Drug : O-6-Benzylguanine

CTRP2 Name : O-6-benzylguanine

Dataset : All
Synonyms :
Targets : MGMT
Pathways : inhibitor of O(6)-alkylguanine DNA alkyltransferases

Information Cards

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Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
O-6-benzylguanine C2BBE1 CTRP2 0.0020 66.0000
O-6-benzylguanine CHAGO-K-1 CTRP2 0.0020 66.0000
O-6-benzylguanine COLO668 CTRP2 0.0020 66.0000
O-6-benzylguanine COV362 CTRP2 0.0020 66.0000
O-6-benzylguanine DV-90 CTRP2 0.0020 66.0000
O-6-benzylguanine EFO-27 CTRP2 0.0020 66.0000
O-6-benzylguanine HD-MY-Z CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H2170 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H647 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H810 CTRP2 0.0020 66.0000
O-6-benzylguanine OCI-AML-3 CTRP2 0.0020 66.0000
O-6-benzylguanine PATU8988S CTRP2 0.0020 66.0000
O-6-benzylguanine MIAPACA-3 CTRP2 0.0020 66.0000
O-6-benzylguanine TE-5 CTRP2 0.0020 66.0000
O-6-benzylguanine UACC-257 CTRP2 0.0020 66.0000
O-6-benzylguanine UACC-62 CTRP2 0.0020 66.0000
O-6-benzylguanine BICR6 CTRP2 0.0020 66.0000
O-6-benzylguanine BT145 CTRP2 0.0020 66.0000
O-6-benzylguanine BT179 CTRP2 0.0020 66.0000
O-6-benzylguanine EC-GI-10 CTRP2 0.0020 66.0000
O-6-benzylguanine EFO-21 CTRP2 0.0020 66.0000
O-6-benzylguanine FTC-133 CTRP2 0.0020 66.0000
O-6-benzylguanine JHUEM-3 CTRP2 0.0020 66.0000
O-6-benzylguanine LK2 CTRP2 0.0020 66.0000
O-6-benzylguanine LNCAPCLONEFGC CTRP2 0.0020 66.0000
O-6-benzylguanine LS1034 CTRP2 0.0020 66.0000
O-6-benzylguanine MKN7 CTRP2 0.0020 66.0000
O-6-benzylguanine HCC1428 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H2029 CTRP2 0.0020 66.0000
O-6-benzylguanine OE21 CTRP2 0.0020 66.0000
O-6-benzylguanine MKN74 CTRP2 0.0020 66.0000
O-6-benzylguanine SH-10-TC CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-449 CTRP2 0.0020 66.0000
O-6-benzylguanine T3M-10 CTRP2 0.0020 66.0000
O-6-benzylguanine BT112 CTRP2 0.0020 66.0000
O-6-benzylguanine BT164 CTRP2 0.0020 66.0000
O-6-benzylguanine CCF-STTG1 CTRP2 0.0020 66.0000
O-6-benzylguanine COLO800 CTRP2 0.0020 66.0000
O-6-benzylguanine DK-MG CTRP2 0.0020 66.0000
O-6-benzylguanine GP2D CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1869 CTRP2 0.0020 66.0000
O-6-benzylguanine HCC38 CTRP2 0.0020 66.0000
O-6-benzylguanine JHOM-1 CTRP2 0.0020 66.0000
O-6-benzylguanine JHUEM-7 CTRP2 0.0020 66.0000
O-6-benzylguanine JL-1 CTRP2 0.0020 66.0000
O-6-benzylguanine KYSE-450 CTRP2 0.0020 66.0000
O-6-benzylguanine LC-1-SQ-SF CTRP2 0.0020 66.0000
O-6-benzylguanine RCM-1[HUMANESC] CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-685 CTRP2 0.0020 66.0000
O-6-benzylguanine VMRC-LCD CTRP2 0.0020 66.0000
O-6-benzylguanine BT224 CTRP2 0.0020 66.0000
O-6-benzylguanine BT-549 CTRP2 0.0020 66.0000
O-6-benzylguanine HELA CTRP2 0.0020 66.0000
O-6-benzylguanine HCC202 CTRP2 0.0020 66.0000
O-6-benzylguanine H-STS CTRP2 0.0020 66.0000
O-6-benzylguanine K029AX CTRP2 0.0020 66.0000
O-6-benzylguanine KYSE-520 CTRP2 0.0020 66.0000
O-6-benzylguanine LOX-IMVI CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1623 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H716 CTRP2 0.0020 66.0000
O-6-benzylguanine OE19 CTRP2 0.0020 66.0000
O-6-benzylguanine OE33 CTRP2 0.0020 66.0000
O-6-benzylguanine N2A-PK1 CTRP2 0.0020 66.0000
O-6-benzylguanine PK-45H CTRP2 0.0020 66.0000
O-6-benzylguanine P-STS CTRP2 0.0020 66.0000
O-6-benzylguanine RERF-LC-AD2 CTRP2 0.0020 66.0000
O-6-benzylguanine U-CH1 CTRP2 0.0020 66.0000
O-6-benzylguanine 697 CTRP2 0.0020 66.0000
O-6-benzylguanine CA46 CTRP2 0.0020 66.0000
O-6-benzylguanine NAMALWA CTRP2 0.0020 66.0000
O-6-benzylguanine TOLEDO CTRP2 0.0020 66.0000
O-6-benzylguanine COLO829 CTRP2 0.0020 66.0000
O-6-benzylguanine DAN-G CTRP2 0.0020 66.0000
O-6-benzylguanine EJM CTRP2 0.0020 66.0000
O-6-benzylguanine GRANTA-519 CTRP2 0.0020 66.0000
O-6-benzylguanine HCC1500 CTRP2 0.0020 66.0000
O-6-benzylguanine IGR-1 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H841 CTRP2 0.0020 66.0000
O-6-benzylguanine OCI-LY19 CTRP2 0.0020 66.0000
O-6-benzylguanine OCI-LY3 CTRP2 0.0020 66.0000
O-6-benzylguanine U-118MG CTRP2 0.0020 66.0000
O-6-benzylguanine LU-65 CTRP2 0.0020 66.0000
O-6-benzylguanine A-172 CTRP2 0.0020 66.0000
O-6-benzylguanine COV644 CTRP2 0.0020 66.0000
O-6-benzylguanine IM95 CTRP2 0.0020 66.0000
O-6-benzylguanine J82 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H23 CTRP2 0.0020 66.0000
O-6-benzylguanine RD CTRP2 0.0020 66.0000
O-6-benzylguanine SK-UT-1 CTRP2 0.0020 66.0000
O-6-benzylguanine T98G CTRP2 0.0020 66.0000
O-6-benzylguanine BECKER CTRP2 0.0020 66.0000
O-6-benzylguanine HS611.T CTRP2 0.0020 66.0000
O-6-benzylguanine JHH-4 CTRP2 0.0020 66.0000
O-6-benzylguanine KARPAS-422 CTRP2 0.0020 66.0000
O-6-benzylguanine KMRC-1 CTRP2 0.0020 66.0000
O-6-benzylguanine LP-1 CTRP2 0.0020 66.0000
O-6-benzylguanine SH4 CTRP2 0.0041 66.0000
O-6-benzylguanine SK-HEP-1 CTRP2 0.0020 66.0000
O-6-benzylguanine SUP-HD1 CTRP2 0.0020 66.0000
O-6-benzylguanine AN3-CA CTRP2 0.0020 66.0000
O-6-benzylguanine ACHN CTRP2 0.0020 66.0000
O-6-benzylguanine CMK CTRP2 0.0020 66.0000
O-6-benzylguanine EN CTRP2 0.0020 66.0000
O-6-benzylguanine KASUMI-1 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H2342 CTRP2 0.0020 66.0000
O-6-benzylguanine OV-90 CTRP2 0.0020 66.0000
O-6-benzylguanine RERF-LC-MS CTRP2 0.0020 66.0000
O-6-benzylguanine RPMI-6666 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-N-MC CTRP2 0.0020 66.0000
O-6-benzylguanine A-253 CTRP2 0.0020 66.0000
O-6-benzylguanine BC-3C CTRP2 0.0020 66.0000
O-6-benzylguanine C32[HUMANMELANOMA] CTRP2 0.0020 66.0000
O-6-benzylguanine CAL-85-1 CTRP2 0.0020 66.0000
O-6-benzylguanine COLO684 CTRP2 0.0020 66.0000
O-6-benzylguanine HS746.T CTRP2 0.0020 66.0000
O-6-benzylguanine HSC-2 CTRP2 0.0020 66.0000
O-6-benzylguanine HT-144 CTRP2 0.0020 66.0000
O-6-benzylguanine VMRC-RCZ CTRP2 0.0020 66.0000
O-6-benzylguanine MES-SA CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1105 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H322 CTRP2 0.0020 66.0000
O-6-benzylguanine OAW42 CTRP2 0.0020 66.0000
O-6-benzylguanine PSN1 CTRP2 0.0020 66.0000
O-6-benzylguanine T24 CTRP2 0.0020 66.0000
O-6-benzylguanine TE441.T CTRP2 0.0020 66.0000
O-6-benzylguanine TT2609-C02 CTRP2 0.0020 66.0000
O-6-benzylguanine CAKI-1 CTRP2 0.0020 66.0000
O-6-benzylguanine COR-L105 CTRP2 0.0020 66.0000
O-6-benzylguanine DMS273 CTRP2 0.0020 66.0000
O-6-benzylguanine ESS-1 CTRP2 0.0020 66.0000
O-6-benzylguanine G-402 CTRP2 0.0020 66.0000
O-6-benzylguanine HOS CTRP2 0.0020 66.0000
O-6-benzylguanine HS294T CTRP2 0.0020 66.0000
O-6-benzylguanine JHH-6 CTRP2 0.0020 66.0000
O-6-benzylguanine MFE-319 CTRP2 0.0020 66.0000
O-6-benzylguanine MOLP-8 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1339 CTRP2 0.0020 66.0000
O-6-benzylguanine OV7 CTRP2 0.0020 66.0000
O-6-benzylguanine PANC03.27 CTRP2 0.0020 66.0000
O-6-benzylguanine PLC-PRF-5 CTRP2 0.0020 66.0000
O-6-benzylguanine SCC-9 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-LMS-1 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-MEL-2 CTRP2 0.0020 66.0000
O-6-benzylguanine JHH-2 CTRP2 0.0020 66.0000
O-6-benzylguanine HLF CTRP2 0.0020 66.0000
O-6-benzylguanine JHH-1 CTRP2 0.0020 66.0000
O-6-benzylguanine OAW28 CTRP2 0.0020 66.0000
O-6-benzylguanine OV56 CTRP2 0.0020 66.0000
O-6-benzylguanine PANC02.03 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-475 CTRP2 0.0020 66.0000
O-6-benzylguanine TOV-21G CTRP2 0.0020 66.0000
O-6-benzylguanine 647V CTRP2 0.0020 66.0000
O-6-benzylguanine 8-MG-BA CTRP2 0.0020 66.0000
O-6-benzylguanine A101D CTRP2 0.0020 66.0000
O-6-benzylguanine A2058 CTRP2 0.0020 66.0000
O-6-benzylguanine ASPC-1 CTRP2 0.0020 66.0000
O-6-benzylguanine CAKI-2 CTRP2 0.0020 66.0000
O-6-benzylguanine CAL-27 CTRP2 0.0020 66.0000
O-6-benzylguanine COLO792 CTRP2 0.0020 66.0000
O-6-benzylguanine FTC-238 CTRP2 0.0020 66.0000
O-6-benzylguanine GMS-10 CTRP2 0.0020 66.0000
O-6-benzylguanine GOS-3 CTRP2 0.0020 66.0000
O-6-benzylguanine HMCB CTRP2 0.0020 66.0000
O-6-benzylguanine HUH-1 CTRP2 0.0020 66.0000
O-6-benzylguanine IGR-39 CTRP2 0.0020 66.0000
O-6-benzylguanine IST-MES1 CTRP2 0.0020 66.0000
O-6-benzylguanine M059K CTRP2 0.0020 66.0000
O-6-benzylguanine PATU8988T CTRP2 0.0020 66.0000
O-6-benzylguanine SCABER CTRP2 0.0020 66.0000
O-6-benzylguanine SK-N-SH CTRP2 0.0020 66.0000
O-6-benzylguanine TM-31 CTRP2 0.0020 66.0000
O-6-benzylguanine YH-13 CTRP2 0.0020 66.0000
O-6-benzylguanine A-673 CTRP2 0.0020 66.0000
O-6-benzylguanine DU145 CTRP2 0.0020 66.0000
O-6-benzylguanine FADU CTRP2 0.0020 66.0000
O-6-benzylguanine HCC4006 CTRP2 0.0020 66.0000
O-6-benzylguanine HS683 CTRP2 0.0020 66.0000
O-6-benzylguanine HS729.T CTRP2 0.0020 66.0000
O-6-benzylguanine HT-1080 CTRP2 0.0020 66.0000
O-6-benzylguanine JHH-5 CTRP2 0.0020 66.0000
O-6-benzylguanine JHUEM-1 CTRP2 0.0020 66.0000
O-6-benzylguanine MEWO CTRP2 0.0020 66.0000
O-6-benzylguanine MIAPACA-2 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-MES-1 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-N-DZ CTRP2 0.0020 66.0000
O-6-benzylguanine SW579 CTRP2 0.0020 66.0000
O-6-benzylguanine WM115 CTRP2 0.0020 66.0000
O-6-benzylguanine WM266-4 CTRP2 0.0020 66.0000
O-6-benzylguanine BT-20 CTRP2 0.0020 66.0000
O-6-benzylguanine CAL-54 CTRP2 0.0020 66.0000
O-6-benzylguanine CAPAN-1 CTRP2 0.0020 66.0000
O-6-benzylguanine CHP-212 CTRP2 0.0020 66.0000
O-6-benzylguanine HS895.T CTRP2 0.0020 66.0000
O-6-benzylguanine KATOIII CTRP2 0.0020 66.0000
O-6-benzylguanine KMRC-2 CTRP2 0.0020 66.0000
O-6-benzylguanine KNS-42 CTRP2 0.0020 66.0000
O-6-benzylguanine MPP89 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1693 CTRP2 0.0020 66.0000
O-6-benzylguanine PANC04.03 CTRP2 0.0020 66.0000
O-6-benzylguanine PE-CA-PJ49 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-MEL-24 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-N-AS CTRP2 0.0020 66.0000
O-6-benzylguanine TE617.T CTRP2 0.0020 66.0000
O-6-benzylguanine YKG-1 CTRP2 0.0020 66.0000
O-6-benzylguanine BL-70 CTRP2 0.0020 66.0000
O-6-benzylguanine COR-L95 CTRP2 0.0020 66.0000
O-6-benzylguanine D283MED CTRP2 0.0020 66.0000
O-6-benzylguanine HL-60 CTRP2 0.0020 66.0000
O-6-benzylguanine HUP-T3 CTRP2 0.0020 66.0000
O-6-benzylguanine IMR-32 CTRP2 0.0020 66.0000
O-6-benzylguanine KO52 CTRP2 0.0020 66.0000
O-6-benzylguanine MEC1 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1092 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H2171 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H2196 CTRP2 0.0020 66.0000
O-6-benzylguanine NH-6 CTRP2 0.0020 66.0000
O-6-benzylguanine OCI-M1 CTRP2 0.0020 66.0000
O-6-benzylguanine SIG-M5 CTRP2 0.0020 66.0000
O-6-benzylguanine TF-1 CTRP2 0.0020 66.0000
O-6-benzylguanine UACC-812 CTRP2 0.0020 66.0000
O-6-benzylguanine 786-O CTRP2 0.0020 66.0000
O-6-benzylguanine A4-FUKUDA CTRP2 0.0020 66.0000
O-6-benzylguanine HCT15 CTRP2 0.0020 66.0000
O-6-benzylguanine HEL92.1.7 CTRP2 0.0020 66.0000
O-6-benzylguanine HUNS1 CTRP2 0.0020 66.0000
O-6-benzylguanine JHOS-2 CTRP2 0.0020 66.0000
O-6-benzylguanine K-562 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1341 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1568 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1703 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H838 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-N-FI CTRP2 0.0020 66.0000
O-6-benzylguanine TE-11 CTRP2 0.0020 66.0000
O-6-benzylguanine BDCM CTRP2 0.0020 66.0000
O-6-benzylguanine DAUDI CTRP2 0.0020 66.0000
O-6-benzylguanine HH[HUMANLYMPHOMA] CTRP2 0.0020 66.0000
O-6-benzylguanine HT-1197 CTRP2 0.0020 0.2600
O-6-benzylguanine LUDLU-1 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H146 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1915 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1944 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H520 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H522 CTRP2 0.0020 66.0000
O-6-benzylguanine PE-CA-PJ41(CLONED2) CTRP2 0.0020 66.0000
O-6-benzylguanine PE-CA-PJ15 CTRP2 0.0020 66.0000
O-6-benzylguanine RVH-421 CTRP2 0.0020 66.0000
O-6-benzylguanine SET-2 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-16 CTRP2 0.0020 66.0000
O-6-benzylguanine TOV-112D CTRP2 0.0020 66.0000
O-6-benzylguanine DB CTRP2 0.0020 66.0000
O-6-benzylguanine HCC1419 CTRP2 0.0020 66.0000
O-6-benzylguanine HCC-56 CTRP2 0.0020 66.0000
O-6-benzylguanine HS839.T CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H2110 CTRP2 0.0020 66.0000
O-6-benzylguanine PE-CA-PJ34(CLONEC12) CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-387 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-503 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-869 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-C1 CTRP2 0.0020 66.0000
O-6-benzylguanine SW1990 CTRP2 0.0020 66.0000
O-6-benzylguanine SW948 CTRP2 0.0020 66.0000
O-6-benzylguanine TE15 CTRP2 0.0020 66.0000
O-6-benzylguanine UM-UC-1 CTRP2 0.0020 66.0000
O-6-benzylguanine WM88 CTRP2 0.0020 66.0000
O-6-benzylguanine WM983B CTRP2 0.0020 66.0000
O-6-benzylguanine ZR-75-30 CTRP2 0.0020 66.0000
O-6-benzylguanine CI-1 CTRP2 0.0020 66.0000
O-6-benzylguanine CJM[HUMANMELANOMA] CTRP2 0.0020 66.0000
O-6-benzylguanine HUG1-N CTRP2 0.0020 66.0000
O-6-benzylguanine JEKO-1 CTRP2 0.0020 66.0000
O-6-benzylguanine JM1 CTRP2 0.0020 66.0000
O-6-benzylguanine KP-2 CTRP2 0.0020 66.0000
O-6-benzylguanine LMSU CTRP2 0.0020 66.0000
O-6-benzylguanine MG-63 CTRP2 0.0020 66.0000
O-6-benzylguanine MINO CTRP2 0.0020 66.0000
O-6-benzylguanine MJ CTRP2 0.0020 66.0000
O-6-benzylguanine MOTN-1 CTRP2 0.0020 66.0000
O-6-benzylguanine RL CTRP2 0.0020 66.0000
O-6-benzylguanine SK-MEL-3 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-1 CTRP2 0.0020 66.0000
O-6-benzylguanine ST486 CTRP2 0.0020 66.0000
O-6-benzylguanine SUP-B15 CTRP2 0.0020 66.0000
O-6-benzylguanine TC71 CTRP2 0.0020 66.0000
O-6-benzylguanine BICR18 CTRP2 0.0020 66.0000
O-6-benzylguanine BICR22 CTRP2 0.0020 66.0000
O-6-benzylguanine BICR31 CTRP2 0.0020 66.0000
O-6-benzylguanine COLO678 CTRP2 0.0020 66.0000
O-6-benzylguanine G-401 CTRP2 0.0020 66.0000
O-6-benzylguanine HS888.LU CTRP2 0.0020 66.0000
O-6-benzylguanine KP-N-YN CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1395 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-423 CTRP2 0.0020 66.0000
O-6-benzylguanine SW1417 CTRP2 0.0020 66.0000
O-6-benzylguanine SW1783 CTRP2 0.0020 66.0000
O-6-benzylguanine VCAP CTRP2 0.0020 66.0000
O-6-benzylguanine KE-39 CTRP2 0.0020 66.0000
O-6-benzylguanine DMS454 CTRP2 0.0020 66.0000
O-6-benzylguanine GCT CTRP2 0.0020 66.0000
O-6-benzylguanine HCC2935 CTRP2 0.0020 66.0000
O-6-benzylguanine HOP-62 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H747 CTRP2 0.0020 66.0000
O-6-benzylguanine OVCAR-5 CTRP2 0.0020 66.0000
O-6-benzylguanine SF268 CTRP2 0.0020 66.0000
O-6-benzylguanine SF539 CTRP2 0.0020 66.0000
O-6-benzylguanine TUHR14TKB CTRP2 0.0020 66.0000
O-6-benzylguanine U-251MG CTRP2 0.0020 66.0000
O-6-benzylguanine DMS53 CTRP2 0.0020 66.0000
O-6-benzylguanine HEC-1-A CTRP2 0.0020 66.0000
O-6-benzylguanine IGR-37 CTRP2 0.0020 66.0000
O-6-benzylguanine KNS-62 CTRP2 0.0020 66.0000
O-6-benzylguanine MDA-MB-157 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1563 CTRP2 0.0020 66.0000
O-6-benzylguanine OC314 CTRP2 0.0020 66.0000
O-6-benzylguanine UO-31 CTRP2 0.0020 66.0000
O-6-benzylguanine BICR56 CTRP2 0.0020 66.0000
O-6-benzylguanine CAL-33 CTRP2 0.0020 66.0000
O-6-benzylguanine CALU-1 CTRP2 0.0020 66.0000
O-6-benzylguanine CAPAN-2 CTRP2 0.0020 66.0000
O-6-benzylguanine DMS114 CTRP2 0.0020 66.0000
O-6-benzylguanine EKVX CTRP2 0.0020 66.0000
O-6-benzylguanine HCC1438 CTRP2 0.0020 66.0000
O-6-benzylguanine HCT8 CTRP2 0.0020 66.0000
O-6-benzylguanine HOP-92 CTRP2 0.0020 66.0000
O-6-benzylguanine KYM-1 CTRP2 0.0020 66.0000
O-6-benzylguanine KYSE-30 CTRP2 0.0020 66.0000
O-6-benzylguanine KYSE-510 CTRP2 0.0020 66.0000
O-6-benzylguanine L-428 CTRP2 0.0020 66.0000
O-6-benzylguanine MDA-MB-361 CTRP2 0.0020 66.0000
O-6-benzylguanine MFE-296 CTRP2 0.0020 66.0000
O-6-benzylguanine NU-DHL-1 CTRP2 0.0020 66.0000
O-6-benzylguanine SNB-75 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-216 CTRP2 0.0020 66.0000
O-6-benzylguanine BICR16 CTRP2 0.0020 66.0000
O-6-benzylguanine F-36P CTRP2 0.0020 66.0000
O-6-benzylguanine JJN-3 CTRP2 0.0020 66.0000
O-6-benzylguanine KASUMI-2 CTRP2 0.0020 66.0000
O-6-benzylguanine KG-1-C CTRP2 0.0020 66.0000
O-6-benzylguanine KMS-20 CTRP2 0.0020 66.0000
O-6-benzylguanine KYSE-150 CTRP2 0.0020 66.0000
O-6-benzylguanine OCI-AML-5 CTRP2 0.0020 66.0000
O-6-benzylguanine PANC08.13 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-601 CTRP2 0.0020 66.0000
O-6-benzylguanine SNU-C4 CTRP2 0.0020 66.0000
O-6-benzylguanine T-47D CTRP2 0.0020 66.0000
O-6-benzylguanine T84 CTRP2 0.0020 66.0000
O-6-benzylguanine TE-14 CTRP2 0.0020 66.0000
O-6-benzylguanine U266B1 CTRP2 0.0020 66.0000
O-6-benzylguanine 42-MG-BA CTRP2 0.0020 66.0000
O-6-benzylguanine BT139 CTRP2 0.0020 66.0000
O-6-benzylguanine BT159 CTRP2 0.0020 66.0000
O-6-benzylguanine BT187 CTRP2 0.0020 66.0000
O-6-benzylguanine BT228 CTRP2 0.0020 66.0000
O-6-benzylguanine BT231 CTRP2 0.0020 66.0000
O-6-benzylguanine BT239 CTRP2 0.0020 66.0000
O-6-benzylguanine BT-474 CTRP2 0.0020 66.0000
O-6-benzylguanine COV434 CTRP2 0.0020 66.0000
O-6-benzylguanine DND-41 CTRP2 0.0020 66.0000
O-6-benzylguanine G-292CLONEA141B1 CTRP2 0.0020 66.0000
O-6-benzylguanine HCC2218 CTRP2 0.0020 66.0000
O-6-benzylguanine HS766T CTRP2 0.0020 66.0000
O-6-benzylguanine M-07E CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1651 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-BR-3 CTRP2 0.0020 66.0000
O-6-benzylguanine A-204 CTRP2 0.0020 66.0000
O-6-benzylguanine AML-193 CTRP2 0.0020 66.0000
O-6-benzylguanine HGC-27 CTRP2 0.0020 66.0000
O-6-benzylguanine HS578BST CTRP2 0.0020 66.0000
O-6-benzylguanine HS688(A).T CTRP2 0.0020 66.0000
O-6-benzylguanine HUT78 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1793 CTRP2 0.0020 66.0000
O-6-benzylguanine SCC-4 CTRP2 0.0020 66.0000
O-6-benzylguanine SK-ES-1 CTRP2 0.0020 66.0000
O-6-benzylguanine HS888.T CTRP2 0.0020 66.0000
O-6-benzylguanine MDA-MB-453 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H660 CTRP2 0.0020 66.0000
O-6-benzylguanine SAOS-2 CTRP2 0.0020 66.0000
O-6-benzylguanine U-BLC1 CTRP2 0.0020 66.0000
O-6-benzylguanine BT248 CTRP2 0.0020 66.0000
O-6-benzylguanine NCI-H1694 CTRP2 0.0020 66.0000
O-6-benzylguanine SEM CTRP2 0.0020 66.0000
O-6-benzylguanine HS822.T CTRP2 0.0020 66.0000
O-6-benzylguanine HS940.T CTRP2 0.0020 66.0000
O-6-benzylguanine KMBC-2 CTRP2 0.0020 66.0000
O-6-benzylguanine RCC10RGB CTRP2 0.0020 66.0000
O-6-benzylguanine SK-N-BE(2) CTRP2 0.0020 66.0000
O-6-benzylguanine AU565 CTRP2 0.0020 66.0000
O-6-benzylguanine COLO320 CTRP2 0.0020 66.0000
O-6-benzylguanine MDA-MB-415 CTRP2 0.0020 66.0000
O-6-benzylguanine PANC10.05 CTRP2 0.0020 66.0000
O-6-benzylguanine BT131 CTRP2 0.0020 66.0000
O-6-benzylguanine BT147 CTRP2 0.0020 66.0000
O-6-benzylguanine BT172 CTRP2 0.0020 66.0000
O-6-benzylguanine BT216 CTRP2 0.0020 66.0000
O-6-benzylguanine BT232 CTRP2 0.0020 66.0000
O-6-benzylguanine BT245 CTRP2 0.0020 66.0000
O-6-benzylguanine BT271 CTRP2 0.0020 66.0000
O-6-benzylguanine BT286 CTRP2 0.0020 66.0000
O-6-benzylguanine BT320 CTRP2 0.0020 66.0000
O-6-benzylguanine BT328 CTRP2 0.0020 66.0000
O-6-benzylguanine BT330 CTRP2 0.0020 66.0000
O-6-benzylguanine BT333 CTRP2 0.0020 66.0000
O-6-benzylguanine BT340 CTRP2 0.0020 66.0000
O-6-benzylguanine BT359 CTRP2 0.0020 66.0000
O-6-benzylguanine BT416 CTRP2 0.0020 66.0000
O-6-benzylguanine BT422 CTRP2 0.0020 66.0000
O-6-benzylguanine BT428 CTRP2 0.0020 66.0000
O-6-benzylguanine BT440 CTRP2 0.0020 66.0000
O-6-benzylguanine BT444 CTRP2 0.0020 66.0000
O-6-benzylguanine BT482 CTRP2 0.0020 66.0000
O-6-benzylguanine BT498 CTRP2 0.0020 66.0000
O-6-benzylguanine BT504 CTRP2 0.0020 66.0000
O-6-benzylguanine 2004 CTRP2 0.0020 66.0000
O-6-benzylguanine ASKA-SS CTRP2 0.0020 66.0000
O-6-benzylguanine BT-12 CTRP2 0.0020 66.0000
O-6-benzylguanine BT-16 CTRP2 0.0020 66.0000
O-6-benzylguanine SW982 CTRP2 0.0020 66.0000
O-6-benzylguanine SYO-1 CTRP2 0.0020 66.0000
O-6-benzylguanine TM87-16 CTRP2 0.0020 66.0000
O-6-benzylguanine TTC-709 CTRP2 0.0020 66.0000
O-6-benzylguanine YAMATO-SS CTRP2 0.0020 66.0000

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.