Drug : Pf-4800567 Hydrochloride

CTRP2 Name : PF-4800567 hydrochloride

Dataset : All
Synonyms :
Targets : CSNK1D;CSNK1E
Pathways : inhibitor of casein kinase isoforms delta and epsilon

Information Cards

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Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
PF-4800567 hydrochloride C2BBE1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CHAGO-K-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COLO668 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COV362 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DV-90 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EFO-27 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HD-MY-Z CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H2170 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H647 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H810 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OCI-AML-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PATU8988S CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MIAPACA-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TE-5 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride UACC-257 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride UACC-62 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BICR6 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT145 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT179 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EC-GI-10 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EFO-21 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride FTC-133 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHUEM-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LK2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LNCAPCLONEFGC CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LS1034 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MKN7 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC1428 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H2029 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OE21 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MKN74 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SH-10-TC CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-449 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride T3M-10 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT112 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT164 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CCF-STTG1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COLO800 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DK-MG CTRP2 0.0020 66.0000
PF-4800567 hydrochloride GP2D CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1869 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC38 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride IA-LM CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHOM-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHUEM-7 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JL-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KYSE-450 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LC-1-SQ-SF CTRP2 0.0020 66.0000
PF-4800567 hydrochloride RCM-1[HUMANESC] CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-685 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride VMRC-LCD CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT224 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT-549 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HELA CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC202 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride H-STS CTRP2 0.0020 66.0000
PF-4800567 hydrochloride K029AX CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KYSE-520 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LOX-IMVI CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1623 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H716 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OE19 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OE33 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride N2A-PK1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PK-45H CTRP2 0.0020 66.0000
PF-4800567 hydrochloride P-STS CTRP2 0.0020 66.0000
PF-4800567 hydrochloride RERF-LC-AD2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride U-CH1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride 697 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride A3-KAWAKAMI CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CA46 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COR-L51 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DU4475 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EB1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EOL-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride GA-10 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MOLT-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NAMALWA CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OPM-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PFEIFFER CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SUP-M2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TOLEDO CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COLO829 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DAN-G CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EJM CTRP2 0.0020 66.0000
PF-4800567 hydrochloride GRANTA-519 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC1500 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride IGR-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H841 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OCI-LY19 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OCI-LY3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride U-118MG CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LU-65 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H2081 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride A-172 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COV644 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride IM95 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride J82 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H23 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride RD CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-UT-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride T98G CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BECKER CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS578T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS611.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHH-4 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KARPAS-422 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KMRC-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LP-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MDA-MB-468 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SH4 CTRP2 0.1300 66.0000
PF-4800567 hydrochloride SK-HEP-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SUP-HD1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride AN3-CA CTRP2 0.0020 66.0000
PF-4800567 hydrochloride ACHN CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CMK CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EN CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KASUMI-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H2342 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OV-90 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride RERF-LC-MS CTRP2 0.0020 66.0000
PF-4800567 hydrochloride RPMI-6666 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-N-MC CTRP2 0.0020 66.0000
PF-4800567 hydrochloride A-253 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BC-3C CTRP2 0.0020 66.0000
PF-4800567 hydrochloride C32[HUMANMELANOMA] CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CAL-85-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COLO684 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS746.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HSC-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HT-144 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride VMRC-RCZ CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MES-SA CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1105 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H322 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OAW42 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PSN1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride T24 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TE441.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TT2609-C02 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CAKI-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COR-L105 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DMS273 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride ESS-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride G-402 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HOS CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS294T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHH-6 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MFE-319 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MOLP-8 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1339 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OV7 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PANC03.27 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PLC-PRF-5 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SCC-9 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-LMS-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-MEL-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHH-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HLF CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHH-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OAW28 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OV56 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PANC02.03 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-475 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride 647V CTRP2 0.0020 66.0000
PF-4800567 hydrochloride 8-MG-BA CTRP2 0.0020 66.0000
PF-4800567 hydrochloride A101D CTRP2 0.0041 66.0000
PF-4800567 hydrochloride A2058 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride ASPC-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CAKI-2 CTRP2 0.0041 66.0000
PF-4800567 hydrochloride CAL-27 CTRP2 0.0041 66.0000
PF-4800567 hydrochloride COLO792 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride FTC-238 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride GMS-10 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride GOS-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HMCB CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HUH-1 CTRP2 0.0041 66.0000
PF-4800567 hydrochloride IGR-39 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride IST-MES1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride M059K CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PATU8988T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SCABER CTRP2 0.0041 66.0000
PF-4800567 hydrochloride SK-N-SH CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TM-31 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride YH-13 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride A-673 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DU145 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride FADU CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC4006 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS683 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS729.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HT-1080 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHH-5 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHUEM-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MEWO CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MIAPACA-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-MES-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-N-DZ CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SW579 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride WM115 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride WM266-4 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT-20 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CAL-54 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CAPAN-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CHP-212 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS895.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KATOIII CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KMRC-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KNS-42 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MPP89 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1693 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PANC04.03 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PE-CA-PJ49 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-MEL-24 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-N-AS CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TE617.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride YKG-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BL-70 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COR-L95 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride D283MED CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HL-60 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HUP-T3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride IMR-32 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KO52 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MEC1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H2196 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NH-6 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OCI-M1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SIG-M5 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TF-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride UACC-812 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride 786-O CTRP2 0.0020 66.0000
PF-4800567 hydrochloride A4-FUKUDA CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCT15 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HEL92.1.7 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HUNS1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JHOS-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride K-562 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1341 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1568 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1703 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H838 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TE-11 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DAUDI CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HH[HUMANLYMPHOMA] CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HT-1197 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LUDLU-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1915 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1944 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H520 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H522 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PE-CA-PJ41(CLONED2) CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PE-CA-PJ15 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride RVH-421 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SET-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-16 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TOV-112D CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DB CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC1419 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC-56 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS839.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H2110 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PE-CA-PJ34(CLONEC12) CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-387 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-503 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-869 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-C1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SW1990 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SW948 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TE15 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride UM-UC-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride WM88 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride WM983B CTRP2 0.0020 66.0000
PF-4800567 hydrochloride ZR-75-30 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CI-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CJM[HUMANMELANOMA] CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HUG1-N CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JEKO-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JM1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KP-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride LMSU CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MG-63 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MINO CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MJ CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MOTN-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride RL CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-MEL-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride ST486 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SUP-B15 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TC71 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BICR18 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BICR22 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BICR31 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COLO678 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EFM-192A CTRP2 0.0020 66.0000
PF-4800567 hydrochloride G-401 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS888.LU CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KP-N-YN CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1395 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-423 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SW1417 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SW1783 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride VCAP CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KE-39 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DMS454 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride GCT CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC2935 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HOP-62 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H747 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OVCAR-5 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SF268 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SF539 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TUHR14TKB CTRP2 0.5200 66.0000
PF-4800567 hydrochloride U-251MG CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DMS53 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HEC-1-A CTRP2 0.0020 66.0000
PF-4800567 hydrochloride IGR-37 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KNS-62 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MDA-MB-157 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1563 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OC314 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride UO-31 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BICR56 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CAL-33 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CALU-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride CAPAN-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DMS114 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride EKVX CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC1438 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCT8 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HOP-92 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KYM-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KYSE-30 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KYSE-510 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride L-428 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MDA-MB-361 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MFE-296 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NU-DHL-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNB-75 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-216 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BICR16 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride F-36P CTRP2 0.0020 66.0000
PF-4800567 hydrochloride JJN-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KASUMI-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KG-1-C CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KMS-20 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KYSE-150 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride OCI-AML-5 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PANC08.13 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-601 CTRP2 0.5200 66.0000
PF-4800567 hydrochloride SNU-C4 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride T-47D CTRP2 0.0020 66.0000
PF-4800567 hydrochloride T84 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TE-14 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride U266B1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride 42-MG-BA CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT139 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT159 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT228 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT231 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT239 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT-474 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COV434 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride DND-41 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride G-292CLONEA141B1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HCC2218 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS766T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KMRC-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1651 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-BR-3 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SNU-1033 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride A-204 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride AML-193 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HGC-27 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS578BST CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS934.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS688(A).T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HUT78 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1793 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SCC-4 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-ES-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS888.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MDA-MB-453 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H660 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SAOS-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride U-BLC1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT248 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride NCI-H1694 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SEM CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS822.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride HS940.T CTRP2 0.0020 66.0000
PF-4800567 hydrochloride KMBC-2 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride RCC10RGB CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SK-N-BE(2) CTRP2 0.0020 66.0000
PF-4800567 hydrochloride AU565 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride COLO320 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride MDA-MB-415 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride PANC10.05 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT131 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT147 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT172 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT216 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT232 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT245 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT271 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT286 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT320 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT328 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT330 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT333 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT340 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT359 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT416 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT422 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT428 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT440 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT444 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT482 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT498 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT504 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride 2004 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride ASKA-SS CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT-12 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride BT-16 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SW982 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride SYO-1 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TM87-16 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride TTC-709 CTRP2 0.0020 66.0000
PF-4800567 hydrochloride YAMATO-SS CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.