Drug : Bafilomycin A1

CTRP2 Name : bafilomycin A1

Dataset : All
Synonyms :
Targets : ATP6V0A1
Pathways : inhibitor of the vacuolar-type H+-ATPase

Information Cards

Click to show/hide information cards below or download all drug response information.

           
     

Information cards below will change according to the dataset selected. The default dataset is “All”, which means information in the cards is based on the integration. If “All” is not selected, information cards will contain drug response information preprocessed for each dataset independently.

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Experimental information

Experimental information from All dataset, including drug name, cell line name, and minimum and maximum dosages used in each experiment. Click on Dose-response to query more detail for each experiment.

Drug name Cellosaurus ID Original Dataset(s) Min Dose Max Dose Dose-response
bafilomycin A1 KE-39 CTRP2 0.0000 0.3300
bafilomycin A1 DMS454 CTRP2 0.0000 0.3300
bafilomycin A1 GCT CTRP2 0.0000 0.3300
bafilomycin A1 HCC2935 CTRP2 0.0000 0.3300
bafilomycin A1 HOP-62 CTRP2 0.0000 0.3300
bafilomycin A1 NCI-H747 CTRP2 0.0000 0.3300
bafilomycin A1 OVCAR-5 CTRP2 0.0000 0.3300
bafilomycin A1 SF268 CTRP2 0.0000 0.3300
bafilomycin A1 SF539 CTRP2 0.0000 0.3300
bafilomycin A1 TUHR14TKB CTRP2 0.0026 0.3300
bafilomycin A1 U-251MG CTRP2 0.0000 0.3300
bafilomycin A1 DMS53 CTRP2 0.0000 0.3300
bafilomycin A1 HEC-1-A CTRP2 0.0000 0.3300
bafilomycin A1 IGR-37 CTRP2 0.0000 0.3300
bafilomycin A1 KNS-62 CTRP2 0.0000 0.3300
bafilomycin A1 NCI-H1563 CTRP2 0.0000 0.3300
bafilomycin A1 OC314 CTRP2 0.0000 0.3300
bafilomycin A1 UO-31 CTRP2 0.0000 0.3300
bafilomycin A1 BICR56 CTRP2 0.0000 0.0013
bafilomycin A1 CAL-33 CTRP2 0.0000 0.3300
bafilomycin A1 CALU-1 CTRP2 0.0000 0.3300
bafilomycin A1 CAPAN-2 CTRP2 0.0000 0.3300
bafilomycin A1 DMS114 CTRP2 0.0000 0.3300
bafilomycin A1 EKVX CTRP2 0.0000 0.3300
bafilomycin A1 HCC1438 CTRP2 0.0000 0.3300
bafilomycin A1 HCT8 CTRP2 0.0000 0.3300
bafilomycin A1 HOP-92 CTRP2 0.0026 0.3300
bafilomycin A1 KYM-1 CTRP2 0.0000 0.3300
bafilomycin A1 KYSE-30 CTRP2 0.0000 0.3300
bafilomycin A1 KYSE-510 CTRP2 0.0000 0.3300
bafilomycin A1 L-428 CTRP2 0.0000 0.3300
bafilomycin A1 MDA-MB-361 CTRP2 0.0000 0.3300
bafilomycin A1 MFE-296 CTRP2 0.0000 0.3300
bafilomycin A1 NU-DHL-1 CTRP2 0.0000 0.3300
bafilomycin A1 SNB-75 CTRP2 0.0000 0.3300
bafilomycin A1 SNU-216 CTRP2 0.0000 0.3300
bafilomycin A1 BICR16 CTRP2 0.0000 0.3300
bafilomycin A1 F-36P CTRP2 0.0000 0.3300
bafilomycin A1 JJN-3 CTRP2 0.0000 0.3300
bafilomycin A1 KASUMI-2 CTRP2 0.0000 0.3300
bafilomycin A1 KG-1-C CTRP2 0.0000 0.3300
bafilomycin A1 KMS-20 CTRP2 0.0000 0.3300
bafilomycin A1 KYSE-150 CTRP2 0.0000 0.3300
bafilomycin A1 OCI-AML-5 CTRP2 0.0000 0.3300
bafilomycin A1 PANC08.13 CTRP2 0.0000 0.3300
bafilomycin A1 SNU-601 CTRP2 0.0026 0.3300
bafilomycin A1 SNU-C4 CTRP2 0.0000 0.3300
bafilomycin A1 T-47D CTRP2 0.0000 0.3300
bafilomycin A1 T84 CTRP2 0.0000 0.3300
bafilomycin A1 TE-14 CTRP2 0.0000 0.3300
bafilomycin A1 U266B1 CTRP2 0.0000 0.3300
bafilomycin A1 42-MG-BA CTRP2 0.0000 0.3300
bafilomycin A1 BT139 CTRP2 0.0000 0.3300
bafilomycin A1 BT159 CTRP2 0.0000 0.3300
bafilomycin A1 BT187 CTRP2 0.0000 0.3300
bafilomycin A1 BT228 CTRP2 0.0000 0.3300
bafilomycin A1 BT231 CTRP2 0.0000 0.3300
bafilomycin A1 BT239 CTRP2 0.0000 0.3300
bafilomycin A1 BT-474 CTRP2 0.0000 0.3300
bafilomycin A1 COV434 CTRP2 0.0000 0.3300
bafilomycin A1 G-292CLONEA141B1 CTRP2 0.0000 0.3300
bafilomycin A1 HS766T CTRP2 0.0000 0.3300
bafilomycin A1 KMRC-3 CTRP2 0.0000 0.3300
bafilomycin A1 M-07E CTRP2 0.0000 0.3300
bafilomycin A1 NCI-H1651 CTRP2 0.0000 0.3300
bafilomycin A1 SK-BR-3 CTRP2 0.0000 0.3300
bafilomycin A1 SNU-1033 CTRP2 0.0000 0.3300
bafilomycin A1 SNU-245 CTRP2 0.0000 0.3300
bafilomycin A1 A-204 CTRP2 0.0000 0.3300
bafilomycin A1 AML-193 CTRP2 0.0000 0.3300
bafilomycin A1 HGC-27 CTRP2 0.0000 0.3300
bafilomycin A1 HS578BST CTRP2 0.0000 0.3300
bafilomycin A1 HS688(A).T CTRP2 0.0000 0.3300
bafilomycin A1 HUT78 CTRP2 0.0000 0.3300
bafilomycin A1 NCI-H1793 CTRP2 0.0000 0.3300
bafilomycin A1 SCC-4 CTRP2 0.0000 0.3300
bafilomycin A1 SK-ES-1 CTRP2 0.0000 0.3300
bafilomycin A1 HS888.T CTRP2 0.0000 0.3300
bafilomycin A1 MDA-MB-453 CTRP2 0.0000 0.3300
bafilomycin A1 SAOS-2 CTRP2 0.0000 0.3300
bafilomycin A1 U-BLC1 CTRP2 0.0000 0.3300
bafilomycin A1 BT248 CTRP2 0.0000 0.3300
bafilomycin A1 NCI-H1694 CTRP2 0.0000 0.3300
bafilomycin A1 SEM CTRP2 0.0000 0.3300
bafilomycin A1 HS822.T CTRP2 0.0000 0.3300
bafilomycin A1 HS940.T CTRP2 0.0000 0.3300
bafilomycin A1 KMBC-2 CTRP2 0.0000 0.3300
bafilomycin A1 RCC10RGB CTRP2 0.0000 0.3300
bafilomycin A1 SK-N-BE(2) CTRP2 0.0000 0.3300
bafilomycin A1 AU565 CTRP2 0.0000 0.3300
bafilomycin A1 COLO320 CTRP2 0.0000 0.3300
bafilomycin A1 MDA-MB-415 CTRP2 0.0000 0.3300
bafilomycin A1 PANC10.05 CTRP2 0.0000 0.3300
bafilomycin A1 BT131 CTRP2 0.0000 0.3300
bafilomycin A1 BT147 CTRP2 0.0000 0.3300
bafilomycin A1 BT172 CTRP2 0.0000 0.3300
bafilomycin A1 BT216 CTRP2 0.0000 0.3300
bafilomycin A1 BT232 CTRP2 0.0000 0.3300
bafilomycin A1 BT245 CTRP2 0.0000 0.3300
bafilomycin A1 BT271 CTRP2 0.0000 0.3300
bafilomycin A1 BT286 CTRP2 0.0000 0.3300
bafilomycin A1 BT320 CTRP2 0.0000 0.3300
bafilomycin A1 BT328 CTRP2 0.0000 0.3300
bafilomycin A1 BT330 CTRP2 0.0000 0.3300
bafilomycin A1 BT333 CTRP2 0.0000 0.3300
bafilomycin A1 BT340 CTRP2 0.0000 0.3300
bafilomycin A1 BT359 CTRP2 0.0000 0.3300
bafilomycin A1 BT416 CTRP2 0.0000 0.3300
bafilomycin A1 BT422 CTRP2 0.0000 0.3300
bafilomycin A1 BT428 CTRP2 0.0000 0.3300
bafilomycin A1 BT440 CTRP2 0.0000 0.3300
bafilomycin A1 BT444 CTRP2 0.0000 0.3300
bafilomycin A1 BT482 CTRP2 0.0000 0.3300
bafilomycin A1 BT504 CTRP2 0.0000 0.3300
bafilomycin A1 2004 CTRP2 0.0000 0.3300
bafilomycin A1 ASKA-SS CTRP2 0.0000 0.3300
bafilomycin A1 BT-12 CTRP2 0.0000 0.3300
bafilomycin A1 BT-16 CTRP2 0.0000 0.3300
bafilomycin A1 SW982 CTRP2 0.0000 0.3300
bafilomycin A1 SYO-1 CTRP2 0.0000 0.3300
bafilomycin A1 TM87-16 CTRP2 0.0000 0.3300
bafilomycin A1 TTC-709 CTRP2 0.0000 0.3300
bafilomycin A1 YAMATO-SS CTRP2 0.0000 0.3300

IC50

IC50 indicates how much drug dosage is needed to inhibit the cells by 50%, in vitro, compared to the control well.

Cell lines with highest and lowest IC50

IC90

IC90 indicates how much drug dosage is needed to inhibit the cells by 90%, in vitro, compared to the control well.

Cell lines with highest and lowest IC90

AUC

AUC represents the area under a dose-response curve, where 0% indicates no activity and 100% indicates that a drug completely inhibits the cells across testing dosages.

Cell lines with highest and lowest AUC

Associated Genes (Mutation)

Genes with the largest and lowest Racksum’s effect sizes, calculated by comparing IC50 between the mutant and wide type cell lines using cell lines from pancan data.

Associated Genes (Gene Expression)

Genes with the highest and lowest Spearman correlations, calculated by comparing gene expression and IC50 across cell lines from pancan data.