Drug : Istradefylline

CTRP2 Name : istradefylline

Dataset : All
Synonyms :
Targets : ADORA2A
Pathways : antagonist of the adenosine A2A receptor

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

:


Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
istradefylline C2BBE1 CTRP2 0.0010 33.0000
istradefylline CHAGO-K-1 CTRP2 0.0010 33.0000
istradefylline COLO668 CTRP2 0.0010 33.0000
istradefylline COV362 CTRP2 0.0010 33.0000
istradefylline DV-90 CTRP2 0.0010 33.0000
istradefylline EFO-27 CTRP2 0.0010 33.0000
istradefylline HD-MY-Z CTRP2 0.0010 33.0000
istradefylline NCI-H2170 CTRP2 0.0010 33.0000
istradefylline NCI-H647 CTRP2 0.0010 33.0000
istradefylline NCI-H810 CTRP2 0.0010 33.0000
istradefylline OCI-AML-3 CTRP2 0.0010 33.0000
istradefylline PATU8988S CTRP2 0.0010 33.0000
istradefylline MIAPACA-3 CTRP2 0.0010 33.0000
istradefylline TE-5 CTRP2 0.0010 33.0000
istradefylline UACC-257 CTRP2 0.0010 33.0000
istradefylline UACC-62 CTRP2 0.0010 33.0000
istradefylline BICR6 CTRP2 0.0010 33.0000
istradefylline BT145 CTRP2 0.0010 33.0000
istradefylline BT179 CTRP2 0.0010 33.0000
istradefylline EC-GI-10 CTRP2 0.0010 33.0000
istradefylline EFO-21 CTRP2 0.0010 33.0000
istradefylline FTC-133 CTRP2 0.0010 33.0000
istradefylline JHUEM-3 CTRP2 0.0010 33.0000
istradefylline LK2 CTRP2 0.0010 33.0000
istradefylline LNCAPCLONEFGC CTRP2 0.0010 33.0000
istradefylline LS1034 CTRP2 0.0010 33.0000
istradefylline MKN7 CTRP2 0.0010 33.0000
istradefylline HCC1428 CTRP2 0.0010 33.0000
istradefylline NCI-H2029 CTRP2 0.0010 33.0000
istradefylline OE21 CTRP2 0.0010 33.0000
istradefylline MKN74 CTRP2 0.0010 33.0000
istradefylline SH-10-TC CTRP2 0.0010 33.0000
istradefylline SNU-449 CTRP2 0.0010 33.0000
istradefylline T3M-10 CTRP2 0.0010 33.0000
istradefylline BT112 CTRP2 0.0010 33.0000
istradefylline BT164 CTRP2 0.0010 33.0000
istradefylline CCF-STTG1 CTRP2 0.0010 33.0000
istradefylline COLO800 CTRP2 0.0010 33.0000
istradefylline DK-MG CTRP2 0.0010 33.0000
istradefylline GP2D CTRP2 0.0010 33.0000
istradefylline NCI-H1869 CTRP2 0.0010 33.0000
istradefylline HCC38 CTRP2 0.0010 33.0000
istradefylline IA-LM CTRP2 0.0010 33.0000
istradefylline JHOM-1 CTRP2 0.0010 33.0000
istradefylline JHUEM-7 CTRP2 0.0010 33.0000
istradefylline JL-1 CTRP2 0.0010 33.0000
istradefylline KYSE-450 CTRP2 0.0010 33.0000
istradefylline LC-1-SQ-SF CTRP2 0.0010 33.0000
istradefylline RCM-1[HUMANESC] CTRP2 0.0010 33.0000
istradefylline SNU-685 CTRP2 0.0010 33.0000
istradefylline VMRC-LCD CTRP2 0.0010 33.0000
istradefylline BT224 CTRP2 0.0010 33.0000
istradefylline BT-549 CTRP2 0.0010 33.0000
istradefylline HELA CTRP2 0.0010 33.0000
istradefylline HCC202 CTRP2 0.0010 33.0000
istradefylline H-STS CTRP2 0.0010 33.0000
istradefylline K029AX CTRP2 0.0010 33.0000
istradefylline KYSE-520 CTRP2 0.0010 33.0000
istradefylline LOX-IMVI CTRP2 0.0010 33.0000
istradefylline NCI-H1623 CTRP2 0.0010 33.0000
istradefylline NCI-H716 CTRP2 0.0010 33.0000
istradefylline OE19 CTRP2 0.0010 33.0000
istradefylline OE33 CTRP2 0.0010 33.0000
istradefylline N2A-PK1 CTRP2 0.0010 33.0000
istradefylline PK-45H CTRP2 0.0010 33.0000
istradefylline P-STS CTRP2 0.0010 33.0000
istradefylline RERF-LC-AD2 CTRP2 0.0010 33.0000
istradefylline U-CH1 CTRP2 0.0010 33.0000
istradefylline 697 CTRP2 0.0010 33.0000
istradefylline A3-KAWAKAMI CTRP2 0.0010 33.0000
istradefylline CA46 CTRP2 0.0010 33.0000
istradefylline COR-L51 CTRP2 0.0010 33.0000
istradefylline DU4475 CTRP2 0.0010 33.0000
istradefylline EB1 CTRP2 0.0010 33.0000
istradefylline EOL-1 CTRP2 0.0010 33.0000
istradefylline GA-10 CTRP2 0.0010 33.0000
istradefylline MOLT-3 CTRP2 0.0010 33.0000
istradefylline NAMALWA CTRP2 0.0010 33.0000
istradefylline OPM-2 CTRP2 0.0010 33.0000
istradefylline PFEIFFER CTRP2 0.0010 33.0000
istradefylline SUP-M2 CTRP2 0.0010 33.0000
istradefylline TOLEDO CTRP2 0.0010 33.0000
istradefylline COLO829 CTRP2 0.0010 33.0000
istradefylline DAN-G CTRP2 0.0010 33.0000
istradefylline EJM CTRP2 0.0010 33.0000
istradefylline GRANTA-519 CTRP2 0.0010 33.0000
istradefylline HCC1500 CTRP2 0.0010 33.0000
istradefylline IGR-1 CTRP2 0.0010 33.0000
istradefylline NCI-H841 CTRP2 0.0010 33.0000
istradefylline OCI-LY10 CTRP2 0.0010 33.0000
istradefylline OCI-LY19 CTRP2 0.0010 33.0000
istradefylline OCI-LY3 CTRP2 0.0010 33.0000
istradefylline U-118MG CTRP2 0.0010 33.0000
istradefylline COR-L88 CTRP2 0.0010 33.0000
istradefylline LU-65 CTRP2 0.0010 33.0000
istradefylline NCI-H2081 CTRP2 0.0010 33.0000
istradefylline NCI-H2141 CTRP2 0.0010 33.0000
istradefylline A-172 CTRP2 0.0010 33.0000
istradefylline COV644 CTRP2 0.0010 33.0000
istradefylline IM95 CTRP2 0.0010 33.0000
istradefylline J82 CTRP2 0.0010 33.0000
istradefylline RD CTRP2 0.0010 33.0000
istradefylline SK-UT-1 CTRP2 0.0010 33.0000
istradefylline T98G CTRP2 0.0010 33.0000
istradefylline BECKER CTRP2 0.0010 33.0000
istradefylline HS578T CTRP2 0.0010 33.0000
istradefylline JHH-4 CTRP2 0.0010 33.0000
istradefylline KARPAS-422 CTRP2 0.0010 33.0000
istradefylline KMRC-1 CTRP2 0.0010 33.0000
istradefylline LP-1 CTRP2 0.0010 33.0000
istradefylline MDA-MB-468 CTRP2 0.0010 33.0000
istradefylline SH4 CTRP2 0.0010 33.0000
istradefylline SK-HEP-1 CTRP2 0.0010 33.0000
istradefylline SUP-HD1 CTRP2 0.0010 33.0000
istradefylline AN3-CA CTRP2 0.0010 33.0000
istradefylline ACHN CTRP2 0.0010 33.0000
istradefylline CMK CTRP2 0.0010 33.0000
istradefylline EN CTRP2 0.0010 33.0000
istradefylline KASUMI-1 CTRP2 0.0010 33.0000
istradefylline NCI-H2342 CTRP2 0.0010 33.0000
istradefylline OV-90 CTRP2 0.0010 33.0000
istradefylline RERF-LC-MS CTRP2 0.0010 33.0000
istradefylline RPMI-6666 CTRP2 0.0010 33.0000
istradefylline SK-N-MC CTRP2 0.0010 33.0000
istradefylline A-253 CTRP2 0.0010 33.0000
istradefylline BC-3C CTRP2 0.0010 33.0000
istradefylline C32[HUMANMELANOMA] CTRP2 0.0010 33.0000
istradefylline CAL-85-1 CTRP2 0.0010 33.0000
istradefylline COLO684 CTRP2 0.0010 33.0000
istradefylline HS746.T CTRP2 0.0010 33.0000
istradefylline HSC-2 CTRP2 0.0010 33.0000
istradefylline HT-144 CTRP2 0.0010 33.0000
istradefylline VMRC-RCZ CTRP2 0.0010 33.0000
istradefylline MES-SA CTRP2 0.0010 33.0000
istradefylline NCI-H1105 CTRP2 0.0010 33.0000
istradefylline NCI-H322 CTRP2 0.0010 33.0000
istradefylline OAW42 CTRP2 0.0010 33.0000
istradefylline PSN1 CTRP2 0.0010 33.0000
istradefylline T24 CTRP2 0.0010 33.0000
istradefylline TE441.T CTRP2 0.0010 33.0000
istradefylline TT2609-C02 CTRP2 0.0010 33.0000
istradefylline CAKI-1 CTRP2 0.0010 33.0000
istradefylline COR-L105 CTRP2 0.0010 33.0000
istradefylline DMS273 CTRP2 0.0010 33.0000
istradefylline ESS-1 CTRP2 0.0010 33.0000
istradefylline G-402 CTRP2 0.0010 33.0000
istradefylline HS294T CTRP2 0.0010 33.0000
istradefylline JHH-6 CTRP2 0.0010 33.0000
istradefylline MFE-319 CTRP2 0.0010 33.0000
istradefylline NCI-H1339 CTRP2 0.0010 33.0000
istradefylline PLC-PRF-5 CTRP2 0.0010 33.0000
istradefylline SCC-9 CTRP2 0.0010 33.0000
istradefylline SK-LMS-1 CTRP2 0.0010 33.0000
istradefylline SK-MEL-2 CTRP2 0.0010 33.0000
istradefylline JHH-2 CTRP2 0.0010 33.0000
istradefylline A-498 CTRP2 0.0010 33.0000
istradefylline HLF CTRP2 0.0010 33.0000
istradefylline JHH-1 CTRP2 0.0010 33.0000
istradefylline OAW28 CTRP2 0.0010 33.0000
istradefylline OV56 CTRP2 0.0010 33.0000
istradefylline PANC02.03 CTRP2 0.0010 33.0000
istradefylline SNU-475 CTRP2 0.0010 33.0000
istradefylline TOV-21G CTRP2 0.0010 33.0000
istradefylline 647V CTRP2 0.0010 33.0000
istradefylline 8-MG-BA CTRP2 0.0010 33.0000
istradefylline A101D CTRP2 0.0010 33.0000
istradefylline A2058 CTRP2 0.0010 33.0000
istradefylline ASPC-1 CTRP2 0.0010 33.0000
istradefylline CAKI-2 CTRP2 0.0010 33.0000
istradefylline CAL-27 CTRP2 0.0010 33.0000
istradefylline COLO792 CTRP2 0.0010 33.0000
istradefylline FTC-238 CTRP2 0.0010 33.0000
istradefylline GMS-10 CTRP2 0.0010 33.0000
istradefylline GOS-3 CTRP2 0.0010 33.0000
istradefylline HMCB CTRP2 0.0010 33.0000
istradefylline HUH-1 CTRP2 0.0010 33.0000
istradefylline IGR-39 CTRP2 0.0010 33.0000
istradefylline IST-MES1 CTRP2 0.0010 33.0000
istradefylline M059K CTRP2 0.0010 33.0000
istradefylline PATU8988T CTRP2 0.0010 33.0000
istradefylline SCABER CTRP2 0.0010 33.0000
istradefylline SK-N-SH CTRP2 0.0010 33.0000
istradefylline TM-31 CTRP2 0.0010 33.0000
istradefylline YH-13 CTRP2 0.0010 33.0000
istradefylline A-673 CTRP2 0.0010 33.0000
istradefylline DU145 CTRP2 0.0010 33.0000
istradefylline FADU CTRP2 0.0010 33.0000
istradefylline HCC4006 CTRP2 0.0010 33.0000
istradefylline HS683 CTRP2 0.0010 33.0000
istradefylline HS729.T CTRP2 0.0010 33.0000
istradefylline HT-1080 CTRP2 0.0010 33.0000
istradefylline JHH-5 CTRP2 0.0010 33.0000
istradefylline JHUEM-1 CTRP2 0.0010 33.0000
istradefylline MEWO CTRP2 0.0010 33.0000
istradefylline MIAPACA-2 CTRP2 0.0010 33.0000
istradefylline NCC-STC-K140 CTRP2 0.2600 33.0000
istradefylline SK-MES-1 CTRP2 0.0010 33.0000
istradefylline SK-N-DZ CTRP2 0.0010 33.0000
istradefylline SW579 CTRP2 0.0010 33.0000
istradefylline WM115 CTRP2 0.0010 33.0000
istradefylline WM266-4 CTRP2 0.0010 33.0000
istradefylline BT-20 CTRP2 0.0010 33.0000
istradefylline CAL-54 CTRP2 0.0010 33.0000
istradefylline CAPAN-1 CTRP2 0.0010 33.0000
istradefylline CHP-212 CTRP2 0.0010 33.0000
istradefylline HS895.T CTRP2 0.0010 33.0000
istradefylline KATOIII CTRP2 0.0010 33.0000
istradefylline KMRC-2 CTRP2 0.0010 33.0000
istradefylline KNS-42 CTRP2 0.0010 33.0000
istradefylline MPP89 CTRP2 0.0010 33.0000
istradefylline NCI-H1693 CTRP2 0.0010 33.0000
istradefylline PANC04.03 CTRP2 0.0010 33.0000
istradefylline PE-CA-PJ49 CTRP2 0.0010 33.0000
istradefylline SK-MEL-24 CTRP2 0.0010 33.0000
istradefylline SK-N-AS CTRP2 0.0010 33.0000
istradefylline TE617.T CTRP2 0.0010 33.0000
istradefylline YKG-1 CTRP2 0.0010 33.0000
istradefylline BL-70 CTRP2 0.0010 33.0000
istradefylline COR-L95 CTRP2 0.0010 33.0000
istradefylline D283MED CTRP2 0.0010 33.0000
istradefylline HL-60 CTRP2 0.0010 33.0000
istradefylline HUP-T3 CTRP2 0.0010 33.0000
istradefylline KO52 CTRP2 0.0010 33.0000
istradefylline MEC1 CTRP2 0.0010 33.0000
istradefylline NCI-H1092 CTRP2 0.0010 33.0000
istradefylline NCI-H2196 CTRP2 0.0010 33.0000
istradefylline NH-6 CTRP2 0.0010 33.0000
istradefylline OCI-M1 CTRP2 0.0010 33.0000
istradefylline SIG-M5 CTRP2 0.0010 33.0000
istradefylline TF-1 CTRP2 0.0010 33.0000
istradefylline UACC-812 CTRP2 0.0010 33.0000
istradefylline 786-O CTRP2 0.0010 33.0000
istradefylline A4-FUKUDA CTRP2 0.0010 33.0000
istradefylline HCT15 CTRP2 0.0010 33.0000
istradefylline HEL92.1.7 CTRP2 0.0010 33.0000
istradefylline JHOS-2 CTRP2 0.0010 33.0000
istradefylline K-562 CTRP2 0.0010 33.0000
istradefylline NCI-H1341 CTRP2 0.0010 33.0000
istradefylline NCI-H1568 CTRP2 0.0010 33.0000
istradefylline NCI-H1703 CTRP2 0.0010 33.0000
istradefylline NCI-H838 CTRP2 0.0010 33.0000
istradefylline TE-11 CTRP2 0.0010 33.0000
istradefylline DAUDI CTRP2 0.0010 33.0000
istradefylline HH[HUMANLYMPHOMA] CTRP2 0.0010 33.0000
istradefylline HT-1197 CTRP2 0.0010 33.0000
istradefylline LUDLU-1 CTRP2 0.0010 33.0000
istradefylline NCI-H146 CTRP2 0.0010 33.0000
istradefylline NCI-H1915 CTRP2 0.0010 33.0000
istradefylline NCI-H1944 CTRP2 0.0010 33.0000
istradefylline NCI-H520 CTRP2 0.0010 33.0000
istradefylline NCI-H522 CTRP2 0.0010 33.0000
istradefylline PE-CA-PJ41(CLONED2) CTRP2 0.0010 33.0000
istradefylline PE-CA-PJ15 CTRP2 0.0010 33.0000
istradefylline RVH-421 CTRP2 0.0010 33.0000
istradefylline SET-2 CTRP2 0.0010 33.0000
istradefylline SNU-16 CTRP2 0.0010 33.0000
istradefylline TOV-112D CTRP2 0.0010 33.0000
istradefylline DB CTRP2 0.0010 33.0000
istradefylline HCC1419 CTRP2 0.0010 33.0000
istradefylline HCC-56 CTRP2 0.0010 33.0000
istradefylline HS839.T CTRP2 0.0010 33.0000
istradefylline NCI-H2110 CTRP2 0.0010 33.0000
istradefylline PE-CA-PJ34(CLONEC12) CTRP2 0.0010 33.0000
istradefylline SNU-387 CTRP2 0.0010 33.0000
istradefylline SNU-503 CTRP2 0.0010 33.0000
istradefylline SNU-869 CTRP2 0.0010 33.0000
istradefylline SNU-C1 CTRP2 0.0010 33.0000
istradefylline SW1990 CTRP2 0.0010 33.0000
istradefylline SW948 CTRP2 0.0010 33.0000
istradefylline TE15 CTRP2 0.0010 33.0000
istradefylline UM-UC-1 CTRP2 0.0010 33.0000
istradefylline WM88 CTRP2 0.0010 33.0000
istradefylline WM983B CTRP2 0.0010 33.0000
istradefylline ZR-75-30 CTRP2 0.0010 33.0000
istradefylline CI-1 CTRP2 0.0010 33.0000
istradefylline CJM[HUMANMELANOMA] CTRP2 0.0010 33.0000
istradefylline HUG1-N CTRP2 0.0010 33.0000
istradefylline JEKO-1 CTRP2 0.0010 33.0000
istradefylline JM1 CTRP2 0.0010 33.0000
istradefylline KP-2 CTRP2 0.0010 33.0000
istradefylline LMSU CTRP2 0.0010 33.0000
istradefylline MG-63 CTRP2 0.0010 33.0000
istradefylline MINO CTRP2 0.0010 33.0000
istradefylline MOTN-1 CTRP2 0.0010 33.0000
istradefylline RL CTRP2 0.0010 33.0000
istradefylline SK-MEL-3 CTRP2 0.0010 33.0000
istradefylline SNU-1 CTRP2 0.0010 33.0000
istradefylline ST486 CTRP2 0.0010 33.0000
istradefylline SUP-B15 CTRP2 0.0010 33.0000
istradefylline TC71 CTRP2 0.0010 33.0000
istradefylline BICR18 CTRP2 0.0010 33.0000
istradefylline BICR22 CTRP2 0.0010 33.0000
istradefylline BICR31 CTRP2 0.0010 33.0000
istradefylline COLO678 CTRP2 0.0010 33.0000
istradefylline EFM-192A CTRP2 0.0010 33.0000
istradefylline G-401 CTRP2 0.0010 33.0000
istradefylline HS888.LU CTRP2 0.0010 33.0000
istradefylline KP-N-YN CTRP2 0.0010 33.0000
istradefylline NCI-H1395 CTRP2 0.0010 33.0000
istradefylline SNU-423 CTRP2 0.0010 33.0000
istradefylline SW1417 CTRP2 0.0010 33.0000
istradefylline SW1783 CTRP2 0.0010 33.0000
istradefylline VCAP CTRP2 0.0010 33.0000
istradefylline KE-39 CTRP2 0.0010 33.0000
istradefylline DMS454 CTRP2 0.0010 33.0000
istradefylline GCT CTRP2 0.0010 33.0000
istradefylline HCC2935 CTRP2 0.0010 33.0000
istradefylline HOP-62 CTRP2 0.0010 33.0000
istradefylline NCI-H747 CTRP2 0.0010 33.0000
istradefylline OVCAR-5 CTRP2 0.0010 33.0000
istradefylline SF268 CTRP2 0.0010 33.0000
istradefylline SF539 CTRP2 0.0010 33.0000
istradefylline TUHR14TKB CTRP2 0.0010 33.0000
istradefylline U-251MG CTRP2 0.0010 33.0000
istradefylline DMS53 CTRP2 0.0010 33.0000
istradefylline HEC-1-A CTRP2 0.0010 33.0000
istradefylline IGR-37 CTRP2 0.0010 33.0000
istradefylline KNS-62 CTRP2 0.0010 33.0000
istradefylline MDA-MB-157 CTRP2 0.0010 33.0000
istradefylline NCI-H1563 CTRP2 0.0010 33.0000
istradefylline OC314 CTRP2 0.0010 33.0000
istradefylline UO-31 CTRP2 0.0010 33.0000
istradefylline BICR56 CTRP2 0.0010 33.0000
istradefylline CAL-33 CTRP2 0.0010 33.0000
istradefylline CALU-1 CTRP2 0.0010 33.0000
istradefylline CAPAN-2 CTRP2 0.0010 33.0000
istradefylline DMS114 CTRP2 0.0010 33.0000
istradefylline EKVX CTRP2 0.0010 33.0000
istradefylline HCC1438 CTRP2 0.0010 33.0000
istradefylline HCT8 CTRP2 0.0010 33.0000
istradefylline HOP-92 CTRP2 0.0010 33.0000
istradefylline KYM-1 CTRP2 0.0010 33.0000
istradefylline KYSE-30 CTRP2 0.0010 33.0000
istradefylline KYSE-510 CTRP2 0.0010 33.0000
istradefylline L-428 CTRP2 0.0010 33.0000
istradefylline MDA-MB-361 CTRP2 0.0010 33.0000
istradefylline MFE-296 CTRP2 0.0010 33.0000
istradefylline NU-DHL-1 CTRP2 0.0010 33.0000
istradefylline SNB-75 CTRP2 0.0010 33.0000
istradefylline SNU-216 CTRP2 0.0010 33.0000
istradefylline BICR16 CTRP2 0.0010 33.0000
istradefylline F-36P CTRP2 0.0010 33.0000
istradefylline JJN-3 CTRP2 0.0010 33.0000
istradefylline KASUMI-2 CTRP2 0.0010 33.0000
istradefylline KG-1-C CTRP2 0.0010 33.0000
istradefylline KMS-20 CTRP2 0.0010 33.0000
istradefylline KYSE-150 CTRP2 0.0010 33.0000
istradefylline OCI-AML-5 CTRP2 0.0010 33.0000
istradefylline PANC08.13 CTRP2 0.0010 33.0000
istradefylline SNU-601 CTRP2 0.0010 33.0000
istradefylline SNU-C4 CTRP2 0.0010 33.0000
istradefylline T-47D CTRP2 0.0010 33.0000
istradefylline T84 CTRP2 0.0010 33.0000
istradefylline TE-14 CTRP2 0.0010 33.0000
istradefylline U266B1 CTRP2 0.0010 33.0000
istradefylline 42-MG-BA CTRP2 0.0010 33.0000
istradefylline BT139 CTRP2 0.0010 33.0000
istradefylline BT159 CTRP2 0.0010 33.0000
istradefylline BT228 CTRP2 0.0010 33.0000
istradefylline BT231 CTRP2 0.0010 33.0000
istradefylline BT239 CTRP2 0.0010 33.0000
istradefylline BT-474 CTRP2 0.0010 33.0000
istradefylline COV434 CTRP2 0.0010 33.0000
istradefylline DND-41 CTRP2 0.0010 33.0000
istradefylline G-292CLONEA141B1 CTRP2 0.0010 33.0000
istradefylline HCC2218 CTRP2 0.0010 33.0000
istradefylline HS766T CTRP2 0.0010 33.0000
istradefylline KMRC-3 CTRP2 0.0010 33.0000
istradefylline M-07E CTRP2 0.0010 33.0000
istradefylline NCI-H1651 CTRP2 0.0010 33.0000
istradefylline SK-BR-3 CTRP2 0.0010 33.0000
istradefylline SNU-1033 CTRP2 0.0010 33.0000
istradefylline A-204 CTRP2 0.0010 33.0000
istradefylline AML-193 CTRP2 0.0010 33.0000
istradefylline HGC-27 CTRP2 0.0010 33.0000
istradefylline HS578BST CTRP2 0.0010 33.0000
istradefylline HS934.T CTRP2 0.0010 33.0000
istradefylline HS688(A).T CTRP2 0.0010 33.0000
istradefylline HUT78 CTRP2 0.0010 33.0000
istradefylline NCI-H1793 CTRP2 0.0010 33.0000
istradefylline SCC-4 CTRP2 0.0010 33.0000
istradefylline SK-ES-1 CTRP2 0.0010 33.0000
istradefylline HS888.T CTRP2 0.0010 33.0000
istradefylline MDA-MB-453 CTRP2 0.0010 33.0000
istradefylline NCI-H660 CTRP2 0.0010 33.0000
istradefylline SAOS-2 CTRP2 0.0010 33.0000
istradefylline U-BLC1 CTRP2 0.0010 33.0000
istradefylline BT248 CTRP2 0.0010 33.0000
istradefylline NCI-H1694 CTRP2 0.0010 33.0000
istradefylline SEM CTRP2 0.0010 33.0000
istradefylline HS822.T CTRP2 0.0010 33.0000
istradefylline HS940.T CTRP2 0.0010 33.0000
istradefylline KMBC-2 CTRP2 0.0010 33.0000
istradefylline RCC10RGB CTRP2 0.0010 33.0000
istradefylline SK-N-BE(2) CTRP2 0.0010 33.0000
istradefylline AU565 CTRP2 0.0010 33.0000
istradefylline COLO320 CTRP2 0.0010 33.0000
istradefylline MDA-MB-415 CTRP2 0.0010 33.0000
istradefylline PANC10.05 CTRP2 0.0010 33.0000
istradefylline BT131 CTRP2 0.0010 33.0000
istradefylline BT147 CTRP2 0.0010 33.0000
istradefylline BT172 CTRP2 0.0010 33.0000
istradefylline BT216 CTRP2 0.0010 33.0000
istradefylline BT232 CTRP2 0.0010 33.0000
istradefylline BT245 CTRP2 0.0010 33.0000
istradefylline BT271 CTRP2 0.0010 33.0000
istradefylline BT286 CTRP2 0.0010 33.0000
istradefylline BT320 CTRP2 0.0010 33.0000
istradefylline BT328 CTRP2 0.0010 33.0000
istradefylline BT330 CTRP2 0.0010 33.0000
istradefylline BT333 CTRP2 0.0010 33.0000
istradefylline BT340 CTRP2 0.0010 33.0000
istradefylline BT359 CTRP2 0.0010 33.0000
istradefylline BT416 CTRP2 0.0010 33.0000
istradefylline BT422 CTRP2 0.0010 33.0000
istradefylline BT440 CTRP2 0.0010 33.0000
istradefylline BT444 CTRP2 0.0010 33.0000
istradefylline BT482 CTRP2 0.0010 33.0000
istradefylline BT498 CTRP2 0.0010 33.0000
istradefylline BT504 CTRP2 0.0010 33.0000
istradefylline 2004 CTRP2 0.0010 33.0000
istradefylline ASKA-SS CTRP2 0.0010 33.0000
istradefylline BT-12 CTRP2 0.0010 33.0000
istradefylline BT-16 CTRP2 0.0010 33.0000
istradefylline SW982 CTRP2 0.0010 33.0000
istradefylline SYO-1 CTRP2 0.0010 33.0000
istradefylline TM87-16 CTRP2 0.0010 33.0000
istradefylline TTC-709 CTRP2 0.0010 33.0000
istradefylline YAMATO-SS CTRP2 0.0010 33.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.