP2 0.0041 33.0000
MLN2480 8-MG-BA CTRP2 0.0041 33.0000
MLN2480 A101D CTRP2 0.0041 33.0000
MLN2480 A2058 CTRP2 0.0041 33.0000
MLN2480 ASPC-1 CTRP2 0.0020 66.0000
MLN2480 CAKI-2 CTRP2 0.0041 33.0000
MLN2480 CAL-27 CTRP2 0.0041 33.0000
MLN2480 COLO792 CTRP2 0.0041 33.0000
MLN2480 FTC-238 CTRP2 0.0041 33.0000
MLN2480 GMS-10 CTRP2 0.0041 33.0000
MLN2480 GOS-3 CTRP2 0.0041 33.0000
MLN2480 HMCB CTRP2 0.0041 33.0000
MLN2480 HUH-1 CTRP2 0.0041 33.0000
MLN2480 IST-MES1 CTRP2 0.0041 33.0000
MLN2480 M059K CTRP2 0.0041 33.0000
MLN2480 PATU8988T CTRP2 0.0041 33.0000
MLN2480 SCABER CTRP2 0.0041 33.0000
MLN2480 SK-N-SH CTRP2 0.0041 33.0000
MLN2480 TM-31 CTRP2 0.0041 33.0000
MLN2480 YH-13 CTRP2 0.0041 33.0000
MLN2480 A-673 CTRP2 0.0020 66.0000
MLN2480 DU145 CTRP2 0.0020 66.0000
MLN2480 FADU CTRP2 0.0020 66.0000
MLN2480 HCC4006 CTRP2 0.0020 66.0000
MLN2480 HS683 CTRP2 0.0020 66.0000
MLN2480 HS729.T CTRP2 0.0020 66.0000
MLN2480 HT-1080 CTRP2 0.0020 66.0000
MLN2480 JHH-5 CTRP2 0.0020 66.0000
MLN2480 JHUEM-1 CTRP2 0.0020 66.0000
MLN2480 MEWO CTRP2 0.0020 66.0000
MLN2480 MIAPACA-2 CTRP2 0.0020 66.0000
MLN2480 NCC-STC-K140 CTRP2 0.0020 66.0000
MLN2480 SK-MES-1 CTRP2 0.0020 66.0000
MLN2480 SK-N-DZ CTRP2 0.0020 66.0000
MLN2480 SW579 CTRP2 0.0020 66.0000
MLN2480 WM115 CTRP2 0.0020 66.0000
MLN2480 WM266-4 CTRP2 0.0020 66.0000
MLN2480 BT-20 CTRP2 0.0020 66.0000
MLN2480 CAL-54 CTRP2 0.0020 66.0000
MLN2480 CAPAN-1 CTRP2 0.0020 66.0000
MLN2480 CHP-212 CTRP2 0.0020 66.0000
MLN2480 HS895.T CTRP2 0.0020 66.0000
MLN2480 KATOIII CTRP2 0.0020 66.0000
MLN2480 KMRC-2 CTRP2 0.0020 66.0000
MLN2480 KNS-42 CTRP2 0.0020 66.0000
MLN2480 MPP89 CTRP2 0.0020 66.0000
MLN2480 NCI-H1693 CTRP2 0.0020 66.0000
MLN2480 PANC04.03 CTRP2 0.0020 66.0000
MLN2480 PE-CA-PJ49 CTRP2 0.0020 66.0000
MLN2480 SK-MEL-24 CTRP2 0.0020 66.0000
MLN2480 SK-N-AS CTRP2 0.0020 66.0000
MLN2480 TE617.T CTRP2 0.0020 66.0000
MLN2480 YKG-1 CTRP2 0.0020 66.0000
MLN2480 BL-70 CTRP2 0.0020 66.0000
MLN2480 COR-L95 CTRP2 0.0020 66.0000
MLN2480 D283MED CTRP2 0.0020 66.0000
MLN2480 HL-60 CTRP2 0.0020 66.0000
MLN2480 HUP-T3 CTRP2 0.0020 66.0000
MLN2480 IMR-32 CTRP2 0.0020 66.0000
MLN2480 KO52 CTRP2 0.0020 66.0000
MLN2480 MEC1 CTRP2 0.0020 66.0000
MLN2480 NCI-H1092 CTRP2 0.0020 66.0000
MLN2480 NCI-H2196 CTRP2 0.0020 66.0000
MLN2480 NH-6 CTRP2 0.0020 66.0000
MLN2480 OCI-M1 CTRP2 0.0020 66.0000
MLN2480 SIG-M5 CTRP2 0.0020 66.0000
MLN2480 TF-1 CTRP2 0.0020 66.0000
MLN2480 UACC-812 CTRP2 0.0020 66.0000
MLN2480 786-O CTRP2 0.0020 66.0000
MLN2480 A4-FUKUDA CTRP2 0.0020 66.0000
MLN2480 HCT15 CTRP2 0.0020 66.0000
MLN2480 HEL92.1.7 CTRP2 0.0020 66.0000
MLN2480 HUNS1 CTRP2 0.0020 66.0000
MLN2480 JHOS-2 CTRP2 0.0020 66.0000
MLN2480 K-562 CTRP2 0.0020 66.0000
MLN2480 NCI-H1341 CTRP2 0.0020 66.0000
MLN2480 NCI-H1568 CTRP2 0.0020 66.0000
MLN2480 NCI-H1703 CTRP2 0.0020 66.0000
MLN2480 NCI-H838 CTRP2 0.0020 66.0000
MLN2480 TE-11 CTRP2 0.0020 66.0000
MLN2480 DAUDI CTRP2 0.0020 66.0000
MLN2480 HH[HUMANLYMPHOMA] CTRP2 0.0020 66.0000
MLN2480 HT-1197 CTRP2 0.0020 66.0000
MLN2480 LUDLU-1 CTRP2 0.0020 66.0000
MLN2480 NCI-H146 CTRP2 0.0020 66.0000
MLN2480 NCI-H1915 CTRP2 0.0020 66.0000
MLN2480 NCI-H1944 CTRP2 0.0020 66.0000
MLN2480 NCI-H520 CTRP2 0.0020 66.0000
MLN2480 NCI-H522 CTRP2 0.0020 66.0000
MLN2480 PE-CA-PJ41(CLONED2) CTRP2 0.0020 66.0000
MLN2480 PE-CA-PJ15 CTRP2 0.0020 66.0000
MLN2480 RVH-421 CTRP2 0.0020 66.0000
MLN2480 SET-2 CTRP2 0.0020 66.0000
MLN2480 SNU-16 CTRP2 0.0020 66.0000
MLN2480 TOV-112D CTRP2 0.0020 66.0000
MLN2480 DB CTRP2 0.0020 66.0000
MLN2480 HCC1419 CTRP2 0.0020 66.0000
MLN2480 HCC-56 CTRP2 0.0020 66.0000
MLN2480 HS839.T CTRP2 0.0020 66.0000
MLN2480 NCI-H2110 CTRP2 0.0020 66.0000
MLN2480 PE-CA-PJ34(CLONEC12) CTRP2 0.0020 66.0000
MLN2480 SNU-387 CTRP2 0.0020 66.0000
MLN2480 SNU-503 CTRP2 0.0020 66.0000
MLN2480 SNU-869 CTRP2 0.0020 66.0000
MLN2480 SNU-C1 CTRP2 0.0020 66.0000
MLN2480 SW1990 CTRP2 0.0020 66.0000
MLN2480 SW948 CTRP2 0.0020 66.0000
MLN2480 TE15 CTRP2 0.0020 66.0000
MLN2480 UM-UC-1 CTRP2 0.0020 66.0000
MLN2480 WM88 CTRP2 0.0020 66.0000
MLN2480 WM983B CTRP2 0.0020 66.0000
MLN2480 ZR-75-30 CTRP2 0.0020 66.0000
MLN2480 CI-1 CTRP2 0.0020 66.0000
MLN2480 CJM[HUMANMELANOMA] CTRP2 0.0020 66.0000
MLN2480 HUG1-N CTRP2 0.0020 66.0000
MLN2480 JEKO-1 CTRP2 0.0020 66.0000
MLN2480 JM1 CTRP2 0.0020 66.0000
MLN2480 KP-2 CTRP2 0.0020 66.0000
MLN2480 LMSU CTRP2 0.0020 66.0000
MLN2480 MG-63 CTRP2 0.0020 66.0000
MLN2480 MINO CTRP2 0.0020 66.0000
MLN2480 MJ CTRP2 0.0020 66.0000
MLN2480 MOTN-1 CTRP2 0.0020 66.0000
MLN2480 RL CTRP2 0.0020 66.0000
MLN2480 SK-MEL-3 CTRP2 0.0020 66.0000
MLN2480 SNU-1 CTRP2 0.0020 66.0000
MLN2480 ST486 CTRP2 0.0020 66.0000
MLN2480 SUP-B15 CTRP2 0.0020 66.0000
MLN2480 TC71 CTRP2 0.0020 66.0000
MLN2480 BICR18 CTRP2 0.0020 66.0000
MLN2480 BICR22 CTRP2 0.0020 66.0000
MLN2480 BICR31 CTRP2 0.0020 66.0000
MLN2480 COLO678 CTRP2 0.0020 66.0000
MLN2480 EFM-192A CTRP2 0.0020 66.0000
MLN2480 G-401 CTRP2 0.0020 66.0000
MLN2480 HS888.LU CTRP2 0.0020 66.0000
MLN2480 KP-N-YN CTRP2 0.0020 66.0000
MLN2480 NCI-H1395 CTRP2 0.0020 66.0000
MLN2480 SNU-423 CTRP2 0.0020 66.0000
MLN2480 SW1417 CTRP2 0.0020 66.0000
MLN2480 SW1783 CTRP2 0.0020 66.0000
MLN2480 VCAP CTRP2 0.0020 66.0000
MLN2480 KE-39 CTRP2 0.0020 66.0000
MLN2480 DMS454 CTRP2 0.0020 66.0000
MLN2480 GCT CTRP2 0.0020 66.0000
MLN2480 HCC2935 CTRP2 0.0020 66.0000
MLN2480 HOP-62 CTRP2 0.0020 66.0000
MLN2480 NCI-H747 CTRP2 0.0020 66.0000
MLN2480 OVCAR-5 CTRP2 0.0020 66.0000
MLN2480 SF268 CTRP2 0.0020 66.0000
MLN2480 SF539 CTRP2 0.0020 66.0000
MLN2480 TUHR14TKB CTRP2 0.5200 66.0000
MLN2480 U-251MG CTRP2 0.0020 66.0000
MLN2480 DMS53 CTRP2 0.0020 66.0000
MLN2480 HEC-1-A CTRP2 0.0020 66.0000
MLN2480 IGR-37 CTRP2 0.0020 66.0000
MLN2480 KNS-62 CTRP2 0.0020 66.0000
MLN2480 MDA-MB-157 CTRP2 0.0020 66.0000
MLN2480 NCI-H1563 CTRP2 0.0020 66.0000
MLN2480 OC314 CTRP2 0.0020 66.0000
MLN2480 UO-31 CTRP2 0.0020 66.0000
MLN2480 BICR56 CTRP2 0.0020 66.0000
MLN2480 CAL-33 CTRP2 0.0020 66.0000
MLN2480 CALU-1 CTRP2 0.0020 66.0000
MLN2480 CAPAN-2 CTRP2 0.0020 66.0000
MLN2480 DMS114 CTRP2 0.0020 66.0000
MLN2480 EKVX CTRP2 0.0020 66.0000
MLN2480 HCC1438 CTRP2 0.0020 66.0000
MLN2480 HCT8 CTRP2 0.0020 66.0000
MLN2480 HOP-92 CTRP2 0.0020 66.0000
MLN2480 KYM-1 CTRP2 0.0020 66.0000
MLN2480 KYSE-30 CTRP2 0.0020 66.0000
MLN2480 KYSE-510 CTRP2 0.0020 66.0000
MLN2480 L-428 CTRP2 0.0020 66.0000
MLN2480 MDA-MB-361 CTRP2 0.0020 66.0000
MLN2480 MFE-296 CTRP2 0.0020 66.0000
MLN2480 NU-DHL-1 CTRP2 0.0020 66.0000
MLN2480 SNB-75 CTRP2 0.0020 66.0000
MLN2480 SNU-216 CTRP2 0.0020 66.0000
MLN2480 BICR16 CTRP2 0.0020 66.0000
MLN2480 F-36P CTRP2 0.0020 66.0000
MLN2480 JJN-3 CTRP2 0.0020 66.0000
MLN2480 KASUMI-2 CTRP2 0.0020 66.0000
MLN2480 KG-1-C CTRP2 0.0020 66.0000
MLN2480 KMS-20 CTRP2 0.0020 66.0000
MLN2480 KYSE-150 CTRP2 0.0020 66.0000
MLN2480 OCI-AML-5 CTRP2 0.0020 66.0000
MLN2480 PANC08.13 CTRP2 0.0020 66.0000
MLN2480 SNU-601 CTRP2 0.0020 66.0000
MLN2480 SNU-C4 CTRP2 0.0020 66.0000
MLN2480 T-47D CTRP2 0.0020 66.0000
MLN2480 T84 CTRP2 0.0020 66.0000
MLN2480 TE-14 CTRP2 0.0020 66.0000
MLN2480 U266B1 CTRP2 0.0020 66.0000
MLN2480 42-MG-BA CTRP2 0.0020 66.0000
MLN2480 BT139 CTRP2 0.0020 66.0000
MLN2480 BT159 CTRP2 0.0020 66.0000
MLN2480 BT228 CTRP2 0.0020 66.0000
MLN2480 BT231 CTRP2 0.0020 66.0000
MLN2480 BT239 CTRP2 0.0020 66.0000
MLN2480 BT-474 CTRP2 0.0020 66.0000
MLN2480 COV434 CTRP2 0.0020 66.0000
MLN2480 DND-41 CTRP2 0.0020 66.0000
MLN2480 G-292CLONEA141B1 CTRP2 0.0020 66.0000
MLN2480 HCC2218 CTRP2 0.0020 66.0000
MLN2480 HS766T CTRP2 0.0020 66.0000
MLN2480 KMRC-3 CTRP2 0.0020 66.0000
MLN2480 M-07E CTRP2 0.0020 66.0000
MLN2480 NCI-H1651 CTRP2 0.0020 66.0000
MLN2480 SK-BR-3 CTRP2 0.0020 66.0000
MLN2480 SNU-1033 CTRP2 0.0020 66.0000
MLN2480 A-204 CTRP2 0.0020 66.0000
MLN2480 AML-193 CTRP2 0.0020 66.0000
MLN2480 HGC-27 CTRP2 0.0020 66.0000
MLN2480 HS578BST CTRP2 0.0020 66.0000
MLN2480 MALME-3M CTRP2 0.0020 66.0000
MLN2480 HS934.T CTRP2 0.0020 66.0000
MLN2480 HS688(A).T CTRP2 0.0020 66.0000
MLN2480 HUT78 CTRP2 0.0020 66.0000
MLN2480 NCI-H1793 CTRP2 0.0020 66.0000
MLN2480 SCC-4 CTRP2 0.0020 66.0000
MLN2480 SK-ES-1 CTRP2 0.0020 66.0000
MLN2480 HS888.T CTRP2 0.0020 66.0000
MLN2480 MDA-MB-453 CTRP2 0.0020 66.0000
MLN2480 NCI-H660 CTRP2 0.0020 66.0000
MLN2480 SAOS-2 CTRP2 0.0020 66.0000
MLN2480 U-BLC1 CTRP2 0.0020 66.0000
MLN2480 BT248 CTRP2 0.0020 66.0000
MLN2480 NCI-H1694 CTRP2 0.0020 66.0000
MLN2480 SEM CTRP2 0.0020 66.0000
MLN2480 HS822.T CTRP2 0.0020 66.0000
MLN2480 HS940.T CTRP2 0.0020 66.0000
MLN2480 KMBC-2 CTRP2 0.0020 66.0000
MLN2480 RCC10RGB CTRP2 0.0020 66.0000
MLN2480 SK-N-BE(2) CTRP2 0.0020 66.0000
MLN2480 AU565 CTRP2 0.0020 66.0000
MLN2480 COLO320 CTRP2 0.0020 66.0000
MLN2480 MDA-MB-415 CTRP2 0.0020 66.0000
MLN2480 PANC10.05 CTRP2 0.0020 66.0000
MLN2480 BT131 CTRP2 0.0020 66.0000
MLN2480 BT147 CTRP2 0.0020 66.0000
MLN2480 BT172 CTRP2 0.0020 66.0000
MLN2480 BT216 CTRP2 0.0020 66.0000
MLN2480 BT232 CTRP2 0.0020 66.0000
MLN2480 BT245 CTRP2 0.0020 66.0000
MLN2480 BT271 CTRP2 0.0020 66.0000
MLN2480 BT286 CTRP2 0.0020 66.0000
MLN2480 BT320 CTRP2 0.0020 66.0000
MLN2480 BT328 CTRP2 0.0020 66.0000
MLN2480 BT330 CTRP2 0.0020 66.0000
MLN2480 BT333 CTRP2 0.0020 66.0000
MLN2480 BT340 CTRP2 0.0020 66.0000
MLN2480 BT359 CTRP2 0.0020 66.0000
MLN2480 BT416 CTRP2 0.0020 66.0000
MLN2480 BT422 CTRP2 0.0020 66.0000
MLN2480 BT428 CTRP2 0.0020 66.0000
MLN2480 BT440 CTRP2 0.0020 66.0000
MLN2480 BT444 CTRP2 0.0020 66.0000
MLN2480 BT482 CTRP2 0.0020 66.0000
MLN2480 BT498 CTRP2 0.0020 66.0000
MLN2480 BT504 CTRP2 0.0020 66.0000
MLN2480 2004 CTRP2 0.0020 66.0000
MLN2480 ASKA-SS CTRP2 0.0020 66.0000
MLN2480 BT-12 CTRP2 0.0020 66.0000
MLN2480 BT-16 CTRP2 0.0020 66.0000
MLN2480 SW982 CTRP2 0.0020 66.0000
MLN2480 SYO-1 CTRP2 0.0020 66.0000
MLN2480 TM87-16 CTRP2 0.0020 66.0000
MLN2480 TTC-709 CTRP2 0.0020 66.0000
MLN2480 YAMATO-SS CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.